Compile Data Set for Download or QSAR
maximum 50k data
Found 631 with Last Name = 'ahmad' and Initial = 'm'
TargetGlutamine--fructose-6-phosphate aminotransferase [isomerizing] 1(Homo sapiens (Human))
Hoffmann-La Roche

Curated by ChEMBL
LigandPNGBDBM50356009(CHEMBL1911368)
Affinity DataKi:  300nMAssay Description:Competitive inhibition of GFAT in presence of glutamineMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamine--fructose-6-phosphate aminotransferase [isomerizing] 1(Homo sapiens (Human))
Hoffmann-La Roche

Curated by ChEMBL
LigandPNGBDBM50356009(CHEMBL1911368)
Affinity DataKi:  300nMAssay Description:Noncompetitive inhibition of GFAT in presence of fructose-6-phosphateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin G/H synthase 2(Homo sapiens (Human))TBA
LigandPNGBDBM50611064(CHEMBL316846)
Affinity DataIC50:  2nMAssay Description:Inhibition of COX-2 (unknown origin) using arachidonic acid as substrate incubated for 1 min by absorbance based analysisMore data for this Ligand-Target Pair
Ligand Info
In DepthDetails PubMed
TargetProstaglandin G/H synthase 2(Homo sapiens (Human))TBA
LigandPNGBDBM50611065(CHEMBL5267453)
Affinity DataIC50:  2nMAssay Description:Inhibition of COX-2 (unknown origin) using arachidonic acid as substrate incubated for 1 min by absorbance based analysisMore data for this Ligand-Target Pair
Ligand Info
In DepthDetails PubMed
TargetProstaglandin G/H synthase 2(Homo sapiens (Human))TBA
LigandPNGBDBM50611066(CHEMBL5279940)
Affinity DataIC50:  2nMAssay Description:Inhibition of COX-2 (unknown origin) using arachidonic acid as substrate incubated for 1 min by absorbance based analysisMore data for this Ligand-Target Pair
Ligand Info
In DepthDetails PubMed
TargetProstaglandin G/H synthase 2(Homo sapiens (Human))TBA
LigandPNGBDBM50611067(CHEMBL5277168)
Affinity DataIC50:  2nMAssay Description:Inhibition of COX-2 (unknown origin) using arachidonic acid as substrate incubated for 1 min by absorbance based analysisMore data for this Ligand-Target Pair
Ligand Info
In DepthDetails PubMed
TargetProstaglandin G/H synthase 2(Homo sapiens (Human))TBA
LigandPNGBDBM50611068(CHEMBL5280463)
Affinity DataIC50:  2nMAssay Description:Inhibition of COX-2 (unknown origin) using arachidonic acid as substrate incubated for 1 min by absorbance based analysisMore data for this Ligand-Target Pair
Ligand Info
In DepthDetails PubMed
TargetProstaglandin G/H synthase 2(Homo sapiens (Human))TBA
LigandPNGBDBM50611069(CHEMBL5265839)
Affinity DataIC50:  2nMAssay Description:Inhibition of COX-2 (unknown origin) using arachidonic acid as substrate incubated for 1 min by absorbance based analysisMore data for this Ligand-Target Pair
Ligand Info
In DepthDetails PubMed
TargetProstaglandin G/H synthase 2(Homo sapiens (Human))TBA
LigandPNGBDBM50611070(CHEMBL5289245)
Affinity DataIC50:  2nMAssay Description:Inhibition of COX-2 (unknown origin) using arachidonic acid as substrate incubated for 1 min by absorbance based analysisMore data for this Ligand-Target Pair
Ligand Info
In DepthDetails PubMed
TargetProstaglandin G/H synthase 2(Homo sapiens (Human))TBA
LigandPNGBDBM50611071(CHEMBL5269974)
Affinity DataIC50:  2nMAssay Description:Inhibition of COX-2 (unknown origin) using arachidonic acid as substrate incubated for 1 min by absorbance based analysisMore data for this Ligand-Target Pair
Ligand Info
In DepthDetails PubMed
TargetProstaglandin G/H synthase 2(Homo sapiens (Human))TBA
LigandPNGBDBM50611072(CHEMBL5290253)
Affinity DataIC50:  2nMAssay Description:Inhibition of COX-2 (unknown origin) using arachidonic acid as substrate incubated for 1 min by absorbance based analysisMore data for this Ligand-Target Pair
Ligand Info
In DepthDetails PubMed
TargetProstaglandin G/H synthase 2(Homo sapiens (Human))TBA
LigandPNGBDBM50611073(CHEMBL5276070)
Affinity DataIC50:  2nMAssay Description:Inhibition of COX-2 (unknown origin) using arachidonic acid as substrate incubated for 1 min by absorbance based analysisMore data for this Ligand-Target Pair
Ligand Info
In DepthDetails PubMed
TargetProstaglandin G/H synthase 2(Homo sapiens (Human))TBA
LigandPNGBDBM50611074(CHEMBL5278033)
Affinity DataIC50:  2nMAssay Description:Inhibition of COX-2 (unknown origin) using arachidonic acid as substrate incubated for 1 min by absorbance based analysisMore data for this Ligand-Target Pair
Ligand Info
In DepthDetails PubMed
TargetProstaglandin G/H synthase 2(Homo sapiens (Human))TBA
LigandPNGBDBM50611232(CHEMBL5283867)
Affinity DataIC50:  2nMAssay Description:Inhibition of human COX-2 using arachidonic acid as substrate incubated for 30 secs by ELISAMore data for this Ligand-Target Pair
Ligand Info
In DepthDetails PubMed
TargetAmine oxidase [flavin-containing] A(Rattus norvegicus (rat))
Government College University

