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Found 177 with Last Name = 'alewood' and Initial = 'pf'
TargetKappa-type opioid receptor(Homo sapiens (Human))TBA
LigandPNGBDBM50613517(CHEMBL5273346)
Affinity DataKi:  0.0700nMAssay Description:Displacement of [3H]U69593 from human kappa opioid receptor expressed in CHO-K1 cells incubated for 1 hr by 1450 microbeta scintillation counter anal...More data for this Ligand-Target Pair
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TargetKappa-type opioid receptor(Homo sapiens (Human))TBA
LigandPNGBDBM50613518(CHEMBL5289754)
Affinity DataKi:  0.130nMAssay Description:Displacement of [3H]U69593 from human kappa opioid receptor expressed in CHO-K1 cells incubated for 1 hr by 1450 microbeta scintillation counter anal...More data for this Ligand-Target Pair
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TargetKappa-type opioid receptor(Homo sapiens (Human))TBA
LigandPNGBDBM50613552(CHEMBL5281808)
Affinity DataKi:  0.160nMAssay Description:Displacement of [3H]U69593 from human kappa opioid receptor expressed in CHO-K1 cells incubated for 1 hr by 1450 microbeta scintillation counter anal...More data for this Ligand-Target Pair
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TargetKappa-type opioid receptor(Homo sapiens (Human))TBA
LigandPNGBDBM50613546(CHEMBL5273114)
Affinity DataKi:  0.230nMAssay Description:Displacement of [3H]U69593 from human kappa opioid receptor expressed in CHO-K1 cells incubated for 1 hr by 1450 microbeta scintillation counter anal...More data for this Ligand-Target Pair
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TargetKappa-type opioid receptor(Homo sapiens (Human))TBA
LigandPNGBDBM50613519(CHEMBL5281912)
Affinity DataKi:  0.25nMAssay Description:Displacement of [3H]U69593 from human kappa opioid receptor expressed in CHO-K1 cells incubated for 1 hr by 1450 microbeta scintillation counter anal...More data for this Ligand-Target Pair
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TargetKappa-type opioid receptor(Homo sapiens (Human))TBA
LigandPNGBDBM50613478(CHEMBL5273273)
Affinity DataKi:  0.280nMAssay Description:Displacement of [3H]U69593 from human kappa opioid receptor expressed in CHO-K1 cells incubated for 1 hr by 1450 microbeta scintillation counter anal...More data for this Ligand-Target Pair
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TargetKappa-type opioid receptor(Homo sapiens (Human))TBA
LigandPNGBDBM50613548(CHEMBL5286081)
Affinity DataKi:  0.290nMAssay Description:Displacement of [3H]U69593 from human kappa opioid receptor expressed in CHO-K1 cells incubated for 1 hr by 1450 microbeta scintillation counter anal...More data for this Ligand-Target Pair
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TargetOxytocin receptor(Homo sapiens (Human))
The University Of Queensland

Curated by ChEMBL
LigandPNGBDBM50332720((S)-1-((4R,7S,10S,13S,16S,19R)-4-amino-16-(2-amino...)
Affinity DataKi:  0.290nMAssay Description:Displacement of [3H]OT from oxytocin receptor expressed in COS1 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
The University Of Queensland

Curated by ChEMBL
LigandPNGBDBM50369584(CHEMBL1790230)
Affinity DataKi:  0.300nMAssay Description:Inhibitory constant against HIV-1 proteaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Homo sapiens (Human))TBA
LigandPNGBDBM50002184(CHEMBL415330 | H-Tyr-Gly-Gly-Phe-Leu-Arg-Arg-Ile-A...)
Affinity DataKi:  0.400nMAssay Description:Displacement of [3H]U69593 from human kappa opioid receptor expressed in CHO-K1 cells incubated for 1 hr by 1450 microbeta scintillation counter anal...More data for this Ligand-Target Pair
In DepthDetails PubMed
TargetKappa-type opioid receptor(Homo sapiens (Human))TBA
LigandPNGBDBM50613550(CHEMBL5279208)
Affinity DataKi:  0.420nMAssay Description:Displacement of [3H]U69593 from human kappa opioid receptor expressed in CHO-K1 cells incubated for 1 hr by 1450 microbeta scintillation counter anal...More data for this Ligand-Target Pair
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TargetKappa-type opioid receptor(Homo sapiens (Human))TBA
LigandPNGBDBM50613528(CHEMBL5282326)
Affinity DataKi:  0.480nMAssay Description:Displacement of [3H]U69593 from human kappa opioid receptor expressed in CHO-K1 cells incubated for 1 hr by 1450 microbeta scintillation counter anal...More data for this Ligand-Target Pair
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In DepthDetails PubMed
TargetKappa-type opioid receptor(Homo sapiens (Human))TBA
LigandPNGBDBM50613551(CHEMBL5283035)
Affinity DataKi:  0.590nMAssay Description:Displacement of [3H]U69593 from human kappa opioid receptor expressed in CHO-K1 cells incubated for 1 hr by 1450 microbeta scintillation counter anal...More data for this Ligand-Target Pair
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TargetKappa-type opioid receptor(Homo sapiens (Human))TBA
LigandPNGBDBM50613520(CHEMBL5283811)
Affinity DataKi:  0.590nMAssay Description:Displacement of [3H]U69593 from human kappa opioid receptor expressed in CHO-K1 cells incubated for 1 hr by 1450 microbeta scintillation counter anal...More data for this Ligand-Target Pair
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In DepthDetails PubMed
TargetKappa-type opioid receptor(Homo sapiens (Human))TBA
LigandPNGBDBM50613547(CHEMBL5278935)
Affinity DataKi:  0.590nMAssay Description:Displacement of [3H]U69593 from human kappa opioid receptor expressed in CHO-K1 cells incubated for 1 hr by 1450 microbeta scintillation counter anal...More data for this Ligand-Target Pair
Ligand Info
In DepthDetails PubMed
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
The University Of Queensland

Curated by ChEMBL
LigandPNGBDBM50092152(2-Benzyl-5-(10-sec-butyl-9,12-dioxo-2-oxa-8,11-dia...)
Affinity DataKi:  0.600nMAssay Description:Inhibitory constant against HIV-1 proteaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDimer of Gag-Pol polyprotein [501-599,Q508K,L534I,L564I,C568A,C596A](Human immunodeficiency virus type 1)
University of Queensland

LigandPNGBDBM13928(2-[(8S,11S)-11-[(1R)-2-[benzene(3-methylbutyl)sulf...)
Affinity DataKi:  0.600nM ΔG°:  -54.8kJ/molepH: 6.5 T: 2°CAssay Description:he Ki values were determined using fluorogenic substrate, 2-(aminobenzoyl)-Thr-Ile-Nle-Phe(p-NO2)-Gln-ArgNH2. A standard curve relating changes in fl...More data for this Ligand-Target Pair
TargetKappa-type opioid receptor(Homo sapiens (Human))TBA
LigandPNGBDBM50613545(CHEMBL5288658)
Affinity DataKi:  0.610nMAssay Description:Displacement of [3H]U69593 from human kappa opioid receptor expressed in CHO-K1 cells incubated for 1 hr by 1450 microbeta scintillation counter anal...More data for this Ligand-Target Pair
Ligand Info
In DepthDetails PubMed
TargetKappa-type opioid receptor(Homo sapiens (Human))TBA
LigandPNGBDBM50613513(CHEMBL5280997)
Affinity DataKi:  0.640nMAssay Description:Displacement of [3H]U69593 from human kappa opioid receptor expressed in CHO-K1 cells incubated for 1 hr by 1450 microbeta scintillation counter anal...More data for this Ligand-Target Pair
Ligand Info
In DepthDetails PubMed
TargetKappa-type opioid receptor(Homo sapiens (Human))TBA
LigandPNGBDBM50613514(CHEMBL5284775)
Affinity DataKi:  0.710nMAssay Description:Displacement of [3H]U69593 from human kappa opioid receptor expressed in CHO-K1 cells incubated for 1 hr by 1450 microbeta scintillation counter anal...More data for this Ligand-Target Pair
Ligand Info
In DepthDetails PubMed
TargetOxytocin receptor(Homo sapiens (Human))
The University Of Queensland

Curated by ChEMBL
LigandPNGBDBM50332721((S)-N-((S)-1-(2-amino-2-oxoethylamino)-3-methylbut...)
Affinity DataKi:  0.720nMAssay Description:Displacement of [3H]OT from oxytocin receptor expressed in COS1 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOxytocin receptor(Homo sapiens (Human))
The University Of Queensland

Curated by ChEMBL
LigandPNGBDBM50205990(CHEMBL395429 | OXYTOCIN)
Affinity DataKi:  0.790nMAssay Description:Displacement of [3H]OT from oxytocin receptor expressed in COS1 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Homo sapiens (Human))TBA
LigandPNGBDBM50613515(CHEMBL5276702)
Affinity DataKi:  0.910nMAssay Description:Displacement of [3H]U69593 from human kappa opioid receptor expressed in CHO-K1 cells incubated for 1 hr by 1450 microbeta scintillation counter anal...More data for this Ligand-Target Pair
Ligand Info
In DepthDetails PubMed
TargetKappa-type opioid receptor(Homo sapiens (Human))TBA
LigandPNGBDBM50613521(CHEMBL5285730)
Affinity DataKi:  0.980nMAssay Description:Displacement of [3H]U69593 from human kappa opioid receptor expressed in CHO-K1 cells incubated for 1 hr by 1450 microbeta scintillation counter anal...More data for this Ligand-Target Pair
Ligand Info
In DepthDetails PubMed
TargetKappa-type opioid receptor(Homo sapiens (Human))TBA
LigandPNGBDBM50613511(CHEMBL5278992)
Affinity DataKi:  1.20nMAssay Description:Displacement of [3H]U69593 from human kappa opioid receptor expressed in CHO-K1 cells incubated for 1 hr by 1450 microbeta scintillation counter anal...More data for this Ligand-Target Pair
Ligand Info
In DepthDetails PubMed
TargetKappa-type opioid receptor(Homo sapiens (Human))TBA
LigandPNGBDBM50613522(CHEMBL5270523)
Affinity DataKi:  1.20nMAssay Description:Displacement of [3H]U69593 from human kappa opioid receptor expressed in CHO-K1 cells incubated for 1 hr by 1450 microbeta scintillation counter anal...More data for this Ligand-Target Pair
Ligand Info
In DepthDetails PubMed
TargetKappa-type opioid receptor(Homo sapiens (Human))TBA
LigandPNGBDBM50613516(CHEMBL5275165)
Affinity DataKi:  1.20nMAssay Description:Displacement of [3H]U69593 from human kappa opioid receptor expressed in CHO-K1 cells incubated for 1 hr by 1450 microbeta scintillation counter anal...More data for this Ligand-Target Pair
Ligand Info
In DepthDetails PubMed
TargetKappa-type opioid receptor(Homo sapiens (Human))TBA
LigandPNGBDBM50613510(CHEMBL5282859)
Affinity DataKi:  1.20nMAssay Description:Displacement of [3H]U69593 from human kappa opioid receptor expressed in CHO-K1 cells incubated for 1 hr by 1450 microbeta scintillation counter anal...More data for this Ligand-Target Pair
Ligand Info
In DepthDetails PubMed
TargetKappa-type opioid receptor(Homo sapiens (Human))TBA
LigandPNGBDBM50613494(CHEMBL5280066)
Affinity DataKi:  1.30nMAssay Description:Displacement of [3H]U69593 from human kappa opioid receptor expressed in CHO-K1 cells incubated for 1 hr by 1450 microbeta scintillation counter anal...More data for this Ligand-Target Pair
Ligand Info
In DepthDetails PubMed
TargetKappa-type opioid receptor(Homo sapiens (Human))TBA
LigandPNGBDBM50613524(CHEMBL5289642)
Affinity DataKi:  1.30nMAssay Description:Displacement of [3H]U69593 from human kappa opioid receptor expressed in CHO-K1 cells incubated for 1 hr by 1450 microbeta scintillation counter anal...More data for this Ligand-Target Pair
Ligand Info
In DepthDetails PubMed
TargetKappa-type opioid receptor(Homo sapiens (Human))TBA
LigandPNGBDBM50613549(CHEMBL5283084)
Affinity DataKi:  1.40nMAssay Description:Displacement of [3H]U69593 from human kappa opioid receptor expressed in CHO-K1 cells incubated for 1 hr by 1450 microbeta scintillation counter anal...More data for this Ligand-Target Pair
Ligand Info
In DepthDetails PubMed
TargetOxytocin receptor(Homo sapiens (Human))
The University Of Queensland

Curated by ChEMBL
LigandPNGBDBM50332723(CHEMBL1630531 | Cystathionine Oxytocin)
Affinity DataKi:  1.5nMAssay Description:Displacement of [3H]OT from oxytocin receptor expressed in COS1 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
The University Of Queensland

Curated by ChEMBL
LigandPNGBDBM50092151((10S,13S,1'R)-13-[1'-HYDROXY-2'-(N-P-AMINOBENZENES...)
Affinity DataKi:  1.70nMAssay Description:Inhibitory constant against HIV-1 proteaseMore data for this Ligand-Target Pair
TargetDimer of Gag-Pol polyprotein [501-599,Q508K,L534I,L564I,C568A,C596A](Human immunodeficiency virus type 1)
University of Queensland

LigandPNGBDBM13931((2S)-N-[(2S,3R)-4-{[(8S,11S)-8-[(2R)-butan-2-yl]-7...)
Affinity DataKi:  1.80nM ΔG°:  -51.9kJ/molepH: 6.5 T: 2°CAssay Description:he Ki values were determined using fluorogenic substrate, 2-(aminobenzoyl)-Thr-Ile-Nle-Phe(p-NO2)-Gln-ArgNH2. A standard curve relating changes in fl...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Homo sapiens (Human))TBA
LigandPNGBDBM50613512(CHEMBL5276129)
Affinity DataKi:  2.10nMAssay Description:Displacement of [3H]U69593 from human kappa opioid receptor expressed in CHO-K1 cells incubated for 1 hr by 1450 microbeta scintillation counter anal...More data for this Ligand-Target Pair
Ligand Info
In DepthDetails PubMed
TargetKappa-type opioid receptor(Homo sapiens (Human))TBA
LigandPNGBDBM50613523(CHEMBL5279518)
Affinity DataKi:  2.20nMAssay Description:Displacement of [3H]U69593 from human kappa opioid receptor expressed in CHO-K1 cells incubated for 1 hr by 1450 microbeta scintillation counter anal...More data for this Ligand-Target Pair
Ligand Info
In DepthDetails PubMed
TargetKappa-type opioid receptor(Homo sapiens (Human))TBA
LigandPNGBDBM50613532(CHEMBL5288155)
Affinity DataKi:  2.40nMAssay Description:Displacement of [3H]U69593 from human kappa opioid receptor expressed in CHO-K1 cells incubated for 1 hr by 1450 microbeta scintillation counter anal...More data for this Ligand-Target Pair
Ligand Info
In DepthDetails PubMed
TargetKappa-type opioid receptor(Homo sapiens (Human))TBA
LigandPNGBDBM50613496(CHEMBL5266718)
Affinity DataKi:  2.90nMAssay Description:Displacement of [3H]U69593 from human kappa opioid receptor expressed in CHO-K1 cells incubated for 1 hr by 1450 microbeta scintillation counter anal...More data for this Ligand-Target Pair
Ligand Info
In DepthDetails PubMed
TargetDimer of Gag-Pol polyprotein [501-599,Q508K,L534I,L564I,C568A,C596A](Human immunodeficiency virus type 1)
University of Queensland

LigandPNGBDBM13933((2S)-N-[(2S,3R)-4-{[(8S,11S)-8-[(2S)-butan-2-yl]-7...)
Affinity DataKi:  3nM ΔG°:  -50.6kJ/molepH: 6.5 T: 2°CAssay Description:he Ki values were determined using fluorogenic substrate, 2-(aminobenzoyl)-Thr-Ile-Nle-Phe(p-NO2)-Gln-ArgNH2. A standard curve relating changes in fl...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Homo sapiens (Human))TBA
LigandPNGBDBM50613506(CHEMBL5268886)
Affinity DataKi:  3.90nMAssay Description:Displacement of [3H]U69593 from human kappa opioid receptor expressed in CHO-K1 cells incubated for 1 hr by 1450 microbeta scintillation counter anal...More data for this Ligand-Target Pair
Ligand Info
In DepthDetails PubMed
TargetDimer of Gag-Pol polyprotein [501-599,Q508K,L534I,L564I,C568A,C596A](Human immunodeficiency virus type 1)
University of Queensland

LigandPNGBDBM13929((2R)-2-[(8S,11S)-6,9-dioxo-8-(propan-2-yl)-2-oxa-7...)
Affinity DataKi:  4nM ΔG°:  -49.9kJ/molepH: 6.5 T: 2°CAssay Description:he Ki values were determined using fluorogenic substrate, 2-(aminobenzoyl)-Thr-Ile-Nle-Phe(p-NO2)-Gln-ArgNH2. A standard curve relating changes in fl...More data for this Ligand-Target Pair
TargetDimer of Gag-Pol polyprotein [501-599,Q508K,L534I,L564I,C568A,C596A](Human immunodeficiency virus type 1)
University of Queensland

LigandPNGBDBM13932(Macrocyclic Peptidomimetic Inhibitor 6 | tert-buty...)
Affinity DataKi:  4nM ΔG°:  -49.9kJ/molepH: 6.5 T: 2°CAssay Description:he Ki values were determined using fluorogenic substrate, 2-(aminobenzoyl)-Thr-Ile-Nle-Phe(p-NO2)-Gln-ArgNH2. A standard curve relating changes in fl...More data for this Ligand-Target Pair
TargetDimer of Gag-Pol polyprotein [501-599,Q508K,L534I,L564I,C568A,C596A](Human immunodeficiency virus type 1)
University of Queensland

LigandPNGBDBM13930((2S)-N-tert-butyl-1-[(2R)-2-[(8S,11S)-8-(carbamoyl...)
Affinity DataKi:  5nM ΔG°:  -49.3kJ/molepH: 6.5 T: 2°CAssay Description:he Ki values were determined using fluorogenic substrate, 2-(aminobenzoyl)-Thr-Ile-Nle-Phe(p-NO2)-Gln-ArgNH2. A standard curve relating changes in fl...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMedMMDB

TargetKappa-type opioid receptor(Homo sapiens (Human))TBA
LigandPNGBDBM50613508(CHEMBL5288478)
Affinity DataKi:  5.30nMAssay Description:Displacement of [3H]U69593 from human kappa opioid receptor expressed in CHO-K1 cells incubated for 1 hr by 1450 microbeta scintillation counter anal...More data for this Ligand-Target Pair
Ligand Info
In DepthDetails PubMed
TargetKappa-type opioid receptor(Homo sapiens (Human))TBA
LigandPNGBDBM50613507(CHEMBL5280357)
Affinity DataKi:  5.40nMAssay Description:Displacement of [3H]U69593 from human kappa opioid receptor expressed in CHO-K1 cells incubated for 1 hr by 1450 microbeta scintillation counter anal...More data for this Ligand-Target Pair
Ligand Info
In DepthDetails PubMed
TargetKappa-type opioid receptor(Homo sapiens (Human))TBA
LigandPNGBDBM50613503(CHEMBL5267287)
Affinity DataKi:  6.70nMAssay Description:Displacement of [3H]U69593 from human kappa opioid receptor expressed in CHO-K1 cells incubated for 1 hr by 1450 microbeta scintillation counter anal...More data for this Ligand-Target Pair
Ligand Info
In DepthDetails PubMed
TargetKappa-type opioid receptor(Homo sapiens (Human))TBA
LigandPNGBDBM50613509(CHEMBL5271178)
Affinity DataKi:  6.70nMAssay Description:Displacement of [3H]U69593 from human kappa opioid receptor expressed in CHO-K1 cells incubated for 1 hr by 1450 microbeta scintillation counter anal...More data for this Ligand-Target Pair
Ligand Info
In DepthDetails PubMed
TargetOxytocin receptor(Homo sapiens (Human))
The University Of Queensland

Curated by ChEMBL
LigandPNGBDBM50332724((S)-N-((S)-1-(2-amino-2-oxoethylamino)-3-methylbut...)
Affinity DataKi:  7.60nMAssay Description:Displacement of [3H]OT from oxytocin receptor expressed in COS1 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Homo sapiens (Human))TBA
LigandPNGBDBM50613533(CHEMBL5276505)
Affinity DataKi:  7.80nMAssay Description:Displacement of [3H]U69593 from human kappa opioid receptor expressed in CHO-K1 cells incubated for 1 hr by 1450 microbeta scintillation counter anal...More data for this Ligand-Target Pair
Ligand Info
In DepthDetails PubMed
TargetKappa-type opioid receptor(Homo sapiens (Human))TBA
LigandPNGBDBM50613553(CHEMBL5276565)
Affinity DataKi:  10nMAssay Description:Displacement of [3H]U69593 from human kappa opioid receptor expressed in CHO-K1 cells incubated for 1 hr by 1450 microbeta scintillation counter anal...More data for this Ligand-Target Pair
Ligand Info
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