Compile Data Set for Download or QSAR
maximum 50k data
Found 43 with Last Name = 'boländer' and Initial = 'a'
TargetMicrotubule-associated protein tau(Homo sapiens (Human))
Technische Universit£T Darmstadt

Curated by ChEMBL
LigandPNGBDBM50398203(CHEMBL2181533)
Affinity DataIC50:  2nMAssay Description:Displacement of thiazene red from tau aggregateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMicrotubule-associated protein tau(Homo sapiens (Human))
Technische Universit£T Darmstadt

Curated by ChEMBL
LigandPNGBDBM50398204(CHEMBL2181532)
Affinity DataIC50:  2nMAssay Description:Displacement of thiazene red from tau aggregateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMicrotubule-associated protein tau(Homo sapiens (Human))
Technische Universit£T Darmstadt

Curated by ChEMBL
LigandPNGBDBM50398207(CHEMBL2181045)
Affinity DataIC50:  4nMAssay Description:Displacement of thiazene red from tau aggregateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMicrotubule-associated protein tau(Homo sapiens (Human))
Technische Universit£T Darmstadt

Curated by ChEMBL
LigandPNGBDBM50398209(CHEMBL2181041)
Affinity DataIC50:  6nMAssay Description:Displacement of thiazene red from tau aggregateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMicrotubule-associated protein tau(Homo sapiens (Human))
Technische Universit£T Darmstadt

Curated by ChEMBL
LigandPNGBDBM50398210(CHEMBL2181039)
Affinity DataIC50:  13nMAssay Description:Displacement of thiazene red from tau aggregateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMicrotubule-associated protein tau(Homo sapiens (Human))
Technische Universit£T Darmstadt

Curated by ChEMBL
LigandPNGBDBM50398205(CHEMBL2181531)
Affinity DataIC50:  17nMAssay Description:Displacement of thiazene red from tau aggregateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMicrotubule-associated protein tau(Homo sapiens (Human))
Technische Universit£T Darmstadt

Curated by ChEMBL
LigandPNGBDBM50398208(CHEMBL2181042)
Affinity DataIC50:  42nMAssay Description:Displacement of thiazene red from tau aggregateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlycogen synthase kinase-3 beta(Homo sapiens (Human))
Technische Universit£T Darmstadt

Curated by ChEMBL
LigandPNGBDBM50352490(CHEMBL1824331)
Affinity DataIC50:  98nMAssay Description:Inhibition of human GSK3-beta activity using Ser/Thr 9 peptide as substrate by FRET assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMicrotubule-associated protein tau(Homo sapiens (Human))
Technische Universit£T Darmstadt

Curated by ChEMBL
LigandPNGBDBM50398211(CHEMBL2181036)
Affinity DataIC50:  246nMAssay Description:Displacement of thiazene red from tau aggregateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMicrotubule-associated protein tau(Homo sapiens (Human))
Technische Universit£T Darmstadt

Curated by ChEMBL
LigandPNGBDBM50398200(CHEMBL2181538)
Affinity DataIC50:  1.25E+3nMAssay Description:Displacement of thiazene red from tau aggregateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMicrotubule-associated protein tau(Homo sapiens (Human))
Technische Universit£T Darmstadt

Curated by ChEMBL
LigandPNGBDBM50398201(CHEMBL2181537)
Affinity DataIC50:  1.59E+3nMAssay Description:Displacement of thiazene red from tau aggregateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMicrotubule-associated protein tau(Homo sapiens (Human))
Technische Universit£T Darmstadt

Curated by ChEMBL
LigandPNGBDBM50398202(CHEMBL2181535)
Affinity DataIC50:  4.71E+3nMAssay Description:Displacement of thiazene red from tau aggregateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMicrotubule-associated protein tau(Homo sapiens (Human))
Technische Universit£T Darmstadt

Curated by ChEMBL
LigandPNGBDBM50398206(CHEMBL2181047)
Affinity DataIC50:  7.47E+3nMAssay Description:Displacement of thiazene red from tau aggregateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlycogen synthase kinase-3 alpha(Homo sapiens (Human))
Technische Universit£T Darmstadt

Curated by ChEMBL
LigandPNGBDBM50229962(1-(4-methoxybenzyl)-3-(5-nitrothiazol-2-yl)urea | ...)
Affinity DataIC50:  7.00E+4nMAssay Description:Inhibition of human GSK3alpha activity using Ser/Thr 11 peptide as substrate by FRET assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlycogen synthase kinase-3 alpha(Homo sapiens (Human))
Technische Universit£T Darmstadt

Curated by ChEMBL
LigandPNGBDBM50352494(CHEMBL1824332)
Affinity DataIC50:  1.30E+5nMAssay Description:Inhibition of human GSK3alpha activity using Ser/Thr 11 peptide as substrate by FRET assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlycogen synthase kinase-3 beta(Homo sapiens (Human))
Technische Universit£T Darmstadt

Curated by ChEMBL
LigandPNGBDBM50352494(CHEMBL1824332)
Affinity DataIC50:  1.40E+5nMAssay Description:Inhibition of human GSK3-beta activity using Ser/Thr 9 peptide as substrate by FRET assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlycogen synthase kinase-3 alpha(Homo sapiens (Human))
Technische Universit£T Darmstadt

Curated by ChEMBL
LigandPNGBDBM50352492(CHEMBL1824540)
Affinity DataIC50:  2.20E+5nMAssay Description:Inhibition of human GSK3alpha activity using Ser/Thr 11 peptide as substrate by FRET assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlycogen synthase kinase-3 beta(Homo sapiens (Human))
Technische Universit£T Darmstadt

Curated by ChEMBL
LigandPNGBDBM50229962(1-(4-methoxybenzyl)-3-(5-nitrothiazol-2-yl)urea | ...)
Affinity DataIC50:  3.30E+5nMAssay Description:Inhibition of human GSK3-beta activity using Ser/Thr 9 peptide as substrate by FRET assayMore data for this Ligand-Target Pair
TargetGlycogen synthase kinase-3 alpha(Homo sapiens (Human))
Technische Universit£T Darmstadt

Curated by ChEMBL
LigandPNGBDBM50352493(CHEMBL1824334)
Affinity DataIC50:  3.70E+5nMAssay Description:Inhibition of human GSK3alpha activity using Ser/Thr 11 peptide as substrate by FRET assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlycogen synthase kinase-3 beta(Homo sapiens (Human))
Technische Universit£T Darmstadt

Curated by ChEMBL
LigandPNGBDBM50352493(CHEMBL1824334)
Affinity DataIC50:  5.10E+5nMAssay Description:Inhibition of human GSK3-beta activity using Ser/Thr 9 peptide as substrate by FRET assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlycogen synthase kinase-3 alpha(Homo sapiens (Human))
Technische Universit£T Darmstadt

Curated by ChEMBL
LigandPNGBDBM50352491(CHEMBL1824539)
Affinity DataIC50:  1.12E+6nMAssay Description:Inhibition of human GSK3alpha activity using Ser/Thr 11 peptide as substrate by FRET assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlycogen synthase kinase-3 beta(Homo sapiens (Human))
Technische Universit£T Darmstadt

Curated by ChEMBL
LigandPNGBDBM50352491(CHEMBL1824539)
Affinity DataIC50:  1.43E+6nMAssay Description:Inhibition of human GSK3-beta activity using Ser/Thr 9 peptide as substrate by FRET assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlycogen synthase kinase-3 beta(Homo sapiens (Human))
Technische Universit£T Darmstadt

Curated by ChEMBL
LigandPNGBDBM50352492(CHEMBL1824540)
Affinity DataIC50:  3.64E+6nMAssay Description:Inhibition of human GSK3-beta activity using Ser/Thr 9 peptide as substrate by FRET assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAurora kinase A(Homo sapiens (Human))
Technische Universit£T Darmstadt

Curated by ChEMBL
LigandPNGBDBM50352494(CHEMBL1824332)
Affinity DataIC50:  4.80E+6nMAssay Description:Inhibition of human AURKA activity using Ser/Thr 1 peptide as substrate by FRET assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCasein kinase I isoform epsilon(Homo sapiens (Human))
Technische Universit£T Darmstadt

Curated by ChEMBL
LigandPNGBDBM50352494(CHEMBL1824332)
Affinity DataIC50:  1.53E+7nMAssay Description:Inhibition of human CKI epsilon activity using Ser/Thr 11 peptide as substrate by FRET assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C alpha type(Homo sapiens (Human))
Technische Universit£T Darmstadt

Curated by ChEMBL
LigandPNGBDBM50352494(CHEMBL1824332)
Affinity DataIC50:  2.42E+7nMAssay Description:Inhibition of human PKCalpha activity using Ser/Thr 7 peptide as substrate by FRET assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCyclin-dependent kinase 5 activator 1(Homo sapiens (Human))
Technische Universit£T Darmstadt

Curated by ChEMBL
LigandPNGBDBM50352494(CHEMBL1824332)
Affinity DataIC50:  2.64E+7nMAssay Description:Inhibition of human CDK5/p35 activity using Ser/Thr 12 peptide as substrate by FRET assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAurora kinase A(Homo sapiens (Human))
Technische Universit£T Darmstadt

Curated by ChEMBL
LigandPNGBDBM50352493(CHEMBL1824334)
Affinity DataIC50: >1.00E+8nMAssay Description:Inhibition of human AURKA activity using Ser/Thr 1 peptide as substrate by FRET assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAurora kinase A(Homo sapiens (Human))
Technische Universit£T Darmstadt

Curated by ChEMBL
LigandPNGBDBM50352491(CHEMBL1824539)
Affinity DataIC50: >1.00E+8nMAssay Description:Inhibition of human AURKA activity using Ser/Thr 1 peptide as substrate by FRET assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCasein kinase I isoform epsilon(Homo sapiens (Human))
Technische Universit£T Darmstadt

Curated by ChEMBL
LigandPNGBDBM50352493(CHEMBL1824334)
Affinity DataIC50: >1.00E+8nMAssay Description:Inhibition of human CKI epsilon activity using Ser/Thr 11 peptide as substrate by FRET assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCasein kinase I isoform epsilon(Homo sapiens (Human))
Technische Universit£T Darmstadt

Curated by ChEMBL
LigandPNGBDBM50352491(CHEMBL1824539)
Affinity DataIC50: >1.00E+8nMAssay Description:Inhibition of human CKI epsilon activity using Ser/Thr 11 peptide as substrate by FRET assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAurora kinase A(Homo sapiens (Human))
Technische Universit£T Darmstadt

Curated by ChEMBL
LigandPNGBDBM50229962(1-(4-methoxybenzyl)-3-(5-nitrothiazol-2-yl)urea | ...)
Affinity DataIC50: >1.00E+8nMAssay Description:Inhibition of human AURKA activity using Ser/Thr 1 peptide as substrate by FRET assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCasein kinase I isoform epsilon(Homo sapiens (Human))
Technische Universit£T Darmstadt

Curated by ChEMBL
LigandPNGBDBM50229962(1-(4-methoxybenzyl)-3-(5-nitrothiazol-2-yl)urea | ...)
Affinity DataIC50: >1.00E+8nMAssay Description:Inhibition of human CKI epsilon activity using Ser/Thr 11 peptide as substrate by FRET assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCyclin-dependent kinase 5 activator 1(Homo sapiens (Human))
Technische Universit£T Darmstadt

Curated by ChEMBL
LigandPNGBDBM50352491(CHEMBL1824539)
Affinity DataIC50: >1.00E+8nMAssay Description:Inhibition of human CDK5/p35 activity using Ser/Thr 12 peptide as substrate by FRET assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCyclin-dependent kinase 5 activator 1(Homo sapiens (Human))
Technische Universit£T Darmstadt

Curated by ChEMBL
LigandPNGBDBM50352492(CHEMBL1824540)
Affinity DataIC50: >1.00E+8nMAssay Description:Inhibition of human CDK5/p35 activity using Ser/Thr 12 peptide as substrate by FRET assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C alpha type(Homo sapiens (Human))
Technische Universit£T Darmstadt

Curated by ChEMBL
LigandPNGBDBM50229962(1-(4-methoxybenzyl)-3-(5-nitrothiazol-2-yl)urea | ...)
Affinity DataIC50: >1.00E+8nMAssay Description:Inhibition of human PKCalpha activity using Ser/Thr 7 peptide as substrate by FRET assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C alpha type(Homo sapiens (Human))
Technische Universit£T Darmstadt

Curated by ChEMBL
LigandPNGBDBM50352493(CHEMBL1824334)
Affinity DataIC50: >1.00E+8nMAssay Description:Inhibition of human PKCalpha activity using Ser/Thr 7 peptide as substrate by FRET assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C alpha type(Homo sapiens (Human))
Technische Universit£T Darmstadt

Curated by ChEMBL
LigandPNGBDBM50352492(CHEMBL1824540)
Affinity DataIC50: >1.00E+8nMAssay Description:Inhibition of human PKCalpha activity using Ser/Thr 7 peptide as substrate by FRET assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCyclin-dependent kinase 5 activator 1(Homo sapiens (Human))
Technische Universit£T Darmstadt

Curated by ChEMBL
LigandPNGBDBM50352493(CHEMBL1824334)
Affinity DataIC50: >1.00E+8nMAssay Description:Inhibition of human CDK5/p35 activity using Ser/Thr 12 peptide as substrate by FRET assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C alpha type(Homo sapiens (Human))
Technische Universit£T Darmstadt

Curated by ChEMBL
LigandPNGBDBM50352491(CHEMBL1824539)
Affinity DataIC50: >1.00E+8nMAssay Description:Inhibition of human PKCalpha activity using Ser/Thr 7 peptide as substrate by FRET assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCyclin-dependent kinase 5 activator 1(Homo sapiens (Human))
Technische Universit£T Darmstadt

Curated by ChEMBL
LigandPNGBDBM50229962(1-(4-methoxybenzyl)-3-(5-nitrothiazol-2-yl)urea | ...)
Affinity DataIC50: >1.00E+8nMAssay Description:Inhibition of human CDK5/p35 activity using Ser/Thr 12 peptide as substrate by FRET assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAurora kinase A(Homo sapiens (Human))
Technische Universit£T Darmstadt

Curated by ChEMBL
LigandPNGBDBM50352492(CHEMBL1824540)
Affinity DataIC50: >1.00E+8nMAssay Description:Inhibition of human AURKA activity using Ser/Thr 1 peptide as substrate by FRET assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCasein kinase I isoform epsilon(Homo sapiens (Human))
Technische Universit£T Darmstadt

Curated by ChEMBL
LigandPNGBDBM50352492(CHEMBL1824540)
Affinity DataIC50: >1.00E+8nMAssay Description:Inhibition of human CKI epsilon activity using Ser/Thr 11 peptide as substrate by FRET assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed