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Found 91 with Last Name = 'daniels' and Initial = 'aj'
TargetBombesin receptor subtype-3(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50275902(CHEMBL525577 | D-Phe-Gln-Trp-Ala-Val-b-Ala-His-Phe...)
Affinity DataKi:  0.360nMAssay Description:Binding affinity to BRS-3 receptor (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGastrin-releasing peptide receptor(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50275902(CHEMBL525577 | D-Phe-Gln-Trp-Ala-Val-b-Ala-His-Phe...)
Affinity DataKi:  0.990nMAssay Description:Binding affinity to gastrin releasing peptide receptor (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuromedin-B receptor(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50275902(CHEMBL525577 | D-Phe-Gln-Trp-Ala-Val-b-Ala-His-Phe...)
Affinity DataKi:  8.90nMAssay Description:Binding affinity to neuromedin B receptor (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptide Y receptor type 2(RAT)
Burroughs Wellcome

Curated by ChEMBL
LigandPNGBDBM50034128(CHEMBL441396 | Neuropeptide Y(NPY) | Tyr-Pro-Ser-L...)
Affinity DataIC50:  0.450nMAssay Description:50% displacement of specifically bound [3H]-NPY2 from rat brain membranes.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanin-concentrating hormone receptor 1(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50241083(6-(4-chlorophenyl)-3-(3-methoxy-4-(2-(pyrrolidin-1...)
Affinity DataIC50:  0.5nMAssay Description:Antagonist activity against human MCHR1 expressed in CHO cells by luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanin-concentrating hormone receptor 1(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50422940(CHEMBL213008)
Affinity DataIC50:  1nMAssay Description:Antagonist activity against human MCHR1 expressed in CHO cells by luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanin-concentrating hormone receptor 1(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50422936(CHEMBL212657)
Affinity DataIC50:  1.30nMAssay Description:Antagonist activity against human MCHR1 expressed in CHO cells by luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanin-concentrating hormone receptor 1(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50422927(CHEMBL441368)
Affinity DataIC50:  1.60nMAssay Description:Antagonist activity against human MCHR1 expressed in CHO cells by luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanin-concentrating hormone receptor 1(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50422930(CHEMBL214276)
Affinity DataIC50:  2nMAssay Description:Antagonist activity against human MCHR1 expressed in CHO cells by luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanin-concentrating hormone receptor 1(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50422924(CHEMBL214416)
Affinity DataIC50:  2.5nMAssay Description:Antagonist activity against human MCHR1 expressed in CHO cells by luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanin-concentrating hormone receptor 1(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50422926(CHEMBL215565)
Affinity DataIC50:  3.20nMAssay Description:Antagonist activity against human MCHR1 expressed in CHO cells by luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanin-concentrating hormone receptor 1(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50422939(CHEMBL439146)
Affinity DataIC50:  5nMAssay Description:Antagonist activity against human MCHR1 expressed in CHO cells by luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanin-concentrating hormone receptor 1(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50422932(CHEMBL212958)
Affinity DataIC50:  5nMAssay Description:Antagonist activity against human MCHR1 expressed in CHO cells by luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanin-concentrating hormone receptor 1(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50422933(CHEMBL212137)
Affinity DataIC50:  6.30nMAssay Description:Antagonist activity against human MCHR1 expressed in CHO cells by luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanin-concentrating hormone receptor 1(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50422922(CHEMBL384113)
Affinity DataIC50:  6.30nMAssay Description:Antagonist activity against human MCHR1 expressed in CHO cells by luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptide Y receptor type 2(RAT)
Burroughs Wellcome

Curated by ChEMBL
LigandPNGBDBM50034111(CHEMBL269515 | Tyr-Ile-Asn-Leu-Ile-Tyr-Arg-Leu-Arg...)
Affinity DataIC50:  8nMAssay Description:50% displacement of specifically bound [3H]-NPY2 from rat brain membranes.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptide Y receptor type 2(RAT)
Burroughs Wellcome

Curated by ChEMBL
LigandPNGBDBM50034118(CHEMBL274850 | His-Tyr-Ile-Asn-Leu-Ile-Tyr-Arg-Leu...)
Affinity DataIC50:  12nMAssay Description:50% displacement of specifically bound [3H]-NPY2 from rat brain membranes.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptide Y receptor type 2(RAT)
Burroughs Wellcome

Curated by ChEMBL
LigandPNGBDBM50034116(Arg-His-Tyr-Ile-Asn-Leu-Ile-Tyr-Arg-Leu-Arg-Tyr-NH...)
Affinity DataIC50:  12nMAssay Description:50% displacement of specifically bound [3H]-NPY2 from rat brain membranes.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanin-concentrating hormone receptor 1(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50422938(CHEMBL215862)
Affinity DataIC50:  13nMAssay Description:Antagonist activity against human MCHR1 expressed in CHO cells by luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptide Y receptor type 2(RAT)
Burroughs Wellcome

Curated by ChEMBL
LigandPNGBDBM50034125(CHEMBL265849 | Neuropeptide Y(NPY)(13-36) | Pro-Al...)
Affinity DataIC50:  15nMAssay Description:50% displacement of specifically bound [3H]-NPY2 from rat brain membranes.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanin-concentrating hormone receptor 1(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50422921(CHEMBL214429)
Affinity DataIC50:  20nMAssay Description:Antagonist activity against human MCHR1 expressed in CHO cells by luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanin-concentrating hormone receptor 1(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50422929(CHEMBL212883)
Affinity DataIC50:  25nMAssay Description:Antagonist activity against human MCHR1 expressed in CHO cells by luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanin-concentrating hormone receptor 1(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50422935(CHEMBL215334)
Affinity DataIC50:  25nMAssay Description:Antagonist activity against human MCHR1 expressed in CHO cells by luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptide Y receptor type 2(RAT)
Burroughs Wellcome

Curated by ChEMBL
LigandPNGBDBM50034127(CHEMBL409457 | Ile-Asn-Leu-Ile-Tyr-Arg-Leu-Arg-Tyr...)
Affinity DataIC50:  37nMAssay Description:50% displacement of specifically bound [3H]-NPY2 from rat brain membranes.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptide Y receptor type 2(RAT)
Burroughs Wellcome

Curated by ChEMBL
LigandPNGBDBM50034113(CHEMBL385246 | Tyr-Ile-Asn-Pro-Ile-Tyr-Arg-Leu-Arg...)
Affinity DataIC50:  44nMAssay Description:50% displacement of specifically bound [3H]-NPY2 from rat brain membranes.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptide Y receptor type 2(RAT)
Burroughs Wellcome

Curated by ChEMBL
LigandPNGBDBM50034123(CHEMBL439534 | NPY[Tyr32,Leu34])
Affinity DataIC50:  83nMAssay Description:50% displacement of specifically bound [3H]-NPY2 from rat brain membranes.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanin-concentrating hormone receptor 1(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50422923(CHEMBL387195)
Affinity DataIC50:  100nMAssay Description:Antagonist activity against human MCHR1 expressed in CHO cells by luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanin-concentrating hormone receptor 1(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50422928(CHEMBL214427)
Affinity DataIC50:  126nMAssay Description:Antagonist activity against human MCHR1 expressed in CHO cells by luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptide Y receptor type 2(RAT)
Burroughs Wellcome

Curated by ChEMBL
LigandPNGBDBM50034121(CHEMBL386823 | Ile-Asn-Pro-Ile-Tyr-Arg-Leu-Arg-Tyr...)
Affinity DataIC50:  174nMAssay Description:50% displacement of specifically bound [3H]-NPY2 from rat brain membranes.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanin-concentrating hormone receptor 1(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50422941(CHEMBL213154)
Affinity DataIC50:  200nMAssay Description:Antagonist activity against human MCHR1 expressed in CHO cells by luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptide Y receptor type 2(RAT)
Burroughs Wellcome

Curated by ChEMBL
LigandPNGBDBM50034120(Asn-Leu-Ile-Tyr-Arg-Leu-Arg-Tyr-NH2 | CHEMBL428097)
Affinity DataIC50:  310nMAssay Description:50% displacement of specifically bound [3H]-NPY2 from rat brain membranes.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptide Y receptor type 2(RAT)
Burroughs Wellcome

Curated by ChEMBL
LigandPNGBDBM50034126(CHEMBL439356 | Tyr-Ile-Asn-Leu-Leu-Tyr-Arg-Gln-Arg...)
Affinity DataIC50:  370nMAssay Description:50% displacement of specifically bound [3H]-NPY2 from rat brain membranes.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptide Y receptor type 2(RAT)
Burroughs Wellcome

Curated by ChEMBL
LigandPNGBDBM50034124(1N-[1-[4-amino(imino)methylamino-1-(1-{4-amino(imi...)
Affinity DataIC50:  400nMAssay Description:50% displacement of specifically bound [3H]-NPY2 from rat brain membranes.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanin-concentrating hormone receptor 1(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50422931(CHEMBL266415)
Affinity DataIC50:  1.26E+3nMAssay Description:Antagonist activity against human MCHR1 expressed in CHO cells by luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptide Y receptor type 2(RAT)
Burroughs Wellcome

Curated by ChEMBL
LigandPNGBDBM50034114(Arg-His-Tyr-Ile-Asn-Leu-Ile-Thr-Arg-Gln-Arg-Tyr-NH...)
Affinity DataIC50:  1.30E+3nMAssay Description:50% displacement of specifically bound [3H]-NPY2 from rat brain membranes.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanin-concentrating hormone receptor 1(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50422925(CHEMBL212963)
Affinity DataIC50:  1.59E+3nMAssay Description:Antagonist activity against human MCHR1 expressed in CHO cells by luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptide Y receptor type 2(RAT)
Burroughs Wellcome

