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Found 480 with Last Name = 'araki' and Initial = 't'
TargetGrowth factor receptor-bound protein 2(Homo sapiens (Human))
National Cancer Institute-Frederick

Curated by ChEMBL
LigandPNGBDBM50139763(CHEMBL306657 | [(E)-(9S,10S,14S,18S)-18-Carbamoylm...)
Affinity DataIC50:  1.40nMAssay Description:In vitro Growth factor receptor bound protein 2-binding affinity of the compound was determined in in surface plasmon resonance (SPR) methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGrowth factor receptor-bound protein 2(Homo sapiens (Human))
National Cancer Institute-Frederick

Curated by ChEMBL
LigandPNGBDBM50139763(CHEMBL306657 | [(E)-(9S,10S,14S,18S)-18-Carbamoylm...)
Affinity DataIC50:  1.40nMAssay Description:In vitro Growth factor receptor bound protein 2-binding affinity of the compound was determined in in surface plasmon resonance (SPR) methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-X-C chemokine receptor type 4(Homo sapiens (Human))
Kyoto University

Curated by ChEMBL
LigandPNGBDBM50202356(CHEMBL218806 | cyclo(-D-Tyr-D-MeArg-L-Arg-L-Nal-Gl...)
Affinity DataIC50:  3nMAssay Description:Inhibition of [125I]SDF1 binding to CXCR4 transfected in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-X-C chemokine receptor type 4(Homo sapiens (Human))
Kyoto University

Curated by ChEMBL
LigandPNGBDBM50202350(CHEMBL219474 | cyclo(-D-Tyr-L-Arg-L-Arg-L-Nal-Gly-...)
Affinity DataIC50:  4nMAssay Description:Inhibition of [125I]SDF1 binding to CXCR4 transfected in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-X-C chemokine receptor type 4(Homo sapiens (Human))
Kyoto University

Curated by ChEMBL
LigandPNGBDBM50166087(CHEMBL436097 | N-{3-[(2R,5S,8S,14R)-5-(3-Guanidino...)
Affinity DataIC50:  4.30nMAssay Description:Inhibition of [125I]-SDF-1 binding to C-X-C chemokine receptor type 4 (CXCR4) expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGrowth factor receptor-bound protein 2(Homo sapiens (Human))
National Cancer Institute-Frederick

Curated by ChEMBL
LigandPNGBDBM50143944(2-[4-((E)-(9S,10S,14S,18S)-18-Carbamoylmethyl-9-ca...)
Affinity DataIC50:  4.30nMAssay Description:In vitro Growth factor receptor bound protein 2-binding affinity of the compound was determined in ELISA methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-X-C chemokine receptor type 4(Homo sapiens (Human))
Kyoto University

Curated by ChEMBL
LigandPNGBDBM50202346(CHEMBL219339 | cyclo(-D-Tyr-D-Arg-L-Arg-L-Nal-Gly-...)
Affinity DataIC50:  8nMAssay Description:Inhibition of [125I]SDF1 binding to CXCR4 transfected in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-X-C chemokine receptor type 4(Homo sapiens (Human))
Kyoto University

Curated by ChEMBL
LigandPNGBDBM50166106(CHEMBL436283 | N-{3-[(2S,5S,8S,14R)-5-(3-Guanidino...)
Affinity DataIC50:  8.40nMAssay Description:Inhibition of [125I]-SDF-1 binding to C-X-C chemokine receptor type 4 (CXCR4) expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-X-C chemokine receptor type 4(Homo sapiens (Human))
Kyoto University

Curated by ChEMBL
LigandPNGBDBM50166096(CHEMBL372874 | N-[(2S,5R,11S,14S,16aS)-14-(3-Guani...)
Affinity DataIC50:  9.90nMAssay Description:Inhibition of [125I]-SDF-1 binding to C-X-C chemokine receptor type 4 (CXCR4) expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin G/H synthase 1(Ovis aries (Sheep))
Hokkaido University

Curated by ChEMBL
LigandPNGBDBM50326129(Indometacin)
Affinity DataIC50:  10nMAssay Description:Inhibition of ovine COX1 by colorimetric assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-X-C chemokine receptor type 4(Homo sapiens (Human))
Kyoto University

Curated by ChEMBL
LigandPNGBDBM50166079(CHEMBL192183 | N-[(2R,5R,11S,14S,16aS)-14-(3-Guani...)
Affinity DataIC50:  10nMAssay Description:Inhibition of [125I]-SDF-1 binding to C-X-C chemokine receptor type 4 (CXCR4) expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGrowth factor receptor-bound protein 2(Homo sapiens (Human))
National Cancer Institute-Frederick

Curated by ChEMBL
LigandPNGBDBM50072865(CHEMBL55627 | N-[(S)-1-{1-[(S)-2-Carbamoyl-1-(3-na...)
Affinity DataIC50:  10nMAssay Description:In vitro Growth factor receptor bound protein 2-binding affinity of the compound was determined in ELISA methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-X-C chemokine receptor type 4(Homo sapiens (Human))
Kyoto University

Curated by ChEMBL
LigandPNGBDBM50202359(CHEMBL375990 | cyclo(-D-Tyr-L-Arg-L-Arg-L-Nal-D-Al...)
Affinity DataIC50:  11nMAssay Description:Inhibition of [125I]SDF1 binding to CXCR4 transfected in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-X-C chemokine receptor type 4(Homo sapiens (Human))
Kyoto University

Curated by ChEMBL
LigandPNGBDBM50202345(CHEMBL373636 | cyclo(-D-Tyr-D-Arg-L-Arg-L-Nal-D-Al...)
Affinity DataIC50:  11nMAssay Description:Inhibition of [125I]SDF1 binding to CXCR4 transfected in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGrowth factor receptor-bound protein 2(Homo sapiens (Human))
National Cancer Institute-Frederick

Curated by ChEMBL
LigandPNGBDBM50143944(2-[4-((E)-(9S,10S,14S,18S)-18-Carbamoylmethyl-9-ca...)
Affinity DataIC50:  12.1nMAssay Description:In vitro Growth factor receptor bound protein 2-binding affinity of the compound was determined in in surface plasmon resonance (SPR) methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-X-C chemokine receptor type 4(Homo sapiens (Human))
Kyoto University

Curated by ChEMBL
LigandPNGBDBM50166101(CHEMBL372422 | N-{3-[(2S,5S,11R)-14-(2-Amino-ethyl...)
Affinity DataIC50:  16nMAssay Description:Inhibition of [125I]-SDF-1 binding to C-X-C chemokine receptor type 4 (CXCR4) expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-X-C chemokine receptor type 4(Homo sapiens (Human))
Kyoto University

Curated by ChEMBL
LigandPNGBDBM50166086(CHEMBL192594 | N-{3-[(2S,5S,11R)-14-(3-Amino-propy...)
Affinity DataIC50:  19nMAssay Description:Inhibition of [125I]-SDF-1 binding to C-X-C chemokine receptor type 4 (CXCR4) expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-X-C chemokine receptor type 4(Homo sapiens (Human))
Kyoto University

Curated by ChEMBL
LigandPNGBDBM50202347(CHEMBL376219 | cyclo(-D-Tyr-D-Arg-L-MeArg-L-Nal-Gl...)
Affinity DataIC50:  21nMAssay Description:Inhibition of [125I]SDF1 binding to CXCR4 transfected in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGrowth factor receptor-bound protein 2(Homo sapiens (Human))
National Cancer Institute-Frederick

Curated by ChEMBL
LigandPNGBDBM50085867(2-(4-((S)-3-(1-((S)-4-amino-1-(3-(naphthalen-1-yl)...)
Affinity DataIC50:  22.1nMAssay Description:In vitro Growth factor receptor bound protein 2-binding affinity of the compound was determined in ELISA methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-X-C chemokine receptor type 4(Homo sapiens (Human))
Kyoto University

Curated by ChEMBL
LigandPNGBDBM50202365(CHEMBL374421 | cyclo(-D-Tyr-L-MeArg-L-Arg-L-Nal-Gl...)
Affinity DataIC50:  23nMAssay Description:Inhibition of [125I]SDF1 binding to CXCR4 transfected in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-X-C chemokine receptor type 4(Homo sapiens (Human))
Kyoto University

Curated by ChEMBL
LigandPNGBDBM50166093(CHEMBL193217 | N-{3-[(2S,5S,11R,14S)-14-(2-Guanidi...)
Affinity DataIC50:  24nMAssay Description:Inhibition of [125I]-SDF-1 binding to C-X-C chemokine receptor type 4 (CXCR4) expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-X-C chemokine receptor type 4(Homo sapiens (Human))
Kyoto University

Curated by ChEMBL
LigandPNGBDBM50166080(CHEMBL192368 | N-{4-[(2S,5S,8S,14R)-5-(3-Guanidino...)
Affinity DataIC50:  33nMAssay Description:Inhibition of [125I]-SDF-1 binding to C-X-C chemokine receptor type 4 (CXCR4) expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-X-C chemokine receptor type 4(Homo sapiens (Human))
Kyoto University

Curated by ChEMBL
LigandPNGBDBM50166094(CHEMBL373155 | N-{3-[(2S,5S,11R,14S)-11-(4-Hydroxy...)
Affinity DataIC50:  42nMAssay Description:Inhibition of [125I]-SDF-1 binding to C-X-C chemokine receptor type 4 (CXCR4) expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-X-C chemokine receptor type 4(Homo sapiens (Human))
Kyoto University

Curated by ChEMBL
LigandPNGBDBM50202344(CHEMBL375991 | cyclo(-D-Tyr-L-Arg-L-Arg-L-Nal-beta...)
Affinity DataIC50:  47nMAssay Description:Inhibition of [125I]SDF1 binding to CXCR4 transfected in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-X-C chemokine receptor type 4(Homo sapiens (Human))
Kyoto University

Curated by ChEMBL
LigandPNGBDBM50166108(CHEMBL364295 | N-{3-[(3R,6S,9S,14S)-6-(3-Guanidino...)
Affinity DataIC50:  54nMAssay Description:Inhibition of [125I]-SDF-1 binding to C-X-C chemokine receptor type 4 (CXCR4) expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-X-C chemokine receptor type 4(Homo sapiens (Human))
Kyoto University

Curated by ChEMBL
LigandPNGBDBM50202367(CHEMBL374108 | cyclo(-D-Tyr-L-Ala-L-Arg-L-Nal-Gly-...)
Affinity DataIC50:  63nMAssay Description:Inhibition of [125I]SDF1 binding to CXCR4 transfected in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-X-C chemokine receptor type 4(Homo sapiens (Human))
Kyoto University

Curated by ChEMBL
LigandPNGBDBM50166088(CHEMBL191687 | N-{3-[(2S,5S,11R,14R)-11-(4-Hydroxy...)
Affinity DataIC50:  63nMAssay Description:Inhibition of [125I]-SDF-1 binding to C-X-C chemokine receptor type 4 (CXCR4) expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-X-C chemokine receptor type 4(Homo sapiens (Human))
Kyoto University

Curated by ChEMBL
LigandPNGBDBM50202360(CHEMBL376811 | cyclo(-D-Tyr-D-Arg-L-Arg-L-Nal-L-Al...)
Affinity DataIC50:  92nMAssay Description:Inhibition of [125I]SDF1 binding to CXCR4 transfected in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-X-C chemokine receptor type 4(Homo sapiens (Human))
Kyoto University

Curated by ChEMBL
LigandPNGBDBM50166109(CHEMBL365952 | N-{3-[(2S,5S,11R,14R)-14-(4-Amino-b...)
Affinity DataIC50:  97nMAssay Description:Inhibition of [125I]-SDF-1 binding to C-X-C chemokine receptor type 4 (CXCR4) expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-X-C chemokine receptor type 4(Homo sapiens (Human))
Kyoto University

Curated by ChEMBL
LigandPNGBDBM50202351(CHEMBL436536 | cyclo(-D-Tyr-L-Arg-L-MeArg-L-Nal-Gl...)
Affinity DataIC50:  99nMAssay Description:Inhibition of [125I]SDF1 binding to CXCR4 transfected in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin G/H synthase 1(Ovis aries (Sheep))
Hokkaido University

Curated by ChEMBL
LigandPNGBDBM17638(2-{1-[(4-chlorophenyl)carbonyl]-5-methoxy-2-methyl...)
Affinity DataIC50:  120nMAssay Description:Inhibition of ovine COX1 by colorimetric assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin G/H synthase 1(Ovis aries (Sheep))
Hokkaido University

Curated by ChEMBL
LigandPNGBDBM17638(2-{1-[(4-chlorophenyl)carbonyl]-5-methoxy-2-methyl...)
Affinity DataIC50:  120nMAssay Description:Inhibition of ovine COX1 by colorimetric assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-X-C chemokine receptor type 4(Homo sapiens (Human))
Kyoto University

Curated by ChEMBL
LigandPNGBDBM50202366(CHEMBL219096 | cyclo(-D-MeTyr-L-Arg-L-Arg-L-Nal-Gl...)
Affinity DataIC50:  128nMAssay Description:Inhibition of [125I]SDF1 binding to CXCR4 transfected in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-X-C chemokine receptor type 4(Homo sapiens (Human))
Kyoto University

Curated by ChEMBL
LigandPNGBDBM50202357(CHEMBL373440 | cyclo(-D-Ala-D-Arg-L-Arg-L-Nal-Gly-...)
Affinity DataIC50:  130nMAssay Description:Inhibition of [125I]SDF1 binding to CXCR4 transfected in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-X-C chemokine receptor type 4(Homo sapiens (Human))
Kyoto University

Curated by ChEMBL
LigandPNGBDBM50202348(CHEMBL375993 | cyclo(-D-MeTyr-D-Arg-L-Arg-L-Nal-Gl...)
Affinity DataIC50:  157nMAssay Description:Inhibition of [125I]SDF1 binding to CXCR4 transfected in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-X-C chemokine receptor type 4(Homo sapiens (Human))
Kyoto University

Curated by ChEMBL
LigandPNGBDBM50202373(CHEMBL219075 | cyclo(-D-Tyr-L-Arg-L-Arg-L-Ala-Sar-...)
Affinity DataIC50:  167nMAssay Description:Inhibition of [125I]SDF1 binding to CXCR4 transfected in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-X-C chemokine receptor type 4(Homo sapiens (Human))
Kyoto University

Curated by ChEMBL
LigandPNGBDBM50166098(3-[(2R,5S,8S,14R)-5-(3-Guanidino-propyl)-14-(4-hyd...)
Affinity DataIC50:  170nMAssay Description:Inhibition of [125I]-SDF-1 binding to C-X-C chemokine receptor type 4 (CXCR4) expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-X-C chemokine receptor type 4(Homo sapiens (Human))
Kyoto University

Curated by ChEMBL
LigandPNGBDBM50202361(CHEMBL387120 | cyclo(-D-Tyr-L-Arg-L-Arg-L-Nal-L-Al...)
Affinity DataIC50:  170nMAssay Description:Inhibition of [125I]SDF1 binding to CXCR4 transfected in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-X-C chemokine receptor type 4(Homo sapiens (Human))
Kyoto University

Curated by ChEMBL
LigandPNGBDBM50202343(CHEMBL384429 | cyclo(-D-Tyr-D-Ala-L-Arg-L-Nal-Gly-...)
Affinity DataIC50:  230nMAssay Description:Inhibition of [125I]SDF1 binding to CXCR4 transfected in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-X-C chemokine receptor type 4(Homo sapiens (Human))
Kyoto University

Curated by ChEMBL
LigandPNGBDBM50166105(CHEMBL192685 | N-{3-[(2S,5S,11R,14S)-11-(4-Hydroxy...)
Affinity DataIC50:  230nMAssay Description:Inhibition of [125I]-SDF-1 binding to C-X-C chemokine receptor type 4 (CXCR4) expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-X-C chemokine receptor type 4(Homo sapiens (Human))
Kyoto University

Curated by ChEMBL
LigandPNGBDBM50202368(CHEMBL375850 | cyclo(-D-Tyr-L-Arg-L-Arg-L-MeNal-Gl...)
Affinity DataIC50:  250nMAssay Description:Inhibition of [125I]SDF1 binding to CXCR4 transfected in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-X-C chemokine receptor type 4(Homo sapiens (Human))
Kyoto University

Curated by ChEMBL
LigandPNGBDBM50202362(CHEMBL374862 | cyclo(-D-Tyr-D-Arg-L-Arg-L-Nal-Sar-...)
Affinity DataIC50:  256nMAssay Description:Inhibition of [125I]SDF1 binding to CXCR4 transfected in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-X-C chemokine receptor type 4(Homo sapiens (Human))
Kyoto University

Curated by ChEMBL
LigandPNGBDBM50166092(2-[(2R,5S,8S,14R)-5-(3-Guanidino-propyl)-14-(4-hyd...)
Affinity DataIC50:  270nMAssay Description:Inhibition of [125I]-SDF-1 binding to C-X-C chemokine receptor type 4 (CXCR4) expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-X-C chemokine receptor type 4(Homo sapiens (Human))
Kyoto University

Curated by ChEMBL
LigandPNGBDBM50202355(CHEMBL219135 | cyclo(-D-Tyr-D-Arg-L-Arg-L-Nal-beta...)
Affinity DataIC50:  350nMAssay Description:Inhibition of [125I]SDF1 binding to CXCR4 transfected in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-X-C chemokine receptor type 4(Homo sapiens (Human))
Kyoto University

Curated by ChEMBL
LigandPNGBDBM50166097(CHEMBL424826 | N-{3-[(5R,11S,14S,16aR)-5-(4-Hydrox...)
Affinity DataIC50:  420nMAssay Description:Inhibition of [125I]-SDF-1 binding to C-X-C chemokine receptor type 4 (CXCR4) expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-X-C chemokine receptor type 4(Homo sapiens (Human))
Kyoto University

Curated by ChEMBL
LigandPNGBDBM50166102(CHEMBL371993 | N-{3-[(2S,5S,11R,14R)-11-(4-Hydroxy...)
Affinity DataIC50:  490nMAssay Description:Inhibition of [125I]-SDF-1 binding to C-X-C chemokine receptor type 4 (CXCR4) expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-X-C chemokine receptor type 4(Homo sapiens (Human))
Kyoto University

Curated by ChEMBL
LigandPNGBDBM50166091((4S,7S,10S,13R)-13-(3-Guanidino-propionylamino)-10...)
Affinity DataIC50:  530nMAssay Description:Inhibition of [125I]-SDF-1 binding to C-X-C chemokine receptor type 4 (CXCR4) expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-X-C chemokine receptor type 4(Homo sapiens (Human))
Kyoto University

Curated by ChEMBL
LigandPNGBDBM50202363(CHEMBL426169 | cyclo(-D-Tyr-D-Arg-L-Arg-L-MeNal-Gl...)
Affinity DataIC50:  563nMAssay Description:Inhibition of [125I]SDF1 binding to CXCR4 transfected in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-X-C chemokine receptor type 4(Homo sapiens (Human))
Kyoto University

Curated by ChEMBL
LigandPNGBDBM50166107(3-[(2R,5S,8S,14R)-5-(3-Guanidino-propyl)-14-(4-hyd...)
Affinity DataIC50:  610nMAssay Description:Inhibition of [125I]-SDF-1 binding to C-X-C chemokine receptor type 4 (CXCR4) expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-X-C chemokine receptor type 4(Homo sapiens (Human))
Kyoto University

Curated by ChEMBL
LigandPNGBDBM50202353(CHEMBL373637 | cyclo(-D-Tyr-D-Arg-L-Arg-L-Nal-L-Pi...)
Affinity DataIC50:  640nMAssay Description:Inhibition of [125I]SDF1 binding to CXCR4 transfected in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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