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Found 126 with Last Name = 'boblewski' and Initial = 'k'
LigandPNGBDBM50271255(1-[(Imidazolidin-2-yl)imino]indazole hydrochloride...)
Affinity DataKi:  14nMAssay Description:Displacement of [3H]RX821002 from alpha2-adrenoceptor in Sprague-Dawley rat brain membranes after 45 mins by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50497435(CHEMBL3343699)
Affinity DataKi:  26nMAssay Description:Displacement of [3H]RX821002 from alpha2-adrenoceptor in Sprague-Dawley rat brain membranes after 45 mins by liquid scintillation countingMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
LigandPNGBDBM50497438(CHEMBL3343704)
Affinity DataKi:  30nMAssay Description:Displacement of [3H]RX821002 from alpha2-adrenoceptor in Sprague-Dawley rat brain membranes after 45 mins by liquid scintillation countingMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetNischarin(RAT)
Medical University Of Gdansk

Curated by ChEMBL
LigandPNGBDBM50334197(7-Chloro-3-[(imidazolidin-2-yl)imino]indazole hydr...)
Affinity DataKi:  30.8nMAssay Description:Displacement of [3H]2BFI from imidazoline I1 receptor in Sprague-Dawley rat brain membrane after 45 mins by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50497439(CHEMBL3343700)
Affinity DataKi:  31nMAssay Description:Displacement of [3H]RX821002 from alpha2-adrenoceptor in Sprague-Dawley rat brain membranes after 45 mins by liquid scintillation countingMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetNischarin(RAT)
Medical University Of Gdansk

Curated by ChEMBL
LigandPNGBDBM50164835(CHEMBL3800398)
Affinity DataKi:  32nMAssay Description:Displacement of [3H]clonidine from Imidazoline receptor 1 in Sprague-Dawley rat kidney P2 membranes after 45 hrs by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50497436(CHEMBL3343703)
Affinity DataKi:  32nMAssay Description:Displacement of [3H]RX821002 from alpha2-adrenoceptor in Sprague-Dawley rat brain membranes after 45 mins by liquid scintillation countingMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAlpha-2A adrenergic receptor(Homo sapiens (Human))
Medical University Of Gdansk

Curated by ChEMBL
LigandPNGBDBM50497435(CHEMBL3343699)
Affinity DataKi:  33nMAssay Description:Displacement of [3H]RS-79948-197 from human alpha2A adrenoceptor expressed in CHO-K1 cells after 45 mins by liquid scintillation countingMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetNischarin(RAT)
Medical University Of Gdansk

Curated by ChEMBL
LigandPNGBDBM50334195(4-Chloro-3-[(imidazolidin-2-yl)imino]indazole hydr...)
Affinity DataKi:  45.2nMAssay Description:Displacement of [3H]2BFI from imidazoline I1 receptor in Sprague-Dawley rat brain membrane after 45 mins by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-2A adrenergic receptor(Homo sapiens (Human))
Medical University Of Gdansk

Curated by ChEMBL
LigandPNGBDBM50271255(1-[(Imidazolidin-2-yl)imino]indazole hydrochloride...)
Affinity DataKi:  52nMAssay Description:Displacement of [3H]RS-79948-197 from human alpha2A adrenoceptor expressed in CHO-K1 cells after 45 mins by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50497440(CHEMBL3343698)
Affinity DataKi:  64nMAssay Description:Displacement of [3H]RX821002 from alpha2-adrenoceptor in Sprague-Dawley rat brain membranes after 45 mins by liquid scintillation countingMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAlpha-2A adrenergic receptor(Homo sapiens (Human))
Medical University Of Gdansk

Curated by ChEMBL
LigandPNGBDBM50497439(CHEMBL3343700)
Affinity DataKi:  65nMAssay Description:Displacement of [3H]RS-79948-197 from human alpha2A adrenoceptor expressed in CHO-K1 cells after 45 mins by liquid scintillation countingMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAlpha-2B adrenergic receptor(Homo sapiens (Human))
Medical University Of Gdansk

Curated by ChEMBL
LigandPNGBDBM50497435(CHEMBL3343699)
Affinity DataKi:  72nMAssay Description:Displacement of [3H]RS-79948-197 from human alpha2B adrenoceptor expressed in CHO-K1 cells after 45 mins by liquid scintillation countingMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAlpha-2B adrenergic receptor(Homo sapiens (Human))
Medical University Of Gdansk

Curated by ChEMBL
LigandPNGBDBM50271255(1-[(Imidazolidin-2-yl)imino]indazole hydrochloride...)
Affinity DataKi:  79nMAssay Description:Displacement of [3H]RS-79948-197 from human alpha2B adrenoceptor expressed in CHO-K1 cells after 45 mins by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNischarin(RAT)
Medical University Of Gdansk

Curated by ChEMBL
LigandPNGBDBM50164841(CHEMBL3798191)
Affinity DataKi:  79nMAssay Description:Displacement of [3H]clonidine from Imidazoline receptor 1 in Sprague-Dawley rat kidney P2 membranes after 45 hrs by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNischarin(RAT)
Medical University Of Gdansk

Curated by ChEMBL
LigandPNGBDBM50334196(3-[(Imidazolidin-2-yl)imino]-4-methylindazole hydr...)
Affinity DataKi:  133nMAssay Description:Displacement of [3H]2BFI from imidazoline I1 receptor in Sprague-Dawley rat brain membrane after 45 mins by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNischarin(RAT)
Medical University Of Gdansk

Curated by ChEMBL
LigandPNGBDBM50334194(3-[(Imidazolidin-2-yl)imino]indazole hydrochloride...)
Affinity DataKi:  134nMAssay Description:Displacement of [3H]2BFI from imidazoline I1 receptor in Sprague-Dawley rat brain membrane after 45 mins by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-2B adrenergic receptor(Homo sapiens (Human))
Medical University Of Gdansk

Curated by ChEMBL
LigandPNGBDBM50497439(CHEMBL3343700)
Affinity DataKi:  158nMAssay Description:Displacement of [3H]RS-79948-197 from human alpha2B adrenoceptor expressed in CHO-K1 cells after 45 mins by liquid scintillation countingMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetNischarin(RAT)
Medical University Of Gdansk

Curated by ChEMBL
LigandPNGBDBM50334206(3-[(Imidazolidin-2-yl)imino]-4-methoxyindazole hyd...)
Affinity DataKi:  167nMAssay Description:Displacement of [3H]2BFI from imidazoline I1 receptor in Sprague-Dawley rat brain membrane after 45 mins by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50497433(CHEMBL3343702)
Affinity DataKi:  187nMAssay Description:Displacement of [3H]RX821002 from alpha2-adrenoceptor in Sprague-Dawley rat brain membranes after 45 mins by liquid scintillation countingMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetNischarin(RAT)
Medical University Of Gdansk

Curated by ChEMBL
LigandPNGBDBM50334204(3-[(Imidazolidin-2-yl)imino]-6-methylindazole hydr...)
Affinity DataKi:  325nMAssay Description:Displacement of [3H]2BFI from imidazoline I1 receptor in Sprague-Dawley rat brain membrane after 45 mins by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNischarin(RAT)
Medical University Of Gdansk

Curated by ChEMBL
LigandPNGBDBM50334203(6-Chloro-3-[(imidazolidin-2-yl)imino]indazole hydr...)
Affinity DataKi:  410nMAssay Description:Displacement of [3H]2BFI from imidazoline I1 receptor in Sprague-Dawley rat brain membrane after 45 mins by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50497434(CHEMBL3343697)
Affinity DataKi:  416nMAssay Description:Displacement of [3H]RX821002 from alpha2-adrenoceptor in Sprague-Dawley rat brain membranes after 45 mins by liquid scintillation countingMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetNischarin(RAT)
Medical University Of Gdansk

Curated by ChEMBL
LigandPNGBDBM50164834(CHEMBL3798638)
Affinity DataKi:  468nMAssay Description:Displacement of [3H]clonidine from Imidazoline receptor 1 in Sprague-Dawley rat kidney P2 membranes after 45 hrs by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1A/Alpha-1B/Alpha-1D adrenergic receptor(Rattus norvegicus (rat))
Medical University Of Gdansk

Curated by ChEMBL
LigandPNGBDBM50497436(CHEMBL3343703)
Affinity DataKi:  476nMAssay Description:Displacement of [3H]prazosin from alpha1-adrenoceptor in Sprague-Dawley rat brain membranes after 45 mins by liquid scintillation countingMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAlpha-1A/Alpha-1B/Alpha-1D adrenergic receptor(Rattus norvegicus (rat))
Medical University Of Gdansk

Curated by ChEMBL
LigandPNGBDBM50497438(CHEMBL3343704)
Affinity DataKi:  518nMAssay Description:Displacement of [3H]prazosin from alpha1-adrenoceptor in Sprague-Dawley rat brain membranes after 45 mins by liquid scintillation countingMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAlpha-1A/Alpha-1B/Alpha-1D adrenergic receptor(Rattus norvegicus (rat))
Medical University Of Gdansk

Curated by ChEMBL
LigandPNGBDBM50497433(CHEMBL3343702)
Affinity DataKi:  535nMAssay Description:Displacement of [3H]prazosin from alpha1-adrenoceptor in Sprague-Dawley rat brain membranes after 45 mins by liquid scintillation countingMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAlpha-2C adrenergic receptor(Homo sapiens (Human))
Medical University Of Gdansk

Curated by ChEMBL
LigandPNGBDBM50497435(CHEMBL3343699)
Affinity DataKi:  600nMAssay Description:Displacement of [3H]RS-79948-197 from human alpha2C adrenoceptor expressed in CHO-K1 cells after 45 mins by liquid scintillation countingMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAlpha-2C adrenergic receptor(Homo sapiens (Human))
Medical University Of Gdansk

Curated by ChEMBL
LigandPNGBDBM50271255(1-[(Imidazolidin-2-yl)imino]indazole hydrochloride...)
Affinity DataKi:  640nMAssay Description:Displacement of [3H]RS-79948-197 from human alpha2C adrenoceptor expressed in CHO-K1 cells after 45 mins by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNischarin(RAT)
Medical University Of Gdansk

Curated by ChEMBL
LigandPNGBDBM50164837(CHEMBL3800446)
Affinity DataKi:  789nMAssay Description:Displacement of [3H]clonidine from Imidazoline receptor 1 in Sprague-Dawley rat kidney P2 membranes after 45 hrs by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1A/Alpha-1B/Alpha-1D adrenergic receptor(Rattus norvegicus (rat))
Medical University Of Gdansk

Curated by ChEMBL
LigandPNGBDBM50497435(CHEMBL3343699)
Affinity DataKi:  918nMAssay Description:Displacement of [3H]prazosin from alpha1-adrenoceptor in Sprague-Dawley rat brain membranes after 45 mins by liquid scintillation countingMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetNischarin(RAT)
Medical University Of Gdansk

Curated by ChEMBL
LigandPNGBDBM50164842(CHEMBL3798387)
Affinity DataKi:  1.00E+3nMAssay Description:Displacement of [3H]clonidine from Imidazoline receptor 1 in Sprague-Dawley rat kidney P2 membranes after 45 hrs by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-2C adrenergic receptor(Homo sapiens (Human))
Medical University Of Gdansk

Curated by ChEMBL
LigandPNGBDBM50497439(CHEMBL3343700)
Affinity DataKi:  1.20E+3nMAssay Description:Displacement of [3H]RS-79948-197 from human alpha2C adrenoceptor expressed in CHO-K1 cells after 45 mins by liquid scintillation countingMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAlpha-1A/Alpha-1B/Alpha-1D adrenergic receptor(Rattus norvegicus (rat))
Medical University Of Gdansk

Curated by ChEMBL
LigandPNGBDBM50497439(CHEMBL3343700)
Affinity DataKi:  1.63E+3nMAssay Description:Displacement of [3H]prazosin from alpha1-adrenoceptor in Sprague-Dawley rat brain membranes after 45 mins by liquid scintillation countingMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAlpha-1A/Alpha-1B/Alpha-1D adrenergic receptor(Rattus norvegicus (rat))
Medical University Of Gdansk

Curated by ChEMBL
LigandPNGBDBM50497440(CHEMBL3343698)
Affinity DataKi:  2.32E+3nMAssay Description:Displacement of [3H]prazosin from alpha1-adrenoceptor in Sprague-Dawley rat brain membranes after 45 mins by liquid scintillation countingMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
LigandPNGBDBM50497437(CHEMBL3343701)
Affinity DataKi:  3.72E+3nMAssay Description:Displacement of [3H]RX821002 from alpha2-adrenoceptor in Sprague-Dawley rat brain membranes after 45 mins by liquid scintillation countingMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAlpha-1A/Alpha-1B/Alpha-1D adrenergic receptor(Rattus norvegicus (rat))
Medical University Of Gdansk

Curated by ChEMBL
LigandPNGBDBM50497434(CHEMBL3343697)
Affinity DataKi:  3.81E+3nMAssay Description:Displacement of [3H]prazosin from alpha1-adrenoceptor in Sprague-Dawley rat brain membranes after 45 mins by liquid scintillation countingMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetNischarin(RAT)
Medical University Of Gdansk

Curated by ChEMBL
LigandPNGBDBM50334205(4-Bromo-3-[(imidazolidin-2-yl)imino]indazole hydro...)
Affinity DataKi:  5.38E+3nMAssay Description:Displacement of [3H]2BFI from imidazoline I1 receptor in Sprague-Dawley rat brain membrane after 45 mins by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNischarin(RAT)
Medical University Of Gdansk

Curated by ChEMBL
LigandPNGBDBM50164838(CHEMBL3797854)
Affinity DataKi:  5.58E+3nMAssay Description:Displacement of [3H]clonidine from Imidazoline receptor 1 in Sprague-Dawley rat kidney P2 membranes after 45 hrs by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNischarin(RAT)
Medical University Of Gdansk

Curated by ChEMBL
LigandPNGBDBM50164839(CHEMBL3797661)
Affinity DataKi:  9.63E+3nMAssay Description:Displacement of [3H]clonidine from Imidazoline receptor 1 in Sprague-Dawley rat kidney P2 membranes after 45 hrs by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNischarin(RAT)
Medical University Of Gdansk

Curated by ChEMBL
LigandPNGBDBM50334202(3-[(Imidazolidin-2-ylo)imino]-5-methoxyindazole hy...)
Affinity DataKi:  9.91E+3nMAssay Description:Displacement of [3H]2BFI from imidazoline I1 receptor in Sprague-Dawley rat brain membrane after 45 mins by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNischarin(RAT)
Medical University Of Gdansk

Curated by ChEMBL
LigandPNGBDBM50334208(3-[(Imidazolidin-2-yl)imino]-5-methylindazole hydr...)
Affinity DataKi:  1.02E+4nMAssay Description:Displacement of [3H]2BFI from imidazoline I1 receptor in Sprague-Dawley rat brain membrane after 45 mins by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNischarin(RAT)
Medical University Of Gdansk

Curated by ChEMBL
LigandPNGBDBM50164840(CHEMBL3799780)
Affinity DataKi:  1.03E+4nMAssay Description:Displacement of [3H]clonidine from Imidazoline receptor 1 in Sprague-Dawley rat kidney P2 membranes after 45 hrs by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNischarin(RAT)
Medical University Of Gdansk

Curated by ChEMBL
LigandPNGBDBM50164836(CHEMBL3798967)
Affinity DataKi:  1.05E+4nMAssay Description:Displacement of [3H]clonidine from Imidazoline receptor 1 in Sprague-Dawley rat kidney P2 membranes after 45 hrs by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNischarin(RAT)
Medical University Of Gdansk

Curated by ChEMBL
LigandPNGBDBM50164833(CHEMBL3799346)
Affinity DataKi:  1.46E+4nMAssay Description:Displacement of [3H]clonidine from Imidazoline receptor 1 in Sprague-Dawley rat kidney P2 membranes after 45 hrs by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1A/Alpha-1B/Alpha-1D adrenergic receptor(Rattus norvegicus (rat))
Medical University Of Gdansk

Curated by ChEMBL
LigandPNGBDBM50497437(CHEMBL3343701)
Affinity DataKi:  1.98E+4nMAssay Description:Displacement of [3H]prazosin from alpha1-adrenoceptor in Sprague-Dawley rat brain membranes after 45 mins by liquid scintillation countingMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetNischarin(RAT)
Medical University Of Gdansk

Curated by ChEMBL
LigandPNGBDBM50164845(CHEMBL3799081)
Affinity DataKi:  3.63E+4nMAssay Description:Displacement of [3H]clonidine from Imidazoline receptor 1 in Sprague-Dawley rat kidney P2 membranes after 45 hrs by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNischarin(RAT)
Medical University Of Gdansk

Curated by ChEMBL
LigandPNGBDBM50164843(CHEMBL3800486)
Affinity DataKi:  4.58E+4nMAssay Description:Displacement of [3H]clonidine from Imidazoline receptor 1 in Sprague-Dawley rat kidney P2 membranes after 45 hrs by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNischarin(RAT)
Medical University Of Gdansk

Curated by ChEMBL
LigandPNGBDBM50164832(CHEMBL3797481)
Affinity DataKi:  8.14E+4nMAssay Description:Displacement of [3H]clonidine from Imidazoline receptor 1 in Sprague-Dawley rat kidney P2 membranes after 45 hrs by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNischarin(RAT)
Medical University Of Gdansk

Curated by ChEMBL
LigandPNGBDBM50334207(5-Chloro-3-[(imidazolidin-2-yl)imino]indazole hydr...)
Affinity DataKi:  9.30E+4nMAssay Description:Displacement of [3H]2BFI from imidazoline I1 receptor in Sprague-Dawley rat brain membrane after 45 mins by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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