TargetSigma non-opioid intracellular receptor 1(Homo sapiens (Human))
Warner-Lambert
Curated by ChEMBL
Warner-Lambert
Curated by ChEMBL
Affinity DataKi: 0.330nMAssay Description:Tested for [3H]-(+)-pentazocine binding to sigma-1 receptor in guinea pig brain membraneMore data for this Ligand-Target Pair
Affinity DataKi: 0.440nMAssay Description:Displacement of [3H]-spiperone from CHO-K1 cell membranes expressing human dopamine receptor D2More data for this Ligand-Target Pair
Affinity DataKi: 0.5nMAssay Description:Tested for binding affinity towards human D2L receptor using [3H]-spiperone as radioligandMore data for this Ligand-Target Pair
Affinity DataKi: 0.580nMAssay Description:Inhibition of human ICEMore data for this Ligand-Target Pair
Affinity DataKi: 0.600nMAssay Description:Inhibition of human ICEMore data for this Ligand-Target Pair
TargetD(3) dopamine receptor(Homo sapiens (Human))
Parke-Davis Pharmaceutical Research
Curated by ChEMBL
Parke-Davis Pharmaceutical Research
Curated by ChEMBL
Affinity DataKi: 0.690nMAssay Description:Tested for binding affinity towards human D3 receptor using [3H]-spiperone as radioligandMore data for this Ligand-Target Pair
Affinity DataKi: 0.700nMAssay Description:Inhibition of human ICEMore data for this Ligand-Target Pair
Affinity DataKi: 0.900nMAssay Description:Inhibition of human ICEMore data for this Ligand-Target Pair
Affinity DataKi: 0.950nMAssay Description:Inhibition of human ICEMore data for this Ligand-Target Pair
TargetD(3) dopamine receptor(Homo sapiens (Human))
Parke-Davis Pharmaceutical Research
Curated by ChEMBL
Parke-Davis Pharmaceutical Research
Curated by ChEMBL
Affinity DataKi: 0.960nMAssay Description:Displacemnt of [3H]-spiperone from CHO-K1 cell membranes expressing human dopamine 3 receptorsMore data for this Ligand-Target Pair
Affinity DataKi: 1.26nMAssay Description:Inhibition of human ICEMore data for this Ligand-Target Pair
Affinity DataKi: 1.29nMAssay Description:Inhibition of human ICEMore data for this Ligand-Target Pair
Affinity DataKi: 1.31nMAssay Description:Inhibition of human ICEMore data for this Ligand-Target Pair
TargetSigma non-opioid intracellular receptor 1(Homo sapiens (Human))
Warner-Lambert
Curated by ChEMBL
Warner-Lambert
Curated by ChEMBL
Affinity DataKi: 1.80nMAssay Description:Tested for [3H]-(+)-pentazocine binding to sigma-1 receptor in guinea pig brain membraneMore data for this Ligand-Target Pair
Affinity DataKi: 1.81nMAssay Description:Inhibition of human ICEMore data for this Ligand-Target Pair
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
Parke-Davis Pharmaceutical Research
Curated by ChEMBL
Parke-Davis Pharmaceutical Research
Curated by ChEMBL
Affinity DataKi: 1.86nMAssay Description:Tested for binding affinity towards rat striatal D2 receptor using [3H]-spiperone as radioligandMore data for this Ligand-Target Pair
TargetSigma non-opioid intracellular receptor 1(Homo sapiens (Human))
Warner-Lambert
Curated by ChEMBL
Warner-Lambert
Curated by ChEMBL
Affinity DataKi: 2.20nMAssay Description:Tested for [3H]-(+)-pentazocine binding to sigma-1 receptor in guinea pig brain membraneMore data for this Ligand-Target Pair
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
Parke-Davis Pharmaceutical Research
Curated by ChEMBL
Parke-Davis Pharmaceutical Research
Curated by ChEMBL
Affinity DataKi: 2.20nMAssay Description:Tested for binding affinity towards rat striatal D2 receptor using [3H]-NPA as radioligandMore data for this Ligand-Target Pair
Affinity DataKi: 2.81nMAssay Description:Inhibition of human ICEMore data for this Ligand-Target Pair
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
Parke-Davis Pharmaceutical Research
Curated by ChEMBL
Parke-Davis Pharmaceutical Research
Curated by ChEMBL
Affinity DataKi: 3.30nMAssay Description:Tested for binding affinity towards rat striatal D2 receptor using [3H]-NPA as radioligandMore data for this Ligand-Target Pair
Affinity DataKi: 3.85nMAssay Description:Inhibition of human ICEMore data for this Ligand-Target Pair
Affinity DataKi: 4nMAssay Description:Inhibitory activity against caspase-1More data for this Ligand-Target Pair
Affinity DataKi: 4nMAssay Description:Inhibitory activity against caspase-1More data for this Ligand-Target Pair
Affinity DataKi: 4.03nMAssay Description:Inhibition of human ICEMore data for this Ligand-Target Pair
Affinity DataKi: 4.30nMAssay Description:Inhibition of human ICEMore data for this Ligand-Target Pair
Affinity DataKi: 4.68nMAssay Description:Inhibition of human ICEMore data for this Ligand-Target Pair
Affinity DataKi: 4.85nMAssay Description:Inhibition of human ICEMore data for this Ligand-Target Pair
Affinity DataKi: 5.02nMAssay Description:Inhibition of human ICEMore data for this Ligand-Target Pair
TargetD(3) dopamine receptor(Homo sapiens (Human))
Parke-Davis Pharmaceutical Research
Curated by ChEMBL
Parke-Davis Pharmaceutical Research
Curated by ChEMBL
Affinity DataKi: 7.80nMAssay Description:Tested for binding affinity towards human D3 receptor using [3H]-spiperone as radioligandMore data for this Ligand-Target Pair
Affinity DataKi: 7.90nMAssay Description:Inhibition of human ICEMore data for this Ligand-Target Pair
Affinity DataKi: 9.24nMAssay Description:Inhibition of human ICEMore data for this Ligand-Target Pair
Affinity DataKi: 13.4nMAssay Description:Inhibition of mouse ICEMore data for this Ligand-Target Pair
Affinity DataKi: 14nMAssay Description:Inhibitory activity against caspase-1More data for this Ligand-Target Pair
Affinity DataKi: 14.4nMAssay Description:Inhibition of mouse ICEMore data for this Ligand-Target Pair
Affinity DataKi: 16.7nMAssay Description:Inhibition of human ICEMore data for this Ligand-Target Pair
Affinity DataKi: 16.9nMAssay Description:Inhibition of human ICEMore data for this Ligand-Target Pair
TargetD(3) dopamine receptor(Homo sapiens (Human))
Parke-Davis Pharmaceutical Research
Curated by ChEMBL
Parke-Davis Pharmaceutical Research
Curated by ChEMBL
Affinity DataKi: 17nMAssay Description:Tested for binding affinity towards human D3 receptor using [3H]-spiperone as radioligandMore data for this Ligand-Target Pair
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
Parke-Davis Pharmaceutical Research
Curated by ChEMBL
Parke-Davis Pharmaceutical Research
Curated by ChEMBL
Affinity DataKi: 17nMAssay Description:Tested for binding affinity towards rat striatal D2 receptor using [3H]-spiperone as radioligandMore data for this Ligand-Target Pair
Affinity DataKi: 18.7nMAssay Description:Inhibition of mouse ICEMore data for this Ligand-Target Pair