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Found 33 with Last Name = 'anwar' and Initial = 'a'
TargetSteryl-sulfatase(Rattus norvegicus)TBA
LigandPNGBDBM50148911((3beta)-3-hydroxyurs-12-en-28-oic acid | 3beta-hyd...)
Affinity DataIC50:  0.0600nMAssay Description:Inhibition of estrone sulfatase in homogeneous rat mammary tumorsMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetSteryl-sulfatase(Homo sapiens (Human))TBA
LigandPNGBDBM50148911((3beta)-3-hydroxyurs-12-en-28-oic acid | 3beta-hyd...)
Affinity DataIC50:  0.120nMAssay Description:Inhibition of estrone sulfatase in human MCF7 cell microsomesMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetEstrogen receptor alpha(Bos taurus)TBA
LigandPNGBDBM50610464(CHEMBL5284918)
Affinity DataIC50:  60nMAssay Description:Displacement of [3H]-17beta-estradiol from bovine uterine estrogen receptor by competitive binding assayMore data for this Ligand-Target Pair
Ligand Info
In DepthDetails PubMed
TargetSulfotransferase 1A1(Rattus norvegicus)TBA
LigandPNGBDBM7460(2-(3,4-dihydroxyphenyl)-3,5,7-trihydroxy-4H-chrome...)
Affinity DataIC50:  290nMAssay Description:Inhibition of rat liver SULT1A1-mediated oestradiol sulfonation incubated for 20 minsMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetSulfotransferase 1A1(Rattus norvegicus)TBA
LigandPNGBDBM19459(5,7-dihydroxy-3-(4-hydroxyphenyl)-4H-chromen-4-one...)
Affinity DataIC50:  290nMAssay Description:Inhibition of rat liver SULT1A1-mediated oestradiol sulfonation incubated for 20 minsMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetSulfotransferase 1A1(Rattus norvegicus)TBA
LigandPNGBDBM23420(7,4′-Dihydroxy-isoflavone (3a) | 7-hydroxy-3...)
Affinity DataIC50:  290nMAssay Description:Inhibition of rat liver SULT1A1-mediated oestradiol sulfonation incubated for 20 minsMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetSulfotransferase 1A1(Rattus norvegicus)TBA
LigandPNGBDBM7462(3,5,7-trihydroxy-2-(4-hydroxyphenyl)-4H-chromen-4-...)
Affinity DataIC50:  290nMAssay Description:Inhibition of rat liver SULT1A1-mediated oestradiol sulfonation incubated for 20 minsMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetEstrogen receptor alpha(Bos taurus)TBA
LigandPNGBDBM50610463(CHEBI:67889 | NYASOL)
Affinity DataIC50:  400nMAssay Description:Displacement of [3H]-17beta-estradiol from bovine uterine estrogen receptor by competitive binding assayMore data for this Ligand-Target Pair
Ligand Info
In DepthDetails PubMed
TargetUrease(Canavalia ensiformis (Jack bean) (Horse bean))
Universiti Teknologi Mara Puncak Alam Campus

Curated by ChEMBL
LigandPNGBDBM50106604(CHEMBL3600575)
Affinity DataIC50:  1.30E+4nMAssay Description:Inhibition of jack bean urease using urea as substrate assessed as ammonia production after 15 mins by Weatherburn assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUrease(Canavalia ensiformis (Jack bean) (Horse bean))
Universiti Teknologi Mara Puncak Alam Campus

Curated by ChEMBL
LigandPNGBDBM50106617(CHEMBL3600581)
Affinity DataIC50:  1.92E+4nMAssay Description:Inhibition of jack bean urease using urea as substrate assessed as ammonia production after 15 mins by Weatherburn assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUrease(Canavalia ensiformis (Jack bean) (Horse bean))
Universiti Teknologi Mara Puncak Alam Campus

Curated by ChEMBL
LigandPNGBDBM50229993(2-thiourea | CHEMBL260876 | Thiocarbamid | Thiohar...)
Affinity DataIC50:  2.10E+4nMAssay Description:Inhibition of jack bean urease using urea as substrate assessed as ammonia production after 15 mins by Weatherburn assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSulfotransferase 2A1(Rattus norvegicus)TBA
LigandPNGBDBM7462(3,5,7-trihydroxy-2-(4-hydroxyphenyl)-4H-chromen-4-...)
Affinity DataIC50:  3.40E+4nMAssay Description:Inhibition of rat SULT2A1-mediated dehydroepiandrosterone sulfonation incubated for 20 minsMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetSulfotransferase 2A1(Rattus norvegicus)TBA
LigandPNGBDBM23420(7,4′-Dihydroxy-isoflavone (3a) | 7-hydroxy-3...)
Affinity DataIC50:  3.40E+4nMAssay Description:Inhibition of rat SULT2A1-mediated dehydroepiandrosterone sulfonation incubated for 20 minsMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetSulfotransferase 2A1(Rattus norvegicus)TBA
LigandPNGBDBM7460(2-(3,4-dihydroxyphenyl)-3,5,7-trihydroxy-4H-chrome...)
Affinity DataIC50:  3.40E+4nMAssay Description:Inhibition of rat SULT2A1-mediated dehydroepiandrosterone sulfonation incubated for 20 minsMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetSulfotransferase 2A1(Rattus norvegicus)TBA
LigandPNGBDBM19459(5,7-dihydroxy-3-(4-hydroxyphenyl)-4H-chromen-4-one...)
Affinity DataIC50:  3.40E+4nMAssay Description:Inhibition of rat SULT2A1-mediated dehydroepiandrosterone sulfonation incubated for 20 minsMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetUrease(Canavalia ensiformis (Jack bean) (Horse bean))
Universiti Teknologi Mara Puncak Alam Campus

Curated by ChEMBL
LigandPNGBDBM50106622(CHEMBL3600576)
Affinity DataIC50:  3.54E+4nMAssay Description:Inhibition of jack bean urease using urea as substrate assessed as ammonia production after 15 mins by Weatherburn assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUrease(Canavalia ensiformis (Jack bean) (Horse bean))
Universiti Teknologi Mara Puncak Alam Campus

Curated by ChEMBL
LigandPNGBDBM50099857(ACETOHYDROXAMIC ACID (AHA) | AHA | Acethydroxamsae...)
Affinity DataIC50:  4.20E+4nMAssay Description:Inhibition of jack bean urease using urea as substrate assessed as ammonia production after 15 mins by Weatherburn assayMore data for this Ligand-Target Pair
TargetUrease(Canavalia ensiformis (Jack bean) (Horse bean))
Universiti Teknologi Mara Puncak Alam Campus

Curated by ChEMBL
LigandPNGBDBM50106621(CHEMBL3600577)
Affinity DataIC50:  4.29E+4nMAssay Description:Inhibition of jack bean urease using urea as substrate assessed as ammonia production after 15 mins by Weatherburn assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUrease(Canavalia ensiformis (Jack bean) (Horse bean))
Universiti Teknologi Mara Puncak Alam Campus

Curated by ChEMBL
LigandPNGBDBM50106605(CHEMBL3600652)
Affinity DataIC50:  4.91E+4nMAssay Description:Inhibition of jack bean urease using urea as substrate assessed as ammonia production after 15 mins by Weatherburn assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUrease(Canavalia ensiformis (Jack bean) (Horse bean))
Universiti Teknologi Mara Puncak Alam Campus

Curated by ChEMBL
LigandPNGBDBM50106620(CHEMBL3600578)
Affinity DataIC50:  5.32E+4nMAssay Description:Inhibition of jack bean urease using urea as substrate assessed as ammonia production after 15 mins by Weatherburn assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUrease(Canavalia ensiformis (Jack bean) (Horse bean))
Universiti Teknologi Mara Puncak Alam Campus

Curated by ChEMBL
LigandPNGBDBM50106618(CHEMBL3600580)
Affinity DataIC50:  7.08E+4nMAssay Description:Inhibition of jack bean urease using urea as substrate assessed as ammonia production after 15 mins by Weatherburn assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUrease(Canavalia ensiformis (Jack bean) (Horse bean))
Universiti Teknologi Mara Puncak Alam Campus

Curated by ChEMBL
LigandPNGBDBM50106610(CHEMBL3600646)
Affinity DataIC50:  7.18E+4nMAssay Description:Inhibition of jack bean urease using urea as substrate assessed as ammonia production after 15 mins by Weatherburn assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUrease(Canavalia ensiformis (Jack bean) (Horse bean))
Universiti Teknologi Mara Puncak Alam Campus

Curated by ChEMBL
LigandPNGBDBM50106608(CHEMBL3600648)
Affinity DataIC50:  8.20E+4nMAssay Description:Inhibition of jack bean urease using urea as substrate assessed as ammonia production after 15 mins by Weatherburn assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUrease(Canavalia ensiformis (Jack bean) (Horse bean))
Universiti Teknologi Mara Puncak Alam Campus

Curated by ChEMBL
LigandPNGBDBM50106614(CHEMBL3600642)
Affinity DataIC50:  8.48E+4nMAssay Description:Inhibition of jack bean urease using urea as substrate assessed as ammonia production after 15 mins by Weatherburn assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUrease(Canavalia ensiformis (Jack bean) (Horse bean))
Universiti Teknologi Mara Puncak Alam Campus

Curated by ChEMBL
LigandPNGBDBM50106607(CHEMBL3600649)
Affinity DataIC50:  9.24E+4nMAssay Description:Inhibition of jack bean urease using urea as substrate assessed as ammonia production after 15 mins by Weatherburn assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUrease(Canavalia ensiformis (Jack bean) (Horse bean))
Universiti Teknologi Mara Puncak Alam Campus

Curated by ChEMBL
LigandPNGBDBM50106615(CHEMBL3600583)
Affinity DataIC50:  1.02E+5nMAssay Description:Inhibition of jack bean urease using urea as substrate assessed as ammonia production after 15 mins by Weatherburn assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUrease(Canavalia ensiformis (Jack bean) (Horse bean))
Universiti Teknologi Mara Puncak Alam Campus

Curated by ChEMBL
LigandPNGBDBM50106616(CHEMBL3600582)
Affinity DataIC50:  1.09E+5nMAssay Description:Inhibition of jack bean urease using urea as substrate assessed as ammonia production after 15 mins by Weatherburn assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUrease(Canavalia ensiformis (Jack bean) (Horse bean))
Universiti Teknologi Mara Puncak Alam Campus

Curated by ChEMBL
LigandPNGBDBM50106611(CHEMBL3600645)
Affinity DataIC50:  1.11E+5nMAssay Description:Inhibition of jack bean urease using urea as substrate assessed as ammonia production after 15 mins by Weatherburn assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUrease(Canavalia ensiformis (Jack bean) (Horse bean))
Universiti Teknologi Mara Puncak Alam Campus

Curated by ChEMBL
LigandPNGBDBM50106613(CHEMBL3600643)
Affinity DataIC50:  1.20E+5nMAssay Description:Inhibition of jack bean urease using urea as substrate assessed as ammonia production after 15 mins by Weatherburn assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUrease(Canavalia ensiformis (Jack bean) (Horse bean))
Universiti Teknologi Mara Puncak Alam Campus

Curated by ChEMBL
LigandPNGBDBM50106619(CHEMBL3600579)
Affinity DataIC50:  1.26E+5nMAssay Description:Inhibition of jack bean urease using urea as substrate assessed as ammonia production after 15 mins by Weatherburn assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUrease(Canavalia ensiformis (Jack bean) (Horse bean))
Universiti Teknologi Mara Puncak Alam Campus

Curated by ChEMBL
LigandPNGBDBM50106612(CHEMBL3600644)
Affinity DataIC50:  1.44E+5nMAssay Description:Inhibition of jack bean urease using urea as substrate assessed as ammonia production after 15 mins by Weatherburn assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUrease(Canavalia ensiformis (Jack bean) (Horse bean))
Universiti Teknologi Mara Puncak Alam Campus

Curated by ChEMBL
LigandPNGBDBM50106609(CHEMBL3600647)
Affinity DataIC50:  1.45E+5nMAssay Description:Inhibition of jack bean urease using urea as substrate assessed as ammonia production after 15 mins by Weatherburn assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUrease(Canavalia ensiformis (Jack bean) (Horse bean))
Universiti Teknologi Mara Puncak Alam Campus

Curated by ChEMBL
LigandPNGBDBM50106606(CHEMBL3600650)
Affinity DataIC50:  1.49E+5nMAssay Description:Inhibition of jack bean urease using urea as substrate assessed as ammonia production after 15 mins by Weatherburn assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed