Target5-hydroxytryptamine receptor 1D(Homo sapiens (Human))
Glaxo Research And Development
Curated by ChEMBL
Glaxo Research And Development
Curated by ChEMBL
Affinity DataKi: 0.126nMAssay Description:Binding affinity against 5-hydroxytryptamine 1D receptor betaMore data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 1D(Homo sapiens (Human))
Glaxo Research And Development
Curated by ChEMBL
Glaxo Research And Development
Curated by ChEMBL
Affinity DataKi: 1.30nMAssay Description:Binding affinity against 5-hydroxytryptamine 1D receptor alphaMore data for this Ligand-Target Pair
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
SynthÉLabo Recherche
Curated by PDSP Ki Database
SynthÉLabo Recherche
Curated by PDSP Ki Database
Target5-hydroxytryptamine receptor 2A(Rattus norvegicus (rat))
SynthÉLabo Recherche
Curated by PDSP Ki Database
SynthÉLabo Recherche
Curated by PDSP Ki Database
TargetAlpha-1B adrenergic receptor(Rattus norvegicus (rat))
SynthÉLabo Recherche
Curated by PDSP Ki Database
SynthÉLabo Recherche
Curated by PDSP Ki Database
Affinity DataKi: 3.20nMAssay Description:In vitro binding affinity towards 5-hydroxytryptamine 1D receptor in guinea-pig striatum in presence of BMY-7378 and mesulergineMore data for this Ligand-Target Pair
Affinity DataKi: 3.20nMAssay Description:In vitro binding affinity towards 5-hydroxytryptamine 1D receptor in guinea-pig striatum in presence of BMY-7378 and mesulergineMore data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 1B(Rattus norvegicus (Rat))
Glaxo Research And Development
Curated by ChEMBL
Glaxo Research And Development
Curated by ChEMBL
Affinity DataKi: 3.20nMAssay Description:In vitro binding affinity towards 5-hydroxytryptamine 1B receptor in rat striatal membrane with [125I]- iodocyanopindololMore data for this Ligand-Target Pair
Affinity DataKi: 3.20nMAssay Description:In vitro binding affinity towards 5-hydroxytryptamine 1D receptor in guinea-pig striatum in presence of BMY-7378 and mesulergineMore data for this Ligand-Target Pair
Affinity DataKi: 5nMAssay Description:In vitro binding affinity towards 5-hydroxytryptamine 1D receptor in guinea-pig striatum in presence of BMY-7378 and mesulergineMore data for this Ligand-Target Pair
Affinity DataKi: 5nMAssay Description:In vitro binding affinity towards 5-hydroxytryptamine 1D receptor in guinea-pig striatum in presence of BMY-7378 and mesulergineMore data for this Ligand-Target Pair
Affinity DataKi: 6.30nMAssay Description:In vitro binding affinity towards 5-hydroxytryptamine 1D receptor in guinea-pig striatum in presence of BMY-7378 and mesulergineMore data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 1B(Rattus norvegicus (Rat))
Glaxo Research And Development
Curated by ChEMBL
Glaxo Research And Development
Curated by ChEMBL
Affinity DataKi: 6.30nMAssay Description:In vitro binding affinity towards 5-hydroxytryptamine 1B receptor in rat striatal membrane with [125I]- iodocyanopindololMore data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 1B(Rattus norvegicus (Rat))
Glaxo Research And Development
Curated by ChEMBL
Glaxo Research And Development
Curated by ChEMBL
Affinity DataKi: 6.30nMAssay Description:In vitro binding affinity towards 5-hydroxytryptamine 1B receptor in rat striatal membrane with [125I]- iodocyanopindololMore data for this Ligand-Target Pair
Affinity DataKi: 6.30nMAssay Description:In vitro binding affinity towards 5-hydroxytryptamine 1D receptor in guinea-pig striatum in presence of BMY-7378 and mesulergineMore data for this Ligand-Target Pair
TargetAlpha-1B adrenergic receptor(Rattus norvegicus (rat))
SynthÉLabo Recherche
Curated by PDSP Ki Database
SynthÉLabo Recherche
Curated by PDSP Ki Database
TargetAlpha-1A adrenergic receptor(Rattus norvegicus (Rat))
SynthÉLabo Recherche
Curated by PDSP Ki Database
SynthÉLabo Recherche
Curated by PDSP Ki Database
Affinity DataKi: 10nMAssay Description:In vitro binding affinity towards 5-hydroxytryptamine 1D receptor in guinea-pig striatum in presence of BMY-7378 and mesulergineMore data for this Ligand-Target Pair
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
SynthÉLabo Recherche
Curated by PDSP Ki Database
SynthÉLabo Recherche
Curated by PDSP Ki Database
TargetHistamine H1 receptor(Cavia porcellus (domestic guinea pig))
SynthÉLabo Recherche
Curated by PDSP Ki Database
SynthÉLabo Recherche
Curated by PDSP Ki Database
TargetSigma non-opioid intracellular receptor 1(Mus musculus (Mouse))
SynthÉLabo Recherche
Curated by PDSP Ki Database
SynthÉLabo Recherche
Curated by PDSP Ki Database
TargetAlpha-1A adrenergic receptor(Rattus norvegicus (Rat))
SynthÉLabo Recherche
Curated by PDSP Ki Database
SynthÉLabo Recherche
Curated by PDSP Ki Database
Affinity DataKi: 32nMAssay Description:In vitro binding affinity towards 5-hydroxytryptamine 1D receptor in guinea-pig striatum in presence of BMY-7378 and mesulergineMore data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 2A(Rattus norvegicus (rat))
SynthÉLabo Recherche
Curated by PDSP Ki Database
SynthÉLabo Recherche
Curated by PDSP Ki Database
Target5-hydroxytryptamine receptor 1A(Rattus norvegicus (rat))
Glaxo Research And Development
Curated by ChEMBL
Glaxo Research And Development
Curated by ChEMBL
Affinity DataKi: 251nMAssay Description:Binding affinity towards 5-hydroxytryptamine 1A receptor in rat hippocampus using [3H]8-OH-DPATMore data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 1A(Rattus norvegicus (rat))
Glaxo Research And Development
Curated by ChEMBL
Glaxo Research And Development
Curated by ChEMBL
Affinity DataKi: 316nMAssay Description:Binding affinity towards 5-hydroxytryptamine 1A receptor in rat hippocampus with [3H]8-OH-DPATMore data for this Ligand-Target Pair
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
SynthÉLabo Recherche
Curated by PDSP Ki Database
SynthÉLabo Recherche
Curated by PDSP Ki Database
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
SynthÉLabo Recherche
Curated by PDSP Ki Database
SynthÉLabo Recherche
Curated by PDSP Ki Database
TargetAlpha-1A/Alpha-1B/Alpha-1D adrenergic receptor(Homo sapiens (Human))
Glaxo Research And Development
Curated by ChEMBL
Glaxo Research And Development
Curated by ChEMBL
Affinity DataKi: <1.00E+3nMAssay Description:Binding affinity against alpha-1 adrenoceptorMore data for this Ligand-Target Pair
TargetAlpha-2A/Alpha-2B/Alpha-2C adrenergic receptor(Homo sapiens (Human))
Glaxo Research And Development
Curated by ChEMBL
Glaxo Research And Development
Curated by ChEMBL
Affinity DataKi: <1.00E+3nMAssay Description:Binding affinity against alpha-2 adrenoceptorMore data for this Ligand-Target Pair
TargetMuscarinic acetylcholine receptor M2(Homo sapiens (Human))
Glaxo Research And Development
Curated by ChEMBL
Glaxo Research And Development
Curated by ChEMBL
Affinity DataKi: <1.00E+3nMAssay Description:Binding affinity against muscarinic M2 receptorMore data for this Ligand-Target Pair
TargetMuscarinic acetylcholine receptor M1(Homo sapiens (Human))
Glaxo Research And Development
Curated by ChEMBL
Glaxo Research And Development
Curated by ChEMBL
Affinity DataKi: <1.00E+3nMAssay Description:Binding affinity against muscarinic M1 receptorMore data for this Ligand-Target Pair
TargetMuscarinic acetylcholine receptor M3(Homo sapiens (Human))
Glaxo Research And Development
Curated by ChEMBL
Glaxo Research And Development
Curated by ChEMBL
Affinity DataKi: <1.00E+3nMAssay Description:Binding affinity against muscarinic M3 receptorMore data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 1A(Rattus norvegicus (rat))
Glaxo Research And Development
Curated by ChEMBL
Glaxo Research And Development
Curated by ChEMBL
Affinity DataKi: 1.26E+3nMAssay Description:Binding affinity towards 5-hydroxytryptamine 1A receptor in rat hippocampus with [3H]8-OH-DPATMore data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 1A(Rattus norvegicus (rat))
Glaxo Research And Development
Curated by ChEMBL
Glaxo Research And Development
Curated by ChEMBL
Affinity DataKi: 1.26E+3nMAssay Description:Binding affinity towards 5-hydroxytryptamine 1A receptor in rat hippocampus using [3H]8-OH-DPATMore data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 1B(Rattus norvegicus (Rat))
Glaxo Research And Development
Curated by ChEMBL
Glaxo Research And Development
Curated by ChEMBL
Target5-hydroxytryptamine 1D receptor(Bos taurus (Bovine))
SynthÉLabo Recherche
Curated by PDSP Ki Database
SynthÉLabo Recherche
Curated by PDSP Ki Database
TargetVoltage-dependent L-type calcium channel subunit alpha-1C(RAT)
SynthÉLabo Recherche
Curated by PDSP Ki Database
SynthÉLabo Recherche
Curated by PDSP Ki Database
Target5-hydroxytryptamine receptor 1A(Rattus norvegicus (rat))
Glaxo Research And Development
Curated by ChEMBL
Glaxo Research And Development
Curated by ChEMBL