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Found 118 with Last Name = 'aust' and Initial = 's'
TargetGlutaminyl-peptide cyclotransferase(Homo sapiens (Human))
Probiodrug

Curated by ChEMBL
LigandPNGBDBM50299858(1-(3,4-Dimethoxyphenyl)-N-(3-(5-methyl-1H-imidazol...)
Affinity DataKi:  2.60nMAssay Description:Inhibition of human glutaminyl cyclase expressed in Pichia pastoris by pGAP coupled enzyme assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutaminyl-peptide cyclotransferase(Homo sapiens (Human))
Probiodrug

Curated by ChEMBL
LigandPNGBDBM50299853(1-(3,4-Dimethoxyphenyl)-3-(3-(5-methyl-1H-imidazol...)
Affinity DataKi:  6.30nMAssay Description:Inhibition of human glutaminyl cyclase expressed in Pichia pastoris by pGAP coupled enzyme assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutaminyl-peptide cyclotransferase(Homo sapiens (Human))
Probiodrug

Curated by ChEMBL
LigandPNGBDBM50299845(3-[3-(5-Methyl-1H-imidazol-1-yl)propyl]-2-thioxo-2...)
Affinity DataKi:  17nMAssay Description:Inhibition of human glutaminyl cyclase expressed in Pichia pastoris by pGAP coupled enzyme assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutaminyl-peptide cyclotransferase(Homo sapiens (Human))
Probiodrug

Curated by ChEMBL
LigandPNGBDBM50299844(2,3-Dihydro-3-(3-(5-methyl-1H-imidazol-1-yl)propyl...)
Affinity DataKi:  18nMAssay Description:Inhibition of human glutaminyl cyclase expressed in Pichia pastoris by pGAP coupled enzyme assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutaminyl-peptide cyclotransferase(Homo sapiens (Human))
Probiodrug

Curated by ChEMBL
LigandPNGBDBM50299847(6-Benzyl-2,3-dihydro-3-(3-(5-methyl-1H-imidazol-1-...)
Affinity DataKi:  20nMAssay Description:Inhibition of human glutaminyl cyclase expressed in Pichia pastoris by pGAP coupled enzyme assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutaminyl-peptide cyclotransferase(Homo sapiens (Human))
Probiodrug

Curated by ChEMBL
LigandPNGBDBM50299866(CHEMBL578153 | N-(1-(3-(5-Methyl-1H-imidazol-1-yl)...)
Affinity DataKi:  34nMAssay Description:Inhibition of human glutaminyl cyclase expressed in Pichia pastoris by pGAP coupled enzyme assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutaminyl-peptide cyclotransferase(Homo sapiens (Human))
Probiodrug

Curated by ChEMBL
LigandPNGBDBM50299846(3-[3-(5-Methyl-1H-imidazol-1-yl)propyl]-2-thioxo-2...)
Affinity DataKi:  39nMAssay Description:Inhibition of human glutaminyl cyclase expressed in Pichia pastoris by pGAP coupled enzyme assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutaminyl-peptide cyclotransferase(Homo sapiens (Human))
Probiodrug

Curated by ChEMBL
LigandPNGBDBM50299850(1-(3,4-Dimethoxyphenyl)-N-(3-(4-methyl-1H-imidazol...)
Affinity DataKi:  41nMAssay Description:Inhibition of human glutaminyl cyclase expressed in Pichia pastoris by pGAP coupled enzyme assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutaminyl-peptide cyclotransferase(Homo sapiens (Human))
Probiodrug

Curated by ChEMBL
LigandPNGBDBM50299867(CHEMBL565907 | N-(1-(3-(5-Methyl-1H-imidazol-1-yl)...)
Affinity DataKi:  42nMAssay Description:Inhibition of human glutaminyl cyclase expressed in Pichia pastoris by pGAP coupled enzyme assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutaminyl-peptide cyclotransferase(Homo sapiens (Human))
Probiodrug

Curated by ChEMBL
LigandPNGBDBM50299864(CHEMBL574357 | N-(1-(3-(5-Methyl-1H-imidazol-1-yl)...)
Affinity DataKi:  44nMAssay Description:Inhibition of human glutaminyl cyclase expressed in Pichia pastoris by pGAP coupled enzyme assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutaminyl-peptide cyclotransferase(Homo sapiens (Human))
Probiodrug

Curated by ChEMBL
LigandPNGBDBM50299865(CHEMBL567406 | N-(-1-(3-(5-Methyl-1H-imidazol-1-yl...)
Affinity DataKi:  51nMAssay Description:Inhibition of human glutaminyl cyclase expressed in Pichia pastoris by pGAP coupled enzyme assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutaminyl-peptide cyclotransferase(Homo sapiens (Human))
Probiodrug

Curated by ChEMBL
LigandPNGBDBM50299849(1-(3,4-Dimethoxyphenyl)-3-(3-(4-methyl-1H-imidazol...)
Affinity DataKi:  60nMAssay Description:Inhibition of human glutaminyl cyclase expressed in Pichia pastoris by pGAP coupled enzyme assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutaminyl-peptide cyclotransferase(Homo sapiens (Human))
Probiodrug

Curated by ChEMBL
LigandPNGBDBM7918(1-(3,4-dimethoxyphenyl)-3-[3-(1H-imidazol-1-yl)pro...)
Affinity DataKi:  60nMAssay Description:Inhibition of human glutaminyl cyclase expressed in Pichia pastoris by pGAP coupled enzyme assayMore data for this Ligand-Target Pair
TargetGlutaminyl-peptide cyclotransferase(Homo sapiens (Human))
Probiodrug

Curated by ChEMBL
LigandPNGBDBM50299863(2-Cyano(3,4,5-trimethoxyphenyl)-3-(3-(5-methyl-1H-...)
Affinity DataKi:  61nMAssay Description:Inhibition of human glutaminyl cyclase expressed in Pichia pastoris by pGAP coupled enzyme assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutaminyl-peptide cyclotransferase(Homo sapiens (Human))
Probiodrug

Curated by ChEMBL
LigandPNGBDBM50299861(2-Cyano-1-[3-(5-methyl-1H-imidazol-1-yl)propyl]-4-...)
Affinity DataKi:  65nMAssay Description:Inhibition of human glutaminyl cyclase expressed in Pichia pastoris by pGAP coupled enzyme assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutaminyl-peptide cyclotransferase(Homo sapiens (Human))
Probiodrug

Curated by ChEMBL
LigandPNGBDBM50299868(CHEMBL565908 | N-(1-(3-(5-Methyl-1H-imidazol-1-yl)...)
Affinity DataKi:  67nMAssay Description:Inhibition of human glutaminyl cyclase expressed in Pichia pastoris by pGAP coupled enzyme assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutaminyl-peptide cyclotransferase(Homo sapiens (Human))
Probiodrug

Curated by ChEMBL
LigandPNGBDBM50299859(2-Cyano(3-(5-methyl-1H-imidazol-1-yl)propyl)-3-(3,...)
Affinity DataKi:  82nMAssay Description:Inhibition of human glutaminyl cyclase expressed in Pichia pastoris by pGAP coupled enzyme assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutaminyl-peptide cyclotransferase(Homo sapiens (Human))
Probiodrug

Curated by ChEMBL
LigandPNGBDBM50299848(2,3-Dihydro-6-methyl-3-(3-(5-methyl-1H-imidazol-1-...)
Affinity DataKi:  83nMAssay Description:Inhibition of human glutaminyl cyclase expressed in Pichia pastoris by pGAP coupled enzyme assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutaminyl-peptide cyclotransferase(Homo sapiens (Human))
Probiodrug

Curated by ChEMBL
LigandPNGBDBM7937(1-(3,4-dimethoxyphenyl)-N-[3-(1H-imidazol-1-yl)pro...)
Affinity DataKi:  90nMAssay Description:Inhibition of human glutaminyl cyclase expressed in Pichia pastoris by pGAP coupled enzyme assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTrypanothione reductase(Trypanosoma cruzi)
University Of Manchester

Curated by ChEMBL
LigandPNGBDBM50091160(CHEMBL106127 | [3-(2-Chloro-phenothiazin-10-yl)-pr...)
Affinity DataKi:  120nMAssay Description:Inhibitory activity against Trypanosoma cruzi trypanothione reductaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutaminyl-peptide cyclotransferase(Homo sapiens (Human))
Probiodrug

Curated by ChEMBL
LigandPNGBDBM50299862((3-(5-Methyl-1H-imidazol-1-yl)propyl)-2-cyano-3-(2...)
Affinity DataKi:  130nMAssay Description:Inhibition of human glutaminyl cyclase expressed in Pichia pastoris by pGAP coupled enzyme assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTrypanothione reductase(Trypanosoma cruzi)
University Of Manchester

Curated by ChEMBL
LigandPNGBDBM50178811(CHEMBL199020 | N-(3-aminopropyl)-4-tert-butyl-N,N-...)
Affinity DataKi:  150nMAssay Description:Mixed inhibition of trypanothione reductase from Trypanosoma cruzi using TSST substrateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTrypanothione reductase(Trypanosoma cruzi)
University Of Manchester

Curated by ChEMBL
LigandPNGBDBM50178803(3,4-dichloro-N-(3-(2-chloro-10H-phenothiazin-10-yl...)
Affinity DataKi:  180nMAssay Description:Linear competitive inhibition of trypanothione reductase from Trypanosoma cruzi using TSST substrateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutaminyl-peptide cyclotransferase(Homo sapiens (Human))
Probiodrug

Curated by ChEMBL
LigandPNGBDBM50299843(2,3-Dihydro-3-(3-(4-methyl-1H-imidazol-1-yl)propyl...)
Affinity DataKi:  230nMAssay Description:Inhibition of human glutaminyl cyclase expressed in Pichia pastoris by pGAP coupled enzyme assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutaminyl-peptide cyclotransferase(Homo sapiens (Human))
Probiodrug

Curated by ChEMBL
LigandPNGBDBM50299860((3,4-Dichlorophenyl)-2-cyano-3-(3-(5-methyl-1H-imi...)
Affinity DataKi:  253nMAssay Description:Inhibition of human glutaminyl cyclase expressed in Pichia pastoris by pGAP coupled enzyme assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutaminyl-peptide cyclotransferase(Homo sapiens (Human))
Probiodrug

Curated by ChEMBL
LigandPNGBDBM50299838(3-(3-(1H-Imidazol-1-yl)propyl)-2,3-dihydro-2-thiox...)
Affinity DataKi:  300nMAssay Description:Inhibition of human glutaminyl cyclase expressed in Pichia pastoris by pGAP coupled enzyme assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutaminyl-peptide cyclotransferase(Homo sapiens (Human))
Probiodrug

Curated by ChEMBL
LigandPNGBDBM50299840(3-[3-(1H-Imidazol-1-yl)propyl]-2-thioxo-2,3,5,6,7,...)
Affinity DataKi:  340nMAssay Description:Inhibition of human glutaminyl cyclase expressed in Pichia pastoris by pGAP coupled enzyme assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutaminyl-peptide cyclotransferase(Homo sapiens (Human))
Probiodrug

Curated by ChEMBL
LigandPNGBDBM50299839(3-(3-(1H-Imidazol-1-yl)propyl)-2,3-dihydro-7-methy...)
Affinity DataKi:  360nMAssay Description:Inhibition of human glutaminyl cyclase expressed in Pichia pastoris by pGAP coupled enzyme assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTrypanothione reductase(Trypanosoma cruzi)
University Of Manchester

Curated by ChEMBL
LigandPNGBDBM50178803(3,4-dichloro-N-(3-(2-chloro-10H-phenothiazin-10-yl...)
Affinity DataKi:  440nMAssay Description:Mixed inhibition of trypanothione reductase from Trypanosoma cruzi using TSST substrateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTrypanothione reductase(Trypanosoma cruzi)
University Of Manchester

Curated by ChEMBL
LigandPNGBDBM50091165((4-Benzyloxy-benzyl)-[3-(2-chloro-phenothiazin-10-...)
Affinity DataKi:  470nMAssay Description:Inhibitory activity against Trypanosoma cruzi trypanothione reductaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTrypanothione reductase(Trypanosoma cruzi)
University Of Manchester

Curated by ChEMBL
LigandPNGBDBM50091158(CHEMBL322826 | [3-(2-Chloro-phenothiazin-10-yl)-pr...)
Affinity DataKi:  470nMAssay Description:Inhibitory activity against Trypanosoma cruzi trypanothione reductaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1D adrenergic receptor(Homo sapiens (Human))
Hokkaido University

Curated by ChEMBL
LigandPNGBDBM50326197(1,9-dimethyl-2,8-dioxo-2,3,8,9-tetrahydro-1H-purin...)
Affinity DataKi:  497nMAssay Description:Binding affinity to adrenergic alpha1D receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutaminyl-peptide cyclotransferase(Homo sapiens (Human))
Probiodrug

Curated by ChEMBL
LigandPNGBDBM50299830(CHEMBL577493 | N-(3-(1H-Imidazol-1-yl)propyl)-N-cy...)
Affinity DataKi:  500nMAssay Description:Inhibition of human glutaminyl cyclase expressed in Pichia pastoris by pGAP coupled enzyme assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutaminyl-peptide cyclotransferase(Homo sapiens (Human))
Probiodrug

Curated by ChEMBL
LigandPNGBDBM50299834(CHEMBL565480 | N-(1-(3-(1H-Imidazol-1-yl)propylami...)
Affinity DataKi:  520nMAssay Description:Inhibition of human glutaminyl cyclase expressed in Pichia pastoris by pGAP coupled enzyme assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutaminyl-peptide cyclotransferase(Homo sapiens (Human))
Probiodrug

Curated by ChEMBL
LigandPNGBDBM50299833(CHEMBL565479 | N-(1-(3-(1H-Imidazol-1-yl)propylami...)
Affinity DataKi:  540nMAssay Description:Inhibition of human glutaminyl cyclase expressed in Pichia pastoris by pGAP coupled enzyme assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutaminyl-peptide cyclotransferase(Homo sapiens (Human))
Probiodrug

Curated by ChEMBL
LigandPNGBDBM50299837(CHEMBL565492 | N-(1-(3-(1H-Imidazol-1-yl)propylami...)
Affinity DataKi:  540nMAssay Description:Inhibition of human glutaminyl cyclase expressed in Pichia pastoris by pGAP coupled enzyme assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTrypanothione reductase(Trypanosoma cruzi)
University Of Manchester

Curated by ChEMBL
LigandPNGBDBM50091148(CHEMBL106769 | [3-(2-Chloro-phenothiazin-10-yl)-pr...)
Affinity DataKi:  560nMAssay Description:Inhibitory activity against Trypanosoma cruzi trypanothione reductaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTrypanothione reductase(Trypanosoma cruzi)
University Of Manchester

Curated by ChEMBL
LigandPNGBDBM50178809(4-tert-butyl-N-(3-(2-chloro-10H-phenothiazin-10-yl...)
Affinity DataKi:  570nMAssay Description:Linear competitive inhibition of trypanothione reductase from Trypanosoma cruzi using TSST substrateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutaminyl-peptide cyclotransferase(Homo sapiens (Human))
Probiodrug

Curated by ChEMBL
LigandPNGBDBM50299832(CHEMBL567415 | N-(1-(3-(1H-Imidazol-1-yl)propylami...)
Affinity DataKi:  570nMAssay Description:Inhibition of human glutaminyl cyclase expressed in Pichia pastoris by pGAP coupled enzyme assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutaminyl-peptide cyclotransferase(Homo sapiens (Human))
Probiodrug

Curated by ChEMBL
LigandPNGBDBM50299836(CHEMBL582920 | N-(-1-(3-(1H-Imidazol-1-yl)propylam...)
Affinity DataKi:  610nMAssay Description:Inhibition of human glutaminyl cyclase expressed in Pichia pastoris by pGAP coupled enzyme assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutaminyl-peptide cyclotransferase(Homo sapiens (Human))
Probiodrug

Curated by ChEMBL
LigandPNGBDBM50299828((3-(1H-Imidazol-1-yl)propyl)-2-cyano-3-(2,3-dihydr...)
Affinity DataKi:  620nMAssay Description:Inhibition of human glutaminyl cyclase expressed in Pichia pastoris by pGAP coupled enzyme assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutaminyl-peptide cyclotransferase(Homo sapiens (Human))
Probiodrug

Curated by ChEMBL
LigandPNGBDBM50299841(3-[3-(1H-Imidazol-1-yl)propyl]-2-thioxo-1,2,3,5,6,...)
Affinity DataKi:  620nMAssay Description:Inhibition of human glutaminyl cyclase expressed in Pichia pastoris by pGAP coupled enzyme assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTrypanothione reductase(Trypanosoma cruzi)
University Of Manchester

Curated by ChEMBL
LigandPNGBDBM50091162((4-tert-Butyl-benzyl)-[3-(2-chloro-phenothiazin-10...)
Affinity DataKi:  680nMAssay Description:Inhibitory activity against Trypanosoma cruzi trypanothione reductaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutaminyl-peptide cyclotransferase(Homo sapiens (Human))
Probiodrug

Curated by ChEMBL
LigandPNGBDBM50299826((3-(1H-Imidazol-1-yl)propyl)-2-cyano-3-(4-methoxyp...)
Affinity DataKi:  700nMAssay Description:Inhibition of human glutaminyl cyclase expressed in Pichia pastoris by pGAP coupled enzyme assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTrypanothione reductase(Trypanosoma cruzi)
University Of Manchester

Curated by ChEMBL
LigandPNGBDBM50091163(Benzhydryl-[3-(2-chloro-phenothiazin-10-yl)-propyl...)
Affinity DataKi:  710nMAssay Description:Inhibitory activity against Trypanosoma cruzi trypanothione reductaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1B adrenergic receptor(Homo sapiens (Human))
Hokkaido University

Curated by ChEMBL
LigandPNGBDBM50326197(1,9-dimethyl-2,8-dioxo-2,3,8,9-tetrahydro-1H-purin...)
Affinity DataKi:  758nMAssay Description:Binding affinity to adrenergic alpha1B receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTrypanothione reductase(Trypanosoma cruzi)
University Of Manchester

Curated by ChEMBL
LigandPNGBDBM50091154(CHEMBL106901 | [3-(2-Chloro-phenothiazin-10-yl)-pr...)
Affinity DataKi:  770nMAssay Description:Inhibitory activity against Trypanosoma cruzi trypanothione reductaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutaminyl-peptide cyclotransferase(Homo sapiens (Human))
Probiodrug

Curated by ChEMBL
LigandPNGBDBM50299825((3-(1H-Imidazol-1-yl)propyl)-2-cyano-3-(4-isopropy...)
Affinity DataKi:  830nMAssay Description:Inhibition of human glutaminyl cyclase expressed in Pichia pastoris by pGAP coupled enzyme assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1A adrenergic receptor(Homo sapiens (Human))
Hokkaido University

Curated by ChEMBL
LigandPNGBDBM50326197(1,9-dimethyl-2,8-dioxo-2,3,8,9-tetrahydro-1H-purin...)
Affinity DataKi:  885nMAssay Description:Binding affinity to adrenergic alpha1A receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutaminyl-peptide cyclotransferase(Homo sapiens (Human))
Probiodrug

Curated by ChEMBL
LigandPNGBDBM50299842(3-[3-(1H-Imidazol-1-yl)propyl]-2-thioxo-2,3,5,6,7,...)
Affinity DataKi:  900nMAssay Description:Inhibition of human glutaminyl cyclase expressed in Pichia pastoris by pGAP coupled enzyme assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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