Affinity DataKi: 0.195nMAssay Description:Binding affinity towards rat cortical H3 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 0.490nMAssay Description:Binding affinity for human recombinant H3 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 0.501nMAssay Description:Binding affinity towards Histamine H3 receptor of rat cortical membranes.More data for this Ligand-Target Pair
Affinity DataKi: 0.603nMAssay Description:Binding affinity for human recombinant H3 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 0.676nMAssay Description:Binding affinity at human cloned Histamine H3 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 0.692nMAssay Description:Binding affinity for human recombinant H3 receptorMore data for this Ligand-Target Pair
TargetMelanin-concentrating hormone receptor 1(Homo sapiens (Human))
Neurocrine Biosciences
Curated by ChEMBL
Neurocrine Biosciences
Curated by ChEMBL
Affinity DataKi: 0.700nMAssay Description:Binding affinity to MCHR1 by competitive binding assayMore data for this Ligand-Target Pair
Affinity DataKi: 0.776nMAssay Description:Binding affinity for human recombinant H3 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 0.776nMAssay Description:Binding affinity for human recombinant H3 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 0.851nMAssay Description:Binding affinity for human recombinant H3 receptorMore data for this Ligand-Target Pair
TargetMelanin-concentrating hormone receptor 1(Homo sapiens (Human))
Neurocrine Biosciences
Curated by ChEMBL
Neurocrine Biosciences
Curated by ChEMBL
Affinity DataKi: 0.900nMAssay Description:Binding affinity to MCHR1 by competitive binding assayMore data for this Ligand-Target Pair
Affinity DataKi: 0.977nMAssay Description:Binding affinity for human recombinant H3 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 1nMAssay Description:Binding affinity towards rat cortical H3 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 1.10nMAssay Description:Binding affinity for human recombinant H3 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 1.20nMAssay Description:Binding affinity towards Histamine H3 receptor of rat cortical membranes.More data for this Ligand-Target Pair
Affinity DataKi: 1.30nMAssay Description:Binding affinity towards Histamine H3 receptor of rat cortical membranes.More data for this Ligand-Target Pair
Affinity DataKi: 1.30nMAssay Description:Binding affinity towards Histamine H3 receptor of rat cortical membranes.More data for this Ligand-Target Pair
Affinity DataKi: 1.40nMAssay Description:Binding affinity for the rat cortical Histamine H3 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 1.60nMAssay Description:Binding affinity against rat histamine H3 receptorMore data for this Ligand-Target Pair
TargetMelanin-concentrating hormone receptor 1(Homo sapiens (Human))
Neurocrine Biosciences
Curated by ChEMBL
Neurocrine Biosciences
Curated by ChEMBL
Affinity DataKi: 1.60nMAssay Description:Binding affinity to MCHR1 by competitive binding assayMore data for this Ligand-Target Pair
Affinity DataKi: 1.70nMAssay Description:Binding affinity towards rat cortical H3 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 1.70nMAssay Description:Binding affinity at human cloned Histamine H3 receptorMore data for this Ligand-Target Pair
TargetMelanin-concentrating hormone receptor 1(Homo sapiens (Human))
Neurocrine Biosciences
Curated by ChEMBL
Neurocrine Biosciences
Curated by ChEMBL
Affinity DataKi: 1.90nMAssay Description:Binding affinity to MCHR1 by competitive binding assayMore data for this Ligand-Target Pair
Affinity DataKi: 1.90nMAssay Description:Binding affinity towards Histamine H3 receptor of rat cortical membranes.More data for this Ligand-Target Pair
Affinity DataKi: 1.90nMAssay Description:Binding affinity towards Histamine H3 receptor of rat cortical membranes.More data for this Ligand-Target Pair
Affinity DataKi: 1.95nMAssay Description:Binding affinity towards Histamine H3 receptor of rat cortical membranes.More data for this Ligand-Target Pair
Affinity DataKi: 2nMAssay Description:Binding affinity of the compound towards rats Histamine type 3 (H3) receptorMore data for this Ligand-Target Pair
Affinity DataKi: 2nMAssay Description:Binding affinity towards rat cortical H3 receptorMore data for this Ligand-Target Pair
TargetMelanin-concentrating hormone receptor 1(Homo sapiens (Human))
Neurocrine Biosciences
Curated by ChEMBL
Neurocrine Biosciences
Curated by ChEMBL
Affinity DataKi: 2nMAssay Description:Binding affinity to MCHR1 by competitive binding assayMore data for this Ligand-Target Pair
TargetMelanin-concentrating hormone receptor 1(Homo sapiens (Human))
Neurocrine Biosciences
Curated by ChEMBL
Neurocrine Biosciences
Curated by ChEMBL
Affinity DataKi: 2nMAssay Description:Binding affinity to MCHR1 by competitive binding assayMore data for this Ligand-Target Pair
Affinity DataKi: 2.10nMAssay Description:Binding affinity for human recombinant H3 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 2.10nMAssay Description:Binding affinity for human recombinant H3 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 2.10nMAssay Description:Binding affinity for human recombinant H3 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 2.10nMAssay Description:Binding affinity at human cloned Histamine H3 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 2.10nMAssay Description:Binding affinity for the rat cortical Histamine H3 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 2.10nMAssay Description:Binding affinity towards Histamine H3 receptor of rat cortical membranes.More data for this Ligand-Target Pair
TargetMelanin-concentrating hormone receptor 1(Homo sapiens (Human))
Neurocrine Biosciences
Curated by ChEMBL
Neurocrine Biosciences
Curated by ChEMBL
Affinity DataKi: 2.20nMAssay Description:Binding affinity to MCHR1 by competitive binding assayMore data for this Ligand-Target Pair
Affinity DataKi: 2.30nMAssay Description:Binding affinity towards Histamine H3 receptor of rat cortical membranes.More data for this Ligand-Target Pair
Affinity DataKi: 2.40nMAssay Description:Binding affinity towards Histamine H3 receptor of rat cortical membranes.More data for this Ligand-Target Pair
Affinity DataKi: 2.40nMAssay Description:Binding affinity for human recombinant H3 receptorMore data for this Ligand-Target Pair
TargetMelanin-concentrating hormone receptor 1(Homo sapiens (Human))
Neurocrine Biosciences
Curated by ChEMBL
Neurocrine Biosciences
Curated by ChEMBL
Affinity DataKi: 2.40nMAssay Description:Binding affinity to MCHR1 by competitive binding assayMore data for this Ligand-Target Pair
Affinity DataKi: 2.5nMAssay Description:Binding affinity towards Histamine H3 receptor of rat cortical membranes.More data for this Ligand-Target Pair
Affinity DataKi: 2.70nMAssay Description:Binding affinity against rat histamine H3 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 2.70nMAssay Description:Binding affinity against rat histamine H3 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 2.80nMAssay Description:Binding affinity towards rat cortical H3 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 2.80nMAssay Description:Binding affinity at human cloned Histamine H3 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 2.80nMAssay Description:Binding affinity towards rat cortical H3 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 2.80nMAssay Description:Binding affinity against rat histamine H3 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 2.90nMAssay Description:Binding affinity against rat histamine H3 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 2.90nMAssay Description:Binding affinity for human recombinant H3 receptorMore data for this Ligand-Target Pair