Compile Data Set for Download or QSAR
maximum 50k data
Found 332 with Last Name = 'asano' and Initial = 'd'
TargetSodium channel subunit beta-2(Homo sapiens)TBA
LigandPNGBDBM145285(US8952169, 64 | US9771376, Example 64)
Affinity DataIC50:  0.400nMAssay Description:Inhibition of human Nav1.7/beta1/2 transfected in HEK293-A cells assessed as inhibition of channel current incubated for 5.5 mins by high-throughput ...More data for this Ligand-Target Pair
In DepthDetails PubMed
LigandPNGBDBM50257179(CHEMBL2325622)
Affinity DataIC50:  0.550nMAssay Description:Inhibition of mouse NaV1.7/beta1/beta2 expressed in HEK293A cells by Ionworks high-throughput electrophysiology methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium channel subunit beta-2(Homo sapiens)TBA
LigandPNGBDBM70937(US9546164, 100 | US9694002, 100)
Affinity DataIC50:  0.600nMAssay Description:Inhibition of human Nav1.7/beta1/2 transfected in HEK293-A cells assessed as inhibition of channel current incubated for 5.5 mins by high-throughput ...More data for this Ligand-Target Pair
In DepthDetails PubMed
TargetSodium channel subunit beta-2(Homo sapiens)TBA
LigandPNGBDBM50257179(CHEMBL2325622)
Affinity DataIC50:  1.90nMAssay Description:Inhibition of human NaV1.7/beta1/beta2 expressed in HEK293A cells by Ionworks high-throughput electrophysiology methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium channel subunit beta-2(Mus musculus)
Daiichi Sankyo

Curated by ChEMBL
LigandPNGBDBM50240267(CHEMBL2325014)
Affinity DataIC50:  4.90nMAssay Description:Inhibition of mouse NaV1.7/beta1/beta2 expressed in HEK293A cells by Ionworks high-throughput electrophysiology methodMore data for this Ligand-Target Pair
LigandPNGBDBM145285(US8952169, 64 | US9771376, Example 64)
Affinity DataIC50:  11nMAssay Description:Inhibition of human Nav1.1/beta1/2 transfected in HEK293-A cells assessed as inhibition of channel current incubated for 5.5 mins by high-throughput ...More data for this Ligand-Target Pair
In DepthDetails PubMed
TargetSodium channel subunit beta-2(Homo sapiens)TBA
LigandPNGBDBM258102(US9493448, 4 | US9845313, Example 4)
Affinity DataIC50:  12nMAssay Description:Inhibition of human NaV1.7/beta1/beta2 expressed in HEK293A cells by Ionworks high-throughput electrophysiology methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSodium channel subunit beta-2(Homo sapiens)TBA
LigandPNGBDBM50240267(CHEMBL2325014)
Affinity DataIC50:  13nMAssay Description:Inhibition of human NaV1.7/beta1/beta2 expressed in HEK293A cells by Ionworks high-throughput electrophysiology methodMore data for this Ligand-Target Pair
TargetSodium channel subunit beta-2(Homo sapiens)TBA
LigandPNGBDBM50613335(CHEMBL5288162)
Affinity DataIC50:  14nMAssay Description:Inhibition of human Nav1.7/beta1/2 transfected in HEK293-A cells assessed as inhibition of channel current incubated for 5.5 mins by high-throughput ...More data for this Ligand-Target Pair
Ligand Info
In DepthDetails PubMed
TargetSodium channel subunit beta-2(Mus musculus)
Daiichi Sankyo

Curated by ChEMBL
LigandPNGBDBM50613344(CHEMBL5284082)
Affinity DataIC50:  15nMAssay Description:Inhibition of mouse Nav1.7/beta1/2 transfected in HEK293-A cells assessed as inhibition of channel current incubated for 5.5 mins by high-throughput ...More data for this Ligand-Target Pair
Ligand Info
In DepthDetails PubMed
TargetSodium channel subunit beta-2(Homo sapiens)TBA
LigandPNGBDBM50613342(CHEMBL5286433)
Affinity DataIC50:  15nMAssay Description:Inhibition of human Nav1.7/beta1/2 transfected in HEK293-A cells assessed as inhibition of channel current incubated for 5.5 mins by high-throughput ...More data for this Ligand-Target Pair
Ligand Info
In DepthDetails PubMed
TargetSodium channel subunit beta-2(Mus musculus)
Daiichi Sankyo

Curated by ChEMBL
LigandPNGBDBM258162(US9493448, 64 | US9597330, Example 21 | US9845313,...)
Affinity DataIC50:  15nMAssay Description:Inhibition of mouse NaV1.7/beta1/beta2 expressed in HEK293A cells by Ionworks high-throughput electrophysiology methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSodium channel subunit beta-2(Mus musculus)
Daiichi Sankyo

Curated by ChEMBL
LigandPNGBDBM50613336(CHEMBL5276801)
Affinity DataIC50:  16nMAssay Description:Inhibition of mouse Nav1.7/beta1/2 transfected in HEK293-A cells assessed as inhibition of channel current incubated for 5.5 mins by high-throughput ...More data for this Ligand-Target Pair
Ligand Info
In DepthDetails PubMed
TargetSodium channel subunit beta-2(Homo sapiens)TBA
LigandPNGBDBM258106(US9493448, 8 | US9845313, Example 8)
Affinity DataIC50:  17nMAssay Description:Inhibition of human NaV1.7/beta1/beta2 expressed in HEK293A cells by Ionworks high-throughput electrophysiology methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSodium channel subunit beta-2(Mus musculus)
Daiichi Sankyo

Curated by ChEMBL
LigandPNGBDBM258102(US9493448, 4 | US9845313, Example 4)
Affinity DataIC50:  17nMAssay Description:Inhibition of mouse NaV1.7/beta1/beta2 expressed in HEK293A cells by Ionworks high-throughput electrophysiology methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSodium channel subunit beta-2(Homo sapiens)TBA
LigandPNGBDBM50613336(CHEMBL5276801)
Affinity DataIC50:  19nMAssay Description:Inhibition of human Nav1.7/beta1/2 transfected in HEK293-A cells assessed as inhibition of channel current incubated for 5.5 mins by high-throughput ...More data for this Ligand-Target Pair
Ligand Info
In DepthDetails PubMed
TargetSodium channel protein type 9 subunit alpha(Homo sapiens (Human))
Daiichi Sankyo

Curated by ChEMBL
LigandPNGBDBM258146(US9493448, 122 | US9493448, 154 | US9493448, 48 | ...)
Affinity DataIC50:  23nMAssay Description:Inhibition of human Nav1.7 expressed in CHO cells with -120 mV holding potential by whole cell manual patch clamp methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium channel subunit beta-2(Homo sapiens)TBA
LigandPNGBDBM258141(US9493448, 43 | US9597330, Example 10 | US9845313,...)
Affinity DataIC50:  24nMAssay Description:Inhibition of human NaV1.7/beta1/beta2 expressed in HEK293A cells by Ionworks high-throughput electrophysiology methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSodium channel subunit beta-2(Homo sapiens)TBA
LigandPNGBDBM258146(US9493448, 122 | US9493448, 154 | US9493448, 48 | ...)
Affinity DataIC50:  24.5nMAssay Description:Inhibition of human NaV1.7/beta1/beta2 expressed in HEK293A cells by Ionworks high-throughput electrophysiology methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium channel subunit beta-2(Homo sapiens)TBA
LigandPNGBDBM258146(US9493448, 122 | US9493448, 154 | US9493448, 48 | ...)
Affinity DataIC50:  25nMAssay Description:Inhibition of human NaV1.7/beta1/beta2 expressed in HEK293A cells by Ionworks high-throughput electrophysiology methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium channel subunit beta-2(Mus musculus)
Daiichi Sankyo

