Compile Data Set for Download or QSAR
maximum 50k data
Found 286 with Last Name = 'cirillo' and Initial = 'r'
TargetOxytocin receptor(Homo sapiens (Human))
Lcg Bioscience

Curated by PDSP Ki Database
LigandPNGBDBM86210(CAS_50-56-6 | NSC_439302 | Oxytocin)
Affinity DataKi:  0.5nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOxytocin receptor(Homo sapiens (Human))
Lcg Bioscience

Curated by PDSP Ki Database
LigandPNGBDBM50326722((Z)-3-(4-(N-(4-chlorophenyl)-N-(2-oxo-2-(2-(2-oxoi...)
Affinity DataKi:  0.650nMAssay Description:Displacement of [125I]OVTA antagonist from human oxytocin receptor expressed in HEK293-EBNA cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOxytocin receptor(RAT)
Serono Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50326722((Z)-3-(4-(N-(4-chlorophenyl)-N-(2-oxo-2-(2-(2-oxoi...)
Affinity DataKi:  0.670nMAssay Description:Displacement of [125I]OVTA antagonist from rat oxytocin receptor expressed in HEK293-EBNA cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOxytocin receptor(Homo sapiens (Human))
Lcg Bioscience

Curated by PDSP Ki Database
LigandPNGBDBM86210(CAS_50-56-6 | NSC_439302 | Oxytocin)
Affinity DataKi:  0.710nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOxytocin receptor(Homo sapiens (Human))
Lcg Bioscience

Curated by PDSP Ki Database
LigandPNGBDBM50410616(CHEMBL2113185)
Affinity DataKi:  0.900nMAssay Description:Displacement of [125I]OVTA antagonist from human oxytocin receptor expressed in HEK293-EBNA cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOxytocin receptor(Homo sapiens (Human))
Lcg Bioscience

Curated by PDSP Ki Database
LigandPNGBDBM50410618(CHEMBL2113181)
Affinity DataKi:  0.900nMAssay Description:Displacement of [125I]OVTA antagonist from human oxytocin receptor expressed in HEK293-EBNA cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOxytocin receptor(Homo sapiens (Human))
Lcg Bioscience

Curated by PDSP Ki Database
LigandPNGBDBM50410625(CHEMBL2113201)
Affinity DataKi:  1.10nMAssay Description:Displacement of [125I]OVTA antagonist from human oxytocin receptor expressed in HEK293-EBNA cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOxytocin receptor(Homo sapiens (Human))
Lcg Bioscience

Curated by PDSP Ki Database
LigandPNGBDBM50410634(CHEMBL2113189)
Affinity DataKi:  1.60nMAssay Description:Displacement of [125I]OVTA antagonist from human oxytocin receptor expressed in HEK293-EBNA cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOxytocin receptor(RAT)
Serono Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM86210(CAS_50-56-6 | NSC_439302 | Oxytocin)
Affinity DataKi:  1.90nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOxytocin receptor(Homo sapiens (Human))
Lcg Bioscience

Curated by PDSP Ki Database
LigandPNGBDBM50410622(CHEMBL2113203)
Affinity DataKi:  2.10nMAssay Description:Displacement of [125I]OVTA antagonist from human oxytocin receptor expressed in HEK293-EBNA cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetType-1 angiotensin II receptor A/B(RAT)
Laboratori Guidotti

Curated by ChEMBL
LigandPNGBDBM50470323(CHEMBL327505)
Affinity DataKi:  2.5nMAssay Description:Inhibition of [3H]angiotensin II binding to rat adrenal cortex membrane containing angiotensin II receptor, type 1More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetOxytocin receptor(RAT)
Serono Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50410634(CHEMBL2113189)
Affinity DataKi:  2.70nMAssay Description:Displacement of [125I]OVTA antagonist from rat oxytocin receptor expressed in HEK293-EBNA cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOxytocin receptor(Homo sapiens (Human))
Lcg Bioscience

Curated by PDSP Ki Database
LigandPNGBDBM50410619(CHEMBL2113208)
Affinity DataKi:  3nMAssay Description:Displacement of [125I]OVTA antagonist from human oxytocin receptor expressed in HEK293-EBNA cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V1a receptor(Homo sapiens (Human))
Lcg Bioscience

Curated by PDSP Ki Database
LigandPNGBDBM86209(Atosiban | CAS_90779-69-4 | NSC_0)
Affinity DataKi:  3.5nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOxytocin receptor(Homo sapiens (Human))
Lcg Bioscience

Curated by PDSP Ki Database
LigandPNGBDBM50410640(CHEMBL2113198)
Affinity DataKi:  3.90nMAssay Description:Displacement of [125I]OVTA antagonist from human oxytocin receptor expressed in HEK293-EBNA cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetType-1 angiotensin II receptor(Bos taurus)
Istituto Lusofarmaco

Curated by ChEMBL
LigandPNGBDBM50029893(2-[4-Butyl-5-(2'-carboxy-biphenyl-4-ylmethyl)-2-me...)
Affinity DataKi: >4nMAssay Description:Binding affinity towards Angiotensin II type 2 receptor in bovine cerebellar cortical membranes; InactiveMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetType-1 angiotensin II receptor(Bos taurus)
Istituto Lusofarmaco

Curated by ChEMBL
LigandPNGBDBM50029903(3-Benzyl-6-butyl-2-methyl-5-[2'-(1H-tetrazol-5-yl)...)
Affinity DataKi: >4nMAssay Description:Binding affinity towards Angiotensin II type 2 receptor in bovine cerebellar cortical membranes; InactiveMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetType-1 angiotensin II receptor(Bos taurus)
Istituto Lusofarmaco

Curated by ChEMBL
LigandPNGBDBM50029911(2-{4-Butyl-2-methyl-6-oxo-5-[2'-(1H-tetrazol-5-yl)...)
Affinity DataKi: >4nMAssay Description:Binding affinity towards Angiotensin II type 2 receptor in bovine cerebellar cortical membranes; InactiveMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetType-1 angiotensin II receptor(Bos taurus)
Istituto Lusofarmaco

Curated by ChEMBL
LigandPNGBDBM50029910(4'-(4-Butyl-6-oxo-1,6-dihydro-pyrimidin-5-ylmethyl...)
Affinity DataKi: >4nMAssay Description:Binding affinity towards Angiotensin II type 2 receptor in bovine cerebellar cortical membranes; InactiveMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetType-1 angiotensin II receptor(Bos taurus)
Istituto Lusofarmaco

Curated by ChEMBL
LigandPNGBDBM50029907(4'-(1-Benzyl-4-butyl-6-oxo-1,6-dihydro-pyrimidin-5...)
Affinity DataKi: >4nMAssay Description:Binding affinity towards Angiotensin II type 2 receptor in bovine cerebellar cortical membranes; InactiveMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetType-1 angiotensin II receptor(Bos taurus)
Istituto Lusofarmaco

Curated by ChEMBL
LigandPNGBDBM50029909(4'-[4-Butyl-1-(2-carboxy-benzyl)-6-oxo-1,6-dihydro...)
Affinity DataKi: >4nMAssay Description:Binding affinity towards Angiotensin II type 2 receptor in bovine cerebellar cortical membranes; InactiveMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetType-1 angiotensin II receptor(Bos taurus)
Istituto Lusofarmaco

Curated by ChEMBL
LigandPNGBDBM50029906(2-[4-Butyl-5-(2'-carboxy-biphenyl-4-ylmethyl)-2-me...)
Affinity DataKi: >4nMAssay Description:Binding affinity towards Angiotensin II type 2 receptor in bovine cerebellar cortical membranes; InactiveMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetType-1 angiotensin II receptor(Bos taurus)
Istituto Lusofarmaco

Curated by ChEMBL
LigandPNGBDBM50029908(4'-(4-Butyl-6-oxo-1-thiophen-2-ylmethyl-1,6-dihydr...)
Affinity DataKi: >4nMAssay Description:Binding affinity towards Angiotensin II type 2 receptor in bovine cerebellar cortical membranes; InactiveMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetType-1 angiotensin II receptor(Bos taurus)
Istituto Lusofarmaco

Curated by ChEMBL
LigandPNGBDBM50029899(3-{4-Butyl-2-methyl-6-oxo-5-[2'-(1H-tetrazol-5-yl)...)
Affinity DataKi: >4nMAssay Description:Binding affinity towards Angiotensin II type 2 receptor in bovine cerebellar cortical membranes; InactiveMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetType-1 angiotensin II receptor(Bos taurus)
Istituto Lusofarmaco

Curated by ChEMBL
LigandPNGBDBM50029905(4'-(2-Butyl-4-methyl-6-oxo-6H-pyrimidin-1-ylmethyl...)
Affinity DataKi: >4nMAssay Description:Binding affinity towards Angiotensin II type 2 receptor in bovine cerebellar cortical membranes; InactiveMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetType-1 angiotensin II receptor(Bos taurus)
Istituto Lusofarmaco

Curated by ChEMBL
LigandPNGBDBM50029895(2-{4-Butyl-2-methyl-6-oxo-5-[2'-(1H-tetrazol-5-yl)...)
Affinity DataKi: >4nMAssay Description:Binding affinity towards Angiotensin II type 2 receptor in bovine cerebellar cortical membranes; InactiveMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetType-1 angiotensin II receptor(Bos taurus)
Istituto Lusofarmaco

Curated by ChEMBL
LigandPNGBDBM50029894(4'-(4-Butyl-2-methyl-6-oxo-1,6-dihydro-pyrimidin-5...)
Affinity DataKi: >4nMAssay Description:Binding affinity towards Angiotensin II type 2 receptor in bovine cerebellar cortical membranes; InactiveMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetType-1 angiotensin II receptor(Bos taurus)
Istituto Lusofarmaco

Curated by ChEMBL
LigandPNGBDBM50029904(4'-[4-Butyl-1-(2-carboxy-benzyl)-2-methyl-6-oxo-1,...)
Affinity DataKi: >4nMAssay Description:Binding affinity towards Angiotensin II type 2 receptor in bovine cerebellar cortical membranes; InactiveMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetType-1 angiotensin II receptor(Bos taurus)
Istituto Lusofarmaco

Curated by ChEMBL
LigandPNGBDBM50029902(6-Butyl-2-methyl-5-[2'-(1H-tetrazol-5-yl)-biphenyl...)
Affinity DataKi: >4nMAssay Description:Binding affinity towards Angiotensin II type 2 receptor in bovine cerebellar cortical membranes; InactiveMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetType-1 angiotensin II receptor(Bos taurus)
Istituto Lusofarmaco

Curated by ChEMBL
LigandPNGBDBM50029897(4'-[4-Butyl-1-(4-carboxy-benzyl)-6-oxo-1,6-dihydro...)
Affinity DataKi: >4nMAssay Description:Binding affinity towards Angiotensin II type 2 receptor in bovine cerebellar cortical membranes; InactiveMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetType-1 angiotensin II receptor(Bos taurus)
Istituto Lusofarmaco

Curated by ChEMBL
LigandPNGBDBM50029901(2-{4-Butyl-2-methyl-6-oxo-5-[2'-(1H-tetrazol-5-yl)...)
Affinity DataKi: >4nMAssay Description:Binding affinity towards Angiotensin II type 2 receptor in bovine cerebellar cortical membranes; InactiveMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetType-1 angiotensin II receptor(Bos taurus)
Istituto Lusofarmaco

Curated by ChEMBL
LigandPNGBDBM50029892(2-{4-Butyl-2-methyl-6-oxo-5-[2'-(1H-tetrazol-5-yl)...)
Affinity DataKi: >4nMAssay Description:Binding affinity towards Angiotensin II type 2 receptor in bovine cerebellar cortical membranes; InactiveMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetType-1 angiotensin II receptor(Bos taurus)
Istituto Lusofarmaco

Curated by ChEMBL
LigandPNGBDBM50241501(6-Butyl-2-methyl-5-[2'-(1H-tetrazol-5-yl)-biphenyl...)
Affinity DataKi: >4nMAssay Description:Binding affinity towards Angiotensin II type 2 receptor in bovine cerebellar cortical membranes; InactiveMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetType-1 angiotensin II receptor(Bos taurus)
Istituto Lusofarmaco

Curated by ChEMBL
LigandPNGBDBM50241491(2-{4-Butyl-2-methyl-6-oxo-5-[2'-(1H-tetrazol-5-yl)...)
Affinity DataKi: >4nMAssay Description:Binding affinity towards Angiotensin II type 2 receptor in bovine cerebellar cortical membranes; InactiveMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetType-1 angiotensin II receptor(Bos taurus)
Istituto Lusofarmaco

Curated by ChEMBL
LigandPNGBDBM50029896(4'-(2-Butyl-6-oxo-6H-pyrimidin-1-ylmethyl)-bipheny...)
Affinity DataKi: >4nMAssay Description:Binding affinity towards Angiotensin II type 2 receptor in bovine cerebellar cortical membranes; InactiveMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOxytocin receptor(Homo sapiens (Human))
Lcg Bioscience

Curated by PDSP Ki Database
LigandPNGBDBM50410623(CHEMBL2113179)
Affinity DataKi:  4.10nMAssay Description:Displacement of [125I]OVTA antagonist from human oxytocin receptor expressed in HEK293-EBNA cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetType-1 angiotensin II receptor A/B(RAT)
Laboratori Guidotti

Curated by ChEMBL
LigandPNGBDBM50470328(CHEMBL317300)
Affinity DataKi:  4.40nMAssay Description:Inhibition of [3H]angiotensin II binding to rat adrenal cortex membrane containing angiotensin II receptor, type 1More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetType-1 angiotensin II receptor A/B(RAT)
Laboratori Guidotti

Curated by ChEMBL
LigandPNGBDBM50470310(CHEMBL98592)
Affinity DataKi:  4.5nMAssay Description:Inhibition of [3H]angiotensin II binding to rat adrenal cortex membrane containing angiotensin II receptor, type 1More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetOxytocin receptor(RAT)
Serono Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50410625(CHEMBL2113201)
Affinity DataKi:  4.60nMAssay Description:Displacement of [125I]OVTA antagonist from rat oxytocin receptor expressed in HEK293-EBNA cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOxytocin receptor(Homo sapiens (Human))
Lcg Bioscience

Curated by PDSP Ki Database
LigandPNGBDBM50410635(CHEMBL2113211)
Affinity DataKi:  7nMAssay Description:Displacement of [125I]OVTA antagonist from human oxytocin receptor expressed in HEK293-EBNA cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOxytocin receptor(Homo sapiens (Human))
Lcg Bioscience

Curated by PDSP Ki Database
LigandPNGBDBM50410621(CHEMBL2113177)
Affinity DataKi:  7nMAssay Description:Displacement of [125I]OVTA antagonist from human oxytocin receptor expressed in HEK293-EBNA cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetType-1 angiotensin II receptor A/B(RAT)
Laboratori Guidotti

Curated by ChEMBL
LigandPNGBDBM50470321(CHEMBL99008)
Affinity DataKi:  7.70nMAssay Description:Inhibition of [3H]angiotensin II binding to rat adrenal cortex membrane containing angiotensin II receptor, type 1More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetOxytocin receptor(RAT)
Serono Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50410616(CHEMBL2113185)
Affinity DataKi:  8nMAssay Description:Displacement of [125I]OVTA antagonist from rat oxytocin receptor expressed in HEK293-EBNA cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOxytocin receptor(Homo sapiens (Human))
Lcg Bioscience

Curated by PDSP Ki Database
LigandPNGBDBM50410638(CHEMBL2113207)
Affinity DataKi:  8.70nMAssay Description:Displacement of [125I]OVTA antagonist from human oxytocin receptor expressed in HEK293-EBNA cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetType-1 angiotensin II receptor A/B(RAT)
Laboratori Guidotti

Curated by ChEMBL
LigandPNGBDBM50470340(CHEMBL98370)
Affinity DataKi:  8.80nMAssay Description:Inhibition of [3H]angiotensin II binding to rat adrenal cortex membrane containing angiotensin II receptor, type 1More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetType-1 angiotensin II receptor A/B(RAT)
Laboratori Guidotti

Curated by ChEMBL
LigandPNGBDBM50470326(CHEMBL319990)
Affinity DataKi:  9.10nMAssay Description:Inhibition of [3H]angiotensin II binding to rat adrenal cortex membrane containing angiotensin II receptor, type 1More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetOxytocin receptor(Homo sapiens (Human))
Lcg Bioscience

Curated by PDSP Ki Database
LigandPNGBDBM50410630(CHEMBL2113209)
Affinity DataKi:  10nMAssay Description:Displacement of [125I]OVTA antagonist from human oxytocin receptor expressed in HEK293-EBNA cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetType-1 angiotensin II receptor A/B(RAT)
Laboratori Guidotti

Curated by ChEMBL
LigandPNGBDBM50470313(CHEMBL441640)
Affinity DataKi:  12nMAssay Description:Inhibition of [3H]angiotensin II binding to rat adrenal cortex membrane containing angiotensin II receptor, type 1More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetType-1 angiotensin II receptor A/B(RAT)
Laboratori Guidotti

Curated by ChEMBL
LigandPNGBDBM50470330(CHEMBL318194)
Affinity DataKi:  12nMAssay Description:Inhibition of [3H]angiotensin II binding to rat adrenal cortex membrane containing angiotensin II receptor, type 1More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetOxytocin receptor(RAT)
Serono Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50410619(CHEMBL2113208)
Affinity DataKi:  12nMAssay Description:Displacement of [125I]OVTA antagonist from rat oxytocin receptor expressed in HEK293-EBNA cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Displayed 1 to 50 (of 286 total ) | Next | Last >>
Jump to: