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Found 69 with Last Name = 'arun' and Initial = 's'
TargetKinesin-like protein KIF11(Homo sapiens (Human))
University Of Kwazulu-Natal (Ukzn)

Curated by ChEMBL
LigandPNGBDBM50463302(CHEMBL4239814)
Affinity DataIC50:  0.200nMAssay Description:Inhibition EG5 (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetReverse transcriptase(Human immunodeficiency virus 1)
Gvk Biosciences

Curated by ChEMBL
LigandPNGBDBM50483581(CHEMBL1689301)
Affinity DataIC50:  0.520nMAssay Description:Inhibition of Human immunodeficiency virus 1 reverse transcriptaseMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetReverse transcriptase(Human immunodeficiency virus 1)
Gvk Biosciences

Curated by ChEMBL
LigandPNGBDBM50483589(CHEMBL1689302)
Affinity DataIC50:  1.70nMAssay Description:Inhibition of Human immunodeficiency virus 1 reverse transcriptaseMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetReverse transcriptase(Human immunodeficiency virus 1)
Gvk Biosciences

Curated by ChEMBL
LigandPNGBDBM50483582(CHEMBL1689303)
Affinity DataIC50:  2.20nMAssay Description:Inhibition of Human immunodeficiency virus 1 reverse transcriptaseMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetReverse transcriptase(Human immunodeficiency virus 1)
Gvk Biosciences

Curated by ChEMBL
LigandPNGBDBM50483597(CHEMBL1689304)
Affinity DataIC50:  3.10nMAssay Description:Inhibition of Human immunodeficiency virus 1 reverse transcriptaseMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetReverse transcriptase(Human immunodeficiency virus 1)
Gvk Biosciences

Curated by ChEMBL
LigandPNGBDBM50483583(CHEMBL1689305)
Affinity DataIC50:  4nMAssay Description:Inhibition of Human immunodeficiency virus 1 reverse transcriptaseMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetReverse transcriptase(Human immunodeficiency virus 1)
Gvk Biosciences

Curated by ChEMBL
LigandPNGBDBM50483595(CHEMBL1689306)
Affinity DataIC50:  5.40nMAssay Description:Inhibition of Human immunodeficiency virus 1 reverse transcriptaseMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetKinesin-like protein KIF11(Homo sapiens (Human))
University Of Kwazulu-Natal (Ukzn)

Curated by ChEMBL
LigandPNGBDBM50431893(ARRY-520 | CHEMBL2347655)
Affinity DataIC50:  6nMAssay Description:Inhibition EG5 (unknown origin)More data for this Ligand-Target Pair
TargetReverse transcriptase(Human immunodeficiency virus 1)
Gvk Biosciences

Curated by ChEMBL
LigandPNGBDBM50483584(CHEMBL1689307)
Affinity DataIC50:  6.90nMAssay Description:Inhibition of Human immunodeficiency virus 1 reverse transcriptaseMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetKinesin-like protein KIF11(Homo sapiens (Human))
University Of Kwazulu-Natal (Ukzn)

Curated by ChEMBL
LigandPNGBDBM50463316(KF 89617 | KF-89617 | Kf89617 | LY 2523355 | LY-25...)
Affinity DataIC50:  7nMAssay Description:Inhibition EG5 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReverse transcriptase(Human immunodeficiency virus 1)
Gvk Biosciences

Curated by ChEMBL
LigandPNGBDBM50483593(CHEMBL1687958)
Affinity DataIC50:  20nMAssay Description:Inhibition of Human immunodeficiency virus 1 reverse transcriptaseMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetReverse transcriptase(Human immunodeficiency virus 1)
Gvk Biosciences

Curated by ChEMBL
LigandPNGBDBM50483585(CHEMBL1689308)
Affinity DataIC50:  24nMAssay Description:Inhibition of Human immunodeficiency virus 1 reverse transcriptaseMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetReverse transcriptase(Human immunodeficiency virus 1)
Gvk Biosciences

Curated by ChEMBL
LigandPNGBDBM50483586(CHEMBL1689309)
Affinity DataIC50:  27nMAssay Description:Inhibition of Human immunodeficiency virus 1 reverse transcriptaseMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetReverse transcriptase(Human immunodeficiency virus 1)
Gvk Biosciences

Curated by ChEMBL
LigandPNGBDBM50483574(CHEMBL1689310)
Affinity DataIC50:  31nMAssay Description:Inhibition of Human immunodeficiency virus 1 reverse transcriptaseMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetReverse transcriptase(Human immunodeficiency virus 1)
Gvk Biosciences

Curated by ChEMBL
LigandPNGBDBM50483587(CHEMBL1689312)
Affinity DataIC50:  54nMAssay Description:Inhibition of Human immunodeficiency virus 1 reverse transcriptaseMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetReverse transcriptase(Human immunodeficiency virus 1)
Gvk Biosciences

Curated by ChEMBL
LigandPNGBDBM50483590(CHEMBL1689311)
Affinity DataIC50:  80nMAssay Description:Inhibition of Human immunodeficiency virus 1 reverse transcriptaseMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetReverse transcriptase(Human immunodeficiency virus 1)
Gvk Biosciences

Curated by ChEMBL
LigandPNGBDBM50483596(CHEMBL1689314)
Affinity DataIC50:  100nMAssay Description:Inhibition of Human immunodeficiency virus 1 reverse transcriptaseMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetReverse transcriptase(Human immunodeficiency virus 1)
Gvk Biosciences

Curated by ChEMBL
LigandPNGBDBM50483575(CHEMBL1689313)
Affinity DataIC50:  111nMAssay Description:Inhibition of Human immunodeficiency virus 1 reverse transcriptaseMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetReverse transcriptase(Human immunodeficiency virus 1)
Gvk Biosciences

Curated by ChEMBL
LigandPNGBDBM50483591(CHEMBL1689315)
Affinity DataIC50:  137nMAssay Description:Inhibition of Human immunodeficiency virus 1 reverse transcriptaseMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetReverse transcriptase(Human immunodeficiency virus 1)
Gvk Biosciences

Curated by ChEMBL
LigandPNGBDBM50483576(CHEMBL1689316)
Affinity DataIC50:  210nMAssay Description:Inhibition of Human immunodeficiency virus 1 reverse transcriptaseMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetReverse transcriptase(Human immunodeficiency virus 1)
Gvk Biosciences

Curated by ChEMBL
LigandPNGBDBM50483578(CHEMBL1689318)
Affinity DataIC50:  240nMAssay Description:Inhibition of Human immunodeficiency virus 1 reverse transcriptaseMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetReverse transcriptase(Human immunodeficiency virus 1)
Gvk Biosciences

Curated by ChEMBL
LigandPNGBDBM50483577(CHEMBL1689317)
Affinity DataIC50:  300nMAssay Description:Inhibition of Human immunodeficiency virus 1 reverse transcriptaseMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetReverse transcriptase(Human immunodeficiency virus 1)
Gvk Biosciences

Curated by ChEMBL
LigandPNGBDBM50483592(CHEMBL1689319)
Affinity DataIC50:  375nMAssay Description:Inhibition of Human immunodeficiency virus 1 reverse transcriptaseMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetReverse transcriptase(Human immunodeficiency virus 1)
Gvk Biosciences

Curated by ChEMBL
LigandPNGBDBM50483579(CHEMBL1689321)
Affinity DataIC50:  404nMAssay Description:Inhibition of Human immunodeficiency virus 1 reverse transcriptaseMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetReverse transcriptase(Human immunodeficiency virus 1)
Gvk Biosciences

Curated by ChEMBL
LigandPNGBDBM50483594(CHEMBL1689320)
Affinity DataIC50:  422nMAssay Description:Inhibition of Human immunodeficiency virus 1 reverse transcriptaseMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetReverse transcriptase(Human immunodeficiency virus 1)
Gvk Biosciences

Curated by ChEMBL
LigandPNGBDBM50483580(CHEMBL1689322)
Affinity DataIC50:  473nMAssay Description:Inhibition of Human immunodeficiency virus 1 reverse transcriptaseMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetReverse transcriptase(Human immunodeficiency virus 1)
Gvk Biosciences

Curated by ChEMBL
LigandPNGBDBM50483588(CHEMBL1689323)
Affinity DataIC50:  597nMAssay Description:Inhibition of Human immunodeficiency virus 1 reverse transcriptaseMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetKinesin-like protein KIF11(Homo sapiens (Human))
University Of Kwazulu-Natal (Ukzn)

Curated by ChEMBL
LigandPNGBDBM50431886(CHEMBL1413473)
Affinity DataIC50:  800nMAssay Description:Inhibition of MT-stimulated EG5 ATPase activity (unknown origin) by pyruvate kinase/lactate dehydrogenase enzyme coupled photometric assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKinesin-like protein KIF11(Homo sapiens (Human))
University Of Kwazulu-Natal (Ukzn)

Curated by ChEMBL
LigandPNGBDBM50431886(CHEMBL1413473)
Affinity DataIC50:  1.30E+3nMAssay Description:Inhibition EG5 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Electrophorus electricus (Electric eel))
Ramkhamhaeng University

Curated by ChEMBL
LigandPNGBDBM50433757(CHEMBL2381443)
Affinity DataIC50:  1.34E+3nMAssay Description:Inhibition of electric eel AChE using acetylthiocholine iodide as substrate after 15 mins by Ellman's methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Electrophorus electricus (Electric eel))
Ramkhamhaeng University

Curated by ChEMBL
LigandPNGBDBM10404((1S,12S,14R)-9-methoxy-4-methyl-11-oxa-4-azatetrac...)
Affinity DataIC50:  1.45E+3nMAssay Description:Inhibition of electric eel AChE using acetylthiocholine iodide as substrate after 15 mins by Ellman's methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Electrophorus electricus (Electric eel))
Ramkhamhaeng University

Curated by ChEMBL
LigandPNGBDBM50433756(CHEMBL2381442)
Affinity DataIC50:  2.04E+3nMAssay Description:Inhibition of electric eel AChE using acetylthiocholine iodide as substrate after 15 mins by Ellman's methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKinesin-like protein KIF11(Homo sapiens (Human))
University Of Kwazulu-Natal (Ukzn)

Curated by ChEMBL
LigandPNGBDBM24174(3-N,3-N-diethyl-5,5-dimethyl-2-N-(thiophene-2-)-4,...)
Affinity DataIC50:  3.10E+3nMAssay Description:Inhibition EG5 (unknown origin)More data for this Ligand-Target Pair
TargetKinesin-like protein KIF11(Homo sapiens (Human))
University Of Kwazulu-Natal (Ukzn)

Curated by ChEMBL
LigandPNGBDBM88776(2-[4-[(Z)-[5-(4-chlorophenyl)-6-isopropoxycarbonyl...)
Affinity DataIC50:  4.60E+3nMAssay Description:Inhibition EG5 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Electrophorus electricus (Electric eel))
Ramkhamhaeng University

Curated by ChEMBL
LigandPNGBDBM50433755(CHEMBL2381440)
Affinity DataIC50:  5.78E+3nMAssay Description:Inhibition of electric eel AChE using acetylthiocholine iodide as substrate after 15 mins by Ellman's methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Electrophorus electricus (Electric eel))
Ramkhamhaeng University

Curated by ChEMBL
LigandPNGBDBM50433754(LETESTUIANIN C | Tetrahydrobisdemethoxycurcumin)
Affinity DataIC50:  7.89E+3nMAssay Description:Inhibition of electric eel AChE using acetylthiocholine iodide as substrate after 15 mins by Ellman's methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Electrophorus electricus (Electric eel))
Ramkhamhaeng University

Curated by ChEMBL
LigandPNGBDBM50433753(CHEMBL2381441)
Affinity DataIC50:  9.10E+3nMAssay Description:Inhibition of electric eel AChE using acetylthiocholine iodide as substrate after 15 mins by Ellman's methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Electrophorus electricus (Electric eel))
Ramkhamhaeng University

Curated by ChEMBL
LigandPNGBDBM50433752(CHEMBL2381438)
Affinity DataIC50:  1.07E+4nMAssay Description:Inhibition of electric eel AChE using acetylthiocholine iodide as substrate after 15 mins by Ellman's methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKinesin-like protein KIF11(Homo sapiens (Human))
University Of Kwazulu-Natal (Ukzn)

Curated by ChEMBL
LigandPNGBDBM50463314(CHEMBL4246367)
Affinity DataIC50:  1.32E+4nMAssay Description:Inhibition of MT-stimulated EG5 ATPase activity (unknown origin) by pyruvate kinase/lactate dehydrogenase enzyme coupled photometric assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Electrophorus electricus (Electric eel))
Ramkhamhaeng University

