TargetMu-type opioid receptor(Homo sapiens (Human))
Julius Maximilian University of W£Rzburg
Curated by ChEMBL
Julius Maximilian University of W£Rzburg
Curated by ChEMBL
Affinity DataKi: 0.200nMAssay Description:Displacement of [3H]-Diprenorphine from human mu opioid receptor expressed in HEK293-TSA cell membranes after 4 hrs by scintillation counting methodMore data for this Ligand-Target Pair
TargetCannabinoid receptor 2(Homo sapiens (Human))
Julius Maximilian University of W£Rzburg
Curated by ChEMBL
Julius Maximilian University of W£Rzburg
Curated by ChEMBL
Affinity DataKi: 5.60nMAssay Description:Displacement of [3H]-CP55950 from human CB2 receptor expressed in HEK cell membranes after 90 minsMore data for this Ligand-Target Pair
TargetCannabinoid receptor 2(Homo sapiens (Human))
Julius Maximilian University of W£Rzburg
Curated by ChEMBL
Julius Maximilian University of W£Rzburg
Curated by ChEMBL
Affinity DataKi: 20nMAssay Description:Displacement of [3H]-CP55950 from human CB2 receptor expressed in HEK cell membranes after 3 hrs by scintillation counting methodMore data for this Ligand-Target Pair
TargetCannabinoid receptor 2(Homo sapiens (Human))
Julius Maximilian University of W£Rzburg
Curated by ChEMBL
Julius Maximilian University of W£Rzburg
Curated by ChEMBL
Affinity DataKi: 37nMAssay Description:Displacement of [3H]-CP55950 from human CB2 receptor expressed in HEK cell membranes after 3 hrs by scintillation counting methodMore data for this Ligand-Target Pair
TargetCannabinoid receptor 1(Homo sapiens (Human))
Julius Maximilian University of W£Rzburg
Curated by ChEMBL
Julius Maximilian University of W£Rzburg
Curated by ChEMBL
Affinity DataKi: 143nMAssay Description:Displacement of [3H]-CP55950 from human CB1 receptor expressed in CHO cell membranes after 3 hrs by scintillation counting methodMore data for this Ligand-Target Pair
TargetCannabinoid receptor 2(Homo sapiens (Human))
Julius Maximilian University of W£Rzburg
Curated by ChEMBL
Julius Maximilian University of W£Rzburg
Curated by ChEMBL
Affinity DataKi: 188nMAssay Description:Displacement of [3H]-CP55950 from human CB2 receptor expressed in HEK cell membranes after 3 hrs by scintillation counting methodMore data for this Ligand-Target Pair
TargetCannabinoid receptor 1(Homo sapiens (Human))
Julius Maximilian University of W£Rzburg
Curated by ChEMBL
Julius Maximilian University of W£Rzburg
Curated by ChEMBL
Affinity DataKi: 254nMAssay Description:Displacement of [3H]-CP55950 from human CB1 receptor expressed in CHO cell membranes after 90 minsMore data for this Ligand-Target Pair
TargetCannabinoid receptor 2(Homo sapiens (Human))
Julius Maximilian University of W£Rzburg
Curated by ChEMBL
Julius Maximilian University of W£Rzburg
Curated by ChEMBL
Affinity DataKi: 353nMAssay Description:Displacement of [3H]-CP55950 from human CB2 receptor expressed in HEK cell membranes after 3 hrs by scintillation counting methodMore data for this Ligand-Target Pair
TargetCannabinoid receptor 2(Homo sapiens (Human))
Julius Maximilian University of W£Rzburg
Curated by ChEMBL
Julius Maximilian University of W£Rzburg
Curated by ChEMBL
Affinity DataKi: 385nMAssay Description:Displacement of [3H]-CP55950 from human CB2 receptor expressed in HEK cell membranes after 3 hrs by scintillation counting methodMore data for this Ligand-Target Pair
TargetCannabinoid receptor 2(Homo sapiens (Human))
Julius Maximilian University of W£Rzburg
Curated by ChEMBL
Julius Maximilian University of W£Rzburg
Curated by ChEMBL
Affinity DataKi: 426nMAssay Description:Displacement of [3H]-CP55950 from human CB2 receptor expressed in HEK cell membranes after 3 hrs by scintillation counting methodMore data for this Ligand-Target Pair
TargetMu-type opioid receptor(Homo sapiens (Human))
Julius Maximilian University of W£Rzburg
Curated by ChEMBL
Julius Maximilian University of W£Rzburg
Curated by ChEMBL
Affinity DataKi: 556nMAssay Description:Displacement of [3H]-Diprenorphine from human mu opioid receptor expressed in HEK293-TSA cell membranes after 4 hrs by scintillation counting methodMore data for this Ligand-Target Pair
TargetMu-type opioid receptor(Homo sapiens (Human))
Julius Maximilian University of W£Rzburg
Curated by ChEMBL
Julius Maximilian University of W£Rzburg
Curated by ChEMBL
Affinity DataKi: 556nMAssay Description:Displacement of [3H]-Diprenorphine from human mu opioid receptor expressed in HEK293-TSA cell membranes after 4 hrs by scintillation counting methodMore data for this Ligand-Target Pair
TargetCannabinoid receptor 1(Homo sapiens (Human))
Julius Maximilian University of W£Rzburg
Curated by ChEMBL
Julius Maximilian University of W£Rzburg
Curated by ChEMBL
Affinity DataKi: 687nMAssay Description:Displacement of [3H]-CP55950 from human CB1 receptor expressed in CHO cell membranes after 3 hrs by scintillation counting methodMore data for this Ligand-Target Pair
TargetCannabinoid receptor 2(Homo sapiens (Human))
Julius Maximilian University of W£Rzburg
Curated by ChEMBL
Julius Maximilian University of W£Rzburg
Curated by ChEMBL
Affinity DataKi: 764nMAssay Description:Displacement of [3H]-CP55950 from human CB2 receptor expressed in HEK cell membranes after 3 hrs by scintillation counting methodMore data for this Ligand-Target Pair
TargetCannabinoid receptor 2(Homo sapiens (Human))
Julius Maximilian University of W£Rzburg
Curated by ChEMBL
Julius Maximilian University of W£Rzburg
Curated by ChEMBL
Affinity DataKi: 962nMAssay Description:Displacement of [3H]-CP55950 from human CB2 receptor expressed in HEK cell membranes after 3 hrs by scintillation counting methodMore data for this Ligand-Target Pair
TargetCannabinoid receptor 2(Homo sapiens (Human))
Julius Maximilian University of W£Rzburg
Curated by ChEMBL
Julius Maximilian University of W£Rzburg
Curated by ChEMBL
Affinity DataKi: 1.00E+3nMAssay Description:Displacement of [3H]-CP55950 from human CB2 receptor expressed in HEK cell membranes after 3 hrs by scintillation counting methodMore data for this Ligand-Target Pair
TargetCannabinoid receptor 2(Homo sapiens (Human))
Julius Maximilian University of W£Rzburg
Curated by ChEMBL
Julius Maximilian University of W£Rzburg
Curated by ChEMBL
Affinity DataKi: 1.90E+3nMAssay Description:Displacement of [3H]-CP55950 from human CB2 receptor expressed in HEK cell membranes after 3 hrs by scintillation counting methodMore data for this Ligand-Target Pair
TargetCannabinoid receptor 2(Homo sapiens (Human))
Julius Maximilian University of W£Rzburg
Curated by ChEMBL
Julius Maximilian University of W£Rzburg
Curated by ChEMBL
Affinity DataKi: 1.90E+3nMAssay Description:Displacement of [3H]-CP55950 from human CB2 receptor expressed in HEK cell membranes after 3 hrs by scintillation counting methodMore data for this Ligand-Target Pair
TargetCannabinoid receptor 2(Homo sapiens (Human))
Julius Maximilian University of W£Rzburg
Curated by ChEMBL
Julius Maximilian University of W£Rzburg
Curated by ChEMBL
Affinity DataKi: 4.30E+3nMAssay Description:Displacement of [3H]-CP55950 from human CB2 receptor expressed in HEK cell membranes after 3 hrs by scintillation counting methodMore data for this Ligand-Target Pair
TargetCannabinoid receptor 2(Homo sapiens (Human))
Julius Maximilian University of W£Rzburg
Curated by ChEMBL
Julius Maximilian University of W£Rzburg
Curated by ChEMBL
Affinity DataKi: 4.70E+3nMAssay Description:Displacement of [3H]-CP55950 from human CB2 receptor expressed in HEK cell membranes after 3 hrs by scintillation counting methodMore data for this Ligand-Target Pair
TargetCannabinoid receptor 2(Homo sapiens (Human))
Julius Maximilian University of W£Rzburg
Curated by ChEMBL
Julius Maximilian University of W£Rzburg
Curated by ChEMBL
Affinity DataKi: 4.80E+3nMAssay Description:Displacement of [3H]-CP55950 from human CB2 receptor expressed in HEK cell membranes after 3 hrs by scintillation counting methodMore data for this Ligand-Target Pair
TargetMu-type opioid receptor(Homo sapiens (Human))
Julius Maximilian University of W£Rzburg
Curated by ChEMBL
Julius Maximilian University of W£Rzburg
Curated by ChEMBL
Affinity DataKi: 6.31E+3nMAssay Description:Displacement of [3H]-Diprenorphine from human mu opioid receptor expressed in HEK293-TSA cell membranes after 4 hrs by scintillation counting methodMore data for this Ligand-Target Pair
TargetMu-type opioid receptor(Homo sapiens (Human))
Julius Maximilian University of W£Rzburg
Curated by ChEMBL
Julius Maximilian University of W£Rzburg
Curated by ChEMBL
Affinity DataKi: 6.70E+3nMAssay Description:Displacement of [3H]-Diprenorphine from human mu opioid receptor expressed in HEK293-TSA cell membranes after 4 hrs by scintillation counting methodMore data for this Ligand-Target Pair
TargetCannabinoid receptor 2(Homo sapiens (Human))
Julius Maximilian University of W£Rzburg
Curated by ChEMBL
Julius Maximilian University of W£Rzburg
Curated by ChEMBL
Affinity DataKi: 8.90E+3nMAssay Description:Displacement of [3H]-CP55950 from human CB2 receptor expressed in HEK cell membranes after 3 hrs by scintillation counting methodMore data for this Ligand-Target Pair
TargetCannabinoid receptor 2(Homo sapiens (Human))
Julius Maximilian University of W£Rzburg
Curated by ChEMBL
Julius Maximilian University of W£Rzburg
Curated by ChEMBL
Affinity DataKi: 1.04E+4nMAssay Description:Displacement of [3H]-CP55950 from human CB2 receptor expressed in HEK cell membranes after 3 hrs by scintillation counting methodMore data for this Ligand-Target Pair
TargetCannabinoid receptor 2(Homo sapiens (Human))
Julius Maximilian University of W£Rzburg
Curated by ChEMBL
Julius Maximilian University of W£Rzburg
Curated by ChEMBL
Affinity DataKi: 1.44E+4nMAssay Description:Displacement of [3H]-CP55950 from human CB2 receptor expressed in HEK cell membranes after 3 hrs by scintillation counting methodMore data for this Ligand-Target Pair
TargetCannabinoid receptor 1(Homo sapiens (Human))
Julius Maximilian University of W£Rzburg
Curated by ChEMBL
Julius Maximilian University of W£Rzburg
Curated by ChEMBL
Affinity DataKi: 1.70E+4nMAssay Description:Displacement of [3H]-CP55950 from human CB1 receptor expressed in CHO cell membranes after 3 hrs by scintillation counting methodMore data for this Ligand-Target Pair
TargetCannabinoid receptor 2(Homo sapiens (Human))
Julius Maximilian University of W£Rzburg
Curated by ChEMBL
Julius Maximilian University of W£Rzburg
Curated by ChEMBL
Affinity DataKi: 2.10E+4nMAssay Description:Displacement of [3H]-CP55950 from human CB2 receptor expressed in HEK cell membranes after 3 hrs by scintillation counting methodMore data for this Ligand-Target Pair
TargetMu-type opioid receptor(Homo sapiens (Human))
Julius Maximilian University of W£Rzburg
Curated by ChEMBL
Julius Maximilian University of W£Rzburg
Curated by ChEMBL
Affinity DataKi: 5.01E+4nMAssay Description:Displacement of [3H]-Diprenorphine from human mu opioid receptor expressed in HEK293-TSA cell membranes after 4 hrs by scintillation counting methodMore data for this Ligand-Target Pair
TargetMu-type opioid receptor(Homo sapiens (Human))
Julius Maximilian University of W£Rzburg
Curated by ChEMBL
Julius Maximilian University of W£Rzburg
Curated by ChEMBL
Affinity DataKi: 5.36E+4nMAssay Description:Displacement of [3H]-Diprenorphine from human mu opioid receptor expressed in HEK293-TSA cell membranes after 4 hrs by scintillation counting methodMore data for this Ligand-Target Pair
Affinity DataIC50: 6.40nMAssay Description:Inhibition of human serum BChE using butyrylthiocholine iodide as substrate incubated for 30 mins followed by substrate addition and measured after 2...More data for this Ligand-Target Pair
Affinity DataIC50: 6.5nMAssay Description:Inhibition of human serum BChE using butyrylthiocholine iodide as substrate incubated for 30 mins followed by substrate addition and measured after 2...More data for this Ligand-Target Pair
Affinity DataIC50: 9.10nMAssay Description:Inhibition of human BChE using BTC iodide as substrate preincubated for 4.5 mins followed by substrate addition measured after 2.5 mins by Ellman's m...More data for this Ligand-Target Pair
Affinity DataIC50: 10nMAssay Description:Inhibition of human BChE using BTC iodide as substrate preincubated for 4.5 mins followed by substrate addition measured after 2.5 mins by Ellman's m...More data for this Ligand-Target Pair
TargetAcetylcholinesterase(Homo sapiens (Human))
Julius Maximilian University of W£Rzburg
Curated by ChEMBL
Julius Maximilian University of W£Rzburg
Curated by ChEMBL
Affinity DataIC50: 19nMAssay Description:Tested for binding affinity against human NK-1 receptor transfected on CHO cells using [125I]-Tyr] SP as radioligandMore data for this Ligand-Target Pair
TargetAcetylcholinesterase(Homo sapiens (Human))
Julius Maximilian University of W£Rzburg
Curated by ChEMBL
Julius Maximilian University of W£Rzburg
Curated by ChEMBL
Affinity DataIC50: 20nMAssay Description:Inhibition of human erythrocyte AChE using ATC iodide as substrate preincubated for 4.5 mins followed by substrate addition measured after 2.5 mins b...More data for this Ligand-Target Pair
TargetCannabinoid receptor 2(Homo sapiens (Human))
Julius Maximilian University of W£Rzburg
Curated by ChEMBL
Julius Maximilian University of W£Rzburg
Curated by ChEMBL
Affinity DataIC50: 20nMAssay Description:Displacement of [3H]-CP55950 from human CB2 receptor expressed in HEK cell membranes after 3 hrs by scintillation counting methodMore data for this Ligand-Target Pair
TargetCannabinoid receptor 2(Homo sapiens (Human))
Julius Maximilian University of W£Rzburg
Curated by ChEMBL
Julius Maximilian University of W£Rzburg
Curated by ChEMBL
Affinity DataIC50: 40nMAssay Description:Displacement of [3H]-CP55950 from human CB2 receptor expressed in HEK cell membranes after 3 hrs by scintillation counting methodMore data for this Ligand-Target Pair
Affinity DataIC50: 54nMAssay Description:Inhibition of human BChE using butyrylthiocholine iodide as substrate incubated for 20 mins followed by substrate addition by Ellman's methodMore data for this Ligand-Target Pair
Affinity DataIC50: 54nMAssay Description:Inhibition of human BChE using butyrylthiocholine iodide as substrate incubated for 20 mins followed by substrate addition by Ellman's methodMore data for this Ligand-Target Pair
Affinity DataIC50: 102nMAssay Description:Inhibition of human BChE using butyrylthiocholine iodide as substrate incubated for 20 mins followed by substrate addition by Ellman's methodMore data for this Ligand-Target Pair
Affinity DataIC50: 102nMAssay Description:Inhibition of human BChE using butyrylthiocholine iodide as substrate incubated for 20 mins followed by substrate addition by Ellman's methodMore data for this Ligand-Target Pair
TargetAcetylcholinesterase(Homo sapiens (Human))
Julius Maximilian University of W£Rzburg
Curated by ChEMBL
Julius Maximilian University of W£Rzburg
Curated by ChEMBL
Affinity DataIC50: 110nMAssay Description:Inhibition of human AChE using acetylthiocholine iodide as substrate incubated for 20 mins followed by substrate addition by Ellman's methodMore data for this Ligand-Target Pair
TargetAcetylcholinesterase(Homo sapiens (Human))
Julius Maximilian University of W£Rzburg
Curated by ChEMBL
Julius Maximilian University of W£Rzburg
Curated by ChEMBL
Affinity DataIC50: 111nMAssay Description:Inhibition of human AChE using acetylthiocholine iodide as substrate incubated for 20 mins followed by substrate addition by Ellman's methodMore data for this Ligand-Target Pair
Affinity DataIC50: 126nMAssay Description:Inhibition of human BChE using butyrylthiocholine iodide as substrate incubated for 20 mins followed by substrate addition by Ellman's methodMore data for this Ligand-Target Pair
Affinity DataIC50: 127nMAssay Description:Inhibition of human BChE using butyrylthiocholine iodide as substrate incubated for 20 mins followed by substrate addition by Ellman's methodMore data for this Ligand-Target Pair
Affinity DataIC50: 155nMAssay Description:Inhibition of human BChE using butyrylthiocholine iodide as substrate incubated for 20 mins followed by substrate addition by Ellman's methodMore data for this Ligand-Target Pair
Affinity DataIC50: 155nMAssay Description:Inhibition of human BChE using butyrylthiocholine iodide as substrate incubated for 20 mins followed by substrate addition by Ellman's methodMore data for this Ligand-Target Pair
TargetCannabinoid receptor 1(Homo sapiens (Human))
Julius Maximilian University of W£Rzburg
Curated by ChEMBL
Julius Maximilian University of W£Rzburg
Curated by ChEMBL
Affinity DataIC50: 158nMAssay Description:Displacement of [3H]-CP55950 from human CB1 receptor expressed in CHO cell membranes after 3 hrs by scintillation counting methodMore data for this Ligand-Target Pair
Affinity DataIC50: 166nMAssay Description:Inhibition of human BChE using butyrylthiocholine iodide as substrate incubated for 20 mins followed by substrate addition by Ellman's methodMore data for this Ligand-Target Pair