Curated by ChEMBL
LigandPNGBDBM50034117(CHEMBL406275 | Tyr-Ile-Asn-Leu-Ile-Thr-Arg-Leu-Tyr...)
Affinity DataIC50:  2.10E+3nMAssay Description:50% displacement of specifically bound [3H]-NPY2 from rat brain membranes.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptide Y receptor type 2(RAT)
Burroughs Wellcome

Curated by ChEMBL
LigandPNGBDBM50034112(CHEMBL269544 | Tyr-Ile-Asn-Leu-Leu-Tyr-Arg-Pro-Arg...)
Affinity DataIC50:  2.70E+3nMAssay Description:50% displacement of specifically bound [3H]-NPY2 from rat brain membranes.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptide Y receptor type 2(RAT)
Burroughs Wellcome

Curated by ChEMBL
LigandPNGBDBM50034129(1N-[1-[4-amino(imino)methylamino-1-(1-{4-amino(imi...)
Affinity DataIC50:  2.95E+3nMAssay Description:50% displacement of specifically bound [3H]-NPY2 from rat brain membranes.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanin-concentrating hormone receptor 1(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50422937(CHEMBL377758)
Affinity DataIC50:  3.16E+3nMAssay Description:Antagonist activity against human MCHR1 expressed in CHO cells by luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanin-concentrating hormone receptor 1(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50422934(CHEMBL424723)
Affinity DataIC50:  3.98E+3nMAssay Description:Antagonist activity against human MCHR1 expressed in CHO cells by luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptide Y receptor type 2(RAT)
Burroughs Wellcome

Curated by ChEMBL
LigandPNGBDBM50034119(CHEMBL385245 | Tyr-Ile-Asn-Leu-Ile-Thr-Arg-Gln-Arg...)
Affinity DataIC50:  3.00E+4nMAssay Description:50% displacement of specifically bound [3H]-NPY2 from rat brain membranes.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptide Y receptor type 2(RAT)
Burroughs Wellcome

Curated by ChEMBL
LigandPNGBDBM50034115(1N-[1-carbamoyl-2-phenyl-(1S)-ethyl]-5-amino(imino...)
Affinity DataIC50:  4.00E+4nMAssay Description:50% displacement of specifically bound [3H]-NPY2 from rat brain membranes.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptide Y receptor type 2(RAT)
Burroughs Wellcome

Curated by ChEMBL
LigandPNGBDBM50034122(1N-{4-amino(imino)methylamino-1-[1-carbamoyl-2-(4-...)
Affinity DataIC50: >1.00E+5nMAssay Description:50% displacement of specifically bound [3H]-NPY2 from rat brain membranes.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBombesin receptor subtype-3(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50275736(6-methoxy-2-(naphthalen-2-ylmethylthio)-1H-benzo[d...)
Affinity DataEC50: >3.20E+4nMAssay Description:Agonist activity at recombinant BRS-3 receptor (unknown origin) expressed in baculovirus-transduced HEK293 cells assessed as intracellular calcium mo...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBombesin receptor subtype-3(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50275737(6-methoxy-2-(pyridin-4-ylmethylthio)-1H-benzo[d]im...)
Affinity DataEC50: >3.20E+4nMAssay Description:Agonist activity at recombinant BRS-3 receptor (unknown origin) expressed in baculovirus-transduced HEK293 cells assessed as intracellular calcium mo...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBombesin receptor subtype-3(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50275735(2-(3,5-dimethoxybenzylthio)-6-methoxy-1H-benzo[d]i...)
Affinity DataEC50:  1.60E+3nMAssay Description:Agonist activity at recombinant BRS-3 receptor (unknown origin) expressed in baculovirus-transduced HEK293 cells assessed as intracellular calcium mo...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBombesin receptor subtype-3(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50275689(2-(3,4-difluorobenzylthio)-6-methoxy-1H-benzo[d]im...)
Affinity DataEC50: >3.20E+4nMAssay Description:Agonist activity at recombinant BRS-3 receptor (unknown origin) expressed in baculovirus-transduced HEK293 cells assessed as intracellular calcium mo...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBombesin receptor subtype-3(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50241343((RS)-6-methoxy-2-((4-methoxy-3,5-dimethylpyridin-2...)
Affinity DataEC50:  1.40E+4nMAssay Description:Agonist activity at recombinant BRS-3 receptor (unknown origin) expressed in baculovirus-transduced HEK293 cells assessed as intracellular calcium mo...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBombesin receptor subtype-3(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50275787(2-(2-(6-chlorobenzo[d][1,3]dioxol-5-yl)ethyl)-6-me...)
Affinity DataEC50: >3.20E+4nMAssay Description:Agonist activity at recombinant BRS-3 receptor (unknown origin) expressed in baculovirus-transduced HEK293 cells assessed as intracellular calcium mo...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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