Curated by ChEMBL
LigandPNGBDBM15581(CHEMBL8706 | CLG | CLORGILINE | Clorgyline | N-[3-...)
Affinity DataIC50:  4.5nMAssay Description:Inhibition of MAO-A in rat liver mitochondria using p-tyramine as substrate preincubated for 10 mins followed by substrate addition measured after 30...More data for this Ligand-Target Pair
TargetDiacylglycerol O-acyltransferase 1(Homo sapiens (Human))
Hoffmann-La Roche

Curated by ChEMBL
LigandPNGBDBM50341785((1R,2R)-2-(3'-fluoro-4'-(3-phenylureido)biphenylca...)
Affinity DataIC50:  7nMAssay Description:Inhibition of human DGAT1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin G/H synthase 2(Homo sapiens (Human))TBA
LigandPNGBDBM11639(4-[5-(4-methylphenyl)-3-(trifluoromethyl)-1H-pyraz...)
Affinity DataIC50:  10nMAssay Description:Inhibition of COX-2 (unknown origin) using arachidonic acid as substrate incubated for 1 min by absorbance based analysisMore data for this Ligand-Target Pair
TargetDiacylglycerol O-acyltransferase 1(Homo sapiens (Human))
Hoffmann-La Roche

Curated by ChEMBL
LigandPNGBDBM50341766(2-Phenyl-5-trifluoromethyloxazole-4-carboxylic Aci...)
Affinity DataIC50:  16nMAssay Description:Inhibition of human DGAT1 expressed in baculovirus infected insect cells after 1 hr using palmitoyl-1-14C-coenzyme A by phospholipid flashplate assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholinesterase(Equus caballus (Horse))
Government College Women University

Curated by ChEMBL
LigandPNGBDBM50004244(CHEMBL3237461)
Affinity DataIC50:  17nMAssay Description:Inhibition of BuChE in equine serum using butyrylthiocholine chloride as substrate preincubated with enzyme for 10 mins prior to substrate challenge ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin G/H synthase 2(Homo sapiens (Human))TBA
LigandPNGBDBM69641(1,3-Diphenyl-1H-pyrazole-4-carbaldehyde | 1,3-diph...)
Affinity DataIC50:  17nMAssay Description:Inhibition of human COX-2 using arachidonic acid as substrate incubated for 30 secs by ELISAMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetProstaglandin G/H synthase 2(Homo sapiens (Human))TBA
LigandPNGBDBM50611226(CHEMBL5278905)
Affinity DataIC50:  17nMAssay Description:Inhibition of human COX-2 using arachidonic acid as substrate incubated for 30 secs by ELISAMore data for this Ligand-Target Pair
Ligand Info
In DepthDetails PubMed
TargetProstaglandin G/H synthase 2(Homo sapiens (Human))TBA
LigandPNGBDBM50611227(CHEMBL5288954)
Affinity DataIC50:  17nMAssay Description:Inhibition of human COX-2 using arachidonic acid as substrate incubated for 30 secs by ELISAMore data for this Ligand-Target Pair
Ligand Info
In DepthDetails PubMed
TargetProstaglandin G/H synthase 2(Homo sapiens (Human))TBA
LigandPNGBDBM50611228(CHEMBL5275104)
Affinity DataIC50:  17nMAssay Description:Inhibition of human COX-2 using arachidonic acid as substrate incubated for 30 secs by ELISAMore data for this Ligand-Target Pair
Ligand Info
In DepthDetails PubMed
TargetAmine oxidase [flavin-containing] B(Rattus norvegicus (rat))
Government College University

Curated by ChEMBL
LigandPNGBDBM39862(Deprenyl | METHYL-(1-METHYL-2-PHENYL-ETHYL)-PROP-2...)
Affinity DataIC50:  20nMAssay Description:Inhibition of MAO-B in rat liver mitochondria using p-tyramine as substrate preincubated for 10 mins followed by substrate addition measured after 30...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholinesterase(Equus caballus (Horse))
Government College Women University

Curated by ChEMBL
LigandPNGBDBM50004238(CHEMBL3237453)
Affinity DataIC50:  26nMAssay Description:Inhibition of BuChE in equine serum using butyrylthiocholine chloride as substrate preincubated with enzyme for 10 mins prior to substrate challenge ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDiacylglycerol O-acyltransferase 1(Homo sapiens (Human))
Hoffmann-La Roche

Curated by ChEMBL
LigandPNGBDBM50341768(4-{5-[(2-Phenyl-5-trifluoromethyloxazole-4-carbony...)
Affinity DataIC50:  28nMAssay Description:Inhibition of human DGAT1 expressed in baculovirus infected insect cells after 1 hr using palmitoyl-1-14C-coenzyme A by phospholipid flashplate assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDiacylglycerol O-acyltransferase 1(Homo sapiens (Human))
Hoffmann-La Roche

Curated by ChEMBL
LigandPNGBDBM50341778(4-(4-{5-[(2-Phenyl-5-trifluoromethyloxazole-4-carb...)
Affinity DataIC50:  35nMAssay Description:Inhibition of human DGAT1 expressed in baculovirus infected insect cells after 1 hr using palmitoyl-1-14C-coenzyme A by phospholipid flashplate assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDiacylglycerol O-acyltransferase 1(Homo sapiens (Human))
Hoffmann-La Roche

Curated by ChEMBL
LigandPNGBDBM50341760(2-Phenyl-5-trifluoromethyloxazole-4-carboxylic Aci...)
Affinity DataIC50:  38nMAssay Description:Inhibition of human DGAT1 expressed in baculovirus infected insect cells after 1 hr using palmitoyl-1-14C-coenzyme A by phospholipid flashplate assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDiacylglycerol O-acyltransferase 1(Homo sapiens (Human))
Hoffmann-La Roche

Curated by ChEMBL
LigandPNGBDBM50341760(2-Phenyl-5-trifluoromethyloxazole-4-carboxylic Aci...)
Affinity DataIC50:  38nMAssay Description:Inhibition of human DGAT1 using [14C]palmitic acid by TLC analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDiacylglycerol O-acyltransferase 1(Homo sapiens (Human))
Hoffmann-La Roche

Curated by ChEMBL
LigandPNGBDBM50341760(2-Phenyl-5-trifluoromethyloxazole-4-carboxylic Aci...)
Affinity DataIC50:  38nMAssay Description:Inhibition of human DGAT1 using palmitoyl-1-14C coenzyme A and DAG as substrate after 1 hr by phospholipid flash plate assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin G/H synthase 2(Homo sapiens (Human))TBA
LigandPNGBDBM50611153(CHEMBL5265750)
Affinity DataIC50:  39nMAssay Description:Inhibition of human COX-2 using arachidonic acid as substrate preincubated for 10 mins followed by substrate addition and measured after 2 mins by EL...More data for this Ligand-Target Pair
Ligand Info
In DepthDetails PubMed
TargetProstaglandin G/H synthase 2(Homo sapiens (Human))TBA
LigandPNGBDBM50611154(CHEMBL5278569)
Affinity DataIC50:  39nMAssay Description:Inhibition of human COX-2 using arachidonic acid as substrate preincubated for 10 mins followed by substrate addition and measured after 2 mins by EL...More data for this Ligand-Target Pair
Ligand Info
In DepthDetails PubMed
TargetProstaglandin G/H synthase 2(Homo sapiens (Human))TBA
LigandPNGBDBM50611155(CHEMBL5282152)
Affinity DataIC50:  39nMAssay Description:Inhibition of human COX-2 using arachidonic acid as substrate preincubated for 10 mins followed by substrate addition and measured after 2 mins by EL...More data for this Ligand-Target Pair
Ligand Info
In DepthDetails PubMed
TargetProstaglandin G/H synthase 2(Homo sapiens (Human))TBA
LigandPNGBDBM50611156(CHEMBL5290194)
Affinity DataIC50:  39nMAssay Description:Inhibition of human COX-2 using arachidonic acid as substrate preincubated for 10 mins followed by substrate addition and measured after 2 mins by EL...More data for this Ligand-Target Pair
Ligand Info
In DepthDetails PubMed
TargetProstaglandin G/H synthase 2(Homo sapiens (Human))TBA
LigandPNGBDBM50611157(CHEMBL5283848)
Affinity DataIC50:  39nMAssay Description:Inhibition of human COX-2 using arachidonic acid as substrate preincubated for 10 mins followed by substrate addition and measured after 2 mins by EL...More data for this Ligand-Target Pair
Ligand Info
In DepthDetails PubMed
TargetProstaglandin G/H synthase 2(Homo sapiens (Human))TBA
LigandPNGBDBM50611158(CHEMBL5266071)
Affinity DataIC50:  39nMAssay Description:Inhibition of human COX-2 using arachidonic acid as substrate preincubated for 10 mins followed by substrate addition and measured after 2 mins by EL...More data for this Ligand-Target Pair
Ligand Info
In DepthDetails PubMed
TargetEpidermal growth factor receptor(Homo sapiens (Human))TBA
LigandPNGBDBM5446(CHEMBL553 | ERLOTINIB HYDROCHLORIDE | Erlotinib | ...)
Affinity DataIC50:  40nMAssay Description:Inhibition of EGFR (unknown origin) incubated for 1 hr in presence of ATP by ADP-Glo kinase assayMore data for this Ligand-Target Pair
TargetProstaglandin G/H synthase 2(Homo sapiens (Human))TBA
LigandPNGBDBM50611164(CHEMBL5286186)
Affinity DataIC50:  41nMAssay Description:Inhibition of human COX-2 using arachidonic acid as substrate preincubated for 10 mins followed by substrate addition and measured after 2 mins by EL...More data for this Ligand-Target Pair
Ligand Info
In DepthDetails PubMed
TargetProstaglandin G/H synthase 2(Homo sapiens (Human))TBA
LigandPNGBDBM50611165(CHEMBL5266705)
Affinity DataIC50:  41nMAssay Description:Inhibition of human COX-2 using arachidonic acid as substrate preincubated for 10 mins followed by substrate addition and measured after 2 mins by EL...More data for this Ligand-Target Pair
Ligand Info
In DepthDetails PubMed
TargetProstaglandin G/H synthase 2(Homo sapiens (Human))TBA
LigandPNGBDBM50611166(CHEMBL5269531)
Affinity DataIC50:  41nMAssay Description:Inhibition of human COX-2 using arachidonic acid as substrate preincubated for 10 mins followed by substrate addition and measured after 2 mins by EL...More data for this Ligand-Target Pair
Ligand Info
In DepthDetails PubMed
TargetCholinesterase(Equus caballus (Horse))
Government College Women University

