Affinity DataIC50: 0.600nMAssay Description:Binding affinity at sigma receptor by [3H]-(+)-SKF-10,047 displacement.More data for this Ligand-Target Pair
Affinity DataIC50: 0.800nMAssay Description:Binding affinity at sigma receptor by [3H]-(+)-SKF-10,047 displacement.More data for this Ligand-Target Pair
Affinity DataIC50: 1nMAssay Description:Binding affinity at sigma receptor by [3H]-(+)-SKF-10,047 displacement.More data for this Ligand-Target Pair
Affinity DataIC50: 2nMAssay Description:Binding affinity at sigma receptor by [3H]-(+)-SKF-10,047 displacement.More data for this Ligand-Target Pair
Affinity DataIC50: 4nMAssay Description:Binding affinity at sigma receptor by [3H]-(+)-SKF-10,047 displacement.More data for this Ligand-Target Pair
Affinity DataIC50: 4nMAssay Description:Binding affinity at sigma receptor by [3H]-(+)-SKF-10,047 displacement.More data for this Ligand-Target Pair
Affinity DataIC50: 6nMAssay Description:Binding affinity at sigma receptor by [3H]-(+)-SKF-10,047 displacement.More data for this Ligand-Target Pair
Affinity DataIC50: 6nMAssay Description:Binding affinity at sigma receptor by [3H]-(+)-SKF-10,047 displacement.More data for this Ligand-Target Pair
Affinity DataIC50: 7nMAssay Description:Binding affinity at sigma receptor by [3H]-(+)-SKF-10,047 displacement.More data for this Ligand-Target Pair
Affinity DataIC50: 7nMAssay Description:Binding affinity at sigma receptor by [3H]-(+)-SKF-10,047 displacement.More data for this Ligand-Target Pair
Affinity DataIC50: 10nMAssay Description:Binding affinity at sigma receptor by [3H]-(+)-SKF-10,047 displacement.More data for this Ligand-Target Pair
Affinity DataIC50: 12nMAssay Description:Binding affinity at sigma receptor by [3H]-(+)-SKF-10,047 displacement.More data for this Ligand-Target Pair
Affinity DataIC50: 15nMAssay Description:Binding affinity at sigma receptor by [3H]-(+)-SKF-10,047 displacement.More data for this Ligand-Target Pair
Affinity DataIC50: 15nMAssay Description:Binding affinity at sigma receptor by [3H]-(+)-SKF-10,047 displacement.More data for this Ligand-Target Pair
TargetCholesteryl ester transfer protein(Homo sapiens (Human))
Boehringer Ingelheim Pharma
Curated by ChEMBL
Boehringer Ingelheim Pharma
Curated by ChEMBL
Affinity DataIC50: 18nMAssay Description:Inhibition of human recombinant CETP by fluorescence transfer assayMore data for this Ligand-Target Pair
Affinity DataIC50: 23nMAssay Description:Binding affinity at sigma receptor by [3H]-(+)-SKF-10,047 displacement.More data for this Ligand-Target Pair
Affinity DataIC50: 23nMAssay Description:Binding affinity at sigma receptor by [3H]-(+)-SKF-10,047 displacement.More data for this Ligand-Target Pair
Affinity DataIC50: 27nMAssay Description:Binding affinity at sigma receptor by [3H]-(+)-SKF-10,047 displacement.More data for this Ligand-Target Pair
TargetCholesteryl ester transfer protein(Homo sapiens (Human))
Boehringer Ingelheim Pharma
Curated by ChEMBL
Boehringer Ingelheim Pharma
Curated by ChEMBL
Affinity DataIC50: 29nMAssay Description:Inhibition of human recombinant CETP by fluorescence transfer assayMore data for this Ligand-Target Pair
Affinity DataIC50: 33nMAssay Description:Binding affinity at sigma receptor by [3H]-(+)-SKF-10,047 displacement.More data for this Ligand-Target Pair
TargetCholesteryl ester transfer protein(Homo sapiens (Human))
Boehringer Ingelheim Pharma
Curated by ChEMBL
Boehringer Ingelheim Pharma
Curated by ChEMBL
Affinity DataIC50: 37nMAssay Description:Inhibition of human recombinant CETP by fluorescence transfer assayMore data for this Ligand-Target Pair
Affinity DataIC50: 38nMAssay Description:Binding affinity at sigma receptor by [3H]-(+)-SKF-10,047 displacement.More data for this Ligand-Target Pair
TargetCholesteryl ester transfer protein(Homo sapiens (Human))
Boehringer Ingelheim Pharma
Curated by ChEMBL
Boehringer Ingelheim Pharma
Curated by ChEMBL
Affinity DataIC50: 42nMAssay Description:Inhibition of human recombinant CETP by fluorescence transfer assayMore data for this Ligand-Target Pair
TargetCholesteryl ester transfer protein(Homo sapiens (Human))
Boehringer Ingelheim Pharma
Curated by ChEMBL
Boehringer Ingelheim Pharma
Curated by ChEMBL
Affinity DataIC50: 45nMAssay Description:Inhibition of human recombinant CETP by fluorescence transfer assayMore data for this Ligand-Target Pair
TargetCholesteryl ester transfer protein(Homo sapiens (Human))
Boehringer Ingelheim Pharma
Curated by ChEMBL
Boehringer Ingelheim Pharma
Curated by ChEMBL
Affinity DataIC50: 47nMAssay Description:Inhibition of human recombinant CETP by fluorescence transfer assayMore data for this Ligand-Target Pair
TargetCholesteryl ester transfer protein(Homo sapiens (Human))
Boehringer Ingelheim Pharma
Curated by ChEMBL
Boehringer Ingelheim Pharma
Curated by ChEMBL
Affinity DataIC50: 51nMAssay Description:Inhibition of human recombinant CETP by fluorescence transfer assayMore data for this Ligand-Target Pair
Affinity DataIC50: 64nMAssay Description:Binding affinity at sigma receptor by [3H]-(+)-SKF-10,047 displacement.More data for this Ligand-Target Pair
TargetCholesteryl ester transfer protein(Homo sapiens (Human))
Boehringer Ingelheim Pharma
Curated by ChEMBL
Boehringer Ingelheim Pharma
Curated by ChEMBL
Affinity DataIC50: 96nMAssay Description:Inhibition of human recombinant CETP by fluorescence transfer assayMore data for this Ligand-Target Pair
Affinity DataIC50: 120nMAssay Description:Binding affinity at dopamine D2 receptor in rat striatum by [3H]-Spiperone displacement.More data for this Ligand-Target Pair
TargetCholesteryl ester transfer protein(Homo sapiens (Human))
Boehringer Ingelheim Pharma
Curated by ChEMBL
Boehringer Ingelheim Pharma
Curated by ChEMBL
Affinity DataIC50: 131nMAssay Description:Inhibition of human recombinant CETP by fluorescence transfer assayMore data for this Ligand-Target Pair
TargetCholesteryl ester transfer protein(Homo sapiens (Human))
Boehringer Ingelheim Pharma
Curated by ChEMBL
Boehringer Ingelheim Pharma
Curated by ChEMBL
Affinity DataIC50: 135nMAssay Description:Inhibition of human recombinant CETP by fluorescence transfer assayMore data for this Ligand-Target Pair
Affinity DataIC50: 150nMAssay Description:Binding affinity at dopamine D2 receptor in rat striatum by [3H]-Spiperone displacement.More data for this Ligand-Target Pair
TargetCholesteryl ester transfer protein(Homo sapiens (Human))
Boehringer Ingelheim Pharma
Curated by ChEMBL
Boehringer Ingelheim Pharma
Curated by ChEMBL
Affinity DataIC50: 151nMAssay Description:Inhibition of human recombinant CETP in presence of 88% human plasma by fluorescence transfer assayMore data for this Ligand-Target Pair
Affinity DataIC50: 160nMAssay Description:Binding affinity at dopamine D2 receptor in rat striatum by [3H]-Spiperone displacement.More data for this Ligand-Target Pair
Affinity DataIC50: 180nMAssay Description:Binding affinity at dopamine D2 receptor in rat striatum by [3H]-Spiperone displacement.More data for this Ligand-Target Pair
Affinity DataIC50: 320nMAssay Description:Binding affinity at dopamine D1 receptor in rat striatum by [3H]-SCH-22,390 displacement.More data for this Ligand-Target Pair
TargetCholesteryl ester transfer protein(Homo sapiens (Human))
Boehringer Ingelheim Pharma
Curated by ChEMBL
Boehringer Ingelheim Pharma
Curated by ChEMBL
Affinity DataIC50: 418nMAssay Description:Inhibition of human recombinant CETP by fluorescence transfer assayMore data for this Ligand-Target Pair
Affinity DataIC50: 423nMAssay Description:Binding affinity at sigma receptor by [3H]-(+)-SKF-10,047 displacement.More data for this Ligand-Target Pair
TargetCholesteryl ester transfer protein(Homo sapiens (Human))
Boehringer Ingelheim Pharma
Curated by ChEMBL
Boehringer Ingelheim Pharma
Curated by ChEMBL
Affinity DataIC50: 524nMAssay Description:Inhibition of human recombinant CETP by fluorescence transfer assayMore data for this Ligand-Target Pair
TargetCholesteryl ester transfer protein(Homo sapiens (Human))
Boehringer Ingelheim Pharma
Curated by ChEMBL
Boehringer Ingelheim Pharma
Curated by ChEMBL
Affinity DataIC50: 548nMAssay Description:Inhibition of human recombinant CETP by fluorescence transfer assayMore data for this Ligand-Target Pair
TargetCholesteryl ester transfer protein(Homo sapiens (Human))
Boehringer Ingelheim Pharma
Curated by ChEMBL
Boehringer Ingelheim Pharma
Curated by ChEMBL
Affinity DataIC50: 576nMAssay Description:Inhibition of human recombinant CETP by fluorescence transfer assayMore data for this Ligand-Target Pair
Affinity DataIC50: 630nMAssay Description:Binding affinity at dopamine D1 receptor in rat striatum by [3H]-SCH-22,390 displacement.More data for this Ligand-Target Pair
Affinity DataIC50: 640nMAssay Description:Binding affinity at sigma receptor by [3H]-(+)-SKF-10,047 displacement.More data for this Ligand-Target Pair
TargetCholesteryl ester transfer protein(Homo sapiens (Human))
Boehringer Ingelheim Pharma
Curated by ChEMBL
Boehringer Ingelheim Pharma
Curated by ChEMBL
Affinity DataIC50: 796nMAssay Description:Inhibition of human recombinant CETP by fluorescence transfer assayMore data for this Ligand-Target Pair
Affinity DataIC50: 870nMAssay Description:Binding affinity at dopamine D2 receptor in rat striatum by [3H]-Spiperone displacement.More data for this Ligand-Target Pair
TargetCholesteryl ester transfer protein(Homo sapiens (Human))
Boehringer Ingelheim Pharma
Curated by ChEMBL
Boehringer Ingelheim Pharma
Curated by ChEMBL
Affinity DataIC50: 1.08E+3nMAssay Description:Inhibition of human recombinant CETP by fluorescence transfer assayMore data for this Ligand-Target Pair
Affinity DataIC50: 1.12E+3nMAssay Description:Binding affinity at dopamine D2 receptor in rat striatum by [3H]-Spiperone displacement.More data for this Ligand-Target Pair
Affinity DataIC50: 1.24E+3nMAssay Description:Binding affinity at dopamine D2 receptor in rat striatum by [3H]-Spiperone displacement.More data for this Ligand-Target Pair
Affinity DataIC50: 1.33E+3nMAssay Description:Binding affinity at dopamine D1 receptor in rat striatum by [3H]-SCH-22,390 displacement.More data for this Ligand-Target Pair
TargetCholesteryl ester transfer protein(Homo sapiens (Human))
Boehringer Ingelheim Pharma
Curated by ChEMBL
Boehringer Ingelheim Pharma
Curated by ChEMBL
Affinity DataIC50: 1.43E+3nMAssay Description:Inhibition of human recombinant CETP by fluorescence transfer assayMore data for this Ligand-Target Pair