Affinity DataKi: 1.20nMAssay Description:Displacement of [3H]DAMGO from mu opioid receptor in rat brain membraneMore data for this Ligand-Target Pair
Affinity DataKi: 1.5nMAssay Description:Displacement of [3H]DAMGO from mu opioid receptor in rat brain membraneMore data for this Ligand-Target Pair
Affinity DataKi: 1.70nMAssay Description:50% inhibitory activity against enkephalinase purified from rat kidney with [3H]D-Ala2-Leu-enkephalin (20 nM) as substrate.More data for this Ligand-Target Pair
Affinity DataKi: 1.80nMAssay Description:50% inhibitory activity against enkephalinase purified from rat kidney with [3H]D-Ala2-Leu-enkephalin (20 nM) as substrate.More data for this Ligand-Target Pair
Affinity DataKi: 2.40nMAssay Description:Displacement of [3H]DAMGO from mu opioid receptor in rat brain membraneMore data for this Ligand-Target Pair
Affinity DataKi: 2.90nMAssay Description:Inhibitory activity against aminopeptidase using 10 nM of [3H]Leu-enkephalin as substrateMore data for this Ligand-Target Pair
Affinity DataKi: 3.80nMAssay Description:Inhibitory activity against aminopeptidase using 10 nM of [3H]Leu-enkephalin as substrateMore data for this Ligand-Target Pair
Affinity DataKi: 7.70nMAssay Description:Displacement of [3H]DSLET from delta opioid receptor in rat brain membraneMore data for this Ligand-Target Pair
Affinity DataKi: 17nMAssay Description:Displacement of [3H]DSLET from delta opioid receptor in rat brain membraneMore data for this Ligand-Target Pair
Affinity DataKi: 27nMAssay Description:Displacement of [3H]DSLET from delta opioid receptor in rat brain membraneMore data for this Ligand-Target Pair
Affinity DataIC50: 0.0100nMAssay Description:Displacement of [3H]naloxone from mu opioid receptor in rat brain membranesMore data for this Ligand-Target Pair
Affinity DataIC50: 0.560nMAssay Description:Displacement of [3H]naltrindole from delta opioid receptor in rat brain membranesMore data for this Ligand-Target Pair
Affinity DataIC50: 0.790nMAssay Description:Displacement of [3H]naloxone from mu opioid receptor in rat brain membranesMore data for this Ligand-Target Pair
Affinity DataIC50: 1nMAssay Description:In vitro inhibition of enkephalinase purified from rat kidney.More data for this Ligand-Target Pair
Affinity DataIC50: 1nMAssay Description:Inhibitory activity against rabbit kidney aminopeptidase using 10 nM of [3H]Leu-enkephalin as substrateMore data for this Ligand-Target Pair
Affinity DataIC50: >1nMAssay Description:In vitro inhibition of enkephalinase purified from rat kidney.More data for this Ligand-Target Pair
Affinity DataIC50: 1.20nMAssay Description:In vitro inhibition of enkephalinase purified from rat kidney.More data for this Ligand-Target Pair
TargetPyroglutamylated RF-amide peptide receptor(Homo sapiens (Human))
Institute For Research And Innovation In Biomedicine (Irib)
Curated by ChEMBL
Institute For Research And Innovation In Biomedicine (Irib)
Curated by ChEMBL
Affinity DataIC50: 1.30nMAssay Description:Displacement of [125I]26RFa from human GPR103 expressed in HEK293 cells incubated for 1 h by gamma counter based methodMore data for this Ligand-Target Pair
Affinity DataIC50: 1.40nMAssay Description:In vitro inhibition of enkephalinase purified from rat kidney.More data for this Ligand-Target Pair
Affinity DataIC50: 1.5nMAssay Description:Displacement of [3H]naloxone from mu opioid receptor in rat brain membranesMore data for this Ligand-Target Pair
Affinity DataIC50: 1.5nMAssay Description:In vitro inhibition of enkephalinase purified from rat kidney.More data for this Ligand-Target Pair
Affinity DataIC50: 2nMAssay Description:Inhibitory activity against rabbit kidney aminopeptidase using 10 nM of [3H]Leu-enkephalin as substrateMore data for this Ligand-Target Pair
Affinity DataIC50: 2nMAssay Description:In vitro inhibition of enkephalinase purified from rat kidney.More data for this Ligand-Target Pair
Affinity DataIC50: 2.5nMAssay Description:Inhibitory activity against rabbit kidney aminopeptidase using 10 nM of [3H]Leu-enkephalin as substrateMore data for this Ligand-Target Pair
Affinity DataIC50: 4nMAssay Description:In vitro inhibition of enkephalinase purified from rat kidney.More data for this Ligand-Target Pair
Affinity DataIC50: 5nMAssay Description:Inhibitory activity against rabbit kidney aminopeptidase using 10 nM of [3H]Leu-enkephalin as substrateMore data for this Ligand-Target Pair
Affinity DataIC50: 7.10nMAssay Description:Inhibitory activity against rabbit kidney aminopeptidase using 10 nM of [3H]Leu-enkephalin as substrateMore data for this Ligand-Target Pair
Affinity DataIC50: 7.70nMAssay Description:Displacement of [3H]DSLET from delta opioid receptor in rat brain membranesMore data for this Ligand-Target Pair
Affinity DataIC50: 7.70nMAssay Description:Agonist activity at mu opioid receptor by inhibition of electrically evoked muscle contraction in guinea pig ileumMore data for this Ligand-Target Pair
Affinity DataIC50: 8.5nMAssay Description:Inhibitory activity against rabbit kidney aminopeptidase using 10 nM of [3H]Leu-enkephalin as substrateMore data for this Ligand-Target Pair
Affinity DataIC50: 10nMAssay Description:In vitro inhibition of enkephalinase purified from rat kidney.More data for this Ligand-Target Pair
Affinity DataIC50: 12nMAssay Description:In vitro inhibition of enkephalinase purified from rat kidney.More data for this Ligand-Target Pair
Affinity DataIC50: 15nMAssay Description:Agonist activity at delta opioid receptor by inhibition of electrically evoked muscle contraction in isolated mouse vas deferensMore data for this Ligand-Target Pair
Affinity DataIC50: 16nMAssay Description:Agonist activity at mu opioid receptor by inhibition of electrically evoked muscle contraction in guinea pig ileumMore data for this Ligand-Target Pair
Affinity DataIC50: 17nMAssay Description:Agonist activity at mu opioid receptor by inhibition of electrically evoked muscle contraction in guinea pig ileumMore data for this Ligand-Target Pair
Affinity DataIC50: 20nMAssay Description:Displacement of [3H]naloxone from mu opioid receptor in rat brain membranesMore data for this Ligand-Target Pair
Affinity DataIC50: 26nMAssay Description:Agonist activity at delta opioid receptor by inhibition of electrically evoked muscle contraction in isolated mouse vas deferensMore data for this Ligand-Target Pair
Affinity DataIC50: 30nMAssay Description:In vitro inhibition of enkephalinase purified from rat kidney.More data for this Ligand-Target Pair
Affinity DataIC50: 350nMAssay Description:In vitro inhibition of enkephalinase purified from rat kidney.More data for this Ligand-Target Pair
Affinity DataIC50: 500nMAssay Description:50% Inhibitory potency against enkephalinase from mouse striatum.More data for this Ligand-Target Pair
Affinity DataIC50: 600nMAssay Description:In vitro inhibition of enkephalinase purified from rat kidney.More data for this Ligand-Target Pair
Affinity DataIC50: 700nMAssay Description:In vitro inhibition of enkephalinase purified from rat kidney.More data for this Ligand-Target Pair
Affinity DataIC50: 700nMAssay Description:50% Inhibitory potency against enkephalinase from mouse striatum.More data for this Ligand-Target Pair
Affinity DataIC50: 750nMAssay Description:In vitro inhibition of enkephalinase purified from rat kidney.More data for this Ligand-Target Pair
Affinity DataIC50: 800nMAssay Description:In vitro inhibition of enkephalinase purified from rat kidney.More data for this Ligand-Target Pair
Affinity DataIC50: 800nMAssay Description:50% Inhibitory potency against enkephalinase from mouse striatum.More data for this Ligand-Target Pair
Affinity DataIC50: 800nMAssay Description:In vitro inhibition of enkephalinase purified from rat kidney.More data for this Ligand-Target Pair
Affinity DataIC50: 850nMAssay Description:In vitro inhibition of enkephalinase purified from rat kidney.More data for this Ligand-Target Pair
Affinity DataIC50: 1.00E+3nMAssay Description:50% Inhibitory potency against enkephalinase from mouse striatum.More data for this Ligand-Target Pair
Affinity DataIC50: 1.56E+3nMAssay Description:Displacement of [3H]naloxone from mu opioid receptor in rat brain membranesMore data for this Ligand-Target Pair