Affinity DataKi: 210nMAssay Description:Inhibition of human CYP3A4 assessed as biotransformation of 7-benzyloxyquinolineMore data for this Ligand-Target Pair
Affinity DataKi: 260nMAssay Description:Inhibition of human CYP3A4 assessed as biotransformation of 7-benzyloxyquinolineMore data for this Ligand-Target Pair
Affinity DataKi: 300nMAssay Description:Inhibition of AChE by Ellman's assayMore data for this Ligand-Target Pair
Affinity DataKi: 340nMAssay Description:Inhibition of AChE by Ellman's assayMore data for this Ligand-Target Pair
Affinity DataKi: 390nMAssay Description:Inhibition of AChE by Ellman's assayMore data for this Ligand-Target Pair
Affinity DataKi: 430nMAssay Description:Inhibition of AChE by Ellman's assayMore data for this Ligand-Target Pair
Affinity DataKi: 540nMAssay Description:Inhibition of AChE by Ellman's assayMore data for this Ligand-Target Pair
Affinity DataKi: 630nMAssay Description:Inhibition of human CYP3A4 assessed as biotransformation of 7-benzyloxyquinolineMore data for this Ligand-Target Pair
Affinity DataKi: 860nMAssay Description:Inhibition of AChE by Ellman's assayMore data for this Ligand-Target Pair
Affinity DataKi: 970nMAssay Description:Inhibition of AChE by Ellman's assayMore data for this Ligand-Target Pair
Affinity DataKi: 7.60E+3nMAssay Description:Inhibition of human CYP3A4 assessed as biotransformation of 7-benzyloxyquinolineMore data for this Ligand-Target Pair
Affinity DataKi: 1.10E+4nMAssay Description:Inhibition of human CYP3A4 assessed as biotransformation of 7-benzyloxyquinolineMore data for this Ligand-Target Pair
TargetAcetylcholinesterase(Electrophorus electricus (Electric eel))
Universitat De Barcelona
Curated by ChEMBL
Universitat De Barcelona
Curated by ChEMBL
Affinity DataIC50: 160nMAssay Description:Inhibition of electric eel acetylcholineesteraseMore data for this Ligand-Target Pair
TargetAcetylcholinesterase(Electrophorus electricus (Electric eel))
Universitat De Barcelona
Curated by ChEMBL
Universitat De Barcelona
Curated by ChEMBL
Affinity DataIC50: 180nMAssay Description:Inhibition of electric eel acetylcholineesteraseMore data for this Ligand-Target Pair
TargetAcetylcholinesterase(Electrophorus electricus (Electric eel))
Universitat De Barcelona
Curated by ChEMBL
Universitat De Barcelona
Curated by ChEMBL
Affinity DataIC50: 480nMAssay Description:Inhibition of electric eel AChE using ATCI as substrate preincubated for 30 mins followed by substrate addition measured after 5 mins by DTNB-based s...More data for this Ligand-Target Pair
TargetAcetylcholinesterase(Electrophorus electricus (Electric eel))
Universitat De Barcelona
Curated by ChEMBL
Universitat De Barcelona
Curated by ChEMBL
Affinity DataIC50: 1.82E+3nMAssay Description:Inhibition of electric eel acetylcholineesteraseMore data for this Ligand-Target Pair
Affinity DataIC50: 2.24E+4nMAssay Description:Inhibition of equine serum BuChE using ATCI as substrate preincubated for 30 mins followed by substrate addition measured after 5 mins by DTNB-based ...More data for this Ligand-Target Pair
Affinity DataIC50: 6.73E+4nMAssay Description:Inhibition of equine serum BuChE using ATCI as substrate preincubated for 30 mins followed by substrate addition measured after 5 mins by DTNB-based ...More data for this Ligand-Target Pair
TargetAcetylcholinesterase(Electrophorus electricus (Electric eel))
Universitat De Barcelona
Curated by ChEMBL
Universitat De Barcelona
Curated by ChEMBL
Affinity DataIC50: 1.14E+5nMAssay Description:Inhibition of electric eel AChE using ATCI as substrate preincubated for 30 mins followed by substrate addition measured after 5 mins by DTNB-based s...More data for this Ligand-Target Pair
Affinity DataIC50: >2.00E+5nMAssay Description:Inhibition of equine serum BuChE using ATCI as substrate preincubated for 30 mins followed by substrate addition measured after 5 mins by DTNB-based ...More data for this Ligand-Target Pair
TargetAcetylcholinesterase(Electrophorus electricus (Electric eel))
Universitat De Barcelona
Curated by ChEMBL
Universitat De Barcelona
Curated by ChEMBL
Affinity DataIC50: >2.00E+5nMAssay Description:Inhibition of electric eel AChE using ATCI as substrate preincubated for 30 mins followed by substrate addition measured after 5 mins by DTNB-based s...More data for this Ligand-Target Pair
TargetAcetylcholinesterase(Electrophorus electricus (Electric eel))
Universitat De Barcelona
Curated by ChEMBL
Universitat De Barcelona
Curated by ChEMBL
Affinity DataIC50: >2.00E+5nMAssay Description:Inhibition of electric eel AChE using ATCI as substrate preincubated for 30 mins followed by substrate addition measured after 5 mins by DTNB-based s...More data for this Ligand-Target Pair
Affinity DataIC50: >2.00E+5nMAssay Description:Inhibition of equine serum BuChE using ATCI as substrate preincubated for 30 mins followed by substrate addition measured after 5 mins by DTNB-based ...More data for this Ligand-Target Pair
Affinity DataIC50: >2.00E+5nMAssay Description:Inhibition of equine serum BuChE using ATCI as substrate preincubated for 30 mins followed by substrate addition measured after 5 mins by DTNB-based ...More data for this Ligand-Target Pair
Affinity DataIC50: >2.00E+5nMAssay Description:Inhibition of equine serum BuChE using ATCI as substrate preincubated for 30 mins followed by substrate addition measured after 5 mins by DTNB-based ...More data for this Ligand-Target Pair
TargetAcetylcholinesterase(Electrophorus electricus (Electric eel))
Universitat De Barcelona
Curated by ChEMBL
Universitat De Barcelona
Curated by ChEMBL
Affinity DataIC50: >2.00E+5nMAssay Description:Inhibition of electric eel AChE using ATCI as substrate preincubated for 30 mins followed by substrate addition measured after 5 mins by DTNB-based s...More data for this Ligand-Target Pair
TargetAcetylcholinesterase(Electrophorus electricus (Electric eel))
Universitat De Barcelona
Curated by ChEMBL
Universitat De Barcelona
Curated by ChEMBL
Affinity DataIC50: >2.00E+5nMAssay Description:Inhibition of electric eel AChE using ATCI as substrate preincubated for 30 mins followed by substrate addition measured after 5 mins by DTNB-based s...More data for this Ligand-Target Pair
Affinity DataIC50: >2.00E+5nMAssay Description:Inhibition of equine serum BuChE using ATCI as substrate preincubated for 30 mins followed by substrate addition measured after 5 mins by DTNB-based ...More data for this Ligand-Target Pair
TargetAcetylcholinesterase(Electrophorus electricus (Electric eel))
Universitat De Barcelona
Curated by ChEMBL
Universitat De Barcelona
Curated by ChEMBL
Affinity DataIC50: >2.00E+5nMAssay Description:Inhibition of electric eel AChE using ATCI as substrate preincubated for 30 mins followed by substrate addition measured after 5 mins by DTNB-based s...More data for this Ligand-Target Pair