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Found 177 with Last Name = 'castillo' and Initial = 'm'
TargetLysine--tRNA ligase(Homo sapiens (Human))
RhôNe-Poulenc Rorer

Curated by ChEMBL
LigandPNGBDBM50390557(CHEMBL2069346)
Affinity DataIC50:  0.600nMAssay Description:Inhibition of human recombinant full-length Syk using poly-GT as substrate after 40 mins by radioactive filtration assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLysine--tRNA ligase(Homo sapiens (Human))
RhôNe-Poulenc Rorer

Curated by ChEMBL
LigandPNGBDBM50390556(CHEMBL2069345)
Affinity DataIC50:  1.80nMAssay Description:Inhibition of human recombinant full-length Syk using poly-GT as substrate after 40 mins by radioactive filtration assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin D2 receptor 2(Homo sapiens (Human))
RhôNe-Poulenc Rorer

Curated by ChEMBL
LigandPNGBDBM50154805(CHEMBL3775213)
Affinity DataIC50:  2nMAssay Description:Displacement of [35S]-GTPgammaS from CRTH2 receptor (unknown origin) expressed in CHOK1 cell membrane after 1 hr by liquid scintillation counterMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin D2 receptor 2(Homo sapiens (Human))
RhôNe-Poulenc Rorer

Curated by ChEMBL
LigandPNGBDBM50154763(CHEMBL3774415)
Affinity DataIC50:  2nMAssay Description:Displacement of [35S]-GTPgammaS from CRTH2 receptor (unknown origin) expressed in CHOK1 cell membrane after 1 hr by liquid scintillation counterMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLysine--tRNA ligase(Homo sapiens (Human))
RhôNe-Poulenc Rorer

Curated by ChEMBL
LigandPNGBDBM50390561(CHEMBL2069350)
Affinity DataIC50:  4nMAssay Description:Inhibition of human recombinant full-length Syk using poly-GT as substrate after 40 mins by radioactive filtration assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLysine--tRNA ligase(Homo sapiens (Human))
RhôNe-Poulenc Rorer

Curated by ChEMBL
LigandPNGBDBM50390563(CHEMBL2069352)
Affinity DataIC50:  4nMAssay Description:Inhibition of human recombinant full-length Syk using poly-GT as substrate after 40 mins by radioactive filtration assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin D2 receptor 2(Homo sapiens (Human))
RhôNe-Poulenc Rorer

Curated by ChEMBL
LigandPNGBDBM50154762(CHEMBL3774971)
Affinity DataIC50:  4nMAssay Description:Displacement of [35S]-GTPgammaS from CRTH2 receptor (unknown origin) expressed in CHOK1 cell membrane after 1 hr by liquid scintillation counterMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLysine--tRNA ligase(Homo sapiens (Human))
RhôNe-Poulenc Rorer

Curated by ChEMBL
LigandPNGBDBM50390560(CHEMBL2069349)
Affinity DataIC50:  4nMAssay Description:Inhibition of human recombinant full-length Syk using poly-GT as substrate after 40 mins by radioactive filtration assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLysine--tRNA ligase(Homo sapiens (Human))
RhôNe-Poulenc Rorer

Curated by ChEMBL
LigandPNGBDBM50390568(CHEMBL2069358)
Affinity DataIC50:  4nMAssay Description:Inhibition of human recombinant full-length Syk using poly-GT as substrate after 40 mins by radioactive filtration assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin D2 receptor 2(Homo sapiens (Human))
RhôNe-Poulenc Rorer

Curated by ChEMBL
LigandPNGBDBM50444781(CHEMBL3099118)
Affinity DataIC50:  4nMAssay Description:Antagonist activity at CRTh2 in human RBC assessed as inhibition of PGD2-induced eosinophil shape changeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin D2 receptor 2(Homo sapiens (Human))
RhôNe-Poulenc Rorer

Curated by ChEMBL
LigandPNGBDBM50034809(CHEMBL3338090)
Affinity DataIC50:  5nMAssay Description:Displacement of [35S]-GTPgammaS from CRTH2 receptor (unknown origin) expressed in CHOK1 cell membrane after 1 hr by liquid scintillation counterMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin D2 receptor 2(Homo sapiens (Human))
RhôNe-Poulenc Rorer

Curated by ChEMBL
LigandPNGBDBM50154760(CHEMBL3774449)
Affinity DataIC50:  5nMAssay Description:Displacement of [35S]-GTPgammaS from CRTH2 receptor (unknown origin) expressed in CHOK1 cell membrane after 1 hr by liquid scintillation counterMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin D2 receptor 2(Homo sapiens (Human))
RhôNe-Poulenc Rorer

Curated by ChEMBL
LigandPNGBDBM50434451(CHEMBL2385124)
Affinity DataIC50:  5nMAssay Description:Antagonist activity at CRTh2 in human whole blood assessed as inhibition of PGD2-induced eosinophil shape changeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLysine--tRNA ligase(Homo sapiens (Human))
RhôNe-Poulenc Rorer

Curated by ChEMBL
LigandPNGBDBM50390564(CHEMBL2069353)
Affinity DataIC50:  5nMAssay Description:Inhibition of human recombinant full-length Syk using poly-GT as substrate after 40 mins by radioactive filtration assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin D2 receptor 2(Homo sapiens (Human))
RhôNe-Poulenc Rorer

Curated by ChEMBL
LigandPNGBDBM50154760(CHEMBL3774449)
Affinity DataIC50:  6nMAssay Description:Antagonist activity at CRTH2 receptor in human eosinophils by ESC assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLysine--tRNA ligase(Homo sapiens (Human))
RhôNe-Poulenc Rorer

Curated by ChEMBL
LigandPNGBDBM50390566(CHEMBL2069355)
Affinity DataIC50:  6nMAssay Description:Inhibition of human recombinant full-length Syk using poly-GT as substrate after 40 mins by radioactive filtration assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin D2 receptor 2(Homo sapiens (Human))
RhôNe-Poulenc Rorer

Curated by ChEMBL
LigandPNGBDBM50434456(CHEMBL2387692)
Affinity DataIC50:  7nMAssay Description:Displacement of [35S]-GTPgammaS from CRTH2 receptor (unknown origin) expressed in CHOK1 cell membrane after 1 hr by liquid scintillation counterMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLysine--tRNA ligase(Homo sapiens (Human))
RhôNe-Poulenc Rorer

Curated by ChEMBL
LigandPNGBDBM50390567(CHEMBL2069357)
Affinity DataIC50:  7nMAssay Description:Inhibition of human recombinant full-length Syk using poly-GT as substrate after 40 mins by radioactive filtration assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLysine--tRNA ligase(Homo sapiens (Human))
RhôNe-Poulenc Rorer

Curated by ChEMBL
LigandPNGBDBM50390562(CHEMBL2069351)
Affinity DataIC50:  8nMAssay Description:Inhibition of human recombinant full-length Syk using poly-GT as substrate after 40 mins by radioactive filtration assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLysine--tRNA ligase(Homo sapiens (Human))
RhôNe-Poulenc Rorer

Curated by ChEMBL
LigandPNGBDBM50390569(CHEMBL2069359)
Affinity DataIC50:  8nMAssay Description:Inhibition of human recombinant full-length Syk using poly-GT as substrate after 40 mins by radioactive filtration assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin D2 receptor 2(Homo sapiens (Human))
RhôNe-Poulenc Rorer

Curated by ChEMBL
LigandPNGBDBM50154809(CHEMBL3775081)
Affinity DataIC50:  8nMAssay Description:Displacement of [35S]-GTPgammaS from CRTH2 receptor (unknown origin) expressed in CHOK1 cell membrane after 1 hr by liquid scintillation counterMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLysine--tRNA ligase(Homo sapiens (Human))
RhôNe-Poulenc Rorer

Curated by ChEMBL
LigandPNGBDBM50390573(CHEMBL2069356)
Affinity DataIC50:  9nMAssay Description:Inhibition of human recombinant full-length Syk using poly-GT as substrate after 40 mins by radioactive filtration assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLysine--tRNA ligase(Homo sapiens (Human))
RhôNe-Poulenc Rorer

Curated by ChEMBL
LigandPNGBDBM50390571(CHEMBL2069360)
Affinity DataIC50:  10nMAssay Description:Inhibition of human recombinant full-length Syk using poly-GT as substrate after 40 mins by radioactive filtration assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin D2 receptor 2(Homo sapiens (Human))
RhôNe-Poulenc Rorer

Curated by ChEMBL
LigandPNGBDBM50154639(CHEMBL3774535)
Affinity DataIC50:  12nMAssay Description:Antagonist activity at CRTH2 receptor in human eosinophils by ESC assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin D2 receptor 2(Homo sapiens (Human))
RhôNe-Poulenc Rorer

Curated by ChEMBL
LigandPNGBDBM50154764(CHEMBL3774547)
Affinity DataIC50:  14nMAssay Description:Displacement of [35S]-GTPgammaS from CRTH2 receptor (unknown origin) expressed in CHOK1 cell membrane after 1 hr by liquid scintillation counterMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin D2 receptor 2(Homo sapiens (Human))
RhôNe-Poulenc Rorer

Curated by ChEMBL
LigandPNGBDBM50434451(CHEMBL2385124)
Affinity DataIC50:  14nMAssay Description:Displacement of [35S]-GTPgammaS from CRTH2 receptor (unknown origin) expressed in CHOK1 cell membrane after 1 hr by liquid scintillation counterMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLysine--tRNA ligase(Homo sapiens (Human))
RhôNe-Poulenc Rorer

Curated by ChEMBL
LigandPNGBDBM50390552(CHEMBL2069341)
Affinity DataIC50:  14nMAssay Description:Inhibition of human recombinant full-length Syk using poly-GT as substrate after 40 mins by radioactive filtration assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin D2 receptor 2(Homo sapiens (Human))
RhôNe-Poulenc Rorer

Curated by ChEMBL
LigandPNGBDBM50154761(CHEMBL3775880)
Affinity DataIC50:  18nMAssay Description:Displacement of [35S]-GTPgammaS from CRTH2 receptor (unknown origin) expressed in CHOK1 cell membrane after 1 hr by liquid scintillation counterMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLysine--tRNA ligase(Homo sapiens (Human))
RhôNe-Poulenc Rorer

Curated by ChEMBL
LigandPNGBDBM50390555(CHEMBL2069344)
Affinity DataIC50:  27nMAssay Description:Inhibition of human recombinant full-length Syk using poly-GT as substrate after 40 mins by radioactive filtration assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLysine--tRNA ligase(Homo sapiens (Human))
RhôNe-Poulenc Rorer

Curated by ChEMBL
LigandPNGBDBM50390565(CHEMBL2069354)
Affinity DataIC50:  28nMAssay Description:Inhibition of human recombinant full-length Syk using poly-GT as substrate after 40 mins by radioactive filtration assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin D2 receptor 2(Homo sapiens (Human))
RhôNe-Poulenc Rorer

Curated by ChEMBL
LigandPNGBDBM50154639(CHEMBL3774535)
Affinity DataIC50:  28nMAssay Description:Displacement of [35S]-GTPgammaS from CRTH2 receptor (unknown origin) expressed in CHOK1 cell membrane after 1 hr by liquid scintillation counterMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin D2 receptor 2(Homo sapiens (Human))
RhôNe-Poulenc Rorer

Curated by ChEMBL
LigandPNGBDBM50444781(CHEMBL3099118)
Affinity DataIC50:  30nMAssay Description:Antagonist activity at CRTh2 (unknown origin) expressed in CHO.K1 cells assessed as inhibition of PGD2-induced [35S]-GTPgammaS binding after 2 hrs by...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin D2 receptor 2(Homo sapiens (Human))
RhôNe-Poulenc Rorer

Curated by ChEMBL
LigandPNGBDBM50444782(CHEMBL3099133)
Affinity DataIC50:  40nMAssay Description:Antagonist activity at CRTh2 (unknown origin) expressed in CHO.K1 cells assessed as inhibition of PGD2-induced [35S]-GTPgammaS binding after 2 hrs by...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLysine--tRNA ligase(Homo sapiens (Human))
RhôNe-Poulenc Rorer

Curated by ChEMBL
LigandPNGBDBM50390559(CHEMBL2069348)
Affinity DataIC50:  43nMAssay Description:Inhibition of human recombinant full-length Syk using poly-GT as substrate after 40 mins by radioactive filtration assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin D2 receptor 2(Homo sapiens (Human))
RhôNe-Poulenc Rorer

Curated by ChEMBL
LigandPNGBDBM50154765(CHEMBL3774567)
Affinity DataIC50:  47nMAssay Description:Displacement of [35S]-GTPgammaS from CRTH2 receptor (unknown origin) expressed in CHOK1 cell membrane after 1 hr by liquid scintillation counterMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin D2 receptor 2(Homo sapiens (Human))
RhôNe-Poulenc Rorer

Curated by ChEMBL
LigandPNGBDBM50444780(CHEMBL3099129)
Affinity DataIC50:  50nMAssay Description:Antagonist activity at CRTh2 (unknown origin) expressed in CHO.K1 cells assessed as inhibition of PGD2-induced [35S]-GTPgammaS binding after 2 hrs by...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin D2 receptor 2(Homo sapiens (Human))
RhôNe-Poulenc Rorer

Curated by ChEMBL
LigandPNGBDBM50444782(CHEMBL3099133)
Affinity DataIC50:  50nMAssay Description:Antagonist activity at CRTh2 in human RBC assessed as inhibition of PGD2-induced eosinophil shape changeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin D2 receptor 2(Homo sapiens (Human))
RhôNe-Poulenc Rorer

Curated by ChEMBL
LigandPNGBDBM50444781(CHEMBL3099118)
Affinity DataIC50:  50nMAssay Description:Antagonist activity at CRTh2 in human whole blood assessed as inhibition of PGD2-induced eosinophil shape changeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin D2 receptor 2(Homo sapiens (Human))
RhôNe-Poulenc Rorer

Curated by ChEMBL
LigandPNGBDBM50444806(CHEMBL3099106)
Affinity DataIC50:  60nMAssay Description:Antagonist activity at CRTh2 (unknown origin) expressed in CHO.K1 cells assessed as inhibition of PGD2-induced [35S]-GTPgammaS binding after 2 hrs by...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLysine--tRNA ligase(Homo sapiens (Human))
RhôNe-Poulenc Rorer

Curated by ChEMBL
LigandPNGBDBM50390558(CHEMBL2069347)
Affinity DataIC50:  62nMAssay Description:Inhibition of human recombinant full-length Syk using poly-GT as substrate after 40 mins by radioactive filtration assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin D2 receptor 2(Homo sapiens (Human))
RhôNe-Poulenc Rorer

Curated by ChEMBL
LigandPNGBDBM50154784(CHEMBL3775706)
Affinity DataIC50:  65nMAssay Description:Displacement of [35S]-GTPgammaS from CRTH2 receptor (unknown origin) expressed in CHOK1 cell membrane after 1 hr by liquid scintillation counterMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin D2 receptor 2(Homo sapiens (Human))
RhôNe-Poulenc Rorer

Curated by ChEMBL
LigandPNGBDBM50444811(CHEMBL3099132)
Affinity DataIC50:  70nMAssay Description:Antagonist activity at CRTh2 (unknown origin) expressed in CHO.K1 cells assessed as inhibition of PGD2-induced [35S]-GTPgammaS binding after 2 hrs by...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] A(Rattus norvegicus (rat))
Universidad De Chile

Curated by ChEMBL
LigandPNGBDBM50164336(2-(2-Chloro-4,6-dimethoxy-phenyl)-1-methyl-ethylam...)
Affinity DataIC50:  70nMAssay Description:Inhibitory concentration against monoamine oxidase A in rat brain mitochondrial suspensionMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin D2 receptor 2(Homo sapiens (Human))
RhôNe-Poulenc Rorer

Curated by ChEMBL
LigandPNGBDBM50444804(CHEMBL3099108)
Affinity DataIC50:  70nMAssay Description:Antagonist activity at CRTh2 (unknown origin) expressed in CHO.K1 cells assessed as inhibition of PGD2-induced [35S]-GTPgammaS binding after 2 hrs by...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin D2 receptor 2(Homo sapiens (Human))
RhôNe-Poulenc Rorer

Curated by ChEMBL
LigandPNGBDBM50444781(CHEMBL3099118)
Affinity DataIC50:  70nMAssay Description:Antagonist activity at CRTh2 (unknown origin) expressed in CHO.K1 cells assessed as inhibition of PGD2-induced [35S]-GTPgammaS binding after 2 hrs by...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] A(Rattus norvegicus (rat))
Universidad De Chile

Curated by ChEMBL
LigandPNGBDBM50164326(2-(4-Ethylsulfanyl-2,6-dimethoxy-phenyl)-1-methyl-...)
Affinity DataIC50:  80nMAssay Description:Inhibitory concentration against monoamine oxidase A in rat brain mitochondrial suspensionMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin D2 receptor 2(Homo sapiens (Human))
RhôNe-Poulenc Rorer

Curated by ChEMBL
LigandPNGBDBM50444782(CHEMBL3099133)
Affinity DataIC50:  85nMAssay Description:Displacement of [35S]-GTPgammaS from CRTH2 receptor (unknown origin) expressed in CHOK1 cell membrane after 1 hr by liquid scintillation counterMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin D2 receptor 2(Homo sapiens (Human))
RhôNe-Poulenc Rorer

Curated by ChEMBL
LigandPNGBDBM50444786(CHEMBL3099097)
Affinity DataIC50:  87nMAssay Description:Antagonist activity at CRTh2 (unknown origin) expressed in CHO.K1 cells assessed as inhibition of PGD2-induced [35S]-GTPgammaS binding after 2 hrs by...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLysine--tRNA ligase(Homo sapiens (Human))
RhôNe-Poulenc Rorer

Curated by ChEMBL
LigandPNGBDBM50390570(CHEMBL2069337)
Affinity DataIC50:  91nMAssay Description:Inhibition of human recombinant full-length Syk using poly-GT as substrate after 40 mins by radioactive filtration assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] A(Rattus norvegicus (rat))
Universidad De Chile

Curated by ChEMBL
LigandPNGBDBM50164327(2-(4-Ethylsulfanyl-phenyl)-1-methyl-ethylamine | 2...)
Affinity DataIC50:  100nMAssay Description:Inhibitory concentration against monoamine oxidase A in rat brain mitochondrial suspensionMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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