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Found 53 with Last Name = 'bergeron' and Initial = 'f'
TargetGastrin/cholecystokinin type B receptor(Homo sapiens (Human))
University of Paris

Curated by ChEMBL
LigandPNGBDBM50228604(CHEMBL3350720)
Affinity DataKi:  54nMAssay Description:Apparent affinity to inhibit binding of [3H]pCCK-8 to Cholecystokinin type B receptor of guinea pig brain membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGastrin/cholecystokinin type B receptor(Homo sapiens (Human))
University of Paris

Curated by ChEMBL
LigandPNGBDBM50228605(CHEMBL3350665)
Affinity DataKi:  93nMAssay Description:Apparent affinity to inhibit binding of [3H]-pCCK-8 to Cholecystokinin type B receptor of guinea pig brain membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGastrin/cholecystokinin type B receptor(Homo sapiens (Human))
University of Paris

Curated by ChEMBL
LigandPNGBDBM50228605(CHEMBL3350665)
Affinity DataKi:  93nMAssay Description:Apparent affinity to inhibit binding of [3H]-pCCK-8 to Cholecystokinin type A receptor of guinea pig pancreatic membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholecystokinin receptor type A(Cavia porcellus)
University of Paris

Curated by ChEMBL
LigandPNGBDBM50228603(CHEMBL3350278)
Affinity DataKi:  200nMAssay Description:Apparent affinity to inhibit binding of [3H]pCCK-8 to Cholecystokinin type A receptor of guinea pig pancreatic membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholecystokinin receptor type A(Cavia porcellus)
University of Paris

Curated by ChEMBL
LigandPNGBDBM50228604(CHEMBL3350720)
Affinity DataKi:  230nMAssay Description:Apparent affinity to inhibit binding of [3H]pCCK-8 to Cholecystokinin type A receptor of guinea pig pancreatic membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholecystokinin receptor type A(Cavia porcellus)
University of Paris

Curated by ChEMBL
LigandPNGBDBM50228605(CHEMBL3350665)
Affinity DataKi:  310nMAssay Description:Apparent affinity to inhibit binding of [3H]-pCCK-8 to Cholecystokinin type B receptor of guinea pig brain membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholecystokinin receptor type A(Cavia porcellus)
University of Paris

Curated by ChEMBL
LigandPNGBDBM50228605(CHEMBL3350665)
Affinity DataKi:  340nMAssay Description:Apparent affinity to inhibit binding of [3H]-pCCK-8 to Cholecystokinin type A receptor of guinea pig pancreatic membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholecystokinin receptor type A(Cavia porcellus)
University of Paris

Curated by ChEMBL
LigandPNGBDBM50228602(CHEMBL3350331)
Affinity DataKi:  340nMAssay Description:Apparent affinity to inhibit binding of [3H]-pCCK-8 to Cholecystokinin type B receptor of guinea pig brain membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGastrin/cholecystokinin type B receptor(Homo sapiens (Human))
University of Paris

Curated by ChEMBL
LigandPNGBDBM50228602(CHEMBL3350331)
Affinity DataKi:  580nMAssay Description:Apparent affinity to inhibit binding of [3H]pCCK-8 to Cholecystokinin type B receptor of guinea pig brain membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholecystokinin receptor type A(Cavia porcellus)
University of Paris

Curated by ChEMBL
LigandPNGBDBM50007932(Boc-Tyr(SO3H)NLe-Gly-Trp-Orn(Z)-Asp-NH2 | CHEMBL23...)
Affinity DataKi:  660nMAssay Description:Apparent affinity to inhibit binding of [3H]-pCCK-8 to Cholecystokinin type A receptor of guinea pig pancreatic membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGastrin/cholecystokinin type B receptor(Homo sapiens (Human))
University of Paris

Curated by ChEMBL
LigandPNGBDBM50007932(Boc-Tyr(SO3H)NLe-Gly-Trp-Orn(Z)-Asp-NH2 | CHEMBL23...)
Affinity DataKi:  660nMAssay Description:Apparent affinity to inhibit binding of [3H]-pCCK-8 to Cholecystokinin type B receptor of guinea pig brain membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGastrin/cholecystokinin type B receptor(Homo sapiens (Human))
University of Paris

Curated by ChEMBL
LigandPNGBDBM50007929(3-{5-Amino-2-[2-tert-butoxycarbonylamino-3-(1H-ind...)
Affinity DataKi:  1.40E+3nMAssay Description:Apparent affinity to inhibit binding of [3H]-pCCK-8 to Cholecystokinin type B receptor of guinea pig brain membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGastrin/cholecystokinin type B receptor(Homo sapiens (Human))
University of Paris

Curated by ChEMBL
LigandPNGBDBM50007933(3-{5-tert-Butoxycarbonylamino-2-[2-tert-butoxycarb...)
Affinity DataKi:  2.20E+3nMAssay Description:Apparent affinity to inhibit binding of [3H]-pCCK-8 to Cholecystokinin type B receptor of guinea pig brain membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGastrin/cholecystokinin type B receptor(Homo sapiens (Human))
University of Paris

Curated by ChEMBL
LigandPNGBDBM50228603(CHEMBL3350278)
Affinity DataKi:  4.20E+3nMAssay Description:Apparent affinity to inhibit binding of [3H]pCCK-8 to Cholecystokinin type B receptor of guinea pig brain membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGastrin/cholecystokinin type B receptor(Homo sapiens (Human))
University of Paris

Curated by ChEMBL
LigandPNGBDBM50007930(3-{5-tert-Butoxycarbonylamino-2-[2-tert-butoxycarb...)
Affinity DataKi:  4.30E+3nMAssay Description:Apparent affinity to inhibit binding of [3H]-pCCK-8 to Cholecystokinin type B receptor of guinea pig brain membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholecystokinin receptor type A(Cavia porcellus)
University of Paris

Curated by ChEMBL
LigandPNGBDBM50007933(3-{5-tert-Butoxycarbonylamino-2-[2-tert-butoxycarb...)
Affinity DataKi:  5.20E+3nMAssay Description:Apparent affinity to inhibit binding of [3H]-pCCK-8 to Cholecystokinin type A receptor of guinea pig pancreatic membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholecystokinin receptor type A(Cavia porcellus)
University of Paris

Curated by ChEMBL
LigandPNGBDBM50007929(3-{5-Amino-2-[2-tert-butoxycarbonylamino-3-(1H-ind...)
Affinity DataKi:  1.40E+4nMAssay Description:Apparent affinity to inhibit binding of [3H]-pCCK-8 to Cholecystokinin type A receptor of guinea pig pancreatic membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholecystokinin receptor type A(Cavia porcellus)
University of Paris

Curated by ChEMBL
LigandPNGBDBM50007930(3-{5-tert-Butoxycarbonylamino-2-[2-tert-butoxycarb...)
Affinity DataKi:  2.90E+4nMAssay Description:Apparent affinity to inhibit binding of [3H]-pCCK-8 to Cholecystokinin type A receptor of guinea pig pancreatic membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGastrin/cholecystokinin type B receptor(Homo sapiens (Human))
University of Paris

Curated by ChEMBL
LigandPNGBDBM50421881(CHEMBL2112488)
Affinity DataKi:  1.00E+5nMAssay Description:Apparent affinity to inhibit binding of [3H]-pCCK-8 to Cholecystokinin type B receptor of guinea pig brain membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholecystokinin receptor type A(Cavia porcellus)
University of Paris

Curated by ChEMBL
LigandPNGBDBM50421881(CHEMBL2112488)
Affinity DataKi:  1.00E+6nMAssay Description:Apparent affinity to inhibit binding of [3H]-pCCK-8 to Cholecystokinin type A receptor of guinea pig pancreatic membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-V/beta-3(Homo sapiens (Human))
Shire Biochem

Curated by ChEMBL
LigandPNGBDBM50123247((S)-3-{[5-(3-Guanidino-phenyl)-thiophene-2-carbony...)
Affinity DataIC50:  0.000920nMAssay Description:Inhibition of fibrinogen binding to K562 cells expressing integrin alphaV-beta3More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-IIb/beta-3(Homo sapiens (Human))
Shire Biochem

Curated by ChEMBL
LigandPNGBDBM50123246((S)-2-Benzenesulfonylamino-3-{[5-(4-guanidino-phen...)
Affinity DataIC50:  0.00130nMAssay Description:Inhibition of vitronectin binding to HT-29 cells expressing integrin alphaV-beta5More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-IIb/beta-3(Homo sapiens (Human))
Shire Biochem

Curated by ChEMBL
LigandPNGBDBM50123251((S)-2-Benzenesulfonylamino-3-{[5-(2-guanidinomethy...)
Affinity DataIC50:  0.00580nMAssay Description:Inhibition of fibrinogen binding to integrin alphaV-beta3 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-V/beta-3(Homo sapiens (Human))
Shire Biochem

Curated by ChEMBL
LigandPNGBDBM50123251((S)-2-Benzenesulfonylamino-3-{[5-(2-guanidinomethy...)
Affinity DataIC50:  0.0400nMAssay Description:Inhibition of fibrinogen binding to integrin alphaIIb-beta3More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-IIb/beta-3(Homo sapiens (Human))
Shire Biochem

Curated by ChEMBL
LigandPNGBDBM50123253((S)-3-{[5-(3-Guanidinomethyl-phenyl)-thiophene-2-c...)
Affinity DataIC50:  0.160nMAssay Description:Inhibition of fibrinogen binding to K562 cells expressing integrin alphaV-beta3More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-V/beta-3(Homo sapiens (Human))
Shire Biochem

Curated by ChEMBL
LigandPNGBDBM50123249((S)-2-Benzenesulfonylamino-3-{[5-(3-guanidino-phen...)
Affinity DataIC50:  0.190nMAssay Description:Inhibition of fibrinogen binding to K562 cells expressing integrin alphaV-beta3More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-IIb/beta-3(Homo sapiens (Human))
Shire Biochem

Curated by ChEMBL
LigandPNGBDBM50123252((S)-2-Benzenesulfonylamino-3-{[5-(2-guanidino-phen...)
Affinity DataIC50:  0.25nMAssay Description:Inhibition of fibrinogen binding to K562 cells expressing integrin alpha5-beta1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-IIb/beta-3(Homo sapiens (Human))
Shire Biochem

Curated by ChEMBL
LigandPNGBDBM50123247((S)-3-{[5-(3-Guanidino-phenyl)-thiophene-2-carbony...)
Affinity DataIC50:  0.310nMAssay Description:Inhibition of fibrinogen binding to integrin alphaV-beta3 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-IIb/beta-3(Homo sapiens (Human))
Shire Biochem

Curated by ChEMBL
LigandPNGBDBM50123248((S)-2-Benzenesulfonylamino-3-{[5-(3-guanidinomethy...)
Affinity DataIC50:  0.340nMAssay Description:Inhibition of fibrinogen binding to integrin alphaV-beta3 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-IIb/beta-3(Homo sapiens (Human))
Shire Biochem

Curated by ChEMBL
LigandPNGBDBM50123249((S)-2-Benzenesulfonylamino-3-{[5-(3-guanidino-phen...)
Affinity DataIC50:  0.590nMAssay Description:Inhibition of vitronectin binding to HT-29 cells expressing integrin alphaV-beta5More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-V/beta-3(Homo sapiens (Human))
Shire Biochem

Curated by ChEMBL
LigandPNGBDBM50123248((S)-2-Benzenesulfonylamino-3-{[5-(3-guanidinomethy...)
Affinity DataIC50:  0.740nMAssay Description:Inhibition of fibrinogen binding to integrin alphaIIb-beta3More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-V/beta-3(Homo sapiens (Human))
Shire Biochem

Curated by ChEMBL
LigandPNGBDBM50123249((S)-2-Benzenesulfonylamino-3-{[5-(3-guanidino-phen...)
Affinity DataIC50:  1nMAssay Description:Inhibition of fibrinogen binding to integrin alphaV-beta3 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-V/beta-3(Homo sapiens (Human))
Shire Biochem

Curated by ChEMBL
LigandPNGBDBM50123247((S)-3-{[5-(3-Guanidino-phenyl)-thiophene-2-carbony...)
Affinity DataIC50:  1.40nMAssay Description:Inhibition of fibrinogen binding to K562 cells expressing integrin alphaV-beta3More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-V/beta-3(Homo sapiens (Human))
Shire Biochem

Curated by ChEMBL
LigandPNGBDBM50123250((S)-2-Benzenesulfonylamino-3-{[5-(4-guanidinomethy...)
Affinity DataIC50:  2.10nMAssay Description:Inhibition of fibrinogen binding to K562 cells expressing integrin alpha5-beta1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-V/beta-3(Homo sapiens (Human))
Shire Biochem

Curated by ChEMBL
LigandPNGBDBM50123248((S)-2-Benzenesulfonylamino-3-{[5-(3-guanidinomethy...)
Affinity DataIC50:  2.20nMAssay Description:Inhibition of fibrinogen binding to integrin alphaV-beta3 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-V/beta-5(Homo sapiens (Human))
Shire Biochem

Curated by ChEMBL
LigandPNGBDBM50123251((S)-2-Benzenesulfonylamino-3-{[5-(2-guanidinomethy...)
Affinity DataIC50:  2.20nMAssay Description:Inhibition of fibrinogen binding to integrin alphaV-beta3 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-V/beta-5(Homo sapiens (Human))
Shire Biochem

Curated by ChEMBL
LigandPNGBDBM50123247((S)-3-{[5-(3-Guanidino-phenyl)-thiophene-2-carbony...)
Affinity DataIC50:  2.5nMAssay Description:Inhibition of fibrinogen binding to K562 cells expressing integrin alphaV-beta3More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-V/beta-3(Homo sapiens (Human))
Shire Biochem

Curated by ChEMBL
LigandPNGBDBM50123253((S)-3-{[5-(3-Guanidinomethyl-phenyl)-thiophene-2-c...)
Affinity DataIC50:  3.40nMAssay Description:Inhibition of vitronectin binding to HT-29 cells expressing integrin alphaV-beta5More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-IIb/beta-3(Homo sapiens (Human))
Shire Biochem

Curated by ChEMBL
LigandPNGBDBM50123250((S)-2-Benzenesulfonylamino-3-{[5-(4-guanidinomethy...)
Affinity DataIC50:  6.10nMAssay Description:Inhibition of fibrinogen binding to integrin alphaIIb-beta3More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-V/beta-5(Homo sapiens (Human))
Shire Biochem

Curated by ChEMBL
LigandPNGBDBM50123249((S)-2-Benzenesulfonylamino-3-{[5-(3-guanidino-phen...)
Affinity DataIC50:  6.40nMAssay Description:Inhibition of fibrinogen binding to K562 cells expressing integrin alphaV-beta3More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-V/beta-3(Homo sapiens (Human))
Shire Biochem

Curated by ChEMBL
LigandPNGBDBM50123253((S)-3-{[5-(3-Guanidinomethyl-phenyl)-thiophene-2-c...)
Affinity DataIC50:  11nMAssay Description:Inhibition of fibrinogen binding to integrin alphaV-beta3 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-V/beta-5(Homo sapiens (Human))
Shire Biochem

Curated by ChEMBL
LigandPNGBDBM50123253((S)-3-{[5-(3-Guanidinomethyl-phenyl)-thiophene-2-c...)
Affinity DataIC50:  11nMAssay Description:Inhibition of fibrinogen binding to K562 cells expressing integrin alpha5-beta1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-V/beta-3(Homo sapiens (Human))
Shire Biochem

Curated by ChEMBL
LigandPNGBDBM50123251((S)-2-Benzenesulfonylamino-3-{[5-(2-guanidinomethy...)
Affinity DataIC50:  21nMAssay Description:Inhibition of fibrinogen binding to integrin alphaIIb-beta3More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-5/beta-1(Homo sapiens (Human))
Shire Biochem

Curated by ChEMBL
LigandPNGBDBM50123247((S)-3-{[5-(3-Guanidino-phenyl)-thiophene-2-carbony...)
Affinity DataIC50:  26nMAssay Description:Inhibition of fibrinogen binding to integrin alphaV-beta3 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-5/beta-1(Homo sapiens (Human))
Shire Biochem

Curated by ChEMBL
LigandPNGBDBM50123253((S)-3-{[5-(3-Guanidinomethyl-phenyl)-thiophene-2-c...)
Affinity DataIC50:  71nMAssay Description:Inhibition of fibrinogen binding to K562 cells expressing integrin alpha5-beta1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-V/beta-5(Homo sapiens (Human))
Shire Biochem

Curated by ChEMBL
LigandPNGBDBM50123248((S)-2-Benzenesulfonylamino-3-{[5-(3-guanidinomethy...)
Affinity DataIC50:  72nMAssay Description:Inhibition of fibrinogen binding to K562 cells expressing integrin alphaV-beta3More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-V/beta-3(Homo sapiens (Human))
Shire Biochem

Curated by ChEMBL
LigandPNGBDBM50123246((S)-2-Benzenesulfonylamino-3-{[5-(4-guanidino-phen...)
Affinity DataIC50:  72nMAssay Description:Inhibition of vitronectin binding to HT-29 cells expressing integrin alphaV-beta5More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-5/beta-1(Homo sapiens (Human))
Shire Biochem

Curated by ChEMBL
LigandPNGBDBM50123249((S)-2-Benzenesulfonylamino-3-{[5-(3-guanidino-phen...)
Affinity DataIC50:  95nMAssay Description:Inhibition of fibrinogen binding to integrin alphaIIb-beta3More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-5/beta-1(Homo sapiens (Human))
Shire Biochem

Curated by ChEMBL
LigandPNGBDBM50123248((S)-2-Benzenesulfonylamino-3-{[5-(3-guanidinomethy...)
Affinity DataIC50:  640nMAssay Description:Inhibition of fibrinogen binding to integrin alphaIIb-beta3More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-V/beta-3(Homo sapiens (Human))
Shire Biochem

Curated by ChEMBL
LigandPNGBDBM50123250((S)-2-Benzenesulfonylamino-3-{[5-(4-guanidinomethy...)
Affinity DataIC50:  730nMAssay Description:Inhibition of fibrinogen binding to K562 cells expressing integrin alphaV-beta3More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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