Curated by ChEMBL
LigandPNGBDBM258146(US9493448, 122 | US9493448, 154 | US9493448, 48 | ...)
Affinity DataIC50:  26.5nMAssay Description:Inhibition of mouse NaV1.7/beta1/beta2 expressed in HEK293A cells by Ionworks high-throughput electrophysiology methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium channel subunit beta-2(Mus musculus)
Daiichi Sankyo

Curated by ChEMBL
LigandPNGBDBM258146(US9493448, 122 | US9493448, 154 | US9493448, 48 | ...)
Affinity DataIC50:  27nMAssay Description:Inhibition of mouse NaV1.7/beta1/beta2 expressed in HEK293A cells by Ionworks high-throughput electrophysiology methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium channel subunit beta-2(Mus musculus)
Daiichi Sankyo

Curated by ChEMBL
LigandPNGBDBM258141(US9493448, 43 | US9597330, Example 10 | US9845313,...)
Affinity DataIC50:  28nMAssay Description:Inhibition of mouse NaV1.7/beta1/beta2 expressed in HEK293A cells by Ionworks high-throughput electrophysiology methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSodium channel subunit beta-2(Mus musculus)
Daiichi Sankyo

Curated by ChEMBL
LigandPNGBDBM258118(US9493448, 20 | US9597330, Example 2 | US9845313, ...)
Affinity DataIC50:  28nMAssay Description:Inhibition of mouse NaV1.7/beta1/beta2 expressed in HEK293A cells by Ionworks high-throughput electrophysiology methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSodium channel subunit beta-2(Homo sapiens)TBA
LigandPNGBDBM301817(5-Chloro-2-fluoro-4-{[(1S*,2R*)-2-(1-methyl-1H-pyr...)
Affinity DataIC50:  28nMAssay Description:Inhibition of human NaV1.7/beta1/beta2 expressed in HEK293A cells by Ionworks high-throughput electrophysiology methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSodium channel subunit beta-2(Homo sapiens)TBA
LigandPNGBDBM258113(US9493448, 15 | US9845313, Example 15)
Affinity DataIC50:  28nMAssay Description:Inhibition of human NaV1.7/beta1/beta2 expressed in HEK293A cells by Ionworks high-throughput electrophysiology methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSodium channel subunit beta-2(Homo sapiens)TBA
LigandPNGBDBM258144(US9493448, 46 | US9597330, Example 11 | US9845313,...)
Affinity DataIC50:  30nMAssay Description:Inhibition of human NaV1.7/beta1/beta2 expressed in HEK293A cells by Ionworks high-throughput electrophysiology methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSodium channel subunit beta-2(Homo sapiens)TBA
LigandPNGBDBM258162(US9493448, 64 | US9597330, Example 21 | US9845313,...)
Affinity DataIC50:  31nMAssay Description:Inhibition of human NaV1.7/beta1/beta2 expressed in HEK293A cells by Ionworks high-throughput electrophysiology methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetNicotinamide phosphoribosyltransferase(Homo sapiens (Human))
Daiichi Sankyo

Curated by ChEMBL
LigandPNGBDBM50570846(CHEMBL4847819)
Affinity DataIC50:  32nMAssay Description:Inhibition of human NAMPT assessed as decrease in NMN production by fluorescence based analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSodium channel subunit beta-2(Homo sapiens)TBA
LigandPNGBDBM50613337(CHEMBL5286829)
Affinity DataIC50:  32nMAssay Description:Inhibition of human Nav1.7/beta1/2 transfected in HEK293-A cells assessed as inhibition of channel current incubated for 5.5 mins by high-throughput ...More data for this Ligand-Target Pair
Ligand Info
In DepthDetails PubMed
TargetSodium channel subunit beta-2(Homo sapiens)TBA
LigandPNGBDBM50613334(CHEMBL5270366)
Affinity DataIC50:  34nMAssay Description:Inhibition of human Nav1.7/beta1/2 transfected in HEK293-A cells assessed as inhibition of channel current incubated for 5.5 mins by high-throughput ...More data for this Ligand-Target Pair
Ligand Info
In DepthDetails PubMed
TargetSodium channel subunit beta-2(Homo sapiens)TBA
LigandPNGBDBM50613328(CHEMBL5280425)
Affinity DataIC50:  38nMAssay Description:Inhibition of human Nav1.7/beta1/2 transfected in HEK293-A cells assessed as inhibition of channel current incubated for 5.5 mins by high-throughput ...More data for this Ligand-Target Pair
Ligand Info
In DepthDetails PubMed
TargetSodium channel subunit beta-2(Homo sapiens)TBA
LigandPNGBDBM50613344(CHEMBL5284082)
Affinity DataIC50:  40nMAssay Description:Inhibition of human Nav1.7/beta1/2 transfected in HEK293-A cells assessed as inhibition of channel current incubated for 5.5 mins by high-throughput ...More data for this Ligand-Target Pair
Ligand Info
In DepthDetails PubMed
TargetSodium channel subunit beta-2(Mus musculus)
Daiichi Sankyo

Curated by ChEMBL
LigandPNGBDBM301817(5-Chloro-2-fluoro-4-{[(1S*,2R*)-2-(1-methyl-1H-pyr...)
Affinity DataIC50:  41nMAssay Description:Inhibition of mouse NaV1.7/beta1/beta2 expressed in HEK293A cells by Ionworks high-throughput electrophysiology methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSodium channel subunit beta-2(Homo sapiens)TBA
LigandPNGBDBM258118(US9493448, 20 | US9597330, Example 2 | US9845313, ...)
Affinity DataIC50:  45nMAssay Description:Inhibition of human NaV1.7/beta1/beta2 expressed in HEK293A cells by Ionworks high-throughput electrophysiology methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
LigandPNGBDBM145285(US8952169, 64 | US9771376, Example 64)
Affinity DataIC50:  51nMAssay Description:Inhibition of human Nav1.5/beta1/2 transfected in HEK293-A cells assessed as inhibition of channel current incubated for 5.5 mins by high-throughput ...More data for this Ligand-Target Pair
In DepthDetails PubMed
TargetSodium channel subunit beta-2(Homo sapiens)TBA
LigandPNGBDBM50405441(CHEMBL5286125)
Affinity DataIC50:  52nMAssay Description:Inhibition of human Nav1.7/beta1/2 transfected in HEK293-A cells assessed as inhibition of channel current incubated for 5.5 mins by high-throughput ...More data for this Ligand-Target Pair
In DepthDetails PubMed
TargetSodium channel subunit beta-2(Mus musculus)
Daiichi Sankyo

Curated by ChEMBL
LigandPNGBDBM258144(US9493448, 46 | US9597330, Example 11 | US9845313,...)
Affinity DataIC50:  56nMAssay Description:Inhibition of mouse NaV1.7/beta1/beta2 expressed in HEK293A cells by Ionworks high-throughput electrophysiology methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSodium channel subunit beta-2(Homo sapiens)TBA
LigandPNGBDBM50613332(CHEMBL5285313)
Affinity DataIC50:  58nMAssay Description:Inhibition of human Nav1.7/beta1/2 transfected in HEK293-A cells assessed as inhibition of channel current incubated for 5.5 mins by high-throughput ...More data for this Ligand-Target Pair
Ligand Info
In DepthDetails PubMed
TargetSodium channel subunit beta-2(Mus musculus)
Daiichi Sankyo

Curated by ChEMBL
LigandPNGBDBM258146(US9493448, 122 | US9493448, 154 | US9493448, 48 | ...)
Affinity DataIC50:  59nMAssay Description:Inhibition of mouse Nav1.7/beta1/beta2 expressed in HEK293A cells with -120 mV holding potential by whole cell manual patch clamp methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium channel subunit beta-2(Homo sapiens)TBA
LigandPNGBDBM50613343(CHEMBL5287784)
Affinity DataIC50:  59nMAssay Description:Inhibition of human Nav1.7/beta1/2 transfected in HEK293-A cells assessed as inhibition of channel current incubated for 5.5 mins by high-throughput ...More data for this Ligand-Target Pair
Ligand Info
In DepthDetails PubMed
TargetSodium channel subunit beta-2(Homo sapiens)TBA
LigandPNGBDBM258125(US9493448, 27 | US9597330, Example 4 | US9845313, ...)
Affinity DataIC50:  60nMAssay Description:Inhibition of human NaV1.7/beta1/beta2 expressed in HEK293A cells by Ionworks high-throughput electrophysiology methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSodium channel subunit beta-2(Mus musculus)
Daiichi Sankyo

Curated by ChEMBL
LigandPNGBDBM50613342(CHEMBL5286433)
Affinity DataIC50:  61nMAssay Description:Inhibition of mouse Nav1.7/beta1/2 transfected in HEK293-A cells assessed as inhibition of channel current incubated for 5.5 mins by high-throughput ...More data for this Ligand-Target Pair
Ligand Info
In DepthDetails PubMed
TargetSodium channel subunit beta-2(Homo sapiens)TBA
LigandPNGBDBM50613341(CHEMBL5267728)
Affinity DataIC50:  85nMAssay Description:Inhibition of human Nav1.7/beta1/2 transfected in HEK293-A cells assessed as inhibition of channel current incubated for 5.5 mins by high-throughput ...More data for this Ligand-Target Pair
Ligand Info
In DepthDetails PubMed
TargetSodium channel subunit beta-2(Homo sapiens)TBA
LigandPNGBDBM50613330(CHEMBL5269981)
Affinity DataIC50:  87nMAssay Description:Inhibition of human Nav1.7/beta1/2 transfected in HEK293-A cells assessed as inhibition of channel current incubated for 5.5 mins by high-throughput ...More data for this Ligand-Target Pair
Ligand Info
In DepthDetails PubMed
TargetSodium channel subunit beta-2(Mus musculus)
Daiichi Sankyo

Curated by ChEMBL
LigandPNGBDBM258125(US9493448, 27 | US9597330, Example 4 | US9845313, ...)
Affinity DataIC50:  96nMAssay Description:Inhibition of mouse NaV1.7/beta1/beta2 expressed in HEK293A cells by Ionworks high-throughput electrophysiology methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSodium channel subunit beta-2(Mus musculus)
Daiichi Sankyo

Curated by ChEMBL
LigandPNGBDBM258113(US9493448, 15 | US9845313, Example 15)
Affinity DataIC50:  100nMAssay Description:Inhibition of mouse NaV1.7/beta1/beta2 expressed in HEK293A cells by Ionworks high-throughput electrophysiology methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSodium channel protein type 9 subunit alpha(Mus musculus)
Daiichi Sankyo

Curated by ChEMBL
LigandPNGBDBM50130532(CHEMBL3632692)
Affinity DataIC50:  100nMAssay Description:Inhibition of mouse NaV1.7 by IonWorks quattro automated electrophysiology assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium channel subunit beta-2(Homo sapiens)TBA
LigandPNGBDBM258123(US9493448, 25 | US9597330, Example 3 | US9845313, ...)
Affinity DataIC50:  113nMAssay Description:Inhibition of human NaV1.7/beta1/beta2 expressed in HEK293A cells by Ionworks high-throughput electrophysiology methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSodium channel subunit beta-2(Homo sapiens)TBA
LigandPNGBDBM258112(US9493448, 14 | US9493448, 31 | US9597330, Example...)
Affinity DataIC50:  180nMAssay Description:Inhibition of human NaV1.7/beta1/beta2 expressed in HEK293A cells by Ionworks high-throughput electrophysiology methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
Displayed 1 to 50 (of 332 total ) | Next | Last >>
Jump to: