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Found 170 with Last Name = 'ho' and Initial = 'wb'
TargetBone morphogenetic protein 1(Homo sapiens (Human))
Fibrogen

Curated by ChEMBL
LigandPNGBDBM50402510(CHEMBL2204087)
Affinity DataIC50:  10nMAssay Description:Inhibition of PCP after 1 hr by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBone morphogenetic protein 1(Homo sapiens (Human))
Fibrogen

Curated by ChEMBL
LigandPNGBDBM50402514(CHEMBL2204088)
Affinity DataIC50:  30nMAssay Description:Inhibition of PCP after 1 hr by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor ionotropic, NMDA 1(RAT)
Emory University

Curated by ChEMBL
LigandPNGBDBM50253203((S)-1-(4-Methanesulfonamidophenoxy)-3-(N-(2-bromob...)
Affinity DataIC50:  38nMAssay Description:Inhibition of rat recombinant NR1/NR2B receptor expressed in Xenopus oocytes assessed as inhibition of glutamate and glycine-induced evoked current b...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBone morphogenetic protein 1(Homo sapiens (Human))
Fibrogen

Curated by ChEMBL
LigandPNGBDBM50402519(CHEMBL2204817)
Affinity DataIC50:  42nMAssay Description:Inhibition of PCP after 1 hr by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor ionotropic, NMDA 1(RAT)
Emory University

Curated by ChEMBL
LigandPNGBDBM50252672((S)-1-(4-Methanesulfonamidephenoxy)-3-(3,4-dichlor...)
Affinity DataIC50:  50nMAssay Description:Inhibition of rat recombinant NR1/NR2B receptor expressed in Xenopus oocytes assessed as inhibition of glutamate and glycine-induced evoked current b...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMatrix metalloproteinase-9(Homo sapiens (Human))
Fibrogen

Curated by ChEMBL
LigandPNGBDBM13104(2-{[(4-chlorophenyl)methyl](4-methoxybenzene)sulfo...)
Affinity DataIC50:  50nMAssay Description:Inhibition of para-amino phenylmercuric acetate-activated MMP9 using Mca-P-L-G-L-Dap(Dnp)-A-R-NH2 as substrate after 1 hr by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor ionotropic, NMDA 1(RAT)
Emory University

Curated by ChEMBL
LigandPNGBDBM50253241((S)-1-(4-Methanesulfonamidophenoxy)-3-(N-(2,3,4-tr...)
Affinity DataIC50:  51nMAssay Description:Inhibition of rat recombinant NR1/NR2B receptor expressed in Xenopus oocytes assessed as inhibition of glutamate and glycine-induced evoked current b...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBone morphogenetic protein 1(Homo sapiens (Human))
Fibrogen

Curated by ChEMBL
LigandPNGBDBM50402513(CHEMBL2204089)
Affinity DataIC50:  60nMAssay Description:Inhibition of PCP after 1 hr by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor ionotropic, NMDA 1(RAT)
Emory University

Curated by ChEMBL
LigandPNGBDBM50252889((S)-1-(4-Methanesulfonamidophenoxy)-3-(3-fluoro-4-...)
Affinity DataIC50:  68nMAssay Description:Inhibition of rat recombinant NR1/NR2B receptor expressed in Xenopus oocytes assessed as inhibition of glutamate and glycine-induced evoked current b...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Emory University

Curated by ChEMBL
LigandPNGBDBM50253032((S)-1-(4-Methanesulfonamidophenoxy)-3-(N-butyl-3,4...)
Affinity DataIC50:  70nMAssay Description:Displacement of [3H]astemizole from human ERG expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor ionotropic, NMDA 1(RAT)
Emory University

Curated by ChEMBL
LigandPNGBDBM50252673((S)-1-(4-Methanesulfonamido-2-fluorophenoxy)-3-(3,...)
Affinity DataIC50:  72nMAssay Description:Inhibition of rat recombinant NR1/NR2B receptor expressed in Xenopus oocytes assessed as inhibition of glutamate and glycine-induced evoked current b...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBone morphogenetic protein 1(Homo sapiens (Human))
Fibrogen

Curated by ChEMBL
LigandPNGBDBM50402516(CHEMBL2204085)
Affinity DataIC50:  73nMAssay Description:Inhibition of PCP after 1 hr by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor ionotropic, NMDA 1(RAT)
Emory University

Curated by ChEMBL
LigandPNGBDBM50007674((+)-erythro 4-[2-(4-Benzyl-piperidin-1-yl)-1-hydro...)
Affinity DataIC50:  73nMAssay Description:Inhibition of rat recombinant NR1/NR2B receptor expressed in Xenopus oocytes assessed as inhibition of glutamate and glycine-induced evoked current b...More data for this Ligand-Target Pair
TargetGlutamate receptor ionotropic, NMDA 1(RAT)
Emory University

