TargetD(4) dopamine receptor(Homo sapiens (Human))
Smithkline Beecham Pharmaceuticals
Curated by ChEMBL
Smithkline Beecham Pharmaceuticals
Curated by ChEMBL
Affinity DataKi: 4nMAssay Description:Binding affinity against cloned human Dopamine receptor D4 using [3H]nemonapride as radioligandMore data for this Ligand-Target Pair
TargetD(4) dopamine receptor(Homo sapiens (Human))
Smithkline Beecham Pharmaceuticals
Curated by ChEMBL
Smithkline Beecham Pharmaceuticals
Curated by ChEMBL
Affinity DataKi: 5nMAssay Description:Binding affinity against cloned human Dopamine receptor D4 using [3H]nemonapride as radioligandMore data for this Ligand-Target Pair
TargetD(4) dopamine receptor(Homo sapiens (Human))
Smithkline Beecham Pharmaceuticals
Curated by ChEMBL
Smithkline Beecham Pharmaceuticals
Curated by ChEMBL
Affinity DataKi: 6.30nMAssay Description:Binding affinity against cloned human Dopamine receptor D4 using [3H]nemonapride as radioligandMore data for this Ligand-Target Pair
TargetD(4) dopamine receptor(Homo sapiens (Human))
Smithkline Beecham Pharmaceuticals
Curated by ChEMBL
Smithkline Beecham Pharmaceuticals
Curated by ChEMBL
Affinity DataKi: 20nMAssay Description:Binding affinity against cloned human Dopamine receptor D4 using [3H]nemonapride as radioligandMore data for this Ligand-Target Pair
TargetD(4) dopamine receptor(Homo sapiens (Human))
Smithkline Beecham Pharmaceuticals
Curated by ChEMBL
Smithkline Beecham Pharmaceuticals
Curated by ChEMBL
Affinity DataKi: 20nMAssay Description:Binding affinity against cloned human Dopamine receptor D4 using [3H]nemonapride as radioligandMore data for this Ligand-Target Pair
TargetD(4) dopamine receptor(Homo sapiens (Human))
Smithkline Beecham Pharmaceuticals
Curated by ChEMBL
Smithkline Beecham Pharmaceuticals
Curated by ChEMBL
Affinity DataKi: 25nMAssay Description:Binding affinity against cloned human Dopamine receptor D4 using [3H]nemonapride as radioligandMore data for this Ligand-Target Pair
TargetD(4) dopamine receptor(Homo sapiens (Human))
Smithkline Beecham Pharmaceuticals
Curated by ChEMBL
Smithkline Beecham Pharmaceuticals
Curated by ChEMBL
Affinity DataKi: 25nMAssay Description:Binding affinity against cloned human Dopamine receptor D4 using [3H]nemonapride as radioligandMore data for this Ligand-Target Pair
TargetD(4) dopamine receptor(Homo sapiens (Human))
Smithkline Beecham Pharmaceuticals
Curated by ChEMBL
Smithkline Beecham Pharmaceuticals
Curated by ChEMBL
Affinity DataKi: 32nMAssay Description:Binding affinity against cloned human Dopamine receptor D4 using [3H]nemonapride as radioligandMore data for this Ligand-Target Pair
TargetD(4) dopamine receptor(Homo sapiens (Human))
Smithkline Beecham Pharmaceuticals
Curated by ChEMBL
Smithkline Beecham Pharmaceuticals
Curated by ChEMBL
Affinity DataKi: 32nMAssay Description:Binding affinity against cloned human Dopamine receptor D4 using [3H]nemonapride as radioligandMore data for this Ligand-Target Pair
TargetD(2) dopamine receptor(Homo sapiens (Human))
Smithkline Beecham Pharmaceuticals
Curated by ChEMBL
Smithkline Beecham Pharmaceuticals
Curated by ChEMBL
Affinity DataKi: 40nMAssay Description:Binding affinity against cloned human Dopamine receptor D2 (long) using [125I]iodosulpiride as radioligandMore data for this Ligand-Target Pair
TargetD(2) dopamine receptor(Homo sapiens (Human))
Smithkline Beecham Pharmaceuticals
Curated by ChEMBL
Smithkline Beecham Pharmaceuticals
Curated by ChEMBL
Affinity DataKi: 126nMAssay Description:Binding affinity against cloned human Dopamine receptor D2 (long) using [125I]iodosulpiride as radioligandMore data for this Ligand-Target Pair
TargetD(4) dopamine receptor(Homo sapiens (Human))
Smithkline Beecham Pharmaceuticals
Curated by ChEMBL
Smithkline Beecham Pharmaceuticals
Curated by ChEMBL
Affinity DataKi: 200nMAssay Description:Binding affinity against cloned human Dopamine receptor D4 using [3H]nemonapride as radioligandMore data for this Ligand-Target Pair
TargetPotassium-transporting ATPase alpha chain 1(Sus scrofa (Pig))
Smith Kline & French Research
Curated by ChEMBL
Smith Kline & French Research
Curated by ChEMBL
Affinity DataKi: 290nMAssay Description:In vitro inhibition of H+/K+ ATPase activity was determined in gastric vesicles of pig using ATPase assay with pH 7More data for this Ligand-Target Pair
TargetPotassium-transporting ATPase alpha chain 1(Sus scrofa (Pig))
Smith Kline & French Research
Curated by ChEMBL
Smith Kline & French Research
Curated by ChEMBL
Affinity DataKi: 290nMAssay Description:Binding affinity of compound towards H+/K+ ATPase for activation was determinedMore data for this Ligand-Target Pair
TargetD(2) dopamine receptor(Homo sapiens (Human))
Smithkline Beecham Pharmaceuticals
Curated by ChEMBL
Smithkline Beecham Pharmaceuticals
Curated by ChEMBL
Affinity DataKi: 398nMAssay Description:Binding affinity against cloned human Dopamine receptor D2 (long) using [125I]iodosulpiride as radioligandMore data for this Ligand-Target Pair
TargetD(2) dopamine receptor(Homo sapiens (Human))
Smithkline Beecham Pharmaceuticals
Curated by ChEMBL
Smithkline Beecham Pharmaceuticals
Curated by ChEMBL
Affinity DataKi: 1.00E+3nMAssay Description:Binding affinity against cloned human Dopamine receptor D2 (long) using [125I]iodosulpiride as radioligandMore data for this Ligand-Target Pair
TargetD(2) dopamine receptor(Homo sapiens (Human))
Smithkline Beecham Pharmaceuticals
Curated by ChEMBL
Smithkline Beecham Pharmaceuticals
Curated by ChEMBL
Affinity DataKi: 1.26E+3nMAssay Description:Binding affinity against cloned human Dopamine receptor D2 (long) using [125I]iodosulpiride as radioligandMore data for this Ligand-Target Pair
TargetD(2) dopamine receptor(Homo sapiens (Human))
Smithkline Beecham Pharmaceuticals
Curated by ChEMBL
Smithkline Beecham Pharmaceuticals
Curated by ChEMBL
Affinity DataKi: 1.59E+3nMAssay Description:Binding affinity against cloned human Dopamine receptor D2 (long) using [125I]iodosulpiride as radioligandMore data for this Ligand-Target Pair
TargetD(2) dopamine receptor(Homo sapiens (Human))
Smithkline Beecham Pharmaceuticals
Curated by ChEMBL
Smithkline Beecham Pharmaceuticals
Curated by ChEMBL
Affinity DataKi: 2.00E+3nMAssay Description:Binding affinity against cloned human Dopamine receptor D2 (long) using [125I]iodosulpiride as radioligandMore data for this Ligand-Target Pair
TargetD(2) dopamine receptor(Homo sapiens (Human))
Smithkline Beecham Pharmaceuticals
Curated by ChEMBL
Smithkline Beecham Pharmaceuticals
Curated by ChEMBL
Affinity DataKi: 3.16E+3nMAssay Description:Binding affinity against cloned human Dopamine receptor D2 (long) using [125I]iodosulpiride as radioligandMore data for this Ligand-Target Pair
TargetD(2) dopamine receptor(Homo sapiens (Human))
Smithkline Beecham Pharmaceuticals
Curated by ChEMBL
Smithkline Beecham Pharmaceuticals
Curated by ChEMBL
Affinity DataKi: 7.94E+3nMAssay Description:Binding affinity against cloned human Dopamine receptor D2 (long) using [125I]iodosulpiride as radioligandMore data for this Ligand-Target Pair
TargetD(2) dopamine receptor(Homo sapiens (Human))
Smithkline Beecham Pharmaceuticals
Curated by ChEMBL
Smithkline Beecham Pharmaceuticals
Curated by ChEMBL
Affinity DataKi: 1.00E+4nMAssay Description:Binding affinity against cloned human Dopamine receptor D2 (long) using [125I]iodosulpiride as radioligandMore data for this Ligand-Target Pair
TargetPotassium-transporting ATPase alpha chain 1/subunit beta(Sus scrofa (Pig))
Smithkline Beecham Pharmaceuticals R&D
Curated by ChEMBL
Smithkline Beecham Pharmaceuticals R&D
Curated by ChEMBL
Affinity DataIC50: 18nMAssay Description:Inhibition of K+ stimulated gastric ATPase activityMore data for this Ligand-Target Pair
TargetPotassium-transporting ATPase alpha chain 1/subunit beta(Sus scrofa (Pig))
Smithkline Beecham Pharmaceuticals R&D
Curated by ChEMBL
Smithkline Beecham Pharmaceuticals R&D
Curated by ChEMBL
Affinity DataIC50: 19nMAssay Description:Inhibition of K+ stimulated gastric ATPase activityMore data for this Ligand-Target Pair
TargetPotassium-transporting ATPase alpha chain 1/subunit beta(Sus scrofa (Pig))
Smithkline Beecham Pharmaceuticals R&D
Curated by ChEMBL
Smithkline Beecham Pharmaceuticals R&D
Curated by ChEMBL
Affinity DataIC50: 19nMAssay Description:Inhibition of K+ stimulated gastric ATPase activityMore data for this Ligand-Target Pair
TargetPotassium-transporting ATPase alpha chain 1/subunit beta(Sus scrofa (Pig))
Smithkline Beecham Pharmaceuticals R&D
Curated by ChEMBL
Smithkline Beecham Pharmaceuticals R&D
Curated by ChEMBL
Affinity DataIC50: 21nMAssay Description:Inhibition of K+ stimulated gastric ATPase activityMore data for this Ligand-Target Pair
TargetPotassium-transporting ATPase alpha chain 1/subunit beta(Sus scrofa (Pig))
Smithkline Beecham Pharmaceuticals R&D
Curated by ChEMBL
Smithkline Beecham Pharmaceuticals R&D
Curated by ChEMBL
Affinity DataIC50: 21nMAssay Description:Inhibition of K+ stimulated gastric ATPase activityMore data for this Ligand-Target Pair
TargetPotassium-transporting ATPase alpha chain 1/subunit beta(Sus scrofa (Pig))
Smithkline Beecham Pharmaceuticals R&D
Curated by ChEMBL
Smithkline Beecham Pharmaceuticals R&D
Curated by ChEMBL
Affinity DataIC50: 22nMAssay Description:Inhibition of K+ stimulated gastric ATPase activityMore data for this Ligand-Target Pair
TargetPotassium-transporting ATPase alpha chain 1/subunit beta(Sus scrofa (Pig))
Smithkline Beecham Pharmaceuticals R&D
Curated by ChEMBL
Smithkline Beecham Pharmaceuticals R&D
Curated by ChEMBL
Affinity DataIC50: 24nMAssay Description:Inhibition of K+ stimulated gastric ATPase activityMore data for this Ligand-Target Pair
TargetPotassium-transporting ATPase alpha chain 1/subunit beta(Sus scrofa (Pig))
Smithkline Beecham Pharmaceuticals R&D
Curated by ChEMBL
Smithkline Beecham Pharmaceuticals R&D
Curated by ChEMBL
Affinity DataIC50: 28nMAssay Description:Inhibition of K+ stimulated gastric ATPase activityMore data for this Ligand-Target Pair
TargetPotassium-transporting ATPase alpha chain 1/subunit beta(Sus scrofa (Pig))
Smithkline Beecham Pharmaceuticals R&D
Curated by ChEMBL
Smithkline Beecham Pharmaceuticals R&D
Curated by ChEMBL
Affinity DataIC50: 32nMAssay Description:Inhibition of K+ stimulated gastric ATPase activityMore data for this Ligand-Target Pair
TargetPotassium-transporting ATPase alpha chain 1/subunit beta(Sus scrofa (Pig))
Smithkline Beecham Pharmaceuticals R&D
Curated by ChEMBL
Smithkline Beecham Pharmaceuticals R&D
Curated by ChEMBL
Affinity DataIC50: 34nMAssay Description:Inhibition of K+ stimulated gastric ATPase activityMore data for this Ligand-Target Pair
TargetPotassium-transporting ATPase alpha chain 1/subunit beta(Sus scrofa (Pig))
Smithkline Beecham Pharmaceuticals R&D
Curated by ChEMBL
Smithkline Beecham Pharmaceuticals R&D
Curated by ChEMBL
Affinity DataIC50: 34nMAssay Description:Inhibition of K+ stimulated gastric ATPase activityMore data for this Ligand-Target Pair
TargetPotassium-transporting ATPase alpha chain 1/subunit beta(Sus scrofa (Pig))
Smithkline Beecham Pharmaceuticals R&D
Curated by ChEMBL
Smithkline Beecham Pharmaceuticals R&D
Curated by ChEMBL
Affinity DataIC50: 35nMAssay Description:Inhibition of K+ stimulated gastric ATPase activityMore data for this Ligand-Target Pair
TargetPotassium-transporting ATPase alpha chain 1/subunit beta(Sus scrofa (Pig))
Smithkline Beecham Pharmaceuticals R&D
Curated by ChEMBL
Smithkline Beecham Pharmaceuticals R&D
Curated by ChEMBL
Affinity DataIC50: 36nMpH: 7.0Assay Description:Inhibition of K+ -stimulated gastric ATPase activity was measured using lyophilized gastric vesicles at pH 7More data for this Ligand-Target Pair
TargetPotassium-transporting ATPase alpha chain 1/subunit beta(Sus scrofa (Pig))
Smithkline Beecham Pharmaceuticals R&D
Curated by ChEMBL
Smithkline Beecham Pharmaceuticals R&D
Curated by ChEMBL
Affinity DataIC50: 36nMAssay Description:Inhibition of K+ stimulated gastric ATPase activityMore data for this Ligand-Target Pair
TargetPotassium-transporting ATPase alpha chain 1/subunit beta(Sus scrofa (Pig))
Smithkline Beecham Pharmaceuticals R&D
Curated by ChEMBL
Smithkline Beecham Pharmaceuticals R&D
Curated by ChEMBL
Affinity DataIC50: 41nMAssay Description:Inhibition of K+ stimulated gastric ATPase activityMore data for this Ligand-Target Pair
TargetPotassium-transporting ATPase alpha chain 1/subunit beta(Sus scrofa (Pig))
Smithkline Beecham Pharmaceuticals R&D
Curated by ChEMBL
Smithkline Beecham Pharmaceuticals R&D
Curated by ChEMBL
Affinity DataIC50: 42nMAssay Description:Inhibition of K+ stimulated gastric ATPase activityMore data for this Ligand-Target Pair
TargetPotassium-transporting ATPase alpha chain 1/subunit beta(Sus scrofa (Pig))
Smithkline Beecham Pharmaceuticals R&D
Curated by ChEMBL
Smithkline Beecham Pharmaceuticals R&D
Curated by ChEMBL
Affinity DataIC50: 46nMAssay Description:Inhibition of K+ stimulated gastric ATPase activityMore data for this Ligand-Target Pair
TargetPotassium-transporting ATPase alpha chain 1/subunit beta(Sus scrofa (Pig))
Smithkline Beecham Pharmaceuticals R&D
Curated by ChEMBL
Smithkline Beecham Pharmaceuticals R&D
Curated by ChEMBL
Affinity DataIC50: 50nMAssay Description:Inhibition of K+ stimulated gastric ATPase activityMore data for this Ligand-Target Pair
TargetPotassium-transporting ATPase alpha chain 1/subunit beta(Sus scrofa (Pig))
Smithkline Beecham Pharmaceuticals R&D
Curated by ChEMBL
Smithkline Beecham Pharmaceuticals R&D
Curated by ChEMBL
Affinity DataIC50: 61nMpH: 7.0Assay Description:Inhibition of K+ -stimulated gastric ATPase activity was measured using lyophilized gastric vesicles at pH 7More data for this Ligand-Target Pair
TargetPotassium-transporting ATPase alpha chain 1/subunit beta(Rattus norvegicus)
Smithkline Beecham Pharmaceuticals R&D
Curated by ChEMBL
Smithkline Beecham Pharmaceuticals R&D
Curated by ChEMBL
Affinity DataIC50: 64nMAssay Description:Inhibition of rat isolated gastric(H+/K+)-ATPase.More data for this Ligand-Target Pair
TargetPotassium-transporting ATPase alpha chain 1/subunit beta(Sus scrofa (Pig))
Smithkline Beecham Pharmaceuticals R&D
Curated by ChEMBL
Smithkline Beecham Pharmaceuticals R&D
Curated by ChEMBL
Affinity DataIC50: 65nMAssay Description:Inhibition of K+ stimulated gastric ATPase activityMore data for this Ligand-Target Pair
TargetPotassium-transporting ATPase alpha chain 1/subunit beta(Sus scrofa (Pig))
Smithkline Beecham Pharmaceuticals R&D
Curated by ChEMBL
Smithkline Beecham Pharmaceuticals R&D
Curated by ChEMBL
Affinity DataIC50: 67nMAssay Description:Inhibition of K+ stimulated gastric ATPase activityMore data for this Ligand-Target Pair
TargetPotassium-transporting ATPase alpha chain 1/subunit beta(Sus scrofa (Pig))
Smithkline Beecham Pharmaceuticals R&D
Curated by ChEMBL
Smithkline Beecham Pharmaceuticals R&D
Curated by ChEMBL
Affinity DataIC50: 71nMpH: 7.0Assay Description:Inhibition of K+ -stimulated gastric ATPase activity was measured using lyophilized gastric vesicles at pH 7More data for this Ligand-Target Pair
TargetPotassium-transporting ATPase alpha chain 1/subunit beta(Sus scrofa (Pig))
Smithkline Beecham Pharmaceuticals R&D
Curated by ChEMBL
Smithkline Beecham Pharmaceuticals R&D
Curated by ChEMBL
Affinity DataIC50: 74nMAssay Description:Inhibition of K+ stimulated gastric ATPase activityMore data for this Ligand-Target Pair
TargetPotassium-transporting ATPase alpha chain 1/subunit beta(Sus scrofa (Pig))
Smithkline Beecham Pharmaceuticals R&D
Curated by ChEMBL
Smithkline Beecham Pharmaceuticals R&D
Curated by ChEMBL
Affinity DataIC50: 80nMAssay Description:Inhibition of K+ stimulated gastric ATPase activityMore data for this Ligand-Target Pair
TargetPotassium-transporting ATPase alpha chain 1/subunit beta(Sus scrofa (Pig))
Smithkline Beecham Pharmaceuticals R&D
Curated by ChEMBL
Smithkline Beecham Pharmaceuticals R&D
Curated by ChEMBL
Affinity DataIC50: 95nMAssay Description:Inhibition of K+ stimulated gastric ATPase activityMore data for this Ligand-Target Pair
TargetPotassium-transporting ATPase alpha chain 1/subunit beta(Sus scrofa (Pig))
Smithkline Beecham Pharmaceuticals R&D
Curated by ChEMBL
Smithkline Beecham Pharmaceuticals R&D
Curated by ChEMBL
Affinity DataIC50: 100nMAssay Description:Inhibition of K+ stimulated gastric ATPase activityMore data for this Ligand-Target Pair
TargetPotassium-transporting ATPase alpha chain 1/subunit beta(Sus scrofa (Pig))
Smithkline Beecham Pharmaceuticals R&D
Curated by ChEMBL
Smithkline Beecham Pharmaceuticals R&D
Curated by ChEMBL
Affinity DataIC50: 100nMAssay Description:Concentration required to inhibit the activity of K+ stimulated gastric ATPaseMore data for this Ligand-Target Pair