TargetDNA-dependent protein kinase catalytic subunit(Homo sapiens (Human))
School Of Natural Sciences--Chemistry
Curated by ChEMBL
School Of Natural Sciences--Chemistry
Curated by ChEMBL
Affinity DataKi: 0.650nMAssay Description:Inhibitory activity against DNA-dependent protein kinase receptorMore data for this Ligand-Target Pair
Affinity DataKi: 6nMAssay Description:Evaluated for the binding affinity against thrombinMore data for this Ligand-Target Pair
Affinity DataKi: 6nMAssay Description:Compound was evaluated for its inhibitory activity against ThrombinMore data for this Ligand-Target Pair
Affinity DataKi: 24nMAssay Description:Inhibition of human thrombin (in vitro)More data for this Ligand-Target Pair
Affinity DataKi: 26nMAssay Description:Inhibition of human thrombin (in vitro)More data for this Ligand-Target Pair
Affinity DataKi: 26nMAssay Description:Evaluated for the binding affinity against thrombinMore data for this Ligand-Target Pair
Affinity DataKi: 26nMAssay Description:Compound was evaluated for its inhibitory activity against ThrombinMore data for this Ligand-Target Pair
Affinity DataKi: 27nMAssay Description:Evaluated for the binding affinity against thrombinMore data for this Ligand-Target Pair
Affinity DataKi: 28nMAssay Description:Compound was evaluated for its inhibitory activity against ThrombinMore data for this Ligand-Target Pair
Affinity DataKi: 34nMAssay Description:Evaluated for the binding affinity against thrombinMore data for this Ligand-Target Pair
Affinity DataKi: 34nMAssay Description:Evaluated for the binding affinity against thrombinMore data for this Ligand-Target Pair
Affinity DataKi: 38nMAssay Description:Inhibition of human thrombin (in vitro)More data for this Ligand-Target Pair
Affinity DataKi: 39nMAssay Description:Evaluated for the binding affinity against thrombinMore data for this Ligand-Target Pair
Affinity DataKi: 47nMAssay Description:Evaluated for the binding affinity against thrombinMore data for this Ligand-Target Pair
Affinity DataKi: 52nMAssay Description:Inhibition of human thrombin (in vitro)More data for this Ligand-Target Pair
Affinity DataKi: 56nMAssay Description:Inhibition of human thrombin (in vitro)More data for this Ligand-Target Pair
Affinity DataKi: 57nMAssay Description:Evaluated for the binding affinity against thrombinMore data for this Ligand-Target Pair
Affinity DataKi: 64nMAssay Description:Evaluated for the binding affinity against thrombinMore data for this Ligand-Target Pair
Affinity DataKi: 65nMAssay Description:Inhibition of human thrombin (in vitro)More data for this Ligand-Target Pair
Affinity DataKi: 77nMAssay Description:Evaluated for the binding affinity against thrombinMore data for this Ligand-Target Pair
Affinity DataKi: 79nMAssay Description:Inhibition of human thrombin (in vitro)More data for this Ligand-Target Pair
Affinity DataKi: 82nMAssay Description:Evaluated for the binding affinity against thrombinMore data for this Ligand-Target Pair
Affinity DataKi: 93nMAssay Description:Inhibition of human thrombin (in vitro)More data for this Ligand-Target Pair
Affinity DataKi: 94nMAssay Description:Evaluated for the binding affinity against thrombinMore data for this Ligand-Target Pair
Affinity DataKi: 118nMAssay Description:Compound was evaluated for its inhibitory activity against ThrombinMore data for this Ligand-Target Pair
Affinity DataKi: 118nMAssay Description:Compound was evaluated for its inhibitory activity against ThrombinMore data for this Ligand-Target Pair
Affinity DataKi: 119nMAssay Description:Evaluated for the binding affinity against thrombinMore data for this Ligand-Target Pair
Affinity DataKi: 119nMAssay Description:Inhibition of human thrombin (in vitro)More data for this Ligand-Target Pair
Affinity DataKi: 125nMAssay Description:Evaluated for the binding affinity against thrombinMore data for this Ligand-Target Pair
Affinity DataKi: 126nMAssay Description:Compound was evaluated for its inhibitory activity against ThrombinMore data for this Ligand-Target Pair
Affinity DataKi: 182nMAssay Description:Inhibition of human thrombin (in vitro)More data for this Ligand-Target Pair
Affinity DataKi: 240nMAssay Description:Inhibition of human thrombin (in vitro)More data for this Ligand-Target Pair
Affinity DataKi: 248nMAssay Description:Compound was evaluated for its inhibitory activity against ThrombinMore data for this Ligand-Target Pair
Affinity DataKi: 280nMAssay Description:Compound was evaluated for its inhibitory activity against ThrombinMore data for this Ligand-Target Pair
Affinity DataKi: 350nMAssay Description:Inhibition of human thrombin (in vitro)More data for this Ligand-Target Pair
Affinity DataKi: 359nMAssay Description:Evaluated for the binding affinity against thrombinMore data for this Ligand-Target Pair
Affinity DataKi: 452nMAssay Description:Compound was evaluated for its inhibitory activity against ThrombinMore data for this Ligand-Target Pair
Affinity DataKi: 500nMAssay Description:Evaluated for the binding affinity against thrombinMore data for this Ligand-Target Pair
Affinity DataKi: 654nMAssay Description:Inhibition of human thrombin (in vitro)More data for this Ligand-Target Pair
Affinity DataKi: 723nMAssay Description:Evaluated for the binding affinity against thrombinMore data for this Ligand-Target Pair
Affinity DataKi: 760nMAssay Description:Compound was evaluated for its inhibitory activity against ThrombinMore data for this Ligand-Target Pair
Affinity DataKi: 780nMAssay Description:Compound was evaluated for its inhibitory activity against ThrombinMore data for this Ligand-Target Pair
Affinity DataKi: 810nMAssay Description:Compound was evaluated for its inhibitory activity against ThrombinMore data for this Ligand-Target Pair
Affinity DataKi: 1.00E+3nMAssay Description:Inhibition of human thrombin (in vitro)More data for this Ligand-Target Pair
Affinity DataKi: 1.18E+3nMAssay Description:Inhibition of human thrombin (in vitro)More data for this Ligand-Target Pair
Affinity DataKi: 1.32E+3nMAssay Description:Compound was evaluated for its inhibitory activity against TrypsinMore data for this Ligand-Target Pair
Affinity DataKi: 1.57E+3nMAssay Description:Compound was evaluated for its inhibitory activity against ThrombinMore data for this Ligand-Target Pair
Affinity DataKi: 1.78E+3nMAssay Description:Compound was evaluated for its inhibitory activity against TrypsinMore data for this Ligand-Target Pair
Affinity DataKi: 2.19E+3nMAssay Description:Compound was evaluated for its inhibitory activity against ThrombinMore data for this Ligand-Target Pair
Affinity DataKi: 3.10E+3nMAssay Description:Compound was evaluated for its inhibitory activity against ThrombinMore data for this Ligand-Target Pair