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Found 165 with Last Name = 'dairaghi' and Initial = 'd'
TargetC-C chemokine receptor type 1(Homo sapiens (Human))
Chemocentryx

Curated by ChEMBL
LigandPNGBDBM50427065(CHEMBL2322875)
Affinity DataIC50:  0.800nMAssay Description:Antagonist activity at CCR1 in human THP1 cells assessed as inhibition of CCL5/RANTES-induced chemotaxisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-C chemokine receptor type 1(Homo sapiens (Human))
Chemocentryx

Curated by ChEMBL
LigandPNGBDBM50427065(CHEMBL2322875)
Affinity DataIC50:  1.5nMAssay Description:Antagonist activity at CCR1 in human THP1 cells assessed as inhibition of CCL15/Leukotactin1-induced chemotaxisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-C chemokine receptor type 1(Homo sapiens (Human))
Chemocentryx

Curated by ChEMBL
LigandPNGBDBM50427070(CHEMBL2322853)
Affinity DataIC50:  2nMAssay Description:Displacement of [125I]-CCL3/MIP-1alpha from CCR1 in human THP1 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-C chemokine receptor type 1(Homo sapiens (Human))
Chemocentryx

Curated by ChEMBL
LigandPNGBDBM50427065(CHEMBL2322875)
Affinity DataIC50:  2.5nMAssay Description:Antagonist activity at CCR1 in human THP1 cells assessed as inhibition of CCL23/CKbeta8.1-induced chemotaxisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-C chemokine receptor type 1(Homo sapiens (Human))
Chemocentryx

Curated by ChEMBL
LigandPNGBDBM50427065(CHEMBL2322875)
Affinity DataIC50:  3.90nMAssay Description:Antagonist activity at CCR1 in human THP1 cells assessed as inhibition of CCL3/MIP-1alpha-induced chemotaxisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-C chemokine receptor type 1(Homo sapiens (Human))
Chemocentryx

Curated by ChEMBL
LigandPNGBDBM50427065(CHEMBL2322875)
Affinity DataIC50:  4nMAssay Description:Displacement of [125I]-CCL3/MIP-1alpha from CCR1 in human THP1 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-X-C chemokine receptor type 3(Homo sapiens (Human))
Amgen

Curated by ChEMBL
LigandPNGBDBM50211148((R)-N-(1-(4-oxo-3-(4-(prop-1-ynyl)phenyl)-3,4-dihy...)
Affinity DataIC50:  4nMAssay Description:Displacement of [125I ]IP10 from CXCR3 receptor expressed in PBMCMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-C chemokine receptor type 1(Homo sapiens (Human))
Chemocentryx

Curated by ChEMBL
LigandPNGBDBM50427065(CHEMBL2322875)
Affinity DataIC50:  4.80nMAssay Description:Antagonist activity at CCR1 in human THP1 cells assessed as inhibition of CCL15/Leukotactin1-induced calcium flux by FLIPR assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-C chemokine receptor type 1(Homo sapiens (Human))
Chemocentryx

Curated by ChEMBL
LigandPNGBDBM50427105(CHEMBL2322879)
Affinity DataIC50:  5nMAssay Description:Displacement of [125I]-CCL3/MIP-1alpha from CCR1 in human THP1 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-C chemokine receptor type 1(Homo sapiens (Human))
Chemocentryx

Curated by ChEMBL
LigandPNGBDBM50427095(CHEMBL2322858)
Affinity DataIC50:  5nMAssay Description:Displacement of [125I]-CCL3/MIP-1alpha from CCR1 in human THP1 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-X-C chemokine receptor type 3(Homo sapiens (Human))
Amgen

Curated by ChEMBL
LigandPNGBDBM50211114((-)-(R)-N-(1-(3-(4-ethoxyphenyl)-4-oxo-3,4-dihydro...)
Affinity DataIC50:  5nMAssay Description:Antagonist activity at human CXCR3 assessed as inhibition of ITAC-induced calcium mobilizationMore data for this Ligand-Target Pair
TargetC-C chemokine receptor type 1(Homo sapiens (Human))
Chemocentryx

Curated by ChEMBL
LigandPNGBDBM50427065(CHEMBL2322875)
Affinity DataIC50:  5.5nMAssay Description:Antagonist activity at CCR1 in human THP1 cells assessed as inhibition of CCL3/MIP-1alpha-induced calcium flux by FLIPR assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-X-C chemokine receptor type 3(Homo sapiens (Human))
Amgen

Curated by ChEMBL
LigandPNGBDBM50211130((R)-N-(1-(3-(4-ethoxyphenyl)-4-oxo-3,4-dihydroquin...)
Affinity DataIC50:  6nMAssay Description:Displacement of [125I ]IP10 from CXCR3 receptor expressed in PBMCMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-C chemokine receptor type 1(Homo sapiens (Human))
Chemocentryx

Curated by ChEMBL
LigandPNGBDBM50427092(CHEMBL2322861)
Affinity DataIC50:  6nMAssay Description:Displacement of [125I]-CCL3/MIP-1alpha from CCR1 in human THP1 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-X-C chemokine receptor type 3(Homo sapiens (Human))
Amgen

Curated by ChEMBL
LigandPNGBDBM50211138((R)-N-(1-(3-(4-ethoxyphenyl)-4-oxo-3,4-dihydroquin...)
Affinity DataIC50:  6nMAssay Description:Displacement of [125I ]IP10 from CXCR3 receptor expressed in PBMCMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-C chemokine receptor type 1(Homo sapiens (Human))
Chemocentryx

Curated by ChEMBL
LigandPNGBDBM50427065(CHEMBL2322875)
Affinity DataIC50:  6nMAssay Description:Displacement of [125I]-CCL3/MIP-1alpha from CCR1 in human monocytesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-X-C chemokine receptor type 3(Homo sapiens (Human))
Amgen

Curated by ChEMBL
LigandPNGBDBM50211137((R)-N-(1-(3-(4-nitrophenyl)-4-oxo-3,4-dihydroquina...)
Affinity DataIC50:  7nMAssay Description:Displacement of [125I ]IP10 from CXCR3 receptor expressed in PBMCMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-C chemokine receptor type 1(Homo sapiens (Human))
Chemocentryx

Curated by ChEMBL
LigandPNGBDBM50427093(CHEMBL2322860)
Affinity DataIC50:  7nMAssay Description:Displacement of [125I]-CCL3/MIP-1alpha from CCR1 in human THP1 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-X-C chemokine receptor type 3(Homo sapiens (Human))
Amgen

Curated by ChEMBL
LigandPNGBDBM50211114((-)-(R)-N-(1-(3-(4-ethoxyphenyl)-4-oxo-3,4-dihydro...)
Affinity DataIC50:  8nMAssay Description:Inhibition of IP10-induced CXCR3 mediated cell migrationMore data for this Ligand-Target Pair
TargetC-C chemokine receptor type 1(Homo sapiens (Human))
Chemocentryx

Curated by ChEMBL
LigandPNGBDBM50427080(CHEMBL2322844)
Affinity DataIC50:  8nMAssay Description:Displacement of [125I]-CCL3/MIP-1alpha from CCR1 in human THP1 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-C chemokine receptor type 1(Homo sapiens (Human))
Chemocentryx

Curated by ChEMBL
LigandPNGBDBM50427094(CHEMBL2322859)
Affinity DataIC50:  8nMAssay Description:Displacement of [125I]-CCL3/MIP-1alpha from CCR1 in human THP1 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-X-C chemokine receptor type 3(Homo sapiens (Human))
Amgen

Curated by ChEMBL
LigandPNGBDBM50211114((-)-(R)-N-(1-(3-(4-ethoxyphenyl)-4-oxo-3,4-dihydro...)
Affinity DataIC50:  8nMAssay Description:Displacement of [125I ]IP10 from CXCR3 receptor expressed in PBMCMore data for this Ligand-Target Pair
TargetC-X-C chemokine receptor type 3(Homo sapiens (Human))
Amgen

Curated by ChEMBL
LigandPNGBDBM50211114((-)-(R)-N-(1-(3-(4-ethoxyphenyl)-4-oxo-3,4-dihydro...)
Affinity DataIC50:  8.20nMAssay Description:Displacement of [125I] ITAC from the CXCR3 receptorMore data for this Ligand-Target Pair
TargetC-X-C chemokine receptor type 3(Homo sapiens (Human))
Amgen

Curated by ChEMBL
LigandPNGBDBM50211128(2-biphenyl-4-yl-N-(2-ethoxy-ethyl)-N-{(R)-1-[3-(4-...)
Affinity DataIC50:  9nMAssay Description:Displacement of [125I ]IP10 from CXCR3 receptor expressed in PBMCMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-C chemokine receptor type 1(Homo sapiens (Human))
Chemocentryx

Curated by ChEMBL
LigandPNGBDBM50427104(CHEMBL2322880)
Affinity DataIC50:  10nMAssay Description:Displacement of [125I]-CCL3/MIP-1alpha from CCR1 in human THP1 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-C chemokine receptor type 1(Homo sapiens (Human))
Chemocentryx

Curated by ChEMBL
LigandPNGBDBM50427086(CHEMBL2322867)
Affinity DataIC50:  10nMAssay Description:Displacement of [125I]-CCL3/MIP-1alpha from CCR1 in human THP1 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-C chemokine receptor type 1(Homo sapiens (Human))
Chemocentryx

Curated by ChEMBL
LigandPNGBDBM50427077(CHEMBL2322847)
Affinity DataIC50:  10nMAssay Description:Displacement of [125I]-CCL3/MIP-1alpha from CCR1 in human THP1 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-C chemokine receptor type 1(Homo sapiens (Human))
Chemocentryx

Curated by ChEMBL
LigandPNGBDBM50427076(CHEMBL2321887)
Affinity DataIC50:  10nMAssay Description:Displacement of [125I]-CCL3/MIP-1alpha from CCR1 in human THP1 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-X-C chemokine receptor type 3(Homo sapiens (Human))
Amgen

Curated by ChEMBL
LigandPNGBDBM50211121((R)-N-(1-(3-(4-cyanophenyl)-4-oxo-3,4-dihydroquina...)
Affinity DataIC50:  11nMAssay Description:Displacement of [125I ]IP10 from CXCR3 receptor expressed in PBMCMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-C chemokine receptor type 1(Homo sapiens (Human))
Chemocentryx

Curated by ChEMBL
LigandPNGBDBM50427069(CHEMBL2322854)
Affinity DataIC50:  11nMAssay Description:Displacement of [125I]-CCL3/MIP-1alpha from CCR1 in human THP1 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-C chemokine receptor type 1(Homo sapiens (Human))
Chemocentryx

Curated by ChEMBL
LigandPNGBDBM50427108(CHEMBL2322876)
Affinity DataIC50:  12nMAssay Description:Displacement of [125I]-CCL3/MIP-1alpha from CCR1 in human THP1 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-X-C chemokine receptor type 3(Homo sapiens (Human))
Amgen

Curated by ChEMBL
LigandPNGBDBM50211123((R)-N-(1-(3-(4-fluorophenyl)-4-oxo-3,4-dihydroquin...)
Affinity DataIC50:  12nMAssay Description:Displacement of [125I ]IP10 from CXCR3 receptor expressed in PBMCMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-C chemokine receptor type 1(Homo sapiens (Human))
Chemocentryx

Curated by ChEMBL
LigandPNGBDBM50427098(CHEMBL2322886)
Affinity DataIC50:  12nMAssay Description:Displacement of [125I]-CCL3/MIP-1alpha from CCR1 in human THP1 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-C chemokine receptor type 1(Homo sapiens (Human))
Chemocentryx

Curated by ChEMBL
LigandPNGBDBM50427065(CHEMBL2322875)
Affinity DataIC50:  12nMAssay Description:Displacement of [125I]-CCL15/Leukotactin1 from CCR1 in human THP1 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-C chemokine receptor type 1(Homo sapiens (Human))
Chemocentryx

Curated by ChEMBL
LigandPNGBDBM50427065(CHEMBL2322875)
Affinity DataIC50:  13nMAssay Description:Displacement of [125I]-CCL15/Leukotactin1 from CCR1 in human monocytesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-X-C chemokine receptor type 3(Homo sapiens (Human))
Amgen

Curated by ChEMBL
LigandPNGBDBM50211123((R)-N-(1-(3-(4-fluorophenyl)-4-oxo-3,4-dihydroquin...)
Affinity DataIC50:  13nMAssay Description:Displacement of [125I ]IP10 from CXCR3 receptor expressed in PBMCMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-C chemokine receptor type 4(Homo sapiens (Human))
Amgen

Curated by ChEMBL
LigandPNGBDBM50183119(4-(((2-(trifluoromethyl)benzyl)(cyclohexylmethyl)a...)
Affinity DataIC50:  14nMAssay Description:Displacement of [125I]TARC from CCR4 expressed in human CEM cell lineMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-X-C chemokine receptor type 3(Homo sapiens (Human))
Amgen

Curated by ChEMBL
LigandPNGBDBM50211143((R)-N-(1-(3-(4-methoxyphenyl)-4-oxo-3,4-dihydroqui...)
Affinity DataIC50:  14nMAssay Description:Displacement of [125I ]IP10 from CXCR3 receptor expressed in PBMCMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-C chemokine receptor type 1(Homo sapiens (Human))
Chemocentryx

Curated by ChEMBL
LigandPNGBDBM50427103(CHEMBL2322881)
Affinity DataIC50:  14nMAssay Description:Displacement of [125I]-CCL3/MIP-1alpha from CCR1 in human THP1 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-X-C chemokine receptor type 3(Homo sapiens (Human))
Amgen

Curated by ChEMBL
LigandPNGBDBM50211114((-)-(R)-N-(1-(3-(4-ethoxyphenyl)-4-oxo-3,4-dihydro...)
Affinity DataIC50:  15nMAssay Description:Inhibition of ITAC-induced CXCR3 mediated cell migrationMore data for this Ligand-Target Pair
TargetC-C chemokine receptor type 1(Homo sapiens (Human))
Chemocentryx

Curated by ChEMBL
LigandPNGBDBM50427065(CHEMBL2322875)
Affinity DataIC50:  15nMAssay Description:Antagonist activity at CCR1 in human monocytes assessed as inhibition of CCL15/Leukotactin1-induced chemotaxisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-C chemokine receptor type 1(Homo sapiens (Human))
Chemocentryx

Curated by ChEMBL
LigandPNGBDBM50427097(CHEMBL2322887)
Affinity DataIC50:  16nMAssay Description:Displacement of [125I]-CCL3/MIP-1alpha from CCR1 in human THP1 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-C chemokine receptor type 1(Homo sapiens (Human))
Chemocentryx

Curated by ChEMBL
LigandPNGBDBM50427079(CHEMBL2322845)
Affinity DataIC50:  16nMAssay Description:Displacement of [125I]-CCL3/MIP-1alpha from CCR1 in human THP1 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-C chemokine receptor type 4(Homo sapiens (Human))
Amgen

Curated by ChEMBL
LigandPNGBDBM50183091(4-((bis(cyclohexylmethyl)amino)methyl)-N-(naphthal...)
Affinity DataIC50:  18nMAssay Description:Displacement of [125I]TARC from CCR4 expressed in human CEM cell lineMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-C chemokine receptor type 1(Homo sapiens (Human))
Chemocentryx

Curated by ChEMBL
LigandPNGBDBM50427090(CHEMBL2322863)
Affinity DataIC50:  18nMAssay Description:Displacement of [125I]-CCL3/MIP-1alpha from CCR1 in human THP1 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-C chemokine receptor type 1(Homo sapiens (Human))
Chemocentryx

Curated by ChEMBL
LigandPNGBDBM50427096(CHEMBL2322857)
Affinity DataIC50:  19nMAssay Description:Displacement of [125I]-CCL3/MIP-1alpha from CCR1 in human THP1 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-C chemokine receptor type 1(Homo sapiens (Human))
Chemocentryx

Curated by ChEMBL
LigandPNGBDBM50427078(CHEMBL2322846)
Affinity DataIC50:  20nMAssay Description:Displacement of [125I]-CCL3/MIP-1alpha from CCR1 in human THP1 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-X-C chemokine receptor type 3(Homo sapiens (Human))
Amgen

Curated by ChEMBL
LigandPNGBDBM50211122((R)-N-(1-(3-(4-chlorophenyl)-4-oxo-3,4-dihydroquin...)
Affinity DataIC50:  22nMAssay Description:Displacement of [125I ]IP10 from CXCR3 receptor expressed in PBMCMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-C chemokine receptor type 1(Homo sapiens (Human))
Chemocentryx

Curated by ChEMBL
LigandPNGBDBM50427067(CHEMBL2322856)
Affinity DataIC50:  23nMAssay Description:Displacement of [125I]-CCL3/MIP-1alpha from CCR1 in human THP1 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-X-C chemokine receptor type 3(Homo sapiens (Human))
Amgen

Curated by ChEMBL
LigandPNGBDBM50211115((R)-N-(1-(4-oxo-3-p-tolyl-3,4-dihydroquinazolin-2-...)
Affinity DataIC50:  25nMAssay Description:Displacement of [125I ]IP10 from CXCR3 receptor expressed in PBMCMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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