Curated by ChEMBL
LigandPNGBDBM50004241(CHEMBL3233057)
Affinity DataIC50:  41nMAssay Description:Inhibition of BuChE in equine serum using butyrylthiocholine chloride as substrate preincubated with enzyme for 10 mins prior to substrate challenge ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDiacylglycerol O-acyltransferase 1(Homo sapiens (Human))
Hoffmann-La Roche

Curated by ChEMBL
LigandPNGBDBM50341770(4-{5-[(2-Phenyl-5-trifluoromethyloxazole-4-carbony...)
Affinity DataIC50:  41nMAssay Description:Inhibition of human DGAT1 expressed in baculovirus infected insect cells after 1 hr using palmitoyl-1-14C-coenzyme A by phospholipid flashplate assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin G/H synthase 2(Homo sapiens (Human))TBA
LigandPNGBDBM50611178(CHEMBL5274739)
Affinity DataIC50:  43nMAssay Description:Inhibition of recombinant human COX-2 by enzyme immunoassayMore data for this Ligand-Target Pair
Ligand Info
In DepthDetails PubMed
TargetProstaglandin G/H synthase 2(Homo sapiens (Human))TBA
LigandPNGBDBM50057593(4-[5-(4-Chloro-phenyl)-3-(4-methoxy-phenyl)-pyrazo...)
Affinity DataIC50:  43nMAssay Description:Inhibition of recombinant human COX-2 by enzyme immunoassayMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetProstaglandin G/H synthase 2(Homo sapiens (Human))TBA
LigandPNGBDBM50611179(CHEMBL5283165)
Affinity DataIC50:  43nMAssay Description:Inhibition of recombinant human COX-2 by enzyme immunoassayMore data for this Ligand-Target Pair
Ligand Info
In DepthDetails PubMed
TargetProstaglandin G/H synthase 2(Homo sapiens (Human))TBA
LigandPNGBDBM50611180(CHEMBL5279336)
Affinity DataIC50:  43nMAssay Description:Inhibition of recombinant human COX-2 by enzyme immunoassayMore data for this Ligand-Target Pair
Ligand Info
In DepthDetails PubMed
TargetProstaglandin G/H synthase 2(Homo sapiens (Human))TBA
LigandPNGBDBM50611181(CHEMBL5274403)
Affinity DataIC50:  43nMAssay Description:Inhibition of recombinant human COX-2 by enzyme immunoassayMore data for this Ligand-Target Pair
Ligand Info
In DepthDetails PubMed
TargetProstaglandin G/H synthase 2(Homo sapiens (Human))TBA
LigandPNGBDBM50611182(CHEMBL5276782)
Affinity DataIC50:  43nMAssay Description:Inhibition of recombinant human COX-2 by enzyme immunoassayMore data for this Ligand-Target Pair
Ligand Info
In DepthDetails PubMed
TargetProstaglandin G/H synthase 2(Homo sapiens (Human))TBA
LigandPNGBDBM50611183(CHEMBL5281497)
Affinity DataIC50:  43nMAssay Description:Inhibition of recombinant human COX-2 by enzyme immunoassayMore data for this Ligand-Target Pair
Ligand Info
In DepthDetails PubMed
TargetProstaglandin G/H synthase 2(Homo sapiens (Human))TBA
LigandPNGBDBM50611184(CHEMBL5279090)
Affinity DataIC50:  43nMAssay Description:Inhibition of recombinant human COX-2 by enzyme immunoassayMore data for this Ligand-Target Pair
Ligand Info
In DepthDetails PubMed
Displayed 1 to 50 (of 631 total ) | Next | Last >>
Jump to: