Found 451 with Last Name = 'bakker' and Initial = 'ra' TargetHistamine H1 receptor(Homo sapiens (Human))
University of North Carolina At Chapel Hill
Curated by PDSP Ki Database
University of North Carolina At Chapel Hill
Curated by PDSP Ki Database
TargetHistamine H1 receptor(Cavia porcellus (domestic guinea pig))
University of North Carolina At Chapel Hill
Curated by PDSP Ki Database
University of North Carolina At Chapel Hill
Curated by PDSP Ki Database
TargetHistamine H1 receptor(Cavia porcellus (domestic guinea pig))
University of North Carolina At Chapel Hill
Curated by PDSP Ki Database
University of North Carolina At Chapel Hill
Curated by PDSP Ki Database
Affinity DataKi: 0.300nMAssay Description:Human KLKB1 (1.78 nM or 0.025 U/mL; Enzyme Research Laboratories) was incubated at 24° C. with 0.25 mM fluorogenic substrate H-Pro-Phe-Arg-AMC (11295...More data for this Ligand-Target Pair
Affinity DataKi: 0.300nMAssay Description:Human KLKB1 (1.78 nM or 0.025 U/mL; Enzyme Research Laboratories) was incubated at 24° C. with 0.25 mM fluorogenic substrate H-Pro-Phe-Arg-AMC (11295...More data for this Ligand-Target Pair
Affinity DataKi: 0.300nMAssay Description:Human KLKB1 (1.78 nM or 0.025 U/mL; Enzyme Research Laboratories) was incubated at 24° C. with 0.25 mM fluorogenic substrate H-Pro-Phe-Arg-AMC (11295...More data for this Ligand-Target Pair
Affinity DataKi: 0.300nMAssay Description:Human KLKB1 (1.78 nM or 0.025 U/mL; Enzyme Research Laboratories) was incubated at 24° C. with 0.25 mM fluorogenic substrate H-Pro-Phe-Arg-AMC (11295...More data for this Ligand-Target Pair
TargetHistamine H1 receptor(Homo sapiens (Human))
University of North Carolina At Chapel Hill
Curated by PDSP Ki Database
University of North Carolina At Chapel Hill
Curated by PDSP Ki Database
Affinity DataKi: 0.339nM ΔG°: -54.1kJ/molepH: 7.4 T: 2°CAssay Description:Ligand displacement assays were performed on CHO cells membranes expressing hH3R. Retained radioactivity was determined by liquid scintillation count...More data for this Ligand-Target Pair
Affinity DataKi: 0.400nMAssay Description:Human KLKB1 (1.78 nM or 0.025 U/mL; Enzyme Research Laboratories) was incubated at 24° C. with 0.25 mM fluorogenic substrate H-Pro-Phe-Arg-AMC (11295...More data for this Ligand-Target Pair
Affinity DataKi: 0.400nMAssay Description:Human KLKB1 (1.78 nM or 0.025 U/mL; Enzyme Research Laboratories) was incubated at 24° C. with 0.25 mM fluorogenic substrate H-Pro-Phe-Arg-AMC (11295...More data for this Ligand-Target Pair
Affinity DataKi: 0.400nMAssay Description:Human KLKB1 (1.78 nM or 0.025 U/mL; Enzyme Research Laboratories) was incubated at 24° C. with 0.25 mM fluorogenic substrate H-Pro-Phe-Arg-AMC (11295...More data for this Ligand-Target Pair
Affinity DataKi: 0.400nMAssay Description:Human KLKB1 (1.78 nM or 0.025 U/mL; Enzyme Research Laboratories) was incubated at 24° C. with 0.25 mM fluorogenic substrate H-Pro-Phe-Arg-AMC (11295...More data for this Ligand-Target Pair
Affinity DataKi: 0.400nMAssay Description:Human KLKB1 (1.78 nM or 0.025 U/mL; Enzyme Research Laboratories) was incubated at 24° C. with 0.25 mM fluorogenic substrate H-Pro-Phe-Arg-AMC (11295...More data for this Ligand-Target Pair
Affinity DataKi: 0.407nM ΔG°: -53.6kJ/molepH: 7.4 T: 2°CAssay Description:Ligand displacement assays were performed on CHO cells membranes expressing hH3R. Retained radioactivity was determined by liquid scintillation count...More data for this Ligand-Target Pair
Affinity DataKi: 0.5nMAssay Description:Human KLKB1 (1.78 nM or 0.025 U/mL; Enzyme Research Laboratories) was incubated at 24° C. with 0.25 mM fluorogenic substrate H-Pro-Phe-Arg-AMC (11295...More data for this Ligand-Target Pair
Affinity DataKi: 0.5nMAssay Description:Human KLKB1 (1.78 nM or 0.025 U/mL; Enzyme Research Laboratories) was incubated at 24° C. with 0.25 mM fluorogenic substrate H-Pro-Phe-Arg-AMC (11295...More data for this Ligand-Target Pair
Affinity DataKi: 0.501nMAssay Description:Ligand displacement assays were performed on The SK-N-MC/hH3R cell homogenates. Retained radioactivity was determined by liquid scintillation countin...More data for this Ligand-Target Pair
Affinity DataKi: 0.501nMAssay Description:Displacement of [3H]N-R-methylhistamine binding to SK-N-MC cell membranes expressing human H3 receptorMore data for this Ligand-Target Pair
TargetHistamine H1 receptor(Cavia porcellus (domestic guinea pig))
University of North Carolina At Chapel Hill
Curated by PDSP Ki Database
University of North Carolina At Chapel Hill
Curated by PDSP Ki Database
TargetHistamine H1 receptor(Cavia porcellus (domestic guinea pig))
University of North Carolina At Chapel Hill
Curated by PDSP Ki Database
University of North Carolina At Chapel Hill
Curated by PDSP Ki Database
Affinity DataKi: 0.600nMAssay Description:Human KLKB1 (1.78 nM or 0.025 U/mL; Enzyme Research Laboratories) was incubated at 24° C. with 0.25 mM fluorogenic substrate H-Pro-Phe-Arg-AMC (11295...More data for this Ligand-Target Pair
Affinity DataKi: 0.630nMAssay Description:Ligand displacement assays were performed on The SK-N-MC/hH3R cell homogenates. Retained radioactivity was determined by liquid scintillation countin...More data for this Ligand-Target Pair
TargetHistamine H1 receptor(Cavia porcellus (domestic guinea pig))
University of North Carolina At Chapel Hill
Curated by PDSP Ki Database
University of North Carolina At Chapel Hill
Curated by PDSP Ki Database
TargetHistamine H1 receptor(Cavia porcellus (domestic guinea pig))
University of North Carolina At Chapel Hill
Curated by PDSP Ki Database
University of North Carolina At Chapel Hill
Curated by PDSP Ki Database
TargetHistamine H1 receptor(Cavia porcellus (domestic guinea pig))
University of North Carolina At Chapel Hill
Curated by PDSP Ki Database
University of North Carolina At Chapel Hill
Curated by PDSP Ki Database
Affinity DataKi: 0.794nMAssay Description:Ligand displacement assays were performed on The SK-N-MC/hH3R cell homogenates. Retained radioactivity was determined by liquid scintillation countin...More data for this Ligand-Target Pair
TargetHistamine H1 receptor(Cavia porcellus (domestic guinea pig))
University of North Carolina At Chapel Hill
Curated by PDSP Ki Database
University of North Carolina At Chapel Hill
Curated by PDSP Ki Database
Affinity DataKi: 1nMAssay Description:Displacement of [3H]N-R-methylhistamine binding to SK-N-MC cell membranes expressing human H3 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 1nM ΔG°: -51.4kJ/mole EC50: 2nMpH: 7.4 T: 2°CAssay Description:Ligand displacement assays were performed on CHO cells membranes expressing hH3R. Retained radioactivity was determined by liquid scintillation count...More data for this Ligand-Target Pair
Affinity DataKi: 1nMAssay Description:Ligand displacement assays were performed on The SK-N-MC/hH3R cell homogenates. Retained radioactivity was determined by liquid scintillation countin...More data for this Ligand-Target Pair
TargetHistamine H1 receptor(Homo sapiens (Human))
University of North Carolina At Chapel Hill
Curated by PDSP Ki Database
University of North Carolina At Chapel Hill
Curated by PDSP Ki Database
Affinity DataKi: 1.10nMAssay Description:Human KLKB1 (1.78 nM or 0.025 U/mL; Enzyme Research Laboratories) was incubated at 24° C. with 0.25 mM fluorogenic substrate H-Pro-Phe-Arg-AMC (11295...More data for this Ligand-Target Pair
TargetHistamine H1 receptor(Homo sapiens (Human))
University of North Carolina At Chapel Hill
Curated by PDSP Ki Database
University of North Carolina At Chapel Hill
Curated by PDSP Ki Database
TargetHistamine H1 receptor(Cavia porcellus (domestic guinea pig))
University of North Carolina At Chapel Hill
Curated by PDSP Ki Database
University of North Carolina At Chapel Hill
Curated by PDSP Ki Database
TargetHistamine H1 receptor(Homo sapiens (Human))
University of North Carolina At Chapel Hill
Curated by PDSP Ki Database
University of North Carolina At Chapel Hill
Curated by PDSP Ki Database
TargetHistamine H1 receptor(Cavia porcellus (domestic guinea pig))
University of North Carolina At Chapel Hill
Curated by PDSP Ki Database
University of North Carolina At Chapel Hill
Curated by PDSP Ki Database
TargetHistamine H1 receptor(Cavia porcellus (domestic guinea pig))
University of North Carolina At Chapel Hill
Curated by PDSP Ki Database
University of North Carolina At Chapel Hill
Curated by PDSP Ki Database
Affinity DataKi: 1.5nMAssay Description:Human KLKB1 (1.78 nM or 0.025 U/mL; Enzyme Research Laboratories) was incubated at 24° C. with 0.25 mM fluorogenic substrate H-Pro-Phe-Arg-AMC (11295...More data for this Ligand-Target Pair
TargetHistamine H1 receptor(Homo sapiens (Human))
University of North Carolina At Chapel Hill
Curated by PDSP Ki Database
University of North Carolina At Chapel Hill
Curated by PDSP Ki Database
TargetHistamine H1 receptor(Cavia porcellus (domestic guinea pig))
University of North Carolina At Chapel Hill
Curated by PDSP Ki Database
University of North Carolina At Chapel Hill
Curated by PDSP Ki Database
TargetHistamine H1 receptor(Homo sapiens (Human))
University of North Carolina At Chapel Hill
Curated by PDSP Ki Database
University of North Carolina At Chapel Hill
Curated by PDSP Ki Database
Affinity DataKi: 1.58nMAssay Description:Displacement of [3H]N-alpha-methylhistamine from human histamine H3 receptor expressed in human SK-N-MC cells by liquid scintillation countingMore data for this Ligand-Target Pair
Affinity DataKi: 1.58nMAssay Description:Displacement of [3H]histamine from human histamine H4 receptor expressed in human SK-N-MC cells by liquid scintillation countingMore data for this Ligand-Target Pair
TargetHistamine H1 receptor(Homo sapiens (Human))
University of North Carolina At Chapel Hill
Curated by PDSP Ki Database
University of North Carolina At Chapel Hill
Curated by PDSP Ki Database
TargetHistamine H1 receptor(Homo sapiens (Human))
University of North Carolina At Chapel Hill
Curated by PDSP Ki Database
University of North Carolina At Chapel Hill
Curated by PDSP Ki Database
Affinity DataKi: 1.90nMAssay Description:Human KLKB1 (1.78 nM or 0.025 U/mL; Enzyme Research Laboratories) was incubated at 24° C. with 0.25 mM fluorogenic substrate H-Pro-Phe-Arg-AMC (11295...More data for this Ligand-Target Pair
TargetHistamine H1 receptor(Cavia porcellus (domestic guinea pig))
University of North Carolina At Chapel Hill
Curated by PDSP Ki Database
University of North Carolina At Chapel Hill
Curated by PDSP Ki Database
Affinity DataKi: 2nMAssay Description:Ligand displacement assays were performed on The SK-N-MC/hH3R cell homogenates. Retained radioactivity was determined by liquid scintillation countin...More data for this Ligand-Target Pair
Affinity DataKi: 2nM ΔG°: -49.7kJ/molepH: 7.4 T: 2°CAssay Description:Ligand displacement assays were performed on CHO cells membranes expressing hH3R. Retained radioactivity was determined by liquid scintillation count...More data for this Ligand-Target Pair
