TargetPolycomb protein EED(Homo sapiens (Human))
Sanquan College Of Xinxiang Medical University
Curated by ChEMBL
Sanquan College Of Xinxiang Medical University
Curated by ChEMBL
Affinity DataKi: 0.300nMAssay Description:Binding affinity to GST-tagged EED (unknown origin) assessed as inhibition constant incubated for 1 hr by TR-FRET assayMore data for this Ligand-Target Pair
TargetPolycomb protein EED(Homo sapiens (Human))
Sanquan College Of Xinxiang Medical University
Curated by ChEMBL
Sanquan College Of Xinxiang Medical University
Curated by ChEMBL
Affinity DataKi: 11nMAssay Description:Binding affinity to GST-tagged EED (unknown origin) assessed as inhibition constant incubated for 1 hr by TR-FRET assayMore data for this Ligand-Target Pair
TargetPolycomb protein EED(Homo sapiens (Human))
Sanquan College Of Xinxiang Medical University
Curated by ChEMBL
Sanquan College Of Xinxiang Medical University
Curated by ChEMBL
Affinity DataIC50: 4.5nMAssay Description:Inhibition of His-tagged EED (unknown origin) incubated for 30 mins in presence of biotinylated H3K27me3 peptide (19 to 33 aa) by alpha screening com...More data for this Ligand-Target Pair
TargetPolycomb protein EED(Homo sapiens (Human))
Sanquan College Of Xinxiang Medical University
Curated by ChEMBL
Sanquan College Of Xinxiang Medical University
Curated by ChEMBL
Affinity DataIC50: 4.5nMAssay Description:Inhibition of EED (unknown origin)More data for this Ligand-Target Pair
TargetPolycomb protein EED(Homo sapiens (Human))
Sanquan College Of Xinxiang Medical University
Curated by ChEMBL
Sanquan College Of Xinxiang Medical University
Curated by ChEMBL
Affinity DataIC50: 5nMAssay Description:Inhibition of EED (unknown origin)More data for this Ligand-Target Pair
TargetPolycomb protein EED(Homo sapiens (Human))
Sanquan College Of Xinxiang Medical University
Curated by ChEMBL
Sanquan College Of Xinxiang Medical University
Curated by ChEMBL
Affinity DataIC50: 6.80nMAssay Description:Inhibition of human N-terminal His-6 tagged EED expressed in Escherichia coli strain BL2(DE3) by SPR analysisMore data for this Ligand-Target Pair
TargetPolycomb protein EED(Homo sapiens (Human))
Sanquan College Of Xinxiang Medical University
Curated by ChEMBL
Sanquan College Of Xinxiang Medical University
Curated by ChEMBL
Affinity DataIC50: 7.80nMAssay Description:Inhibition of human N-terminal His-6 tagged EED expressed in Escherichia coli strain BL2(DE3) by SPR analysisMore data for this Ligand-Target Pair
TargetHistone-lysine N-methyltransferase EZH2/Polycomb protein EED/Polycomb protein SUZ12(Homo sapiens (Human))
Sanquan College Of Xinxiang Medical University
Curated by ChEMBL
Sanquan College Of Xinxiang Medical University
Curated by ChEMBL
Affinity DataIC50: 18nMAssay Description:Inhibition of PRC2 complex of EZH2-EED-SUZ12 (unknown origin) using human nucleosome as substrate incubated for 70 mins in presence of [3H]SAMMore data for this Ligand-Target Pair
TargetPolycomb protein EED(Homo sapiens (Human))
Sanquan College Of Xinxiang Medical University
Curated by ChEMBL
Sanquan College Of Xinxiang Medical University
Curated by ChEMBL
Affinity DataIC50: <20nMAssay Description:Inhibition of EED (unknown origin)More data for this Ligand-Target Pair
TargetPolycomb protein EED(Homo sapiens (Human))
Sanquan College Of Xinxiang Medical University
Curated by ChEMBL
Sanquan College Of Xinxiang Medical University
Curated by ChEMBL
Affinity DataIC50: <20nMAssay Description:Inhibition of EED (unknown origin)More data for this Ligand-Target Pair
TargetPolycomb protein EED(Homo sapiens (Human))
Sanquan College Of Xinxiang Medical University
Curated by ChEMBL
Sanquan College Of Xinxiang Medical University
Curated by ChEMBL
Affinity DataIC50: <20nMAssay Description:Inhibition of EED (unknown origin)More data for this Ligand-Target Pair
TargetPolycomb protein EED(Homo sapiens (Human))
Sanquan College Of Xinxiang Medical University
Curated by ChEMBL
Sanquan College Of Xinxiang Medical University
Curated by ChEMBL
Affinity DataIC50: 20nMAssay Description:Inhibition of EED (unknown origin)More data for this Ligand-Target Pair
TargetPolycomb protein EED(Homo sapiens (Human))
Sanquan College Of Xinxiang Medical University
Curated by ChEMBL
Sanquan College Of Xinxiang Medical University
Curated by ChEMBL
Affinity DataIC50: <20nMAssay Description:Inhibition of EED (unknown origin)More data for this Ligand-Target Pair
Affinity DataIC50: 22nMAssay Description:Binding affinity to BRD4 bromodomain 1 in human Ramos cellsMore data for this Ligand-Target Pair
TargetPolycomb protein EED(Homo sapiens (Human))
Sanquan College Of Xinxiang Medical University
Curated by ChEMBL
Sanquan College Of Xinxiang Medical University
Curated by ChEMBL
Affinity DataIC50: 45nMAssay Description:Inhibition of full length N-terminal His-6x tagged EED (1 to 441 residues) (unknown origin) incubated for 1 hr by TR-FRET assayMore data for this Ligand-Target Pair
TargetPolycomb protein EED(Homo sapiens (Human))
Sanquan College Of Xinxiang Medical University
Curated by ChEMBL
Sanquan College Of Xinxiang Medical University
Curated by ChEMBL
Affinity DataIC50: 60nMAssay Description:Inhibition of EED (unknown origin) by alpha screen binding assayMore data for this Ligand-Target Pair
TargetPolycomb protein EED(Homo sapiens (Human))
Sanquan College Of Xinxiang Medical University
Curated by ChEMBL
Sanquan College Of Xinxiang Medical University
Curated by ChEMBL
Affinity DataIC50: <100nMAssay Description:Inhibition of EED (unknown origin)More data for this Ligand-Target Pair
TargetPolycomb protein EED(Homo sapiens (Human))
Sanquan College Of Xinxiang Medical University
Curated by ChEMBL
Sanquan College Of Xinxiang Medical University
Curated by ChEMBL
Affinity DataIC50: <100nMAssay Description:Inhibition of EED (unknown origin)More data for this Ligand-Target Pair
TargetPolycomb protein EED(Homo sapiens (Human))
Sanquan College Of Xinxiang Medical University
Curated by ChEMBL
Sanquan College Of Xinxiang Medical University
Curated by ChEMBL
Affinity DataIC50: <100nMAssay Description:Inhibition of EED (unknown origin)More data for this Ligand-Target Pair
TargetPolycomb protein EED(Homo sapiens (Human))
Sanquan College Of Xinxiang Medical University
Curated by ChEMBL
Sanquan College Of Xinxiang Medical University
Curated by ChEMBL
Affinity DataIC50: <100nMAssay Description:Inhibition of EED (unknown origin)More data for this Ligand-Target Pair
TargetPolycomb protein EED(Homo sapiens (Human))
Sanquan College Of Xinxiang Medical University
Curated by ChEMBL
Sanquan College Of Xinxiang Medical University
Curated by ChEMBL
Affinity DataIC50: <100nMAssay Description:Inhibition of EED (unknown origin)More data for this Ligand-Target Pair
TargetPolycomb protein EED(Homo sapiens (Human))
Sanquan College Of Xinxiang Medical University
Curated by ChEMBL
Sanquan College Of Xinxiang Medical University
Curated by ChEMBL
Affinity DataIC50: <100nMAssay Description:Inhibition of EED (unknown origin)More data for this Ligand-Target Pair
Affinity DataIC50: 190nMAssay Description:Inhibition of electric eel AChE using acetylthiocholine iodide as substrate preincubated with compounds for 20 mins followed by substrate addition an...More data for this Ligand-Target Pair
Affinity DataIC50: 240nMAssay Description:Induction of BRD4 degradation in human 231MFP cellsMore data for this Ligand-Target Pair
TargetPolycomb protein EED(Homo sapiens (Human))
Sanquan College Of Xinxiang Medical University
Curated by ChEMBL
Sanquan College Of Xinxiang Medical University
Curated by ChEMBL
Affinity DataIC50: 247nMAssay Description:Inhibition of full length N-terminal His-6x tagged EED (1 to 441 residues) (unknown origin) incubated for 1 hr by TR-FRET assayMore data for this Ligand-Target Pair
TargetPolycomb protein EED(Homo sapiens (Human))
Sanquan College Of Xinxiang Medical University
Curated by ChEMBL
Sanquan College Of Xinxiang Medical University
Curated by ChEMBL
Affinity DataIC50: 290nMAssay Description:Inhibition of GST-tagged EED in human G-401 cells assessed as inhibition of histone trimethylation by TR-FRET assayMore data for this Ligand-Target Pair
TargetHistone-lysine N-methyltransferase EZH2(Homo sapiens (Human))
Sanquan College Of Xinxiang Medical University
Curated by ChEMBL
Sanquan College Of Xinxiang Medical University
Curated by ChEMBL
Affinity DataIC50: 300nMAssay Description:Inhibition of EZH2 (unknown origin)More data for this Ligand-Target Pair
Affinity DataIC50: 470nMAssay Description:Inhibition of RNF114 (unknown origin)More data for this Ligand-Target Pair
TargetPolycomb protein EED(Homo sapiens (Human))
Sanquan College Of Xinxiang Medical University
Curated by ChEMBL
Sanquan College Of Xinxiang Medical University
Curated by ChEMBL
Affinity DataIC50: 620nMAssay Description:Inhibition of biotinylated H3K27Me3 peptide (19 to 33 aa) binding to EED (1 to 441 residues) (unknown origin) expressed in Escherichia coli BL21-Codo...More data for this Ligand-Target Pair
Affinity DataIC50: 670nMAssay Description:Inhibition of FNIP1 in human HEK293T cellsMore data for this Ligand-Target Pair
TargetPolycomb protein EED(Homo sapiens (Human))
Sanquan College Of Xinxiang Medical University
Curated by ChEMBL
Sanquan College Of Xinxiang Medical University
Curated by ChEMBL
Affinity DataIC50: 1.00E+3nMAssay Description:Inhibition of EED (unknown origin)More data for this Ligand-Target Pair
Affinity DataIC50: 1.00E+3nMAssay Description:Inhibition of electric eel AChE using acetylthiocholine iodide as substrate preincubated with compounds for 20 mins followed by substrate addition an...More data for this Ligand-Target Pair
Affinity DataIC50: 1.50E+3nMAssay Description:Inhibition of electric eel AChE using acetylthiocholine chloride as a substrate incubated for 20 mins followed by substrate addition and measured aft...More data for this Ligand-Target Pair
Affinity DataIC50: 1.70E+3nMAssay Description:Inhibition of electric eel AChE using acetylthiocholine iodide as substrate preincubated with compounds for 20 mins followed by substrate addition an...More data for this Ligand-Target Pair
TargetPolycomb protein EED(Homo sapiens (Human))
Sanquan College Of Xinxiang Medical University
Curated by ChEMBL
Sanquan College Of Xinxiang Medical University
Curated by ChEMBL
Affinity DataIC50: 2.10E+3nMAssay Description:Inhibition of human EED (76 to 441 residues) expressed in Escherichia coli strain BL21(DE3) by alpha screen assayMore data for this Ligand-Target Pair
TargetPolycomb protein EED(Homo sapiens (Human))
Sanquan College Of Xinxiang Medical University
Curated by ChEMBL
Sanquan College Of Xinxiang Medical University
Curated by ChEMBL
Affinity DataIC50: 2.10E+3nMAssay Description:Inhibition of human EED (76 to 441 residues) expressed in Escherichia coli strain BL21(DE3) by alpha screen assayMore data for this Ligand-Target Pair
TargetPolycomb protein EED(Homo sapiens (Human))
Sanquan College Of Xinxiang Medical University
Curated by ChEMBL
Sanquan College Of Xinxiang Medical University
Curated by ChEMBL
Affinity DataIC50: 3.28E+3nMAssay Description:Inhibition of EED in human G-401 cells assessed as reduction of global H3K27Me3 level by ELISAMore data for this Ligand-Target Pair
Affinity DataIC50: 3.60E+3nMAssay Description:Inhibition of electric eel AChE using acetylthiocholine iodide as substrate preincubated with compounds for 20 mins followed by substrate addition an...More data for this Ligand-Target Pair
Affinity DataIC50: 3.90E+3nMAssay Description:Inhibition of electric eel AChE using acetylthiocholine chloride as a substrate incubated for 20 mins followed by substrate addition and measured aft...More data for this Ligand-Target Pair
TargetPolycomb protein EED(Homo sapiens (Human))
Sanquan College Of Xinxiang Medical University
Curated by ChEMBL
Sanquan College Of Xinxiang Medical University
Curated by ChEMBL
Affinity DataIC50: 4.03E+3nMAssay Description:Inhibition of EED (unknown origin)More data for this Ligand-Target Pair
Affinity DataIC50: 4.50E+3nMAssay Description:Inhibition of electric eel AChE using acetylthiocholine chloride as a substrate incubated for 20 mins followed by substrate addition and measured aft...More data for this Ligand-Target Pair
TargetPolycomb protein EED(Homo sapiens (Human))
Sanquan College Of Xinxiang Medical University
Curated by ChEMBL
Sanquan College Of Xinxiang Medical University
Curated by ChEMBL
Affinity DataIC50: 5.60E+3nMAssay Description:Inhibition of human EED (76 to 441 residues) expressed in Escherichia coli strain BL21(DE3) by alpha screen assayMore data for this Ligand-Target Pair
Affinity DataIC50: 7.60E+3nMAssay Description:Binding affinity to BRD4 bromodomain 1 in human Ramos cellsMore data for this Ligand-Target Pair
TargetEpidermal growth factor receptor(Homo sapiens (Human))
Southwest Jiaotong University
Curated by ChEMBL
Southwest Jiaotong University
Curated by ChEMBL
Affinity DataIC50: 1.06E+4nMAssay Description:Inhibition of EGFR (unknown origin)More data for this Ligand-Target Pair
Affinity DataIC50: 1.10E+4nMAssay Description:Inhibition of electric eel AChE using acetylthiocholine chloride as a substrate incubated for 20 mins followed by substrate addition and measured aft...More data for this Ligand-Target Pair
Affinity DataIC50: 1.70E+4nMAssay Description:Inhibition of electric eel AChE using acetylthiocholine iodide as substrate preincubated with compounds for 20 mins followed by substrate addition an...More data for this Ligand-Target Pair
TargetEpidermal growth factor receptor(Homo sapiens (Human))
Southwest Jiaotong University
Curated by ChEMBL
Southwest Jiaotong University
Curated by ChEMBL
Affinity DataIC50: 1.85E+4nMAssay Description:Inhibition of EGFR (unknown origin)More data for this Ligand-Target Pair
TargetEpidermal growth factor receptor(Homo sapiens (Human))
Southwest Jiaotong University
Curated by ChEMBL
Southwest Jiaotong University
Curated by ChEMBL
Affinity DataIC50: 2.10E+4nMAssay Description:Inhibition of EGFR (unknown origin)More data for this Ligand-Target Pair
Affinity DataIC50: 2.70E+4nMAssay Description:Inhibition of electric eel AChE using acetylthiocholine iodide as substrate preincubated with compounds for 20 mins followed by substrate addition an...More data for this Ligand-Target Pair
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Sanquan College Of Xinxiang Medical University
Curated by ChEMBL
Sanquan College Of Xinxiang Medical University
Curated by ChEMBL
Affinity DataIC50: >3.00E+4nMAssay Description:Inhibition of human ERGMore data for this Ligand-Target Pair