Curated by ChEMBL
LigandPNGBDBM50253204((S)-1-(4-Methanesulfonamidophenoxy)-3-(N-(2-fluoro...)
Affinity DataIC50:  80nMAssay Description:Inhibition of rat recombinant NR1/NR2B receptor expressed in Xenopus oocytes assessed as inhibition of glutamate and glycine-induced evoked current b...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBone morphogenetic protein 1(Homo sapiens (Human))
Fibrogen

Curated by ChEMBL
LigandPNGBDBM50402511(CHEMBL2204802)
Affinity DataIC50:  80nMAssay Description:Inhibition of PCP after 1 hr by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBone morphogenetic protein 1(Homo sapiens (Human))
Fibrogen

Curated by ChEMBL
LigandPNGBDBM50402521(CHEMBL2204815)
Affinity DataIC50:  93nMAssay Description:Inhibition of PCP after 1 hr by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor ionotropic, NMDA 1(RAT)
Emory University

Curated by ChEMBL
LigandPNGBDBM50253003((S)-1-(4-Methanesulfonamidophenoxy)-3-(N-ethyl-3,4...)
Affinity DataIC50:  96nMAssay Description:Inhibition of rat recombinant NR1/NR2B receptor expressed in Xenopus oocytes assessed as inhibition of glutamate and glycine-induced evoked current b...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor ionotropic, NMDA 1(RAT)
Emory University

Curated by ChEMBL
LigandPNGBDBM50252886((S)-1-(4-Methanesulfonamidophenoxy)-3-(4-chlorophe...)
Affinity DataIC50:  101nMAssay Description:Inhibition of rat recombinant NR1/NR2B receptor expressed in Xenopus oocytes assessed as inhibition of glutamate and glycine-induced evoked current b...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor ionotropic, NMDA 1(RAT)
Emory University

Curated by ChEMBL
LigandPNGBDBM50253078((S)-1-(4-Methanesulfonamidophenoxy)-3-(N-(4-hydrox...)
Affinity DataIC50:  113nMAssay Description:Inhibition of rat recombinant NR1/NR2B receptor expressed in Xenopus oocytes assessed as inhibition of glutamate and glycine-induced evoked current b...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor ionotropic, NMDA 1(RAT)
Emory University

Curated by ChEMBL
LigandPNGBDBM50253030((S)-1-(4-Methanesulfonamidophenoxy)-3-(N-(2-hydrox...)
Affinity DataIC50:  122nMAssay Description:Inhibition of rat recombinant NR1/NR2B receptor expressed in Xenopus oocytes assessed as inhibition of glutamate and glycine-induced evoked current b...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor ionotropic, NMDA 1(RAT)
Emory University

Curated by ChEMBL
LigandPNGBDBM50253002((S)-1-(4-Methanesulfonamidophenoxy)-3-(N-methyl-3,...)
Affinity DataIC50:  130nMAssay Description:Inhibition of rat recombinant NR1/NR2B receptor expressed in Xenopus oocytes assessed as inhibition of glutamate and glycine-induced evoked current b...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Emory University

Curated by ChEMBL
LigandPNGBDBM50253031((S)-1-(4-Methanesulfonamidophenoxy)3-(N-propyl-3,4...)
Affinity DataIC50:  130nMAssay Description:Displacement of [3H]astemizole from human ERG expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target72 kDa type IV collagenase(Homo sapiens (Human))
Fibrogen

Curated by ChEMBL
LigandPNGBDBM13104(2-{[(4-chlorophenyl)methyl](4-methoxybenzene)sulfo...)
Affinity DataIC50:  140nMAssay Description:Inhibition of para-amino phenylmercuric acetate-activated MMP2 using Mca-P-L-G-L-Dap(Dnp)-A-R-NH2 as substrate after 1 hr by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor ionotropic, NMDA 1(RAT)
Emory University

Curated by ChEMBL
LigandPNGBDBM50253120((S)-1-(4-Methanesulfonamidophenoxy)-3-(N-(2,4-dihy...)
Affinity DataIC50:  146nMAssay Description:Inhibition of rat recombinant NR1/NR2B receptor expressed in Xenopus oocytes assessed as inhibition of glutamate and glycine-induced evoked current b...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Emory University

Curated by ChEMBL
LigandPNGBDBM50253003((S)-1-(4-Methanesulfonamidophenoxy)-3-(N-ethyl-3,4...)
Affinity DataIC50:  170nMAssay Description:Displacement of [3H]astemizole from human ERG expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor ionotropic, NMDA 1(RAT)
Emory University

Curated by ChEMBL
LigandPNGBDBM50252846((R)-1-(4-Methanesulfonamidophenoxy)-3-(N-(2-hydrox...)
Affinity DataIC50:  173nMAssay Description:Inhibition of rat recombinant NR1/NR2B receptor expressed in Xenopus oocytes assessed as inhibition of glutamate and glycine-induced evoked current b...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor ionotropic, NMDA 1(RAT)
Emory University

Curated by ChEMBL
LigandPNGBDBM50253057((S)-1-(4-Methanesulfonamidophenoxy)-3-(N-benzyl-3,...)
Affinity DataIC50:  177nMAssay Description:Inhibition of rat recombinant NR1/NR2B receptor expressed in Xenopus oocytes assessed as inhibition of glutamate and glycine-induced evoked current b...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor ionotropic, NMDA 1(RAT)
Emory University

Curated by ChEMBL
LigandPNGBDBM50252812((R)-1-(4-Methanesulfonamidophenoxy)-3-(3,4-dichlor...)
Affinity DataIC50:  188nMAssay Description:Inhibition of rat recombinant NR1/NR2B receptor expressed in Xenopus oocytes assessed as inhibition of glutamate and glycine-induced evoked current b...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor ionotropic, NMDA 1(RAT)
Emory University

Curated by ChEMBL
LigandPNGBDBM50252999((S)-1-(4-Methanesulfonamidophenoxy)-3-(3,4-dimethy...)
Affinity DataIC50:  207nMAssay Description:Inhibition of rat recombinant NR1/NR2B receptor expressed in Xenopus oocytes assessed as inhibition of glutamate and glycine-induced evoked current b...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor ionotropic, NMDA 1(RAT)
Emory University

Curated by ChEMBL
LigandPNGBDBM50253077((S)-1-(4-Methanesulfonamidophenoxy)-3-(N-(3-hydrox...)
Affinity DataIC50:  238nMAssay Description:Inhibition of rat recombinant NR1/NR2B receptor expressed in Xenopus oocytes assessed as inhibition of glutamate and glycine-induced evoked current b...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor ionotropic, NMDA 1(RAT)
Emory University

Curated by ChEMBL
LigandPNGBDBM50253238((S)-1-(4-Methanesulfonamidophenoxy)-3-(N-(3-fluoro...)
Affinity DataIC50:  249nMAssay Description:Inhibition of rat recombinant NR1/NR2B receptor expressed in Xenopus oocytes assessed as inhibition of glutamate and glycine-induced evoked current b...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor ionotropic, NMDA 1(RAT)
Emory University

Curated by ChEMBL
LigandPNGBDBM50252813((R)-1-(4-Methanesulfonamidophenoxy)3-(N-methyl-3,4...)
Affinity DataIC50:  253nMAssay Description:Inhibition of rat recombinant NR1/NR2B receptor expressed in Xenopus oocytes assessed as inhibition of glutamate and glycine-induced evoked current b...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor ionotropic, NMDA 1(RAT)
Emory University

Curated by ChEMBL
LigandPNGBDBM50253239((S)-1-(4-Methanesulfonamidophenoxy)-3-(N-(4-fluoro...)
Affinity DataIC50:  275nMAssay Description:Inhibition of rat recombinant NR1/NR2B receptor expressed in Xenopus oocytes assessed as inhibition of glutamate and glycine-induced evoked current b...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor ionotropic, NMDA 1(RAT)
Emory University

Curated by ChEMBL
LigandPNGBDBM50252680((S)-1-(4-Methanesulfonamidophenoxy)-3-(N-(3-pridyl...)
Affinity DataIC50:  278nMAssay Description:Inhibition of rat recombinant NR1/NR2B receptor expressed in Xenopus oocytes assessed as inhibition of glutamate and glycine-induced evoked current b...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor ionotropic, NMDA 1(RAT)
Emory University

Curated by ChEMBL
LigandPNGBDBM50253240((S)-1-(4-Methanesulfonamidophenoxy)-3-(N-(2,6-difl...)
Affinity DataIC50:  281nMAssay Description:Inhibition of rat recombinant NR1/NR2B receptor expressed in Xenopus oocytes assessed as inhibition of glutamate and glycine-induced evoked current b...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBone morphogenetic protein 1(Homo sapiens (Human))
Fibrogen

Curated by ChEMBL
LigandPNGBDBM50402512(CHEMBL2204807)
Affinity DataIC50:  290nMAssay Description:Inhibition of PCP after 1 hr by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBone morphogenetic protein 1(Homo sapiens (Human))
Fibrogen

Curated by ChEMBL
LigandPNGBDBM50402515(CHEMBL2204086)
Affinity DataIC50:  300nMAssay Description:Inhibition of PCP after 1 hr by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBone morphogenetic protein 1(Homo sapiens (Human))
Fibrogen

Curated by ChEMBL
LigandPNGBDBM50402520(CHEMBL2204816)
Affinity DataIC50:  350nMAssay Description:Inhibition of PCP after 1 hr by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor ionotropic, NMDA 1(RAT)
Emory University

Curated by ChEMBL
LigandPNGBDBM50252936((S)-1-(4-Methanesulfonamidophenoxy)-3-(3,4-difluor...)
Affinity DataIC50:  357nMAssay Description:Inhibition of rat recombinant NR1/NR2B receptor expressed in Xenopus oocytes assessed as inhibition of glutamate and glycine-induced evoked current b...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor ionotropic, NMDA 1(RAT)
Emory University

Curated by ChEMBL
LigandPNGBDBM50253054((S)-1-(4-Methanesulfonamidophenoxy)-3-(N-isobutyl-...)
Affinity DataIC50:  370nMAssay Description:Inhibition of rat recombinant NR1/NR2B receptor expressed in Xenopus oocytes assessed as inhibition of glutamate and glycine-induced evoked current b...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Emory University

Curated by ChEMBL
LigandPNGBDBM50253002((S)-1-(4-Methanesulfonamidophenoxy)-3-(N-methyl-3,...)
Affinity DataIC50:  370nMAssay Description:Displacement of [3H]astemizole from human ERG expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBone morphogenetic protein 1(Homo sapiens (Human))
Fibrogen

Curated by ChEMBL
LigandPNGBDBM50402518(CHEMBL2204083)
Affinity DataIC50:  380nMAssay Description:Inhibition of PCP after 1 hr by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor ionotropic, NMDA 1(RAT)
Emory University

Curated by ChEMBL
LigandPNGBDBM50252888((S)-1-(4-Methanesulfonamidophenoxy)-3-(3-chloro-4-...)
Affinity DataIC50:  397nMAssay Description:Inhibition of rat recombinant NR1/NR2B receptor expressed in Xenopus oocytes assessed as inhibition of glutamate and glycine-induced evoked current b...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBone morphogenetic protein 1(Homo sapiens (Human))
Fibrogen

Curated by ChEMBL
LigandPNGBDBM50402532(CHEMBL2204803)
Affinity DataIC50:  400nMAssay Description:Inhibition of PCP after 1 hr by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor ionotropic, NMDA 1(RAT)
Emory University

Curated by ChEMBL
LigandPNGBDBM50252849((R)-1-(4-Methanesulfonamidophenoxy)-3-(N-(3-hydrox...)
Affinity DataIC50:  409nMAssay Description:Inhibition of rat recombinant NR1/NR2B receptor expressed in Xenopus oocytes assessed as inhibition of glutamate and glycine-induced evoked current b...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBone morphogenetic protein 1(Homo sapiens (Human))
Fibrogen

Curated by ChEMBL
LigandPNGBDBM50402530(CHEMBL2204805)
Affinity DataIC50:  410nMAssay Description:Inhibition of PCP after 1 hr by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor ionotropic, NMDA 1(RAT)
Emory University

Curated by ChEMBL
LigandPNGBDBM50253032((S)-1-(4-Methanesulfonamidophenoxy)-3-(N-butyl-3,4...)
Affinity DataIC50:  421nMAssay Description:Inhibition of rat recombinant NR1/NR2B receptor expressed in Xenopus oocytes assessed as inhibition of glutamate and glycine-induced evoked current b...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor ionotropic, NMDA 1(RAT)
Emory University

Curated by ChEMBL
LigandPNGBDBM50252674((S)-1-(4-Methanesulfonamido-3-fluorophenoxy)-3-(3,...)
Affinity DataIC50:  427nMAssay Description:Inhibition of rat recombinant NR1/NR2B receptor expressed in Xenopus oocytes assessed as inhibition of glutamate and glycine-induced evoked current b...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor ionotropic, NMDA 1(RAT)
Emory University

Curated by ChEMBL
LigandPNGBDBM50252845((S)-1-(4-Methanesulfonamidophenoxy)-3-(2-chlorophe...)
Affinity DataIC50:  429nMAssay Description:Inhibition of rat recombinant NR1/NR2B receptor expressed in Xenopus oocytes assessed as inhibition of glutamate and glycine-induced evoked current b...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Emory University

Curated by ChEMBL
LigandPNGBDBM50253057((S)-1-(4-Methanesulfonamidophenoxy)-3-(N-benzyl-3,...)
Affinity DataIC50:  430nMAssay Description:Displacement of [3H]astemizole from human ERG expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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