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Found 73 with Last Name = 'choo' and Initial = 'ih'
Target5-hydroxytryptamine receptor 7(Homo sapiens (Human))
Yonsei University

Curated by ChEMBL
LigandPNGBDBM50098551((R)-3-(2-(2-(4-methylpiperidin-1-yl)ethyl)pyrrolid...)
Affinity DataKi:  0.340nMAssay Description:Displacement of [3H]LSD from 5-HT7R (unknown origin) expressed in CHO-K1 cells by liquid scintillation counting methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 1B(Homo sapiens (Human))
Yonsei University

Curated by ChEMBL
LigandPNGBDBM50058069(CHEMBL3326993)
Affinity DataKi:  7nMAssay Description:Binding affinity to 5-HT1B (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 7(Homo sapiens (Human))
Yonsei University

Curated by ChEMBL
LigandPNGBDBM50058214(CHEMBL3326982)
Affinity DataKi:  8.70nMAssay Description:Displacement of [3H]LSD from 5-HT7R (unknown origin) expressed in CHO-K1 cells by liquid scintillation counting methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 1A(Homo sapiens (Human))
Yonsei University

Curated by ChEMBL
LigandPNGBDBM50058069(CHEMBL3326993)
Affinity DataKi:  11nMAssay Description:Binding affinity to 5-HT1A (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 7(Homo sapiens (Human))
Yonsei University

Curated by ChEMBL
LigandPNGBDBM50058069(CHEMBL3326993)
Affinity DataKi:  16nMAssay Description:Displacement of [3H]LSD from 5-HT7R (unknown origin) expressed in CHO-K1 cells by liquid scintillation counting methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 1A(Homo sapiens (Human))
Yonsei University

Curated by ChEMBL
LigandPNGBDBM50058214(CHEMBL3326982)
Affinity DataKi:  20nMAssay Description:Binding affinity to 5-HT1A (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 7(Homo sapiens (Human))
Yonsei University

Curated by ChEMBL
LigandPNGBDBM50058162(CHEMBL3326986)
Affinity DataKi:  22nMAssay Description:Displacement of [3H]LSD from 5-HT7R (unknown origin) expressed in CHO-K1 cells by liquid scintillation counting methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 7(Homo sapiens (Human))
Yonsei University

Curated by ChEMBL
LigandPNGBDBM50058156(CHEMBL3326989)
Affinity DataKi:  26nMAssay Description:Displacement of [3H]LSD from 5-HT7R (unknown origin) expressed in CHO-K1 cells by liquid scintillation counting methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 7(Homo sapiens (Human))
Yonsei University

Curated by ChEMBL
LigandPNGBDBM50058211(CHEMBL3326984)
Affinity DataKi:  26nMAssay Description:Displacement of [3H]LSD from 5-HT7R (unknown origin) expressed in CHO-K1 cells by liquid scintillation counting methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2C(Homo sapiens (Human))
Yonsei University

Curated by ChEMBL
LigandPNGBDBM50058214(CHEMBL3326982)
Affinity DataKi:  26nMAssay Description:Binding affinity to 5-HT2C (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 7(Homo sapiens (Human))
Yonsei University

Curated by ChEMBL
LigandPNGBDBM50058209(CHEMBL3326985)
Affinity DataKi:  31nMAssay Description:Displacement of [3H]LSD from 5-HT7R (unknown origin) expressed in CHO-K1 cells by liquid scintillation counting methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 7(Homo sapiens (Human))
Yonsei University

Curated by ChEMBL
LigandPNGBDBM50058157(CHEMBL3326988)
Affinity DataKi:  32nMAssay Description:Displacement of [3H]LSD from 5-HT7R (unknown origin) expressed in CHO-K1 cells by liquid scintillation counting methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 7(Homo sapiens (Human))
Yonsei University

Curated by ChEMBL
LigandPNGBDBM50058216(CHEMBL3326980)
Affinity DataKi:  35nMAssay Description:Displacement of [3H]LSD from 5-HT7R (unknown origin) expressed in CHO-K1 cells by liquid scintillation counting methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 7(Homo sapiens (Human))
Yonsei University

Curated by ChEMBL
LigandPNGBDBM50058215(CHEMBL3326981)
Affinity DataKi:  35nMAssay Description:Displacement of [3H]LSD from 5-HT7R (unknown origin) expressed in CHO-K1 cells by liquid scintillation counting methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 7(Homo sapiens (Human))
Yonsei University

Curated by ChEMBL
LigandPNGBDBM50058217(CHEMBL3326979)
Affinity DataKi:  37nMAssay Description:Displacement of [3H]LSD from 5-HT7R (unknown origin) expressed in CHO-K1 cells by liquid scintillation counting methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 7(Homo sapiens (Human))
Yonsei University

Curated by ChEMBL
LigandPNGBDBM50058219(CHEMBL3325464)
Affinity DataKi:  38nMAssay Description:Displacement of [3H]LSD from 5-HT7R (unknown origin) expressed in CHO-K1 cells by liquid scintillation counting methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 7(Homo sapiens (Human))
Yonsei University

Curated by ChEMBL
LigandPNGBDBM50058218(CHEMBL3326978)
Affinity DataKi:  44nMAssay Description:Displacement of [3H]LSD from 5-HT7R (unknown origin) expressed in CHO-K1 cells by liquid scintillation counting methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 7(Homo sapiens (Human))
Yonsei University

Curated by ChEMBL
LigandPNGBDBM50058159(CHEMBL3326987)
Affinity DataKi:  44nMAssay Description:Displacement of [3H]LSD from 5-HT7R (unknown origin) expressed in CHO-K1 cells by liquid scintillation counting methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 7(Homo sapiens (Human))
Yonsei University

Curated by ChEMBL
LigandPNGBDBM50058070(CHEMBL3326992)
Affinity DataKi:  47nMAssay Description:Displacement of [3H]LSD from 5-HT7R (unknown origin) expressed in CHO-K1 cells by liquid scintillation counting methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 7(Homo sapiens (Human))
Yonsei University

Curated by ChEMBL
LigandPNGBDBM50058151(CHEMBL3326990)
Affinity DataKi:  48nMAssay Description:Displacement of [3H]LSD from 5-HT7R (unknown origin) expressed in CHO-K1 cells by liquid scintillation counting methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 7(Homo sapiens (Human))
Yonsei University

Curated by ChEMBL
LigandPNGBDBM50058282(CHEMBL3326977)
Affinity DataKi:  65nMAssay Description:Displacement of [3H]LSD from 5-HT7R (unknown origin) expressed in CHO-K1 cells by liquid scintillation counting methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 7(Homo sapiens (Human))
Yonsei University

Curated by ChEMBL
LigandPNGBDBM50058071(CHEMBL3326991)
Affinity DataKi:  66nMAssay Description:Displacement of [3H]LSD from 5-HT7R (unknown origin) expressed in CHO-K1 cells by liquid scintillation counting methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2C(Homo sapiens (Human))
Yonsei University

Curated by ChEMBL
LigandPNGBDBM50058069(CHEMBL3326993)
Affinity DataKi:  70nMAssay Description:Binding affinity to 5-HT2C (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2A(Homo sapiens (Human))
Yonsei University

Curated by ChEMBL
LigandPNGBDBM50058069(CHEMBL3326993)
Affinity DataKi:  77nMAssay Description:Binding affinity to 5-HT2A (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 1D(Homo sapiens (Human))
Yonsei University

Curated by ChEMBL
LigandPNGBDBM50058069(CHEMBL3326993)
Affinity DataKi:  122nMAssay Description:Binding affinity to 5-HT1D (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 1B(Homo sapiens (Human))
Yonsei University

Curated by ChEMBL
LigandPNGBDBM50058214(CHEMBL3326982)
Affinity DataKi:  131nMAssay Description:Binding affinity to 5-HT1B (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 7(Homo sapiens (Human))
Yonsei University

Curated by ChEMBL
LigandPNGBDBM50058284(CHEMBL3326976)
Affinity DataKi:  187nMAssay Description:Displacement of [3H]LSD from 5-HT7R (unknown origin) expressed in CHO-K1 cells by liquid scintillation counting methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 7(Homo sapiens (Human))
Yonsei University

Curated by ChEMBL
LigandPNGBDBM50058213(CHEMBL3326983)
Affinity DataKi:  405nMAssay Description:Displacement of [3H]LSD from 5-HT7R (unknown origin) expressed in CHO-K1 cells by liquid scintillation counting methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 1D(Homo sapiens (Human))
Yonsei University

Curated by ChEMBL
LigandPNGBDBM50058214(CHEMBL3326982)
Affinity DataKi:  418nMAssay Description:Binding affinity to 5-HT1D (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2A(Homo sapiens (Human))
Yonsei University

Curated by ChEMBL
LigandPNGBDBM50058214(CHEMBL3326982)
Affinity DataKi:  478nMAssay Description:Binding affinity to 5-HT2A (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 5A(Homo sapiens (Human))
Yonsei University

Curated by ChEMBL
LigandPNGBDBM50058069(CHEMBL3326993)
Affinity DataKi:  517nMAssay Description:Binding affinity to 5-HT5A (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 5A(Homo sapiens (Human))
Yonsei University

Curated by ChEMBL
LigandPNGBDBM50058214(CHEMBL3326982)
Affinity DataKi:  1.18E+3nMAssay Description:Binding affinity to 5-HT5A (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 6(Homo sapiens (Human))
Yonsei University

Curated by ChEMBL
LigandPNGBDBM50058069(CHEMBL3326993)
Affinity DataKi:  1.32E+3nMAssay Description:Binding affinity to 5-HT6 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 6(Homo sapiens (Human))
Yonsei University

Curated by ChEMBL
LigandPNGBDBM50058214(CHEMBL3326982)
Affinity DataKi:  1.52E+3nMAssay Description:Binding affinity to 5-HT6 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 3A(Homo sapiens (Human))
Yonsei University

Curated by ChEMBL
LigandPNGBDBM50058214(CHEMBL3326982)
Affinity DataKi: >1.00E+4nMAssay Description:Binding affinity to 5-HT3 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 3A(Homo sapiens (Human))
Yonsei University

Curated by ChEMBL
LigandPNGBDBM50058069(CHEMBL3326993)
Affinity DataKi: >1.00E+4nMAssay Description:Binding affinity to 5-HT3 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] B(Homo sapiens (Human))
Korea Institute Of Science And Technology

Curated by ChEMBL
LigandPNGBDBM15579(CHEMBL972 | DEPRENYL | L-Deprenyl | N-methyl-N-[(2...)
Affinity DataIC50:  1.30nMAssay Description:Inhibition of human recombinant MAO-B using benzylamine hydrochloride as substrate assessed as H2O2 synthesis after 1 hr by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMetabotropic glutamate receptor 1(Homo sapiens (Human))
Yonsei University

Curated by ChEMBL
LigandPNGBDBM50345949(3-(4-Methoxy-phenyl)-9-prop-2-ynylamino-3H-pyrido[...)
Affinity DataIC50:  6.70nMAssay Description:Antagonist activity at mGluR1 (unknown origin) expressed in Chem-3 cells assessed as inhibition of glutamate-induced increased intracellular calcium ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] B(Homo sapiens (Human))
Korea Institute Of Science And Technology

Curated by ChEMBL
LigandPNGBDBM50493222(CHEMBL2418211)
Affinity DataIC50:  27nMAssay Description:Inhibition of human recombinant MAO-B using benzylamine hydrochloride as substrate assessed as H2O2 synthesis after 1 hr by fluorescence assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetMetabotropic glutamate receptor 1(Homo sapiens (Human))
Yonsei University

Curated by ChEMBL
LigandPNGBDBM50058042(CHEMBL3330823)
Affinity DataIC50:  45nMAssay Description:Antagonist activity at mGluR1 (unknown origin) expressed in Chem-3 cells assessed as inhibition of glutamate-induced increased intracellular calcium ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMetabotropic glutamate receptor 1(Homo sapiens (Human))
Yonsei University

Curated by ChEMBL
LigandPNGBDBM50058048(CHEMBL3330811)
Affinity DataIC50:  50nMAssay Description:Antagonist activity at mGluR1 (unknown origin) expressed in Chem-3 cells assessed as inhibition of glutamate-induced increased intracellular calcium ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMetabotropic glutamate receptor 1(Homo sapiens (Human))
Yonsei University

Curated by ChEMBL
LigandPNGBDBM50058044(CHEMBL3330817)
Affinity DataIC50:  57nMAssay Description:Antagonist activity at mGluR1 (unknown origin) expressed in Chem-3 cells assessed as inhibition of glutamate-induced increased intracellular calcium ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMetabotropic glutamate receptor 1(Homo sapiens (Human))
Yonsei University

Curated by ChEMBL
LigandPNGBDBM50058056(CHEMBL3330801)
Affinity DataIC50:  58nMAssay Description:Antagonist activity at mGluR1 (unknown origin) expressed in Chem-3 cells assessed as inhibition of glutamate-induced increased intracellular calcium ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMetabotropic glutamate receptor 1(Homo sapiens (Human))
Yonsei University

Curated by ChEMBL
LigandPNGBDBM50058055(CHEMBL3330802)
Affinity DataIC50:  66nMAssay Description:Antagonist activity at mGluR1 (unknown origin) expressed in Chem-3 cells assessed as inhibition of glutamate-induced increased intracellular calcium ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMetabotropic glutamate receptor 1(Homo sapiens (Human))
Yonsei University

Curated by ChEMBL
LigandPNGBDBM50058047(CHEMBL3330812 | US9260448, 29)
Affinity DataIC50:  74nMAssay Description:Antagonist activity at mGluR1 (unknown origin) expressed in Chem-3 cells assessed as inhibition of glutamate-induced increased intracellular calcium ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMetabotropic glutamate receptor 1(Homo sapiens (Human))
Yonsei University

Curated by ChEMBL
LigandPNGBDBM50058049(CHEMBL3330808 | US9260448, 18)
Affinity DataIC50:  112nMAssay Description:Antagonist activity at mGluR1 (unknown origin) expressed in Chem-3 cells assessed as inhibition of glutamate-induced increased intracellular calcium ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMetabotropic glutamate receptor 1(Homo sapiens (Human))
Yonsei University

Curated by ChEMBL
LigandPNGBDBM50058045(CHEMBL3330813)
Affinity DataIC50:  128nMAssay Description:Antagonist activity at mGluR1 (unknown origin) expressed in Chem-3 cells assessed as inhibition of glutamate-induced increased intracellular calcium ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMetabotropic glutamate receptor 1(Homo sapiens (Human))
Yonsei University

Curated by ChEMBL
LigandPNGBDBM50058059(CHEMBL3330800)
Affinity DataIC50:  136nMAssay Description:Antagonist activity at mGluR1 (unknown origin) expressed in Chem-3 cells assessed as inhibition of glutamate-induced increased intracellular calcium ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMetabotropic glutamate receptor 1(Homo sapiens (Human))
Yonsei University

Curated by ChEMBL
LigandPNGBDBM50058052(CHEMBL3330805 | US9260448, 7)
Affinity DataIC50:  162nMAssay Description:Antagonist activity at mGluR1 (unknown origin) expressed in Chem-3 cells assessed as inhibition of glutamate-induced increased intracellular calcium ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] B(Homo sapiens (Human))
Korea Institute Of Science And Technology

Curated by ChEMBL
LigandPNGBDBM50493221(CHEMBL2418212)
Affinity DataIC50:  171nMAssay Description:Inhibition of human recombinant MAO-B using benzylamine hydrochloride as substrate assessed as H2O2 synthesis after 1 hr by fluorescence assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
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