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Found 67 with Last Name = 'cremonesi' and Initial = 'p'
LigandPNGBDBM50289537(1-(3-Phenyl-propyl)-3-((Z)-styryl)-piperidine | CH...)
Affinity DataIC50:  0.600nMAssay Description:Binding affinity at sigma receptor by [3H]-(+)-SKF-10,047 displacement.More data for this Ligand-Target Pair
In DepthDetails Article
LigandPNGBDBM50289553(1-Phenethyl-3-((Z)-styryl)-piperidine | CHEMBL3697...)
Affinity DataIC50:  0.800nMAssay Description:Binding affinity at sigma receptor by [3H]-(+)-SKF-10,047 displacement.More data for this Ligand-Target Pair
In DepthDetails Article
LigandPNGBDBM50289552(1-(3-Methyl-but-2-enyl)-3-((Z)-styryl)-piperidine ...)
Affinity DataIC50:  1nMAssay Description:Binding affinity at sigma receptor by [3H]-(+)-SKF-10,047 displacement.More data for this Ligand-Target Pair
In DepthDetails Article
LigandPNGBDBM50289539(1-Cyclohexyl-3-((Z)-styryl)-piperidine | CHEMBL398...)
Affinity DataIC50:  2nMAssay Description:Binding affinity at sigma receptor by [3H]-(+)-SKF-10,047 displacement.More data for this Ligand-Target Pair
In DepthDetails Article
LigandPNGBDBM50289538(1-Allyl-3-((E)-styryl)-piperidine | CHEMBL39735)
Affinity DataIC50:  4nMAssay Description:Binding affinity at sigma receptor by [3H]-(+)-SKF-10,047 displacement.More data for this Ligand-Target Pair
In DepthDetails Article
LigandPNGBDBM50289541(1-(3-Phenyl-propyl)-3-((E)-styryl)-piperidine | CH...)
Affinity DataIC50:  4nMAssay Description:Binding affinity at sigma receptor by [3H]-(+)-SKF-10,047 displacement.More data for this Ligand-Target Pair
In DepthDetails Article
LigandPNGBDBM50289547(1-Phenethyl-3-((E)-styryl)-piperidine | CHEMBL2879...)
Affinity DataIC50:  6nMAssay Description:Binding affinity at sigma receptor by [3H]-(+)-SKF-10,047 displacement.More data for this Ligand-Target Pair
In DepthDetails Article
LigandPNGBDBM50289549(1-Cyclohexyl-3-((E)-styryl)-piperidine | CHEMBL291...)
Affinity DataIC50:  6nMAssay Description:Binding affinity at sigma receptor by [3H]-(+)-SKF-10,047 displacement.More data for this Ligand-Target Pair
In DepthDetails Article
LigandPNGBDBM50289551(1-(4-Phenyl-butyl)-3-((Z)-styryl)-piperidine | CHE...)
Affinity DataIC50:  7nMAssay Description:Binding affinity at sigma receptor by [3H]-(+)-SKF-10,047 displacement.More data for this Ligand-Target Pair
In DepthDetails Article
LigandPNGBDBM50289545(1-(2-Cyclohexyl-ethyl)-3-((Z)-styryl)-piperidine |...)
Affinity DataIC50:  7nMAssay Description:Binding affinity at sigma receptor by [3H]-(+)-SKF-10,047 displacement.More data for this Ligand-Target Pair
In DepthDetails Article
LigandPNGBDBM50289536(1-Benzyl-3-((E)-styryl)-piperidine | CHEMBL39855)
Affinity DataIC50:  10nMAssay Description:Binding affinity at sigma receptor by [3H]-(+)-SKF-10,047 displacement.More data for this Ligand-Target Pair
In DepthDetails Article
LigandPNGBDBM50289554(1-Pent-4-enyl-3-((E)-styryl)-piperidine | CHEMBL38...)
Affinity DataIC50:  12nMAssay Description:Binding affinity at sigma receptor by [3H]-(+)-SKF-10,047 displacement.More data for this Ligand-Target Pair
In DepthDetails Article
LigandPNGBDBM50289540(1-(3-Phenoxy-propyl)-3-((Z)-styryl)-piperidine | C...)
Affinity DataIC50:  15nMAssay Description:Binding affinity at sigma receptor by [3H]-(+)-SKF-10,047 displacement.More data for this Ligand-Target Pair
In DepthDetails Article
LigandPNGBDBM50289544(1-Phenyl-4-[3-((Z)-styryl)-piperidin-1-yl]-butan-1...)
Affinity DataIC50:  15nMAssay Description:Binding affinity at sigma receptor by [3H]-(+)-SKF-10,047 displacement.More data for this Ligand-Target Pair
In DepthDetails Article
TargetCholesteryl ester transfer protein(Homo sapiens (Human))
Boehringer Ingelheim Pharma

Curated by ChEMBL
LigandPNGBDBM50028965(CHEMBL3360279)
Affinity DataIC50:  18nMAssay Description:Inhibition of human recombinant CETP by fluorescence transfer assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50289557(Adamantane-1-carboxylic acid {4-[3-((Z)-styryl)-pi...)
Affinity DataIC50:  23nMAssay Description:Binding affinity at sigma receptor by [3H]-(+)-SKF-10,047 displacement.More data for this Ligand-Target Pair
In DepthDetails Article
LigandPNGBDBM50289556(1,1-Dioxo-2-{4-[3-((E)-styryl)-piperidin-1-yl]-but...)
Affinity DataIC50:  23nMAssay Description:Binding affinity at sigma receptor by [3H]-(+)-SKF-10,047 displacement.More data for this Ligand-Target Pair
In DepthDetails Article
LigandPNGBDBM50289543(2-{3-[3-((Z)-Styryl)-piperidin-1-yl]-propylsulfany...)
Affinity DataIC50:  27nMAssay Description:Binding affinity at sigma receptor by [3H]-(+)-SKF-10,047 displacement.More data for this Ligand-Target Pair
In DepthDetails Article
TargetCholesteryl ester transfer protein(Homo sapiens (Human))
Boehringer Ingelheim Pharma

Curated by ChEMBL
LigandPNGBDBM50028951(CHEMBL3359665)
Affinity DataIC50:  29nMAssay Description:Inhibition of human recombinant CETP by fluorescence transfer assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50289550(1-(3-Phenoxy-propyl)-3-((E)-styryl)-piperidine | C...)
Affinity DataIC50:  33nMAssay Description:Binding affinity at sigma receptor by [3H]-(+)-SKF-10,047 displacement.More data for this Ligand-Target Pair
In DepthDetails Article
TargetCholesteryl ester transfer protein(Homo sapiens (Human))
Boehringer Ingelheim Pharma

Curated by ChEMBL
LigandPNGBDBM50028958(CHEMBL3360275)
Affinity DataIC50:  37nMAssay Description:Inhibition of human recombinant CETP by fluorescence transfer assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50289546(1-(3-Methyl-but-2-enyl)-3-((E)-styryl)-piperidine ...)
Affinity DataIC50:  38nMAssay Description:Binding affinity at sigma receptor by [3H]-(+)-SKF-10,047 displacement.More data for this Ligand-Target Pair
In DepthDetails Article
TargetCholesteryl ester transfer protein(Homo sapiens (Human))
Boehringer Ingelheim Pharma

Curated by ChEMBL
LigandPNGBDBM50028959(CHEMBL3360276)
Affinity DataIC50:  42nMAssay Description:Inhibition of human recombinant CETP by fluorescence transfer assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholesteryl ester transfer protein(Homo sapiens (Human))
Boehringer Ingelheim Pharma

Curated by ChEMBL
LigandPNGBDBM50028964(CHEMBL3360278)
Affinity DataIC50:  45nMAssay Description:Inhibition of human recombinant CETP by fluorescence transfer assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholesteryl ester transfer protein(Homo sapiens (Human))
Boehringer Ingelheim Pharma

Curated by ChEMBL
LigandPNGBDBM50028950(CHEMBL3359664)
Affinity DataIC50:  47nMAssay Description:Inhibition of human recombinant CETP by fluorescence transfer assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholesteryl ester transfer protein(Homo sapiens (Human))
Boehringer Ingelheim Pharma

Curated by ChEMBL
LigandPNGBDBM50028952(CHEMBL3360269)
Affinity DataIC50:  51nMAssay Description:Inhibition of human recombinant CETP by fluorescence transfer assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50289542(3-((Z)-Styryl)-piperidine | CHEMBL38345)
Affinity DataIC50:  64nMAssay Description:Binding affinity at sigma receptor by [3H]-(+)-SKF-10,047 displacement.More data for this Ligand-Target Pair
In DepthDetails Article
TargetCholesteryl ester transfer protein(Homo sapiens (Human))
Boehringer Ingelheim Pharma

Curated by ChEMBL
LigandPNGBDBM50028955(CHEMBL3360272)
Affinity DataIC50:  96nMAssay Description:Inhibition of human recombinant CETP by fluorescence transfer assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
TBA

Curated by ChEMBL
LigandPNGBDBM50289553(1-Phenethyl-3-((Z)-styryl)-piperidine | CHEMBL3697...)
Affinity DataIC50:  120nMAssay Description:Binding affinity at dopamine D2 receptor in rat striatum by [3H]-Spiperone displacement.More data for this Ligand-Target Pair
In DepthDetails Article
TargetCholesteryl ester transfer protein(Homo sapiens (Human))
Boehringer Ingelheim Pharma

Curated by ChEMBL
LigandPNGBDBM50028954(CHEMBL3360271)
Affinity DataIC50:  131nMAssay Description:Inhibition of human recombinant CETP by fluorescence transfer assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholesteryl ester transfer protein(Homo sapiens (Human))
Boehringer Ingelheim Pharma

Curated by ChEMBL
LigandPNGBDBM50028956(CHEMBL3360273)
Affinity DataIC50:  135nMAssay Description:Inhibition of human recombinant CETP by fluorescence transfer assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
TBA

Curated by ChEMBL
LigandPNGBDBM50289537(1-(3-Phenyl-propyl)-3-((Z)-styryl)-piperidine | CH...)
Affinity DataIC50:  150nMAssay Description:Binding affinity at dopamine D2 receptor in rat striatum by [3H]-Spiperone displacement.More data for this Ligand-Target Pair
In DepthDetails Article
TargetCholesteryl ester transfer protein(Homo sapiens (Human))
Boehringer Ingelheim Pharma

Curated by ChEMBL
LigandPNGBDBM50028965(CHEMBL3360279)
Affinity DataIC50:  151nMAssay Description:Inhibition of human recombinant CETP in presence of 88% human plasma by fluorescence transfer assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
TBA

Curated by ChEMBL
LigandPNGBDBM50289552(1-(3-Methyl-but-2-enyl)-3-((Z)-styryl)-piperidine ...)
Affinity DataIC50:  160nMAssay Description:Binding affinity at dopamine D2 receptor in rat striatum by [3H]-Spiperone displacement.More data for this Ligand-Target Pair
In DepthDetails Article
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
TBA

Curated by ChEMBL
LigandPNGBDBM50289546(1-(3-Methyl-but-2-enyl)-3-((E)-styryl)-piperidine ...)
Affinity DataIC50:  180nMAssay Description:Binding affinity at dopamine D2 receptor in rat striatum by [3H]-Spiperone displacement.More data for this Ligand-Target Pair
In DepthDetails Article
TargetD(1A) dopamine receptor(RAT)
TBA

Curated by ChEMBL
LigandPNGBDBM50289552(1-(3-Methyl-but-2-enyl)-3-((Z)-styryl)-piperidine ...)
Affinity DataIC50:  320nMAssay Description:Binding affinity at dopamine D1 receptor in rat striatum by [3H]-SCH-22,390 displacement.More data for this Ligand-Target Pair
In DepthDetails Article
TargetCholesteryl ester transfer protein(Homo sapiens (Human))
Boehringer Ingelheim Pharma

Curated by ChEMBL
LigandPNGBDBM50028957(CHEMBL3360274)
Affinity DataIC50:  418nMAssay Description:Inhibition of human recombinant CETP by fluorescence transfer assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50289548(3-((E)-Styryl)-piperidine | CHEMBL40056)
Affinity DataIC50:  423nMAssay Description:Binding affinity at sigma receptor by [3H]-(+)-SKF-10,047 displacement.More data for this Ligand-Target Pair
In DepthDetails Article
TargetCholesteryl ester transfer protein(Homo sapiens (Human))
Boehringer Ingelheim Pharma

Curated by ChEMBL
LigandPNGBDBM50028953(CHEMBL3360270)
Affinity DataIC50:  524nMAssay Description:Inhibition of human recombinant CETP by fluorescence transfer assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholesteryl ester transfer protein(Homo sapiens (Human))
Boehringer Ingelheim Pharma

Curated by ChEMBL
LigandPNGBDBM50028960(CHEMBL3360277)
Affinity DataIC50:  548nMAssay Description:Inhibition of human recombinant CETP by fluorescence transfer assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholesteryl ester transfer protein(Homo sapiens (Human))
Boehringer Ingelheim Pharma

Curated by ChEMBL
LigandPNGBDBM50028966(CHEMBL3360280)
Affinity DataIC50:  576nMAssay Description:Inhibition of human recombinant CETP by fluorescence transfer assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(1A) dopamine receptor(RAT)
TBA

Curated by ChEMBL
LigandPNGBDBM50289553(1-Phenethyl-3-((Z)-styryl)-piperidine | CHEMBL3697...)
Affinity DataIC50:  630nMAssay Description:Binding affinity at dopamine D1 receptor in rat striatum by [3H]-SCH-22,390 displacement.More data for this Ligand-Target Pair
In DepthDetails Article
LigandPNGBDBM50289555(CHEMBL289972 | N-Phenyl-2-[3-((Z)-styryl)-piperidi...)
Affinity DataIC50:  640nMAssay Description:Binding affinity at sigma receptor by [3H]-(+)-SKF-10,047 displacement.More data for this Ligand-Target Pair
In DepthDetails Article
TargetCholesteryl ester transfer protein(Homo sapiens (Human))
Boehringer Ingelheim Pharma

Curated by ChEMBL
LigandPNGBDBM50028948(CHEMBL3359662)
Affinity DataIC50:  796nMAssay Description:Inhibition of human recombinant CETP by fluorescence transfer assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
TBA

Curated by ChEMBL
LigandPNGBDBM50289542(3-((Z)-Styryl)-piperidine | CHEMBL38345)
Affinity DataIC50:  870nMAssay Description:Binding affinity at dopamine D2 receptor in rat striatum by [3H]-Spiperone displacement.More data for this Ligand-Target Pair
In DepthDetails Article
TargetCholesteryl ester transfer protein(Homo sapiens (Human))
Boehringer Ingelheim Pharma

Curated by ChEMBL
LigandPNGBDBM50028949(CHEMBL3359663)
Affinity DataIC50:  1.08E+3nMAssay Description:Inhibition of human recombinant CETP by fluorescence transfer assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
TBA

Curated by ChEMBL
LigandPNGBDBM50289539(1-Cyclohexyl-3-((Z)-styryl)-piperidine | CHEMBL398...)
Affinity DataIC50:  1.12E+3nMAssay Description:Binding affinity at dopamine D2 receptor in rat striatum by [3H]-Spiperone displacement.More data for this Ligand-Target Pair
In DepthDetails Article
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
TBA

Curated by ChEMBL
LigandPNGBDBM50289541(1-(3-Phenyl-propyl)-3-((E)-styryl)-piperidine | CH...)
Affinity DataIC50:  1.24E+3nMAssay Description:Binding affinity at dopamine D2 receptor in rat striatum by [3H]-Spiperone displacement.More data for this Ligand-Target Pair
In DepthDetails Article
TargetD(1A) dopamine receptor(RAT)
TBA

Curated by ChEMBL
LigandPNGBDBM50289546(1-(3-Methyl-but-2-enyl)-3-((E)-styryl)-piperidine ...)
Affinity DataIC50:  1.33E+3nMAssay Description:Binding affinity at dopamine D1 receptor in rat striatum by [3H]-SCH-22,390 displacement.More data for this Ligand-Target Pair
In DepthDetails Article
TargetCholesteryl ester transfer protein(Homo sapiens (Human))
Boehringer Ingelheim Pharma

Curated by ChEMBL
LigandPNGBDBM50028946(CHEMBL3359660)
Affinity DataIC50:  1.43E+3nMAssay Description:Inhibition of human recombinant CETP by fluorescence transfer assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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