Affinity DataKi: 0.400nMAssay Description:Compound was evaluated in vitro for the binding of Cysteinyl leukotriene receptor 1 to guinea pig lung membranesMore data for this Ligand-Target Pair
Affinity DataKi: 0.600nMAssay Description:Compound was evaluated in vitro for the binding of Cysteinyl leukotriene receptor 1 to guinea pig lung membranesMore data for this Ligand-Target Pair
Affinity DataKi: 0.700nMAssay Description:Antagonism of Cysteinyl leukotriene receptor 1 from guinea pig lung membranesMore data for this Ligand-Target Pair
Affinity DataKi: 0.800nMAssay Description:Ability to antagonize LTD4 receptors isolated from guinea pig lung membranesMore data for this Ligand-Target Pair
Affinity DataKi: 0.800nMAssay Description:Compound was evaluated in vitro for the binding of Cysteinyl leukotriene receptor 1 to guinea pig lung membranesMore data for this Ligand-Target Pair
Affinity DataKi: 0.800nMAssay Description:Antagonism of Cysteinyl leukotriene receptor 1 from guinea pig lung membranesMore data for this Ligand-Target Pair
Affinity DataKi: 2nMAssay Description:Ability to antagonize LTD4 receptors isolated from guinea pig lung membranesMore data for this Ligand-Target Pair
Affinity DataKi: 2nMAssay Description:Ability to antagonize LTD4 receptors isolated from guinea pig lung membranesMore data for this Ligand-Target Pair
Affinity DataKi: 2nMAssay Description:Ability to antagonize LTD4 receptors isolated from guinea pig lung membranesMore data for this Ligand-Target Pair
Affinity DataKi: 2nMAssay Description:Compound was evaluated in vitro for the binding of cysLT1 receptor to guinea pig lung membranes.More data for this Ligand-Target Pair
Affinity DataKi: 2nMAssay Description:Antagonism of Cysteinyl leukotriene receptor 1 from guinea pig lung membranesMore data for this Ligand-Target Pair
Affinity DataKi: 2nMAssay Description:Antagonism of Cysteinyl leukotriene receptor 1 from guinea pig lung membranesMore data for this Ligand-Target Pair
Affinity DataKi: 3nMAssay Description:Ability to antagonize LTD4 receptors isolated from guinea pig lung membranesMore data for this Ligand-Target Pair
Affinity DataKi: 4nMAssay Description:Antagonism of Cysteinyl leukotriene receptor 1 from guinea pig lung membranesMore data for this Ligand-Target Pair
Affinity DataKi: 4nMAssay Description:Antagonism of Cysteinyl leukotriene receptor 1 from guinea pig lung membranesMore data for this Ligand-Target Pair
Affinity DataKi: 5nMAssay Description:Antagonism of Cysteinyl leukotriene receptor 1 from guinea pig lung membranesMore data for this Ligand-Target Pair
Affinity DataKi: 7nMAssay Description:Antagonism of Cysteinyl leukotriene receptor 1 from guinea pig lung membranesMore data for this Ligand-Target Pair
Affinity DataKi: 14nMAssay Description:Ability to antagonize LTD4 receptors isolated from guinea pig lung membranesMore data for this Ligand-Target Pair
Affinity DataKi: 14nMAssay Description:Antagonism of Cysteinyl leukotriene receptor 1 from guinea pig lung membranesMore data for this Ligand-Target Pair
Affinity DataKi: 19nMAssay Description:Ability to antagonize LTD4 receptors isolated from guinea pig lung membranesMore data for this Ligand-Target Pair
Affinity DataKi: 27nMAssay Description:Ability to antagonize LTD4 receptors isolated from guinea pig lung membranesMore data for this Ligand-Target Pair
Affinity DataKi: 92nMAssay Description:Ability to antagonize LTD4 receptors isolated from guinea pig lung membranesMore data for this Ligand-Target Pair
Affinity DataKi: 434nMAssay Description:Ability to antagonize LTD4 receptors isolated from guinea pig lung membranesMore data for this Ligand-Target Pair
Affinity DataKi: 650nMAssay Description:Inhibition of [3H]-LTD4 binding to LTD4 receptor in guinea pig lung membranesMore data for this Ligand-Target Pair
Affinity DataKi: 1.50E+3nMAssay Description:Inhibition of [3H]-LTD4 binding to LTD4 receptor in guinea pig lung membranesMore data for this Ligand-Target Pair
Affinity DataKi: 6.80E+3nMAssay Description:Inhibition of [3H]-LTD4 binding to LTD4 receptor in guinea pig lung membranesMore data for this Ligand-Target Pair
Affinity DataKi: 8.00E+3nMAssay Description:Inhibition of [3H]-LTD4 binding to LTD4 receptor in guinea pig lung membranesMore data for this Ligand-Target Pair
Affinity DataKi: 2.40E+4nMAssay Description:Inhibition of [3H]-LTD4 binding to LTD4 receptor in guinea pig lung membranesMore data for this Ligand-Target Pair
Affinity DataIC50: 0.200nMAssay Description:Compound was tested for the inhibition of human plasma renin(Hu Renin)More data for this Ligand-Target Pair
Affinity DataIC50: 0.25nMAssay Description:Inhibition of human recombinant sVCAM-1 binding to alpha4-beta1 integrin (VLA-4) in ELISAMore data for this Ligand-Target Pair
Affinity DataIC50: 0.300nMAssay Description:Compound was tested for the inhibition of monkey plasma reninMore data for this Ligand-Target Pair
Affinity DataIC50: 0.400nMAssay Description:Binding affinity against leukotriene D4 receptor in [3H]-LTD4 binding assayMore data for this Ligand-Target Pair
Affinity DataIC50: 0.400nMAssay Description:Binding affinity against leukotriene D4 receptor in [3H]-LTD4 binding assayMore data for this Ligand-Target Pair
Affinity DataIC50: 0.400nMAssay Description:Binding affinity against leukotriene D4 receptor in [3H]-LTD4 binding assayMore data for this Ligand-Target Pair
Affinity DataIC50: 0.5nMAssay Description:Binding affinity against leukotriene D4 receptor in [3H]-LTD4 binding assayMore data for this Ligand-Target Pair
Affinity DataIC50: 0.5nMAssay Description:Binding affinity against leukotriene D4 receptor in [3H]-LTD4 binding assayMore data for this Ligand-Target Pair
Affinity DataIC50: 0.5nMAssay Description:Binding affinity against leukotriene D4 receptor in [3H]-LTD4 binding assayMore data for this Ligand-Target Pair
Affinity DataIC50: 0.5nMAssay Description:Compound was tested for the inhibition of monkey plasma reninMore data for this Ligand-Target Pair
Affinity DataIC50: 0.5nMAssay Description:Compound was tested for the inhibition of guinea pig plasma reninMore data for this Ligand-Target Pair
Affinity DataIC50: 0.5nMAssay Description:Binding affinity against leukotriene D4 receptor in [3H]-LTD4 binding assayMore data for this Ligand-Target Pair
Affinity DataIC50: 0.600nMAssay Description:Compound was tested for the inhibition of human plasma renin(Hu Renin)More data for this Ligand-Target Pair
Affinity DataIC50: 0.690nMAssay Description:Inhibition of Alpha4-beta1 integrin in Jurkat cellsMore data for this Ligand-Target Pair
Affinity DataIC50: 1nMAssay Description:Inhibition of C5a mediated human eosinophil chemotaxisMore data for this Ligand-Target Pair
Affinity DataIC50: 1nMAssay Description:Inhibition of PAF mediated human eosinophil chemotaxisMore data for this Ligand-Target Pair
Affinity DataIC50: 1nMAssay Description:Inhibition of Alpha4-beta1 integrin in Jurkat cellsMore data for this Ligand-Target Pair
Affinity DataIC50: 1nMAssay Description:Binding affinity against leukotriene D4 receptor in [3H]-LTD4 binding assayMore data for this Ligand-Target Pair
Affinity DataIC50: 1nMAssay Description:Binding affinity against leukotriene D4 receptor in [3H]-LTD4 binding assayMore data for this Ligand-Target Pair
Affinity DataIC50: 1nMAssay Description:Binding affinity against leukotriene D4 receptor in [3H]-LTD4 binding assayMore data for this Ligand-Target Pair
Affinity DataIC50: 2nMAssay Description:Ability to inhibit LTB4-induced chemotaxis of isolated human neutrophils.More data for this Ligand-Target Pair