Affinity DataKi: 0.400nMAssay Description:Compound was evaluated in vitro for the binding of Cysteinyl leukotriene receptor 1 to guinea pig lung membranesMore data for this Ligand-Target Pair
Affinity DataKi: 0.600nMAssay Description:Compound was evaluated in vitro for the binding of Cysteinyl leukotriene receptor 1 to guinea pig lung membranesMore data for this Ligand-Target Pair
Affinity DataKi: 0.800nMAssay Description:Compound was evaluated in vitro for the binding of Cysteinyl leukotriene receptor 1 to guinea pig lung membranesMore data for this Ligand-Target Pair
Affinity DataKi: 2nMAssay Description:Compound was evaluated in vitro for the binding of cysLT1 receptor to guinea pig lung membranes.More data for this Ligand-Target Pair
Affinity DataKi: 2.30nMAssay Description:Displacement of [3H]-leukotriene D4 (LTD4) from receptor in guinea pig lung membranesMore data for this Ligand-Target Pair
Affinity DataKi: 5nMAssay Description:Displacement of [3H]-ligand from platelet activating factor (PAF) receptor in rabbit plateletsMore data for this Ligand-Target Pair
Affinity DataKi: 20nMAssay Description:Displacement of [3H]-LTD4 from receptor in guinea pig lung membranesMore data for this Ligand-Target Pair
Affinity DataKi: 24nMAssay Description:Displacement of [3H]-ligand from platelet activating factor (PAF) receptor in rabbit plateletsMore data for this Ligand-Target Pair
Affinity DataKi: 29nMAssay Description:Displacement of [3H]-ligand from platelet activating factor (PAF) receptor in rabbit plateletsMore data for this Ligand-Target Pair
Affinity DataKi: 34nMAssay Description:Displacement of [3H]-leukotriene D4 (LTD4) from receptor in guinea pig lung membranesMore data for this Ligand-Target Pair
Affinity DataKi: 37nMAssay Description:Displacement of [3H]-ligand from platelet activating factor (PAF) receptor in rabbit plateletsMore data for this Ligand-Target Pair
Affinity DataKi: 73nMAssay Description:Displacement of [3H]-leukotriene D4 (LTD4) from receptor in guinea pig lung membranesMore data for this Ligand-Target Pair
Affinity DataKi: 650nMAssay Description:Inhibition of [3H]-LTD4 binding to LTD4 receptor in guinea pig lung membranesMore data for this Ligand-Target Pair
Affinity DataKi: 1.50E+3nMAssay Description:Inhibition of [3H]-LTD4 binding to LTD4 receptor in guinea pig lung membranesMore data for this Ligand-Target Pair
Affinity DataKi: 6.80E+3nMAssay Description:Inhibition of [3H]-LTD4 binding to LTD4 receptor in guinea pig lung membranesMore data for this Ligand-Target Pair
Affinity DataKi: 8.00E+3nMAssay Description:Inhibition of [3H]-LTD4 binding to LTD4 receptor in guinea pig lung membranesMore data for this Ligand-Target Pair
Affinity DataKi: 2.40E+4nMAssay Description:Inhibition of [3H]-LTD4 binding to LTD4 receptor in guinea pig lung membranesMore data for this Ligand-Target Pair
Affinity DataKi: >3.00E+4nMAssay Description:Displacement of [3H]-leukotriene D4 (LTD4) from receptor in guinea pig lung membranesMore data for this Ligand-Target Pair
Affinity DataKi: >5.00E+4nMAssay Description:Displacement of [3H]-ligand from platelet activating factor (PAF) receptor in rabbit plateletsMore data for this Ligand-Target Pair
Affinity DataIC50: 0.400nMAssay Description:Binding affinity against leukotriene D4 receptor in [3H]-LTD4 binding assayMore data for this Ligand-Target Pair
Affinity DataIC50: 0.400nMAssay Description:Binding affinity against leukotriene D4 receptor in [3H]-LTD4 binding assayMore data for this Ligand-Target Pair
Affinity DataIC50: 0.400nMAssay Description:Binding affinity against leukotriene D4 receptor in [3H]-LTD4 binding assayMore data for this Ligand-Target Pair
Affinity DataIC50: 0.5nMAssay Description:Binding affinity against leukotriene D4 receptor in [3H]-LTD4 binding assayMore data for this Ligand-Target Pair
Affinity DataIC50: 0.5nMAssay Description:Binding affinity against leukotriene D4 receptor in [3H]-LTD4 binding assayMore data for this Ligand-Target Pair
Affinity DataIC50: 0.5nMAssay Description:Binding affinity against leukotriene D4 receptor in [3H]-LTD4 binding assayMore data for this Ligand-Target Pair
Affinity DataIC50: 0.5nMAssay Description:Binding affinity against leukotriene D4 receptor in [3H]-LTD4 binding assayMore data for this Ligand-Target Pair
Affinity DataIC50: 1nMAssay Description:Binding affinity against leukotriene D4 receptor in [3H]-LTD4 binding assayMore data for this Ligand-Target Pair
Affinity DataIC50: 1nMAssay Description:Binding affinity against leukotriene D4 receptor in [3H]-LTD4 binding assayMore data for this Ligand-Target Pair
Affinity DataIC50: 1nMAssay Description:Binding affinity against leukotriene D4 receptor in [3H]-LTD4 binding assayMore data for this Ligand-Target Pair
Affinity DataIC50: 2nMAssay Description:Binding affinity against leukotriene D4 receptor in [3H]-LTD4 binding assayMore data for this Ligand-Target Pair
Affinity DataIC50: 2nMAssay Description:Binding affinity against leukotriene D4 receptor in [3H]-LTD4 binding assayMore data for this Ligand-Target Pair
Affinity DataIC50: 3nMAssay Description:Displacement of [3H]rolipram from mouse brain homogenatesMore data for this Ligand-Target Pair
Affinity DataIC50: 3nMAssay Description:Displacement of [3H]rolipram from mouse brain homogenatesMore data for this Ligand-Target Pair
Affinity DataIC50: 4nMAssay Description:Displacement of [3H]rolipram from mouse brain homogenatesMore data for this Ligand-Target Pair
Affinity DataIC50: 5nMAssay Description:Displacement of [3H]rolipram from mouse brain homogenatesMore data for this Ligand-Target Pair
Affinity DataIC50: 9nMAssay Description:Displacement of [3H]rolipram from mouse brain homogenatesMore data for this Ligand-Target Pair
Affinity DataIC50: 15nMAssay Description:Displacement of [3H]rolipram from mouse brain homogenatesMore data for this Ligand-Target Pair
Affinity DataIC50: 15nMAssay Description:Displacement of [3H]rolipram from mouse brain homogenatesMore data for this Ligand-Target Pair
TargetcAMP-specific 3',5'-cyclic phosphodiesterase 4A/4B/4C/4D(Homo sapiens (Human))
Pfizer
Curated by ChEMBL
Pfizer
Curated by ChEMBL
Affinity DataIC50: 81nMAssay Description:Inhibition of Phosphodiesterase 4More data for this Ligand-Target Pair
TargetcAMP-specific 3',5'-cyclic phosphodiesterase 4A/4B/4C/4D(Homo sapiens (Human))
Pfizer
Curated by ChEMBL
Pfizer
Curated by ChEMBL
Affinity DataIC50: 110nMAssay Description:Inhibition of Phosphodiesterase 4More data for this Ligand-Target Pair
Affinity DataIC50: 111nMAssay Description:Displacement of [3H]rolipram from mouse brain homogenatesMore data for this Ligand-Target Pair
Affinity DataIC50: 129nMAssay Description:Displacement of [3H]rolipram from mouse brain homogenatesMore data for this Ligand-Target Pair
Affinity DataIC50: 130nMAssay Description:Displacement of [3H]rolipram from mouse brain homogenatesMore data for this Ligand-Target Pair
TargetcAMP-specific 3',5'-cyclic phosphodiesterase 4A/4B/4C/4D(Homo sapiens (Human))
Pfizer
Curated by ChEMBL
Pfizer
Curated by ChEMBL
Affinity DataIC50: 130nMAssay Description:Inhibition of Phosphodiesterase 4More data for this Ligand-Target Pair
TargetcAMP-specific 3',5'-cyclic phosphodiesterase 4A/4B/4C/4D(Homo sapiens (Human))
Pfizer
Curated by ChEMBL
Pfizer
Curated by ChEMBL
Affinity DataIC50: 130nMAssay Description:Inhibition of Phosphodiesterase 4More data for this Ligand-Target Pair
TargetcAMP-specific 3',5'-cyclic phosphodiesterase 4A/4B/4C/4D(Homo sapiens (Human))
Pfizer
Curated by ChEMBL
Pfizer
Curated by ChEMBL
Affinity DataIC50: 140nMAssay Description:Inhibition of Phosphodiesterase 4More data for this Ligand-Target Pair
Affinity DataIC50: 150nMAssay Description:Inhibition of 5-Lipoxygenase (5-LO) in rat basophilic leukemic cellsMore data for this Ligand-Target Pair
TargetcAMP-specific 3',5'-cyclic phosphodiesterase 4A/4B/4C/4D(Homo sapiens (Human))
Pfizer
Curated by ChEMBL
Pfizer
Curated by ChEMBL
Affinity DataIC50: 160nMAssay Description:Inhibition of Phosphodiesterase 4More data for this Ligand-Target Pair
TargetcAMP-specific 3',5'-cyclic phosphodiesterase 4A/4B/4C/4D(Homo sapiens (Human))
Pfizer
Curated by ChEMBL
Pfizer
Curated by ChEMBL
Affinity DataIC50: 300nMAssay Description:Inhibition of Phosphodiesterase 4More data for this Ligand-Target Pair
Affinity DataIC50: 323nMAssay Description:Displacement of [3H]rolipram from mouse brain homogenatesMore data for this Ligand-Target Pair