Curated by ChEMBL
LigandPNGBDBM50433751(CHEMBL2381434)
Affinity DataIC50:  1.43E+4nMAssay Description:Inhibition of electric eel AChE using acetylthiocholine iodide as substrate after 15 mins by Ellman's methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKinesin-like protein KIF11(Homo sapiens (Human))
University Of Kwazulu-Natal (Ukzn)

Curated by ChEMBL
LigandPNGBDBM50463319(CHEMBL4238439)
Affinity DataIC50:  1.72E+4nMAssay Description:Inhibition of MT-stimulated EG5 ATPase activity (unknown origin) by pyruvate kinase/lactate dehydrogenase enzyme coupled photometric assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Electrophorus electricus (Electric eel))
Ramkhamhaeng University

Curated by ChEMBL
LigandPNGBDBM50433750(CHEMBL2381433)
Affinity DataIC50:  1.73E+4nMAssay Description:Inhibition of electric eel AChE using acetylthiocholine iodide as substrate after 15 mins by Ellman's methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Electrophorus electricus (Electric eel))
Ramkhamhaeng University

Curated by ChEMBL
LigandPNGBDBM50059989((1E,4Z,6E)-5-Hydroxy-1,7-bis-(4-hydroxy-phenyl)-he...)
Affinity DataIC50:  1.83E+4nMAssay Description:Inhibition of electric eel AChE using acetylthiocholine iodide as substrate after 15 mins by Ellman's methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKinesin-like protein KIF11(Homo sapiens (Human))
University Of Kwazulu-Natal (Ukzn)

Curated by ChEMBL
LigandPNGBDBM50463309(CHEMBL4240281)
Affinity DataIC50:  2.02E+4nMAssay Description:Inhibition of MT-stimulated EG5 ATPase activity (unknown origin) by pyruvate kinase/lactate dehydrogenase enzyme coupled photometric assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Electrophorus electricus (Electric eel))
Ramkhamhaeng University

Curated by ChEMBL
LigandPNGBDBM50433749(TETRAHYDRODEMETHOXYCURCUMIN)
Affinity DataIC50:  2.06E+4nMAssay Description:Inhibition of electric eel AChE using acetylthiocholine iodide as substrate after 15 mins by Ellman's methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Electrophorus electricus (Electric eel))
Ramkhamhaeng University

Curated by ChEMBL
LigandPNGBDBM50433748(CHEMBL2381439)
Affinity DataIC50:  2.09E+4nMAssay Description:Inhibition of electric eel AChE using acetylthiocholine iodide as substrate after 15 mins by Ellman's methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKinesin-like protein KIF11(Homo sapiens (Human))
University Of Kwazulu-Natal (Ukzn)

Curated by ChEMBL
LigandPNGBDBM50463308(CHEMBL4241043)
Affinity DataIC50:  2.75E+4nMAssay Description:Inhibition of MT-stimulated EG5 ATPase activity (unknown origin) by pyruvate kinase/lactate dehydrogenase enzyme coupled photometric assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Electrophorus electricus (Electric eel))
Ramkhamhaeng University

Curated by ChEMBL
LigandPNGBDBM50433747(CHEMBL2381430)
Affinity DataIC50:  3.63E+4nMAssay Description:Inhibition of electric eel AChE using acetylthiocholine iodide as substrate after 15 mins by Ellman's methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Electrophorus electricus (Electric eel))
Ramkhamhaeng University

Curated by ChEMBL
LigandPNGBDBM50163744((1E,4Z,6E)-5-Hydroxy-1-(4-hydroxy-3-methoxy-phenyl...)
Affinity DataIC50:  3.77E+4nMAssay Description:Inhibition of electric eel AChE using acetylthiocholine iodide as substrate after 15 mins by Ellman's methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKinesin-like protein KIF11(Homo sapiens (Human))
University Of Kwazulu-Natal (Ukzn)

Curated by ChEMBL
LigandPNGBDBM50463311(CHEMBL4248454)
Affinity DataIC50:  3.92E+4nMAssay Description:Inhibition of MT-stimulated EG5 ATPase activity (unknown origin) by pyruvate kinase/lactate dehydrogenase enzyme coupled photometric assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
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