Compile Data Set for Download or QSAR
maximum 50k data
Found 11 with Last Name = 'damera' and Initial = 'k'
TargetProtein translocase subunit SecA 1(Staphylococcus aureus (strain NCTC 8325))
Georgia State University

Curated by ChEMBL
LigandPNGBDBM50498947(Rose bengal sodium)
Affinity DataIC50:  500nMAssay Description:Inhibition of Staphylococcus aureus ATCC 35556 SecA1 liposomal ion channel activity in Xenopus laevis oocytes incubated for 3 hrs measured by recordi...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein translocase subunit SecA 1(Staphylococcus aureus (strain NCTC 8325))
Georgia State University

Curated by ChEMBL
LigandPNGBDBM50498946(CHEMBL3735815)
Affinity DataIC50:  1.00E+3nMAssay Description:Inhibition of Staphylococcus aureus ATCC 35556 SecA1 liposomal ion channel activity in Xenopus laevis oocytes incubated for 3 hrs measured by recordi...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProtein translocase subunit SecA 1(Staphylococcus aureus (strain NCTC 8325))
Georgia State University

Curated by ChEMBL
LigandPNGBDBM50498947(Rose bengal sodium)
Affinity DataIC50:  1.00E+3nMAssay Description:Inhibition of Staphylococcus aureus ATCC 35556 SecA1 expressed in Escherichia coli BL21-gammaDE3 assessed as reduction in intrinsic ATPase activity i...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein translocase subunit SecA 1(Staphylococcus aureus (strain NCTC 8325))
Georgia State University

Curated by ChEMBL
LigandPNGBDBM50498948(CHEMBL3736159)
Affinity DataIC50:  2.00E+3nMAssay Description:Inhibition of Staphylococcus aureus ATCC 35556 SecA1 liposomal ion channel activity in Xenopus laevis oocytes incubated for 3 hrs measured by recordi...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProtein translocase subunit SecA 2(Staphylococcus aureus (strain NCTC 8325))
Georgia State University

Curated by ChEMBL
LigandPNGBDBM50498947(Rose bengal sodium)
Affinity DataIC50:  2.00E+3nMAssay Description:Inhibition of Staphylococcus aureus ATCC 35556 SecA2 expressed in Escherichia coli BL21-gammaDE3 assessed as reduction in intrinsic ATPase activity i...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein translocase subunit SecA 1(Staphylococcus aureus (strain NCTC 8325))
Georgia State University

Curated by ChEMBL
LigandPNGBDBM50498946(CHEMBL3735815)
Affinity DataIC50:  4.00E+3nMAssay Description:Inhibition of Staphylococcus aureus ATCC 35556 SecA1 liposome dependent proOmpA translocation incubated for 1.5 hrs measured by Western blot analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProtein translocase subunit SecA 2(Staphylococcus aureus (strain NCTC 8325))
Georgia State University

Curated by ChEMBL
LigandPNGBDBM50498946(CHEMBL3735815)
Affinity DataIC50:  1.50E+4nMAssay Description:Inhibition of Staphylococcus aureus ATCC 35556 SecA2 expressed in Escherichia coli BL21-gammaDE3 assessed as reduction in intrinsic ATPase activity i...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProtein translocase subunit SecA 1(Staphylococcus aureus (strain NCTC 8325))
Georgia State University

Curated by ChEMBL
LigandPNGBDBM50498946(CHEMBL3735815)
Affinity DataIC50:  2.00E+4nMAssay Description:Inhibition of Staphylococcus aureus ATCC 35556 SecA1 expressed in Escherichia coli BL21-gammaDE3 assessed as reduction in intrinsic ATPase activity i...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProtein translocase subunit SecA 2(Staphylococcus aureus (strain NCTC 8325))
Georgia State University

Curated by ChEMBL
LigandPNGBDBM50498948(CHEMBL3736159)
Affinity DataIC50:  3.00E+4nMAssay Description:Inhibition of Staphylococcus aureus ATCC 35556 SecA2 expressed in Escherichia coli BL21-gammaDE3 assessed as reduction in intrinsic ATPase activity i...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProtein translocase subunit SecA 1(Staphylococcus aureus (strain NCTC 8325))
Georgia State University

Curated by ChEMBL
LigandPNGBDBM50498948(CHEMBL3736159)
Affinity DataIC50:  3.50E+4nMAssay Description:Inhibition of Staphylococcus aureus ATCC 35556 SecA1 expressed in Escherichia coli BL21-gammaDE3 assessed as reduction in intrinsic ATPase activity i...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetHistone acetyltransferase p300(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50396040(CHEMBL1823895)
Affinity DataKd:  345nMAssay Description:Binding affinity to recombinant P300 CH1 domain assessed as dissociation constant by surface plasmon resonance analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed