Affinity DataKi: 0.150nMAssay Description:Opioid receptor delta 1 binding affinity by displacement of radioligand [3H][D-Pen]-enkephalin (DPDPE) from rat brain membrane synaptosomesMore data for this Ligand-Target Pair
Affinity DataKi: 0.280nMAssay Description:Opioid receptor mu 1 binding affinity by displacement of radioligand [3H][DAla,MePhe,Gly-ol]enkephalin (DAGO) from rat brain membrane synaptosomesMore data for this Ligand-Target Pair
Affinity DataKi: 0.290nMAssay Description:Opioid receptor mu 1 binding affinity by displacement of radioligand [3H][DAla,MePhe,Gly-ol]enkephalin (DAGO) from rat brain membrane synaptosomesMore data for this Ligand-Target Pair
Affinity DataKi: 0.460nMAssay Description:Opioid receptor mu 1 binding affinity by displacement of radioligand [3H][DAla,MePhe,Gly-ol]enkephalin (DAGO) from rat brain membrane synaptosomesMore data for this Ligand-Target Pair
Affinity DataKi: 1.30nMAssay Description:Opioid receptor delta 1 binding affinity by displacement of radioligand [3H][D-Pen]-enkephalin (DPDPE) from rat brain membrane synaptosomesMore data for this Ligand-Target Pair
Affinity DataKi: 1.60nMAssay Description:Opioid receptor delta 1 binding affinity by displacement of radioligand [3H][D-Pen]-enkephalin (DPDPE) from rat brain membrane synaptosomesMore data for this Ligand-Target Pair
Affinity DataKi: 67nMAssay Description:Opioid receptor delta 1 binding affinity by displacement of radioligand [3H][D-Pen]-enkephalin (DPDPE) from rat brain membrane synaptosomesMore data for this Ligand-Target Pair
Affinity DataKi: 83nMAssay Description:Opioid receptor delta 1 binding affinity by displacement of radioligand [3H][D-Pen]-enkephalin (DPDPE) from rat brain membrane synaptosomesMore data for this Ligand-Target Pair
Affinity DataKi: 87nMAssay Description:Opioid receptor delta 1 binding affinity by displacement of radioligand [3H][D-Pen]-enkephalin (DPDPE) from rat brain membrane synaptosomesMore data for this Ligand-Target Pair
Affinity DataKi: 147nMAssay Description:Opioid receptor mu 1 binding affinity by displacement of radioligand [3H][DAla,MePhe,Gly-ol]enkephalin (DAGO) from rat brain membrane synaptosomesMore data for this Ligand-Target Pair
TargetM-phase inducer phosphatase 3(Homo sapiens (Human))
University Of Naples Federico Ii
Curated by ChEMBL
University Of Naples Federico Ii
Curated by ChEMBL
Affinity DataKi: 400nMAssay Description:Inhibition of N-terminal His6-tagged human CDC25C (280 to 454 residues) expressed in Escherichia coli BL21(DE3) cells using OMFP as substrate by doub...More data for this Ligand-Target Pair
Affinity DataKi: 579nMAssay Description:Opioid receptor mu 1 binding affinity by displacement of radioligand [3H][DAla,MePhe,Gly-ol]enkephalin (DAGO) from rat brain membrane synaptosomesMore data for this Ligand-Target Pair
TargetM-phase inducer phosphatase 1(Homo sapiens (Human))
University Of Naples Federico Ii
Curated by ChEMBL
University Of Naples Federico Ii
Curated by ChEMBL
Affinity DataKi: 600nMAssay Description:Inhibition of N-terminal His6-tagged human CDC25A (336 to 508 residues) expressed in Escherichia coli BL21(DE3) cells using OMFP as substrate by doub...More data for this Ligand-Target Pair
TargetM-phase inducer phosphatase 1(Homo sapiens (Human))
University Of Naples Federico Ii
Curated by ChEMBL
University Of Naples Federico Ii
Curated by ChEMBL
Affinity DataKi: 600nMAssay Description:Inhibition of N-terminal His6-tagged human CDC25A (336 to 508 residues) expressed in Escherichia coli BL21(DE3) cells using OMFP as substrate by doub...More data for this Ligand-Target Pair
Affinity DataKi: 635nMAssay Description:Opioid receptor mu 1 binding affinity by displacement of radioligand [3H][DAla,MePhe,Gly-ol]enkephalin (DAGO) from rat brain membrane synaptosomesMore data for this Ligand-Target Pair
TargetM-phase inducer phosphatase 2(Homo sapiens (Human))
University Of Naples Federico Ii
Curated by ChEMBL
University Of Naples Federico Ii
Curated by ChEMBL
Affinity DataKi: 800nMAssay Description:Non-competitive inhibition of N-terminal His6-tagged human CDC25B (377 to 550 residues) expressed in Escherichia coli BL21(DE3) cells using OMFP as s...More data for this Ligand-Target Pair
TargetM-phase inducer phosphatase 2(Homo sapiens (Human))
University Of Naples Federico Ii
Curated by ChEMBL
University Of Naples Federico Ii
Curated by ChEMBL
Affinity DataKi: 1.40E+3nMAssay Description:Non-competitive inhibition of N-terminal His6-tagged human CDC25B (377 to 550 residues) expressed in Escherichia coli BL21(DE3) cells using OMFP as s...More data for this Ligand-Target Pair
Affinity DataKi: 1.52E+3nMAssay Description:Opioid receptor mu 1 binding affinity by displacement of radioligand [3H][DAla,MePhe,Gly-ol]enkephalin (DAGO) from rat brain membrane synaptosomesMore data for this Ligand-Target Pair
Affinity DataKi: 1.70E+3nMAssay Description:Opioid receptor mu 1 binding affinity by displacement of radioligand [3H][DAla,MePhe,Gly-ol]enkephalin (DAGO) from rat brain membrane synaptosomesMore data for this Ligand-Target Pair
Affinity DataKi: 1.76E+3nMAssay Description:Opioid receptor delta 1 binding affinity by displacement of radioligand [3H][D-Pen]-enkephalin (DPDPE) from rat brain membrane synaptosomesMore data for this Ligand-Target Pair
TargetM-phase inducer phosphatase 3(Homo sapiens (Human))
University Of Naples Federico Ii
Curated by ChEMBL
University Of Naples Federico Ii
Curated by ChEMBL
Affinity DataKi: 1.90E+3nMAssay Description:Inhibition of N-terminal His6-tagged human CDC25C (280 to 454 residues) expressed in Escherichia coli BL21(DE3) cells using OMFP as substrate by doub...More data for this Ligand-Target Pair
Affinity DataKi: 1.99E+3nMAssay Description:Opioid receptor mu 1 binding affinity by displacement of radioligand [3H][DAla,MePhe,Gly-ol]enkephalin (DAGO) from rat brain membrane synaptosomesMore data for this Ligand-Target Pair
Affinity DataKi: 2.11E+3nMAssay Description:Opioid receptor delta 1 binding affinity by displacement of radioligand [3H][D-Pen]-enkephalin (DPDPE) from rat brain membrane synaptosomesMore data for this Ligand-Target Pair
TargetM-phase inducer phosphatase 2(Homo sapiens (Human))
University Of Naples Federico Ii
Curated by ChEMBL
University Of Naples Federico Ii
Curated by ChEMBL
Affinity DataKi: 2.70E+3nMAssay Description:Non-competitive inhibition of N-terminal His6-tagged human CDC25B (377 to 550 residues) expressed in Escherichia coli BL21(DE3) cells using OMFP as s...More data for this Ligand-Target Pair
TargetM-phase inducer phosphatase 2(Homo sapiens (Human))
University Of Naples Federico Ii
Curated by ChEMBL
University Of Naples Federico Ii
Curated by ChEMBL
Affinity DataKi: 2.80E+3nMAssay Description:Uncompetitive inhibition of N-terminal His6-tagged human CDC25B (377 to 550 residues) expressed in Escherichia coli BL21(DE3) cells using OMFP as sub...More data for this Ligand-Target Pair
TargetM-phase inducer phosphatase 2(Homo sapiens (Human))
University Of Naples Federico Ii
Curated by ChEMBL
University Of Naples Federico Ii
Curated by ChEMBL
Affinity DataKi: 2.90E+3nMAssay Description:Non-competitive inhibition of N-terminal His6-tagged human CDC25B (377 to 550 residues) expressed in Escherichia coli BL21(DE3) cells using OMFP as s...More data for this Ligand-Target Pair
TargetM-phase inducer phosphatase 1(Homo sapiens (Human))
University Of Naples Federico Ii
Curated by ChEMBL
University Of Naples Federico Ii
Curated by ChEMBL
Affinity DataKi: 3.00E+3nMAssay Description:Inhibition of N-terminal His6-tagged human CDC25A (336 to 508 residues) expressed in Escherichia coli BL21(DE3) cells using OMFP as substrate by doub...More data for this Ligand-Target Pair
TargetM-phase inducer phosphatase 3(Homo sapiens (Human))
University Of Naples Federico Ii
Curated by ChEMBL
University Of Naples Federico Ii
Curated by ChEMBL
Affinity DataKi: 4.00E+3nMAssay Description:Inhibition of N-terminal His6-tagged human CDC25C (280 to 454 residues) expressed in Escherichia coli BL21(DE3) cells using OMFP as substrate by doub...More data for this Ligand-Target Pair
Affinity DataKi: 4.40E+3nMAssay Description:Opioid receptor mu 1 binding affinity by displacement of radioligand [3H][DAla,MePhe,Gly-ol]enkephalin (DAGO) from rat brain membrane synaptosomesMore data for this Ligand-Target Pair
TargetM-phase inducer phosphatase 2(Homo sapiens (Human))
University Of Naples Federico Ii
Curated by ChEMBL
University Of Naples Federico Ii
Curated by ChEMBL
Affinity DataKi: 4.90E+3nMAssay Description:Non-competitive inhibition of N-terminal His6-tagged human CDC25B (377 to 550 residues) expressed in Escherichia coli BL21(DE3) cells using OMFP as s...More data for this Ligand-Target Pair
TargetM-phase inducer phosphatase 2(Homo sapiens (Human))
University Of Naples Federico Ii
Curated by ChEMBL
University Of Naples Federico Ii
Curated by ChEMBL
Affinity DataKi: 5.10E+3nMAssay Description:Non-competitive inhibition of N-terminal His6-tagged human CDC25B (377 to 550 residues) expressed in Escherichia coli BL21(DE3) cells using OMFP as s...More data for this Ligand-Target Pair
TargetM-phase inducer phosphatase 2(Homo sapiens (Human))
University Of Naples Federico Ii
Curated by ChEMBL
University Of Naples Federico Ii
Curated by ChEMBL
Affinity DataKi: 5.30E+3nMAssay Description:Competitive reversible inhibition of N-terminal His6-tagged human CDC25B (377 to 550 residues) expressed in Escherichia coli BL21(DE3) cells using OM...More data for this Ligand-Target Pair
TargetM-phase inducer phosphatase 2(Homo sapiens (Human))
University Of Naples Federico Ii
Curated by ChEMBL
University Of Naples Federico Ii
Curated by ChEMBL
Affinity DataKi: 5.80E+3nMAssay Description:Non-competitive inhibition of N-terminal His6-tagged human CDC25B (377 to 550 residues) expressed in Escherichia coli BL21(DE3) cells using OMFP as s...More data for this Ligand-Target Pair
TargetM-phase inducer phosphatase 2(Homo sapiens (Human))
University Of Naples Federico Ii
Curated by ChEMBL
University Of Naples Federico Ii
Curated by ChEMBL
Affinity DataKi: 6.10E+3nMAssay Description:Uncompetitive inhibition of N-terminal His6-tagged human CDC25B (377 to 550 residues) expressed in Escherichia coli BL21(DE3) cells using OMFP as sub...More data for this Ligand-Target Pair
TargetM-phase inducer phosphatase 2(Homo sapiens (Human))
University Of Naples Federico Ii
Curated by ChEMBL
University Of Naples Federico Ii
Curated by ChEMBL
Affinity DataKi: 6.40E+3nMAssay Description:Uncompetitive inhibition of N-terminal His6-tagged human CDC25B (377 to 550 residues) expressed in Escherichia coli BL21(DE3) cells using OMFP as sub...More data for this Ligand-Target Pair
TargetM-phase inducer phosphatase 2(Homo sapiens (Human))
University Of Naples Federico Ii
Curated by ChEMBL
University Of Naples Federico Ii
Curated by ChEMBL
Affinity DataKi: 6.50E+3nMAssay Description:Non-competitive inhibition of N-terminal His6-tagged human CDC25B (377 to 550 residues) expressed in Escherichia coli BL21(DE3) cells using OMFP as s...More data for this Ligand-Target Pair
TargetM-phase inducer phosphatase 2(Homo sapiens (Human))
University Of Naples Federico Ii
Curated by ChEMBL
University Of Naples Federico Ii
Curated by ChEMBL
Affinity DataKi: 6.90E+3nMAssay Description:Non-competitive inhibition of N-terminal His6-tagged human CDC25B (377 to 550 residues) expressed in Escherichia coli BL21(DE3) cells using OMFP as s...More data for this Ligand-Target Pair
TargetM-phase inducer phosphatase 2(Homo sapiens (Human))
University Of Naples Federico Ii
Curated by ChEMBL
University Of Naples Federico Ii
Curated by ChEMBL
Affinity DataKi: 7.10E+3nMAssay Description:Non-competitive inhibition of N-terminal His6-tagged human CDC25B (377 to 550 residues) expressed in Escherichia coli BL21(DE3) cells using OMFP as s...More data for this Ligand-Target Pair
TargetM-phase inducer phosphatase 2(Homo sapiens (Human))
University Of Naples Federico Ii
Curated by ChEMBL
University Of Naples Federico Ii
Curated by ChEMBL
Affinity DataKi: 7.30E+3nMAssay Description:Uncompetitive inhibition of N-terminal His6-tagged human CDC25B (377 to 550 residues) expressed in Escherichia coli BL21(DE3) cells using OMFP as sub...More data for this Ligand-Target Pair
TargetM-phase inducer phosphatase 2(Homo sapiens (Human))
University Of Naples Federico Ii
Curated by ChEMBL
University Of Naples Federico Ii
Curated by ChEMBL
Affinity DataKi: 7.40E+3nMAssay Description:Non-competitive inhibition of N-terminal His6-tagged human CDC25B (377 to 550 residues) expressed in Escherichia coli BL21(DE3) cells using OMFP as s...More data for this Ligand-Target Pair
TargetM-phase inducer phosphatase 2(Homo sapiens (Human))
University Of Naples Federico Ii
Curated by ChEMBL
University Of Naples Federico Ii
Curated by ChEMBL
Affinity DataKi: 8.50E+3nMAssay Description:Uncompetitive inhibition of N-terminal His6-tagged human CDC25B (377 to 550 residues) expressed in Escherichia coli BL21(DE3) cells using OMFP as sub...More data for this Ligand-Target Pair
Affinity DataKi: 9.50E+3nMAssay Description:Opioid receptor delta 1 binding affinity by displacement of radioligand [3H][D-Pen]-enkephalin (DPDPE) from rat brain membrane synaptosomesMore data for this Ligand-Target Pair
TargetM-phase inducer phosphatase 2(Homo sapiens (Human))
University Of Naples Federico Ii
Curated by ChEMBL
University Of Naples Federico Ii
Curated by ChEMBL
Affinity DataKi: 9.90E+3nMAssay Description:Non-competitive inhibition of N-terminal His6-tagged human CDC25B (377 to 550 residues) expressed in Escherichia coli BL21(DE3) cells using OMFP as s...More data for this Ligand-Target Pair
TargetM-phase inducer phosphatase 2(Homo sapiens (Human))
University Of Naples Federico Ii
Curated by ChEMBL
University Of Naples Federico Ii
Curated by ChEMBL
Affinity DataKi: 1.19E+4nMAssay Description:Non-competitive inhibition of N-terminal His6-tagged human CDC25B (377 to 550 residues) expressed in Escherichia coli BL21(DE3) cells using OMFP as s...More data for this Ligand-Target Pair
TargetM-phase inducer phosphatase 2(Homo sapiens (Human))
University Of Naples Federico Ii
Curated by ChEMBL
University Of Naples Federico Ii
Curated by ChEMBL
Affinity DataKi: 1.25E+4nMAssay Description:Uncompetitive inhibition of N-terminal His6-tagged human CDC25B (377 to 550 residues) expressed in Escherichia coli BL21(DE3) cells using OMFP as sub...More data for this Ligand-Target Pair
TargetM-phase inducer phosphatase 2(Homo sapiens (Human))
University Of Naples Federico Ii
Curated by ChEMBL
University Of Naples Federico Ii
Curated by ChEMBL
Affinity DataKi: 1.34E+4nMAssay Description:Non-competitive inhibition of N-terminal His6-tagged human CDC25B (377 to 550 residues) expressed in Escherichia coli BL21(DE3) cells using OMFP as s...More data for this Ligand-Target Pair
TargetM-phase inducer phosphatase 2(Homo sapiens (Human))
University Of Naples Federico Ii
Curated by ChEMBL
University Of Naples Federico Ii
Curated by ChEMBL
Affinity DataKi: 1.69E+4nMAssay Description:Non-competitive inhibition of N-terminal His6-tagged human CDC25B (377 to 550 residues) expressed in Escherichia coli BL21(DE3) cells using OMFP as s...More data for this Ligand-Target Pair
TargetM-phase inducer phosphatase 2(Homo sapiens (Human))
University Of Naples Federico Ii
Curated by ChEMBL
University Of Naples Federico Ii
Curated by ChEMBL
Affinity DataKi: 2.20E+4nMAssay Description:Uncompetitive inhibition of N-terminal His6-tagged human CDC25B (377 to 550 residues) expressed in Escherichia coli BL21(DE3) cells using OMFP as sub...More data for this Ligand-Target Pair
Affinity DataKi: 2.26E+4nMAssay Description:Opioid receptor delta 1 binding affinity by displacement of radioligand [3H][D-Pen]-enkephalin (DPDPE) from rat brain membrane synaptosomesMore data for this Ligand-Target Pair
TargetM-phase inducer phosphatase 2(Homo sapiens (Human))
University Of Naples Federico Ii
Curated by ChEMBL
University Of Naples Federico Ii
Curated by ChEMBL
Affinity DataKi: 3.00E+4nMAssay Description:Mixed inhibition of N-terminal His6-tagged human CDC25B (377 to 550 residues) expressed in Escherichia coli BL21(DE3) cells using OMFP as substrate b...More data for this Ligand-Target Pair