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Found 248 with Last Name = 'beavers' and Initial = 'mp'
TargetKiSS-1 receptor(Homo sapiens (Human))
University Of Minnesota Health Science Center

Curated by ChEMBL
LigandPNGBDBM50203781((2S)-2-{[(2S)-1-[(2S)-2-amino-4-methylpentanoyl]py...)
Affinity DataKi:  0.800nMAssay Description:Displacement of [125]metastin from metastin receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKiSS-1 receptor(Homo sapiens (Human))
University Of Minnesota Health Science Center

Curated by ChEMBL
LigandPNGBDBM50203803((2S)-2-{[(2S)-1-[(2S)-2-amino-4-methylpentanoyl]py...)
Affinity DataKi:  1.10nMAssay Description:Displacement of [125]metastin from metastin receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKiSS-1 receptor(Homo sapiens (Human))
University Of Minnesota Health Science Center

Curated by ChEMBL
LigandPNGBDBM50203803((2S)-2-{[(2S)-1-[(2S)-2-amino-4-methylpentanoyl]py...)
Affinity DataKi:  1.10nMAssay Description:Displacement of [125]metastin from metastin receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKiSS-1 receptor(Homo sapiens (Human))
University Of Minnesota Health Science Center

Curated by ChEMBL
LigandPNGBDBM26349((2S)-2-[(2S)-2-[(2S)-2-[(2S)-2-amino-3-(4-hydroxyp...)
Affinity DataKi:  1.30nMAssay Description:Displacement of [125]metastin from metastin receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKiSS-1 receptor(Homo sapiens (Human))
University Of Minnesota Health Science Center

Curated by ChEMBL
LigandPNGBDBM50203782((2S)-2-{[(2S)-1-[(2S)-2-amino-4-methylpentanoyl]py...)
Affinity DataKi:  1.60nMAssay Description:Displacement of [125]metastin from metastin receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKiSS-1 receptor(Homo sapiens (Human))
University Of Minnesota Health Science Center

Curated by ChEMBL
LigandPNGBDBM50203794((2S)-2-{[(2S)-1-[(2S)-2-amino-4-methylpentanoyl]py...)
Affinity DataKi:  1.80nMAssay Description:Displacement of [125]metastin from metastin receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKiSS-1 receptor(Homo sapiens (Human))
University Of Minnesota Health Science Center

Curated by ChEMBL
LigandPNGBDBM50203811((2S)-2-{[(2S)-1-[(2S)-2-amino-4-methylpentanoyl]py...)
Affinity DataKi:  2nMAssay Description:Displacement of [125]metastin from metastin receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKiSS-1 receptor(Homo sapiens (Human))
University Of Minnesota Health Science Center

Curated by ChEMBL
LigandPNGBDBM50203802((2S)-2-{[(2S)-1-[(2S)-2-amino-4-methylpentanoyl]py...)
Affinity DataKi:  4.70nMAssay Description:Displacement of [125]metastin from metastin receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKiSS-1 receptor(Homo sapiens (Human))
University Of Minnesota Health Science Center

Curated by ChEMBL
LigandPNGBDBM50203814((2S)-2-{[(2S)-1-[(2S)-2-amino-4-methylpentanoyl]py...)
Affinity DataKi:  5nMAssay Description:Displacement of [125]metastin from metastin receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKiSS-1 receptor(Homo sapiens (Human))
University Of Minnesota Health Science Center

Curated by ChEMBL
LigandPNGBDBM50203813((2S)-2-{[(2S)-1-[(2S)-2-amino-4-methylpentanoyl]py...)
Affinity DataKi:  7.70nMAssay Description:Displacement of [125]metastin from metastin receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKiSS-1 receptor(Homo sapiens (Human))
University Of Minnesota Health Science Center

Curated by ChEMBL
LigandPNGBDBM50203816((2S)-2-{[(2S)-1-[(2S)-2-amino-4-methylpentanoyl]py...)
Affinity DataKi:  9.30nMAssay Description:Displacement of [125]metastin from metastin receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKiSS-1 receptor(Homo sapiens (Human))
University Of Minnesota Health Science Center

Curated by ChEMBL
LigandPNGBDBM50203791((2S)-N-[(1S)-1-{[(1S)-1-{[(1S)-1-{[(1S)-1-{[(1S)-1...)
Affinity DataKi:  9.40nMAssay Description:Displacement of [125]metastin from metastin receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKiSS-1 receptor(Homo sapiens (Human))
University Of Minnesota Health Science Center

Curated by ChEMBL
LigandPNGBDBM50203800((2S)-2-{[(2S)-1-[(2S)-2-amino-4-methylpentanoyl]py...)
Affinity DataKi:  11.1nMAssay Description:Displacement of [125]metastin from metastin receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKiSS-1 receptor(Homo sapiens (Human))
University Of Minnesota Health Science Center

Curated by ChEMBL
LigandPNGBDBM50203779((2S)-2-{[(2S)-1-[(2S)-2-amino-4-methylpentanoyl]py...)
Affinity DataKi:  15.8nMAssay Description:Displacement of [125]metastin from metastin receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKiSS-1 receptor(Homo sapiens (Human))
University Of Minnesota Health Science Center

Curated by ChEMBL
LigandPNGBDBM50203789((2S)-2-{[(2S)-1-[(2S)-2-amino-4-methylpentanoyl]py...)
Affinity DataKi:  16.2nMAssay Description:Displacement of [125]metastin from metastin receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKiSS-1 receptor(Homo sapiens (Human))
University Of Minnesota Health Science Center

Curated by ChEMBL
LigandPNGBDBM50203810((2S)-2-{[(2S)-1-[(2S)-2-amino-4-methylpentanoyl]py...)
Affinity DataKi:  21.1nMAssay Description:Displacement of [125]metastin from metastin receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKiSS-1 receptor(Homo sapiens (Human))
University Of Minnesota Health Science Center

Curated by ChEMBL
LigandPNGBDBM50203780((2S)-2-{[(2S)-1-[(2S)-2-amino-4-methylpentanoyl]py...)
Affinity DataKi:  29.5nMAssay Description:Displacement of [125]metastin from metastin receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKiSS-1 receptor(Homo sapiens (Human))
University Of Minnesota Health Science Center

Curated by ChEMBL
LigandPNGBDBM50203787((2S)-2-{[(2S)-1-[(2S)-2-amino-4-methylpentanoyl]py...)
Affinity DataKi:  33.4nMAssay Description:Displacement of [125]metastin from metastin receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKiSS-1 receptor(Homo sapiens (Human))
University Of Minnesota Health Science Center

Curated by ChEMBL
LigandPNGBDBM50203799((2S)-2-{[(2S)-1-[(2S)-2-amino-4-methylpentanoyl]py...)
Affinity DataKi:  51.5nMAssay Description:Displacement of [125]metastin from metastin receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKiSS-1 receptor(Homo sapiens (Human))
University Of Minnesota Health Science Center

Curated by ChEMBL
LigandPNGBDBM50203797((2S)-2-{[(2S)-1-[(2S)-2-amino-4-methylpentanoyl]py...)
Affinity DataKi:  80.8nMAssay Description:Displacement of [125]metastin from metastin receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKiSS-1 receptor(Homo sapiens (Human))
University Of Minnesota Health Science Center

Curated by ChEMBL
LigandPNGBDBM50203797((2S)-2-{[(2S)-1-[(2S)-2-amino-4-methylpentanoyl]py...)
Affinity DataKi:  80.8nMAssay Description:Displacement of [125]metastin from metastin receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKiSS-1 receptor(Homo sapiens (Human))
University Of Minnesota Health Science Center

Curated by ChEMBL
LigandPNGBDBM50203790((2S)-2-[(2S)-2-[(2S)-2-{[(2S)-1-[(2S)-2-amino-4-me...)
Affinity DataKi:  82.7nMAssay Description:Displacement of [125]metastin from metastin receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKiSS-1 receptor(Homo sapiens (Human))
University Of Minnesota Health Science Center

Curated by ChEMBL
LigandPNGBDBM50203798((2S)-2-[(2S)-2-[(2S)-2-{[(2S)-1-[(2S)-2-amino-4-me...)
Affinity DataKi:  88.1nMAssay Description:Displacement of [125]metastin from metastin receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKiSS-1 receptor(Homo sapiens (Human))
University Of Minnesota Health Science Center

Curated by ChEMBL
LigandPNGBDBM50203807(CHEMBL374077 | LPNYNWNSFGLRF-NH2)
Affinity DataKi:  94.8nMAssay Description:Displacement of [125]metastin from metastin receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKiSS-1 receptor(Homo sapiens (Human))
University Of Minnesota Health Science Center

Curated by ChEMBL
LigandPNGBDBM50203786((2S)-2-{[(2S)-1-[(2S)-2-amino-4-methylpentanoyl]py...)
Affinity DataKi:  110nMAssay Description:Displacement of [125]metastin from metastin receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKiSS-1 receptor(Homo sapiens (Human))
University Of Minnesota Health Science Center

Curated by ChEMBL
LigandPNGBDBM50203795((2S)-2-{[(2S)-1-[(2S)-2-amino-4-methylpentanoyl]py...)
Affinity DataKi:  142nMAssay Description:Displacement of [125]metastin from metastin receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKiSS-1 receptor(Homo sapiens (Human))
University Of Minnesota Health Science Center

Curated by ChEMBL
LigandPNGBDBM50203817((2S)-2-{[(2S)-1-[(2S)-2-amino-4-methylpentanoyl]py...)
Affinity DataKi:  162nMAssay Description:Displacement of [125]metastin from metastin receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKiSS-1 receptor(Homo sapiens (Human))
University Of Minnesota Health Science Center

Curated by ChEMBL
LigandPNGBDBM50203788((2S)-2-{[(2S)-1-[(2S)-2-amino-4-methylpentanoyl]py...)
Affinity DataKi:  197nMAssay Description:Displacement of [125]metastin from metastin receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKiSS-1 receptor(Homo sapiens (Human))
University Of Minnesota Health Science Center

Curated by ChEMBL
LigandPNGBDBM50203796((2S)-2-{[(2S)-1-[(2S)-2-amino-4-methylpentanoyl]py...)
Affinity DataKi:  198nMAssay Description:Displacement of [125]metastin from metastin receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKiSS-1 receptor(Homo sapiens (Human))
University Of Minnesota Health Science Center

Curated by ChEMBL
LigandPNGBDBM50203785((2S)-2-{[(2S)-1-[(2S)-2-amino-4-methylpentanoyl]py...)
Affinity DataKi:  240nMAssay Description:Displacement of [125]metastin from metastin receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKiSS-1 receptor(Homo sapiens (Human))
University Of Minnesota Health Science Center

Curated by ChEMBL
LigandPNGBDBM50203809((2S)-2-[(2S)-2-[(2S)-2-[(2S)-2-[(2S)-2-[(2S)-2-[(2...)
Affinity DataKi:  298nMAssay Description:Displacement of [125]metastin from metastin receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKiSS-1 receptor(Homo sapiens (Human))
University Of Minnesota Health Science Center

Curated by ChEMBL
LigandPNGBDBM50203784((2S)-2-[(2S)-2-[(2S)-2-{2-[(2S)-2-[(2S)-2-[(2S)-2-...)
Affinity DataKi:  495nMAssay Description:Displacement of [125]metastin from metastin receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKiSS-1 receptor(Homo sapiens (Human))
University Of Minnesota Health Science Center

Curated by ChEMBL
LigandPNGBDBM50203805(CHEMBL220853 | LPNYNWNSFGLRF)
Affinity DataKi:  552nMAssay Description:Displacement of [125]metastin from metastin receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKiSS-1 receptor(Homo sapiens (Human))
University Of Minnesota Health Science Center

Curated by ChEMBL
LigandPNGBDBM50203818(3-(1-(3-aminopropyl)-1H-indazol-3-yl)-4-(1-(benzo[...)
Affinity DataKi:  708nMAssay Description:Displacement of [125]metastin from metastin receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKiSS-1 receptor(Homo sapiens (Human))
University Of Minnesota Health Science Center

Curated by ChEMBL
LigandPNGBDBM50203792((2S)-2-{[(2S)-1-[(2S)-2-amino-4-methylpentanoyl]py...)
Affinity DataKi:  775nMAssay Description:Displacement of [125]metastin from metastin receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKiSS-1 receptor(Homo sapiens (Human))
University Of Minnesota Health Science Center

Curated by ChEMBL
LigandPNGBDBM50203812(CHEMBL221753 | benzethonium hydrochloride | cid_84...)
Affinity DataKi:  3.60E+3nMAssay Description:Displacement of [125]metastin from metastin receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKiSS-1 receptor(Homo sapiens (Human))
University Of Minnesota Health Science Center

Curated by ChEMBL
LigandPNGBDBM50203808((2S)-2-{[(2S)-1-[(2S)-2-amino-4-methylpentanoyl]py...)
Affinity DataKi:  1.00E+4nMAssay Description:Displacement of [125]metastin from metastin receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKiSS-1 receptor(Homo sapiens (Human))
University Of Minnesota Health Science Center

Curated by ChEMBL
LigandPNGBDBM50203804((2S)-2-{[(2S)-1-[(2S)-2-amino-4-methylpentanoyl]py...)
Affinity DataKi:  1.00E+4nMAssay Description:Displacement of [125]metastin from metastin receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKiSS-1 receptor(Homo sapiens (Human))
University Of Minnesota Health Science Center

Curated by ChEMBL
LigandPNGBDBM50203793((2S)-2-[(2S)-2-[(2S)-2-{[(2S)-1-[(2S)-2-amino-4-me...)
Affinity DataKi:  1.00E+4nMAssay Description:Displacement of [125]metastin from metastin receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKiSS-1 receptor(Homo sapiens (Human))
University Of Minnesota Health Science Center

Curated by ChEMBL
LigandPNGBDBM50203801((2S)-2-{[(2S)-1-[(2S)-2-amino-4-methylpentanoyl]py...)
Affinity DataKi:  1.00E+4nMAssay Description:Displacement of [125]metastin from metastin receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKiSS-1 receptor(Homo sapiens (Human))
University Of Minnesota Health Science Center

Curated by ChEMBL
LigandPNGBDBM50203815((2S)-2-{[(2S)-1-[(2S)-2-amino-4-methylpentanoyl]py...)
Affinity DataKi:  1.00E+4nMAssay Description:Displacement of [125]metastin from metastin receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKiSS-1 receptor(Homo sapiens (Human))
University Of Minnesota Health Science Center

Curated by ChEMBL
LigandPNGBDBM50203783(CHEMBL262316 | LPNYNWNSFLRF-NH2)
Affinity DataKi:  1.00E+4nMAssay Description:Displacement of [125]metastin from metastin receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKiSS-1 receptor(Homo sapiens (Human))
University Of Minnesota Health Science Center

Curated by ChEMBL
LigandPNGBDBM50203806((2S)-2-{[(2S)-1-[(2S)-2-amino-4-methylpentanoyl]py...)
Affinity DataKi:  1.00E+4nMAssay Description:Displacement of [125]metastin from metastin receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCathepsin S(Homo sapiens (Human))
Johnson & Johnson Pharmaceutical Research And Development

Curated by ChEMBL
LigandPNGBDBM50152984(1-(4-Phenyl-piperazin-1-yl)-3-(3-phenyl-4,5,6,7-te...)
Affinity DataIC50:  5nMAssay Description:Inhibitory concentration against human cysteine protease cathepsin SMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C beta type(Homo sapiens (Human))
Johnson And Johnson Pharmaceutical Research And Development

Curated by ChEMBL
LigandPNGBDBM17055((18S)-18-[(dimethylamino)methyl]-17-oxa-4,14,21-tr...)
Affinity DataIC50:  6nMAssay Description:Inhibition of Protein kinase C beta 2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C beta type(Homo sapiens (Human))
Johnson And Johnson Pharmaceutical Research And Development

Curated by ChEMBL
LigandPNGBDBM50133057(17,20,23-trioxa-4,14,26-triazahexacyclo[24.6.1.17,...)
Affinity DataIC50:  6nMAssay Description:Inhibition of Protein kinase C beta 2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProcathepsin L(Homo sapiens (Human))
University Of Pennsylvania

Curated by ChEMBL
LigandPNGBDBM51395(CHEMBL263634 | N-[(2S)-1-[[[2-(3,4-dihydro-2H-quin...)
Affinity DataIC50:  7nMAssay Description:Inhibition of human cathepsin LMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-IIb/beta-3(Homo sapiens (Human))
R. W. Johnson Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50034690(3-{[(R)-1-((S)-6-Amino-2-tert-butoxycarbonylamino-...)
Affinity DataIC50:  8nMAssay Description:Inhibition of biotinylated fibrinogen binding to isolated alpha IIb beta3 integrinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-IIb/beta-3(Homo sapiens (Human))
R. W. Johnson Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50034703(3-{[1-(3-Piperidin-4-yl-propionyl)-piperidine-3-ca...)
Affinity DataIC50:  9nMAssay Description:Inhibition of biotinylated fibrinogen binding to isolated alpha IIb beta3 integrinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium/glucose cotransporter 2(Homo sapiens (Human))
Johnson & Johnson Pharmaceutical Research And Development

Curated by ChEMBL
LigandPNGBDBM20877(3-(1-benzofuran-5-yl)-1-(2-hydroxy-4-methyl-6-{[(2...)
Affinity DataIC50:  11nMAssay Description:Inhibitory activity aginst SGLT2 expressed in CHO-K1 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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