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Found 277 with Last Name = 'cheetham' and Initial = 's'
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
Boots Pharmaceuticals

Curated by PDSP Ki Database
LigandPNGBDBM22416((3S,4R)-3-[(1,3-benzodioxol-5-yloxy)methyl]-4-(4-f...)
Affinity DataKi:  0.0190nMMore data for this Ligand-Target Pair
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
Boots Pharmaceuticals

Curated by PDSP Ki Database
LigandPNGBDBM82217(CHEMBL284994 | CP-52003 | SERTRALINE | [4-(3,4-Dic...)
Affinity DataKi:  0.0470nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
Boots Pharmaceuticals

Curated by PDSP Ki Database
LigandPNGBDBM50021226(CHEMBL296602 | Indatraline | [3-(3,4-Dichloro-phen...)
Affinity DataKi:  0.130nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
Boots Pharmaceuticals

Curated by PDSP Ki Database
LigandPNGBDBM77970(3-(2-chloranyl-5,6-dihydrobenzo[b][1]benzazepin-11...)
Affinity DataKi:  0.140nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
Boots Pharmaceuticals

Curated by PDSP Ki Database
LigandPNGBDBM22416((3S,4R)-3-[(1,3-benzodioxol-5-yloxy)methyl]-4-(4-f...)
Affinity DataKi:  0.480nMMore data for this Ligand-Target Pair
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
Boots Pharmaceuticals

Curated by PDSP Ki Database
LigandPNGBDBM25870(1-[3-(dimethylamino)propyl]-1-(4-fluorophenyl)-1,3...)
Affinity DataKi:  0.650nMMore data for this Ligand-Target Pair
TargetMelanin-concentrating hormone receptor 1(Homo sapiens (Human))
Amri

Curated by ChEMBL
LigandPNGBDBM50184924(1-((1S,2R,5S)-5-(4-cyanophenyl)bicyclo[3.1.0]hexan...)
Affinity DataKi:  1.20nMAssay Description:Displacement of [3H]GW803430 from MCH-1 receptor expressed in CHO-K1 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
Boots Pharmaceuticals

Curated by PDSP Ki Database
LigandPNGBDBM50021226(CHEMBL296602 | Indatraline | [3-(3,4-Dichloro-phen...)
Affinity DataKi:  1.5nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
Boots Pharmaceuticals

Curated by PDSP Ki Database
LigandPNGBDBM30130(CHEMBL1201082 | CHEMBL41 | Fluoxetin | Fluoxetine ...)
Affinity DataKi:  1.96nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
Boots Pharmaceuticals

Curated by PDSP Ki Database
LigandPNGBDBM50028066(4-(3,4-Dichloro-phenyl)-1,2,3,4-tetrahydro-naphtha...)
Affinity DataKi:  2.29nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanin-concentrating hormone receptor 1(Homo sapiens (Human))
Amri

Curated by ChEMBL
LigandPNGBDBM50331198(1-(5-methyl-2,3,4,5-tetrahydro-1H-pyrido[4,3-b]ind...)
Affinity DataKi:  2.40nMAssay Description:Displacement of [3H]4-(benzyloxy)-1-(1-(2-(pyrrolidin-1-yl)ethyl)-1H-indazol-5-yl)pyridin-2(1H)-one from MCH-1 receptor expressed in CHO-K1 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanin-concentrating hormone receptor 1(Homo sapiens (Human))
Amri

Curated by ChEMBL
LigandPNGBDBM50331161(4-(benzyloxy)-1-(1-(2-(pyrrolidin-1-yl)ethyl)-1H-i...)
Affinity DataKi:  2.60nMAssay Description:Displacement of [3H]4-(benzyloxy)-1-(1-(2-(pyrrolidin-1-yl)ethyl)-1H-indazol-5-yl)pyridin-2(1H)-one from MCH-1 receptor expressed in CHO-K1 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanin-concentrating hormone receptor 1(Homo sapiens (Human))
Amri

Curated by ChEMBL
LigandPNGBDBM50331199(4-(4-methoxyphenyl)-1-(5-methyl-2,3,4,5-tetrahydro...)
Affinity DataKi:  2.60nMAssay Description:Displacement of [3H]4-(benzyloxy)-1-(1-(2-(pyrrolidin-1-yl)ethyl)-1H-indazol-5-yl)pyridin-2(1H)-one from MCH-1 receptor expressed in CHO-K1 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanin-concentrating hormone receptor 1(Homo sapiens (Human))
Amri

Curated by ChEMBL
LigandPNGBDBM50331161(4-(benzyloxy)-1-(1-(2-(pyrrolidin-1-yl)ethyl)-1H-i...)
Affinity DataKi:  2.60nMAssay Description:Displacement of [3H]4-(benzyloxy)-1-(1-(2-(pyrrolidin-1-yl)ethyl)-1H-indazol-5-yl)pyridin-2(1H)-one from MCH-1 receptor expressed in CHO-K1 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanin-concentrating hormone receptor 1(Homo sapiens (Human))
Amri

Curated by ChEMBL
LigandPNGBDBM50331161(4-(benzyloxy)-1-(1-(2-(pyrrolidin-1-yl)ethyl)-1H-i...)
Affinity DataKi:  2.60nMAssay Description:Displacement of [3H]GW803430 from MCH-1 receptor expressed in CHO-K1 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanin-concentrating hormone receptor 1(Homo sapiens (Human))
Amri

Curated by ChEMBL
LigandPNGBDBM50331201(4-(4-chlorophenyl)-1-(5-methyl-2,3,4,5-tetrahydro-...)
Affinity DataKi:  2.70nMAssay Description:Displacement of [3H]4-(benzyloxy)-1-(1-(2-(pyrrolidin-1-yl)ethyl)-1H-indazol-5-yl)pyridin-2(1H)-one from MCH-1 receptor expressed in CHO-K1 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanin-concentrating hormone receptor 1(Homo sapiens (Human))
Amri

Curated by ChEMBL
LigandPNGBDBM50331172(4-(2-chloro-4-methoxyphenyl)-1-(1-(2-(pyrrolidin-1...)
Affinity DataKi:  2.80nMAssay Description:Displacement of [3H]GW803430 from MCH-1 receptor expressed in CHO-K1 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanin-concentrating hormone receptor 1(Homo sapiens (Human))
Amri

Curated by ChEMBL
LigandPNGBDBM50241083(6-(4-chlorophenyl)-3-(3-methoxy-4-(2-(pyrrolidin-1...)
Affinity DataKi:  2.80nMAssay Description:Displacement of [3H]GW803430 from MCH-1 receptor expressed in CHO-K1 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
Boots Pharmaceuticals

Curated by PDSP Ki Database
LigandPNGBDBM82217(CHEMBL284994 | CP-52003 | SERTRALINE | [4-(3,4-Dic...)
Affinity DataKi:  2.80nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanin-concentrating hormone receptor 1(Homo sapiens (Human))
Amri

Curated by ChEMBL
LigandPNGBDBM50331251((R)-4-(benzyloxy)-1-(1-(2-(2-(hydroxymethyl)pyrrol...)
Affinity DataKi:  3.10nMAssay Description:Displacement of [3H]4-(benzyloxy)-1-(1-(2-(pyrrolidin-1-yl)ethyl)-1H-indazol-5-yl)pyridin-2(1H)-one from MCH-1 receptor expressed in CHO-K1 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
Boots Pharmaceuticals

Curated by PDSP Ki Database
LigandPNGBDBM50254790((S)-Norfluoxetine | CHEMBL465123 | NORFLUOXETINE)
Affinity DataKi:  3.15nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanin-concentrating hormone receptor 1(Homo sapiens (Human))
Amri

Curated by ChEMBL
LigandPNGBDBM50331170(4-(2,4-dichlorophenyl)-1-(1-(2-(pyrrolidin-1-yl)et...)
Affinity DataKi:  3.40nMAssay Description:Displacement of [3H]GW803430 from MCH-1 receptor expressed in CHO-K1 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
Boots Pharmaceuticals

Curated by PDSP Ki Database
LigandPNGBDBM25870(1-[3-(dimethylamino)propyl]-1-(4-fluorophenyl)-1,3...)
Affinity DataKi:  3.51nMMore data for this Ligand-Target Pair
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
Boots Pharmaceuticals

Curated by PDSP Ki Database
LigandPNGBDBM50028091((1E)-5-methoxy-1-[4-(trifluoromethyl)phenyl]pentan...)
Affinity DataKi:  3.57nMMore data for this Ligand-Target Pair
TargetMelanin-concentrating hormone receptor 1(Homo sapiens (Human))
Amri

Curated by ChEMBL
LigandPNGBDBM50331212(4-(benzyloxy)-1-(2-(2-hydroxyethyl)-5-methyl-2,3,4...)
Affinity DataKi:  3.60nMAssay Description:Displacement of [3H]4-(benzyloxy)-1-(1-(2-(pyrrolidin-1-yl)ethyl)-1H-indazol-5-yl)pyridin-2(1H)-one from MCH-1 receptor expressed in CHO-K1 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanin-concentrating hormone receptor 1(Homo sapiens (Human))
Amri

Curated by ChEMBL
LigandPNGBDBM50331187(4-(benzyloxy)-1-(2,3,4,5-tetrahydro-1H-pyrido[4,3-...)
Affinity DataKi:  3.80nMAssay Description:Displacement of [3H]4-(benzyloxy)-1-(1-(2-(pyrrolidin-1-yl)ethyl)-1H-indazol-5-yl)pyridin-2(1H)-one from MCH-1 receptor expressed in CHO-K1 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanin-concentrating hormone receptor 1(Homo sapiens (Human))
Amri

Curated by ChEMBL
LigandPNGBDBM50331174(4-(2-methyl-4-(trifluoromethoxy)phenyl)-1-(1-(2-(p...)
Affinity DataKi:  3.90nMAssay Description:Displacement of [3H]GW803430 from MCH-1 receptor expressed in CHO-K1 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
Boots Pharmaceuticals

Curated by PDSP Ki Database
LigandPNGBDBM50028091((1E)-5-methoxy-1-[4-(trifluoromethyl)phenyl]pentan...)
Affinity DataKi:  4.17nMMore data for this Ligand-Target Pair
TargetMelanin-concentrating hormone receptor 1(Homo sapiens (Human))
Amri

Curated by ChEMBL
LigandPNGBDBM50331200(1-(5-methyl-2,3,4,5-tetrahydro-1H-pyrido[4,3-b]ind...)
Affinity DataKi:  4.20nMAssay Description:Displacement of [3H]4-(benzyloxy)-1-(1-(2-(pyrrolidin-1-yl)ethyl)-1H-indazol-5-yl)pyridin-2(1H)-one from MCH-1 receptor expressed in CHO-K1 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanin-concentrating hormone receptor 1(Homo sapiens (Human))
Amri

Curated by ChEMBL
LigandPNGBDBM50331209(4-(4-chlorobenzyloxy)-1-(5-methyl-2,3,4,5-tetrahyd...)
Affinity DataKi:  4.20nMAssay Description:Displacement of [3H]4-(benzyloxy)-1-(1-(2-(pyrrolidin-1-yl)ethyl)-1H-indazol-5-yl)pyridin-2(1H)-one from MCH-1 receptor expressed in CHO-K1 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanin-concentrating hormone receptor 1(Homo sapiens (Human))
Amri

Curated by ChEMBL
LigandPNGBDBM50331242(2-(4-chloro-2-fluorophenyl)-5-(1-(2-(pyrrolidin-1-...)
Affinity DataKi:  4.20nMAssay Description:Displacement of [3H]4-(benzyloxy)-1-(1-(2-(pyrrolidin-1-yl)ethyl)-1H-indazol-5-yl)pyridin-2(1H)-one from MCH-1 receptor expressed in CHO-K1 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanin-concentrating hormone receptor 1(Homo sapiens (Human))
Amri

Curated by ChEMBL
LigandPNGBDBM50331186(4-(benzyloxy)-1-(2,5-dimethyl-2,3,4,5-tetrahydro-1...)
Affinity DataKi:  4.5nMAssay Description:Displacement of [3H]4-(benzyloxy)-1-(1-(2-(pyrrolidin-1-yl)ethyl)-1H-indazol-5-yl)pyridin-2(1H)-one from MCH-1 receptor expressed in CHO-K1 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanin-concentrating hormone receptor 1(Homo sapiens (Human))
Amri

Curated by ChEMBL
LigandPNGBDBM50331234((S)-4-(benzyloxy)-1-(1-(2-(3-hydroxypyrrolidin-1-y...)
Affinity DataKi:  4.70nMAssay Description:Displacement of [3H]4-(benzyloxy)-1-(1-(2-(pyrrolidin-1-yl)ethyl)-1H-indazol-5-yl)pyridin-2(1H)-one from MCH-1 receptor expressed in CHO-K1 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanin-concentrating hormone receptor 1(Homo sapiens (Human))
Amri

Curated by ChEMBL
LigandPNGBDBM50331245(4-(benzyloxy)-1-(1-(2-(dimethylamino)ethyl)-1H-ind...)
Affinity DataKi:  4.70nMAssay Description:Displacement of [3H]4-(benzyloxy)-1-(1-(2-(pyrrolidin-1-yl)ethyl)-1H-indazol-5-yl)pyridin-2(1H)-one from MCH-1 receptor expressed in CHO-K1 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanin-concentrating hormone receptor 1(Homo sapiens (Human))
Amri

Curated by ChEMBL
LigandPNGBDBM50331185(4-(benzyloxy)-1-(9-methyl-2,3,4,9-tetrahydro-1H-py...)
Affinity DataKi:  4.90nMAssay Description:Displacement of [3H]4-(benzyloxy)-1-(1-(2-(pyrrolidin-1-yl)ethyl)-1H-indazol-5-yl)pyridin-2(1H)-one from MCH-1 receptor expressed in CHO-K1 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanin-concentrating hormone receptor 1(Homo sapiens (Human))
Amri

Curated by ChEMBL
LigandPNGBDBM50331168(1-(1-(2-(pyrrolidin-1-yl)ethyl)-1H-indazol-5-yl)-4...)
Affinity DataKi:  5nMAssay Description:Displacement of [3H]GW803430 from MCH-1 receptor expressed in CHO-K1 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanin-concentrating hormone receptor 1(Homo sapiens (Human))
Amri

Curated by ChEMBL
LigandPNGBDBM50331236(2-(4-chlorophenyl)-5-(1-(2-(pyrrolidin-1-yl)ethyl)...)
Affinity DataKi:  5.20nMAssay Description:Displacement of [3H]4-(benzyloxy)-1-(1-(2-(pyrrolidin-1-yl)ethyl)-1H-indazol-5-yl)pyridin-2(1H)-one from MCH-1 receptor expressed in CHO-K1 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanin-concentrating hormone receptor 1(Homo sapiens (Human))
Amri

Curated by ChEMBL
LigandPNGBDBM50331184(4-(benzyloxy)-1-(2,9-dimethyl-2,3,4,9-tetrahydro-1...)
Affinity DataKi:  5.20nMAssay Description:Displacement of [3H]4-(benzyloxy)-1-(1-(2-(pyrrolidin-1-yl)ethyl)-1H-indazol-5-yl)pyridin-2(1H)-one from MCH-1 receptor expressed in CHO-K1 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanin-concentrating hormone receptor 1(Homo sapiens (Human))
Amri

Curated by ChEMBL
LigandPNGBDBM50331196(4-(4-chlorophenyl)-1-(2,9-dimethyl-2,3,4,9-tetrahy...)
Affinity DataKi:  5.60nMAssay Description:Displacement of [3H]4-(benzyloxy)-1-(1-(2-(pyrrolidin-1-yl)ethyl)-1H-indazol-5-yl)pyridin-2(1H)-one from MCH-1 receptor expressed in CHO-K1 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanin-concentrating hormone receptor 1(Homo sapiens (Human))
Amri

Curated by ChEMBL
LigandPNGBDBM50331171(4-(2-chloro-4-(trifluoromethyl)phenyl)-1-(1-(2-(py...)
Affinity DataKi:  5.80nMAssay Description:Displacement of [3H]GW803430 from MCH-1 receptor expressed in CHO-K1 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
Boots Pharmaceuticals

Curated by PDSP Ki Database
LigandPNGBDBM77970(3-(2-chloranyl-5,6-dihydrobenzo[b][1]benzazepin-11...)
Affinity DataKi:  5.80nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanin-concentrating hormone receptor 1(Homo sapiens (Human))
Amri

Curated by ChEMBL
LigandPNGBDBM50331239(2-(4-fluorophenyl)-5-(1-(2-(pyrrolidin-1-yl)ethyl)...)
Affinity DataKi:  6.10nMAssay Description:Displacement of [3H]4-(benzyloxy)-1-(1-(2-(pyrrolidin-1-yl)ethyl)-1H-indazol-5-yl)pyridin-2(1H)-one from MCH-1 receptor expressed in CHO-K1 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanin-concentrating hormone receptor 1(Homo sapiens (Human))
Amri

Curated by ChEMBL
LigandPNGBDBM50331210(1-(5-methyl-2,3,4,5-tetrahydro-1H-pyrido[4,3-b]ind...)
Affinity DataKi:  6.70nMAssay Description:Displacement of [3H]4-(benzyloxy)-1-(1-(2-(pyrrolidin-1-yl)ethyl)-1H-indazol-5-yl)pyridin-2(1H)-one from MCH-1 receptor expressed in CHO-K1 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanin-concentrating hormone receptor 1(Homo sapiens (Human))
Amri

Curated by ChEMBL
LigandPNGBDBM50331206(4-(4-chloro-2-methoxyphenyl)-1-(5-methyl-2,3,4,5-t...)
Affinity DataKi:  7nMAssay Description:Displacement of [3H]4-(benzyloxy)-1-(1-(2-(pyrrolidin-1-yl)ethyl)-1H-indazol-5-yl)pyridin-2(1H)-one from MCH-1 receptor expressed in CHO-K1 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanin-concentrating hormone receptor 1(Homo sapiens (Human))
Amri

Curated by ChEMBL
LigandPNGBDBM50331197(4-(2,4-dichlorophenyl)-1-(5-methyl-2,3,4,5-tetrahy...)
Affinity DataKi:  7.20nMAssay Description:Displacement of [3H]4-(benzyloxy)-1-(1-(2-(pyrrolidin-1-yl)ethyl)-1H-indazol-5-yl)pyridin-2(1H)-one from MCH-1 receptor expressed in CHO-K1 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanin-concentrating hormone receptor 1(Homo sapiens (Human))
Amri

Curated by ChEMBL
LigandPNGBDBM50331205(4-(4-methoxy-2-methylphenyl)-1-(5-methyl-2,3,4,5-t...)
Affinity DataKi:  7.60nMAssay Description:Displacement of [3H]4-(benzyloxy)-1-(1-(2-(pyrrolidin-1-yl)ethyl)-1H-indazol-5-yl)pyridin-2(1H)-one from MCH-1 receptor expressed in CHO-K1 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanin-concentrating hormone receptor 1(Homo sapiens (Human))
Amri

Curated by ChEMBL
LigandPNGBDBM50331203(4-(4-chlorobenzyloxy)-1-(2,9-dimethyl-2,3,4,9-tetr...)
Affinity DataKi:  7.60nMAssay Description:Displacement of [3H]4-(benzyloxy)-1-(1-(2-(pyrrolidin-1-yl)ethyl)-1H-indazol-5-yl)pyridin-2(1H)-one from MCH-1 receptor expressed in CHO-K1 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanin-concentrating hormone receptor 1(Homo sapiens (Human))
Amri

Curated by ChEMBL
LigandPNGBDBM50331207(1-(2,5-dimethyl-2,3,4,5-tetrahydro-1H-pyrido[4,3-b...)
Affinity DataKi:  7.80nMAssay Description:Displacement of [3H]4-(benzyloxy)-1-(1-(2-(pyrrolidin-1-yl)ethyl)-1H-indazol-5-yl)pyridin-2(1H)-one from MCH-1 receptor expressed in CHO-K1 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanin-concentrating hormone receptor 1(Homo sapiens (Human))
Amri

Curated by ChEMBL
LigandPNGBDBM50331193(1-(9-methyl-2,3,4,9-tetrahydro-1H-pyrido[3,4-b]ind...)
Affinity DataKi:  8.40nMAssay Description:Displacement of [3H]4-(benzyloxy)-1-(1-(2-(pyrrolidin-1-yl)ethyl)-1H-indazol-5-yl)pyridin-2(1H)-one from MCH-1 receptor expressed in CHO-K1 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanin-concentrating hormone receptor 1(Homo sapiens (Human))
Amri

Curated by ChEMBL
LigandPNGBDBM50331248((S)-4-(benzyloxy)-1-(1-(2-(3-methoxypyrrolidin-1-y...)
Affinity DataKi:  9.40nMAssay Description:Displacement of [3H]4-(benzyloxy)-1-(1-(2-(pyrrolidin-1-yl)ethyl)-1H-indazol-5-yl)pyridin-2(1H)-one from MCH-1 receptor expressed in CHO-K1 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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