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Found 33 with Last Name = 'charton' and Initial = 'y'
TargetNeuronal acetylcholine receptor subunit alpha-4(Rattus norvegicus (Rat))
Servier, Chemistry Research Division A

Curated by PDSP Ki Database
LigandPNGBDBM86902(1-((5-bromopyridin-3-yloxy)methyl)-N-methylcyclopr...)
Affinity DataKi:  1.07nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuronal acetylcholine receptor subunit alpha-4(Rattus norvegicus (Rat))
Servier, Chemistry Research Division A

Curated by PDSP Ki Database
LigandPNGBDBM86919(CAS_22325164 | N-methyl-1-((pyridin-3-yloxy)methyl...)
In DepthDetails ArticlePubMed
TargetNeuronal acetylcholine receptor subunit alpha-4(Rattus norvegicus (Rat))
Servier, Chemistry Research Division A

Curated by PDSP Ki Database
LigandPNGBDBM50004108((+-)-nicotine | (R,S)-nicotine | (RS)-nicotine | 3...)
TargetNeuronal acetylcholine receptor subunit alpha-4(Rattus norvegicus (Rat))
Servier, Chemistry Research Division A

Curated by PDSP Ki Database
LigandPNGBDBM86899(1-((5-bromo-6-chloropyridin-3-yloxy)methyl)-N-meth...)
Affinity DataKi:  5.37nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuronal acetylcholine receptor subunit alpha-4(Rattus norvegicus (Rat))
Servier, Chemistry Research Division A

Curated by PDSP Ki Database
LigandPNGBDBM86907(1-((5-ethynylpyridin-3-yloxy)methyl)-N-methylcyclo...)
Affinity DataKi:  6.56nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuronal acetylcholine receptor subunit alpha-4(Rattus norvegicus (Rat))
Servier, Chemistry Research Division A

Curated by PDSP Ki Database
LigandPNGBDBM86918(1-((6-chloropyridin-3-yloxy)methyl)-N-methylcyclop...)
Affinity DataKi:  13nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuronal acetylcholine receptor subunit alpha-4(Rattus norvegicus (Rat))
Servier, Chemistry Research Division A

Curated by PDSP Ki Database
LigandPNGBDBM86911(1-(pyridin-3-yloxymethyl)-cyclopropylamine; hydroc...)
Affinity DataKi:  34nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuronal acetylcholine receptor subunit alpha-4(Rattus norvegicus (Rat))
Servier, Chemistry Research Division A

Curated by PDSP Ki Database
LigandPNGBDBM86915(1-((6-bromopyridin-3-yloxy)methyl)-N-methylcyclopr...)
Affinity DataKi:  38.8nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuronal acetylcholine receptor subunit alpha-4(Rattus norvegicus (Rat))
Servier, Chemistry Research Division A

Curated by PDSP Ki Database
LigandPNGBDBM10759(2-acetoxyethyl(trimethyl)ammonium;bromide | 2-acet...)
Affinity DataKi:  39nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuronal acetylcholine receptor subunit alpha-4(Rattus norvegicus (Rat))
Servier, Chemistry Research Division A

Curated by PDSP Ki Database
LigandPNGBDBM86922(CAS_9899400 | N-methyl-1-((6-methylpyridin-3-yloxy...)
Affinity DataKi:  40nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuronal acetylcholine receptor subunit alpha-4(Rattus norvegicus (Rat))
Servier, Chemistry Research Division A

Curated by PDSP Ki Database
LigandPNGBDBM86905(CAS_45263892 | N-methyl-1-((5-vinylpyridin-3-yloxy...)
Affinity DataKi:  70.1nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetNeuronal acetylcholine receptor subunit alpha-4(Rattus norvegicus (Rat))
Servier, Chemistry Research Division A

Curated by PDSP Ki Database
LigandPNGBDBM86916(CAS_22325080 | NSC_22325080 | dimethyl-[1-(pyridin...)
Affinity DataKi:  95nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuronal acetylcholine receptor subunit alpha-4(Rattus norvegicus (Rat))
Servier, Chemistry Research Division A

Curated by PDSP Ki Database
LigandPNGBDBM86908(1-(6-chloro-pyridin-3-yloxymethyl)-cyclopropylamin...)
Affinity DataKi:  98nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuronal acetylcholine receptor subunit alpha-4(Rattus norvegicus (Rat))
Servier, Chemistry Research Division A

Curated by PDSP Ki Database
LigandPNGBDBM86920(CAS_9944441 | NSC_9944441 | methyl-{1-[2-(pyridin-...)
Affinity DataKi:  109nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuronal acetylcholine receptor subunit alpha-4(Rattus norvegicus (Rat))
Servier, Chemistry Research Division A

Curated by PDSP Ki Database
LigandPNGBDBM86912(CAS_45263898 | N-methyl-1-(2-(pyridin-3-yl)ethyl)c...)
Affinity DataKi:  251nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetNeuronal acetylcholine receptor subunit alpha-4(Rattus norvegicus (Rat))
Servier, Chemistry Research Division A

Curated by PDSP Ki Database
LigandPNGBDBM86921(1-((6-methylpyridin-3-yloxy)methyl)cyclopropanamin...)
Affinity DataKi:  266nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuronal acetylcholine receptor subunit alpha-4(Rattus norvegicus (Rat))
Servier, Chemistry Research Division A

Curated by PDSP Ki Database
LigandPNGBDBM86914(CAS_45263712 | NSC_45263712 | [1-(5-bromo-pyridin-...)
Affinity DataKi:  273nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuronal acetylcholine receptor subunit alpha-4(Rattus norvegicus (Rat))
Servier, Chemistry Research Division A

Curated by PDSP Ki Database
LigandPNGBDBM86900(1-((6-chloropyridin-3-yloxy)methyl)-N,N-dimethylcy...)
Affinity DataKi:  304nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuronal acetylcholine receptor subunit alpha-4(Rattus norvegicus (Rat))
Servier, Chemistry Research Division A

Curated by PDSP Ki Database
LigandPNGBDBM86901(1-((6-bromopyridin-3-yloxy)methyl)-N,N-dimethylcyc...)
Affinity DataKi:  394nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuronal acetylcholine receptor subunit alpha-4(Rattus norvegicus (Rat))
Servier, Chemistry Research Division A

Curated by PDSP Ki Database
LigandPNGBDBM86910(CAS_44454126 | N-ethyl-1-((pyridin-3-yloxy)methyl)...)
Affinity DataKi:  1.01E+3nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuronal acetylcholine receptor subunit alpha-4(Rattus norvegicus (Rat))
Servier, Chemistry Research Division A

Curated by PDSP Ki Database
LigandPNGBDBM86909(CAS_45263866 | N,N-dimethyl-1-((6-methylpyridin-3-...)
Affinity DataKi:  1.09E+3nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuronal acetylcholine receptor subunit alpha-4(Rattus norvegicus (Rat))
Servier, Chemistry Research Division A

Curated by PDSP Ki Database
LigandPNGBDBM86903(CAS_45263725 | CAS_45263737 | NSC_45263725 | NSC_4...)
Affinity DataKi:  1.10E+3nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuronal acetylcholine receptor subunit alpha-4(Rattus norvegicus (Rat))
Servier, Chemistry Research Division A

Curated by PDSP Ki Database
LigandPNGBDBM86906(CAS_9922040 | NSC_9922040 | methyl-[1-(2-pyridin-3...)
Affinity DataKi:  1.16E+3nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetNeuronal acetylcholine receptor subunit alpha-4(Rattus norvegicus (Rat))
Servier, Chemistry Research Division A

Curated by PDSP Ki Database
LigandPNGBDBM86913(3-((1-(pyrrolidin-1-yl)cyclopropyl)methoxy)pyridin...)
Affinity DataKi:  1.61E+3nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuronal acetylcholine receptor subunit alpha-4(Rattus norvegicus (Rat))
Servier, Chemistry Research Division A

Curated by PDSP Ki Database
LigandPNGBDBM86903(CAS_45263725 | CAS_45263737 | NSC_45263725 | NSC_4...)
Affinity DataKi:  2.28E+3nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuronal acetylcholine receptor subunit alpha-4(Rattus norvegicus (Rat))
Servier, Chemistry Research Division A

Curated by PDSP Ki Database
LigandPNGBDBM86917(CAS_44454204 | NSC_44454204 | methyl-{1-[3-(pyridi...)
Affinity DataKi:  2.46E+3nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHexokinase-4(Homo sapiens (Human))
Istituto Italiano Di Tecnologia

Curated by ChEMBL
LigandPNGBDBM50346026((R)-2-(3-chloro-4-(methylsulfonyl)phenyl)-3-((R)-3...)
Affinity DataKd:  830nMAssay Description:Displacement of TAFMT from human pancreatic N-terminal His6-tagged glucokinase isoform 1 expressed in Escherichia coli BL21(DE3) by stopped-flow fluo...More data for this Ligand-Target Pair
TargetHexokinase-4(Homo sapiens (Human))
Istituto Italiano Di Tecnologia

Curated by ChEMBL
LigandPNGBDBM50533461(CHEMBL4483049)
Affinity DataKd:  400nMAssay Description:Displacement of TAFMT from human pancreatic N-terminal His6-tagged glucokinase isoform 1 expressed in Escherichia coli BL21(DE3) by stopped-flow fluo...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetHexokinase-4(Homo sapiens (Human))
Istituto Italiano Di Tecnologia

Curated by ChEMBL
LigandPNGBDBM50533462(CHEMBL4534484)
Affinity DataKd:  720nMAssay Description:Displacement of TAFMT from human pancreatic N-terminal His6-tagged glucokinase isoform 1 expressed in Escherichia coli BL21(DE3) by stopped-flow fluo...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetHexokinase-4(Homo sapiens (Human))
Istituto Italiano Di Tecnologia

Curated by ChEMBL
LigandPNGBDBM50533463(CHEMBL4522750)
Affinity DataKd:  2.00E+3nMAssay Description:Displacement of TAFMT from human pancreatic N-terminal His6-tagged glucokinase isoform 1 expressed in Escherichia coli BL21(DE3) by stopped-flow fluo...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetHexokinase-4(Homo sapiens (Human))
Istituto Italiano Di Tecnologia

Curated by ChEMBL
LigandPNGBDBM34071(benzamide derivative, 6)
Affinity DataKd:  360nMAssay Description:Binding affinity to human pancreatic N-terminal His6-tagged glucokinase isoform 1 expressed in Escherichia coli BL21(DE3) by stopped-flow fluorometri...More data for this Ligand-Target Pair
TargetHexokinase-4(Homo sapiens (Human))
Istituto Italiano Di Tecnologia

Curated by ChEMBL
LigandPNGBDBM50320996(6-(3-((S)-1-methoxypropan-2-yloxy)-5-((S)-1-phenyl...)
Affinity DataKd:  3.30E+3nMAssay Description:Displacement of TAFMT from human pancreatic N-terminal His6-tagged glucokinase isoform 1 expressed in Escherichia coli BL21(DE3) by stopped-flow fluo...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHexokinase-4(Homo sapiens (Human))
Istituto Italiano Di Tecnologia

Curated by ChEMBL
LigandPNGBDBM50533464(CHEMBL4457828)
Affinity DataKd:  4.40E+3nMAssay Description:Displacement of TAFMT from human pancreatic N-terminal His6-tagged glucokinase isoform 1 expressed in Escherichia coli BL21(DE3) by stopped-flow fluo...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed