Affinity DataIC50: 2.30nMAssay Description:Binding affinity to human fibrinogen receptorMore data for this Ligand-Target Pair
Affinity DataIC50: 2.60nMAssay Description:Binding affinity to human fibrinogen receptorMore data for this Ligand-Target Pair
Affinity DataIC50: 2.70nMAssay Description:Binding affinity to human fibrinogen receptorMore data for this Ligand-Target Pair
Affinity DataIC50: 2.70nMAssay Description:Binding affinity to human fibrinogen receptorMore data for this Ligand-Target Pair
Affinity DataIC50: 2.70nMAssay Description:Binding affinity to human fibrinogen receptorMore data for this Ligand-Target Pair
Affinity DataIC50: 3.80nMAssay Description:Binding affinity to human fibrinogen receptorMore data for this Ligand-Target Pair
Affinity DataIC50: 4nMAssay Description:Binding affinity to human fibrinogen receptorMore data for this Ligand-Target Pair
Affinity DataIC50: 4.30nMAssay Description:Binding affinity to human fibrinogen receptorMore data for this Ligand-Target Pair
Affinity DataIC50: 5nMAssay Description:Binding affinity to human fibrinogen receptorMore data for this Ligand-Target Pair
Affinity DataIC50: 5.10nMAssay Description:Binding affinity to human fibrinogen receptorMore data for this Ligand-Target Pair
Affinity DataIC50: 5.30nMAssay Description:Binding affinity to human fibrinogen receptorMore data for this Ligand-Target Pair
Affinity DataIC50: 5.40nMAssay Description:Binding affinity to human fibrinogen receptorMore data for this Ligand-Target Pair
Affinity DataIC50: 5.60nMAssay Description:Binding affinity to human fibrinogen receptorMore data for this Ligand-Target Pair
Affinity DataIC50: 5.70nMAssay Description:Binding affinity to human fibrinogen receptorMore data for this Ligand-Target Pair
Affinity DataIC50: 5.80nMAssay Description:Binding affinity to human fibrinogen receptorMore data for this Ligand-Target Pair
Affinity DataIC50: 7nMAssay Description:Binding affinity to human fibrinogen receptorMore data for this Ligand-Target Pair
Affinity DataIC50: 8.60nMAssay Description:Binding affinity to human fibrinogen receptorMore data for this Ligand-Target Pair
Affinity DataIC50: 13nMAssay Description:Binding affinity to human fibrinogen receptorMore data for this Ligand-Target Pair
Affinity DataIC50: 21nMAssay Description:Binding affinity to human fibrinogen receptorMore data for this Ligand-Target Pair
Affinity DataIC50: 21.3nMAssay Description:Binding affinity to human fibrinogen receptorMore data for this Ligand-Target Pair
Affinity DataIC50: 22.3nMAssay Description:Binding affinity to human fibrinogen receptorMore data for this Ligand-Target Pair
Affinity DataIC50: 23.7nMAssay Description:Binding affinity to human fibrinogen receptorMore data for this Ligand-Target Pair
Affinity DataIC50: 25.3nMAssay Description:Binding affinity to human fibrinogen receptorMore data for this Ligand-Target Pair
Affinity DataIC50: 27.3nMAssay Description:Binding affinity to human fibrinogen receptorMore data for this Ligand-Target Pair
Affinity DataIC50: 31.3nMAssay Description:Binding affinity to human fibrinogen receptorMore data for this Ligand-Target Pair
Affinity DataIC50: 34.7nMAssay Description:Binding affinity to human fibrinogen receptorMore data for this Ligand-Target Pair
Affinity DataIC50: 36nMAssay Description:Binding affinity to human fibrinogen receptorMore data for this Ligand-Target Pair
Affinity DataIC50: 47.3nMAssay Description:Binding affinity to human fibrinogen receptorMore data for this Ligand-Target Pair
Affinity DataIC50: 125nMAssay Description:Binding affinity to human fibrinogen receptorMore data for this Ligand-Target Pair
TargetGrowth/differentiation factor 8(Homo sapiens (Human))
Tokyo University Of Pharmacy And Life Sciences
Curated by ChEMBL
Tokyo University Of Pharmacy And Life Sciences
Curated by ChEMBL
Affinity DataIC50: 130nMAssay Description:Inhibition of myostatin (unknown origin) expressed in HEK293 cells incubated for 4 hrs by dual luciferase reporter gene assayMore data for this Ligand-Target Pair
TargetGrowth/differentiation factor 8(Homo sapiens (Human))
Tokyo University Of Pharmacy And Life Sciences
Curated by ChEMBL
Tokyo University Of Pharmacy And Life Sciences
Curated by ChEMBL
Affinity DataIC50: 290nMAssay Description:Inhibition of myostatin (unknown origin) expressed in HEK293 cells incubated for 4 hrs by dual luciferase reporter gene assayMore data for this Ligand-Target Pair
TargetGrowth/differentiation factor 8(Homo sapiens (Human))
Tokyo University Of Pharmacy And Life Sciences
Curated by ChEMBL
Tokyo University Of Pharmacy And Life Sciences
Curated by ChEMBL
Affinity DataIC50: 320nMAssay Description:Inhibition of recombinant myostatin (unknown origin) expressed in HEK293 cells after 4 hrs by dual-luciferase reporter gene assayMore data for this Ligand-Target Pair
Affinity DataIC50: 363nMAssay Description:Binding affinity to human fibrinogen receptorMore data for this Ligand-Target Pair
TargetGrowth/differentiation factor 8(Homo sapiens (Human))
Tokyo University Of Pharmacy And Life Sciences
Curated by ChEMBL
Tokyo University Of Pharmacy And Life Sciences
Curated by ChEMBL
Affinity DataIC50: 1.19E+3nMAssay Description:Inhibition of recombinant myostatin (unknown origin) expressed in HEK293 cells after 4 hrs by dual-luciferase reporter gene assayMore data for this Ligand-Target Pair
TargetGrowth/differentiation factor 8(Homo sapiens (Human))
Tokyo University Of Pharmacy And Life Sciences
Curated by ChEMBL
Tokyo University Of Pharmacy And Life Sciences
Curated by ChEMBL
Affinity DataIC50: 1.20E+3nMAssay Description:Inhibition of human recombinant myostatin expressed in HEK293 cells after 4 hrs by SBE4 based luciferase reporter gene assayMore data for this Ligand-Target Pair
TargetGrowth/differentiation factor 8(Homo sapiens (Human))
Tokyo University Of Pharmacy And Life Sciences
Curated by ChEMBL
Tokyo University Of Pharmacy And Life Sciences
Curated by ChEMBL
Affinity DataIC50: 3.56E+3nMAssay Description:Inhibition of recombinant myostatin (unknown origin) expressed in HEK293 cells after 4 hrs by dual-luciferase reporter gene assayMore data for this Ligand-Target Pair
TargetGrowth/differentiation factor 8(Homo sapiens (Human))
Tokyo University Of Pharmacy And Life Sciences
Curated by ChEMBL
Tokyo University Of Pharmacy And Life Sciences
Curated by ChEMBL
Affinity DataIC50: 4.10E+3nMAssay Description:Inhibition of human recombinant myostatin pre-incubated with compound for 1 hr before addition to human HepG2 cells assessed as reduction in myostati...More data for this Ligand-Target Pair
TargetNeuromedin-U receptor 1(Homo sapiens (Human))
Tokyo University Of Pharmacy And Life Sciences
Curated by ChEMBL
Tokyo University Of Pharmacy And Life Sciences
Curated by ChEMBL
Affinity DataEC50: 1.70nMAssay Description:Partial agonist activity at human NMUR1 expressed in CHO cells by calcium mobilization assayMore data for this Ligand-Target Pair
TargetNeuromedin-U receptor 1(Homo sapiens (Human))
Tokyo University Of Pharmacy And Life Sciences
Curated by ChEMBL
Tokyo University Of Pharmacy And Life Sciences
Curated by ChEMBL
Affinity DataEC50: 30nMAssay Description:Agonist activity at human NMUR1 expressed in CHO cells by calcium mobilization assayMore data for this Ligand-Target Pair
TargetNeuromedin-U receptor 1(Homo sapiens (Human))
Tokyo University Of Pharmacy And Life Sciences
Curated by ChEMBL
Tokyo University Of Pharmacy And Life Sciences
Curated by ChEMBL
Affinity DataEC50: 3.20nMAssay Description:Agonist activity at human NMUR1 expressed in CHO cells by calcium mobilization assayMore data for this Ligand-Target Pair
TargetGrowth/differentiation factor 8(Homo sapiens (Human))
Tokyo University Of Pharmacy And Life Sciences
Curated by ChEMBL
Tokyo University Of Pharmacy And Life Sciences
Curated by ChEMBL
Affinity DataKd: 117nMAssay Description:Binding affinity to recombinant myostatin (unknown origin) by surface plasmon resonance assayMore data for this Ligand-Target Pair
TargetGrowth/differentiation factor 8(Homo sapiens (Human))
Tokyo University Of Pharmacy And Life Sciences
Curated by ChEMBL
Tokyo University Of Pharmacy And Life Sciences
Curated by ChEMBL
Affinity DataKd: 30nMAssay Description:Binding affinity to recombinant myostatin (unknown origin) by surface plasmon resonance assayMore data for this Ligand-Target Pair
TargetGrowth/differentiation factor 8(Homo sapiens (Human))
Tokyo University Of Pharmacy And Life Sciences
Curated by ChEMBL
Tokyo University Of Pharmacy And Life Sciences
Curated by ChEMBL
Affinity DataKd: 36nMAssay Description:Binding affinity to recombinant myostatin (unknown origin) by surface plasmon resonance assayMore data for this Ligand-Target Pair
TargetNeuromedin-U receptor 2(Homo sapiens (Human))
Tokyo University Of Pharmacy And Life Sciences
Curated by ChEMBL
Tokyo University Of Pharmacy And Life Sciences
Curated by ChEMBL
Affinity DataEC50: >1.00E+3nMAssay Description:Agonist activity at human NMUR2 expressed in CHO cells by calcium mobilization assayMore data for this Ligand-Target Pair