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Found 140 with Last Name = 'de frutos' and Initial = 'o'
TargetMelanocortin receptor 4(Homo sapiens (Human))
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50186127(CHEMBL378408 | N-[(R)-2-{4-[2-(acetyl-ethyl-amino)...)
Affinity DataKi:  2nMAssay Description:Inhibition of [125]I-NDP-alpha-MSH binding to human MC4R transfected in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanocortin receptor 4(Homo sapiens (Human))
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50186127(CHEMBL378408 | N-[(R)-2-{4-[2-(acetyl-ethyl-amino)...)
Affinity DataKi:  3nMAssay Description:Inhibition of [125]I-NDP-alpha-MSH binding to human MC4R transfected in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanocortin receptor 4(Homo sapiens (Human))
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50186127(CHEMBL378408 | N-[(R)-2-{4-[2-(acetyl-ethyl-amino)...)
Affinity DataKi:  3nMAssay Description:Inhibition of [125]I-NDP-alpha-MSH binding to human MC4R transfected in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanocortin receptor 4(Homo sapiens (Human))
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50186131((R)-N-((R)-3-(4-chlorophenyl)-1-(4-(1-cyclohexyl-2...)
Affinity DataKi:  4nMAssay Description:Inhibition of [125]I-NDP-alpha-MSH binding to human MC4R transfected in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanocortin receptor 4(Homo sapiens (Human))
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50186121((R)-N-((R)-3-(4-chlorophenyl)-1-(4-(1-cyclopentyl-...)
Affinity DataKi:  4nMAssay Description:Inhibition of [125]I-NDP-alpha-MSH binding to human MC4R transfected in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanocortin receptor 4(Homo sapiens (Human))
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50186128(CHEMBL209990 | N-((R)-3-(4-chlorophenyl)-1-(4-(1-c...)
Affinity DataKi:  5nMAssay Description:Inhibition of [125]I-NDP-alpha-MSH binding to human MC4R transfected in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanocortin receptor 4(Homo sapiens (Human))
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50186125(CHEMBL377825 | N-((R)-3-(4-chlorophenyl)-1-(4-(3-c...)
Affinity DataKi:  5nMAssay Description:Inhibition of [125]I-NDP-alpha-MSH binding to human MC4R transfected in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanocortin receptor 4(Homo sapiens (Human))
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50186128(CHEMBL209990 | N-((R)-3-(4-chlorophenyl)-1-(4-(1-c...)
Affinity DataKi:  5nMAssay Description:Inhibition of [125]I-NDP-alpha-MSH binding to human MC4R transfected in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanocortin receptor 4(Homo sapiens (Human))
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50186124(CHEMBL410087 | N-((R)-3-(4-chlorophenyl)-1-(4-(1-c...)
Affinity DataKi:  6nMAssay Description:Inhibition of [125]I-NDP-alpha-MSH binding to human MC4R transfected in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanocortin receptor 4(Homo sapiens (Human))
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50186124(CHEMBL410087 | N-((R)-3-(4-chlorophenyl)-1-(4-(1-c...)
Affinity DataKi:  6nMAssay Description:Inhibition of [125]I-NDP-alpha-MSH binding to human MC4R transfected in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanocortin receptor 4(Homo sapiens (Human))
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50186138(CHEMBL425609 | N-((R)-3-(4-chlorophenyl)-1-(4-(1-c...)
Affinity DataKi:  7nMAssay Description:Inhibition of [125]I-NDP-alpha-MSH binding to human MC4R transfected in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanocortin receptor 4(Homo sapiens (Human))
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50186122(CHEMBL377313 | N-((R)-3-(4-chlorophenyl)-1-(4-(3-c...)
Affinity DataKi:  10nMAssay Description:Inhibition of [125]I-NDP-alpha-MSH binding to human MC4R transfected in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanocortin receptor 4(Homo sapiens (Human))
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50186120(CHEMBL380391 | N-((R)-3-(4-chlorophenyl)-1-(4-(1-(...)
Affinity DataKi:  12nMAssay Description:Inhibition of [125]I-NDP-alpha-MSH binding to human MC4R transfected in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanocortin receptor 4(Homo sapiens (Human))
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50186135((R)-N-((R)-3-(4-chlorophenyl)-1-(4-(3-cyclohexyl-1...)
Affinity DataKi:  13nMAssay Description:Inhibition of [125]I-NDP-alpha-MSH binding to human MC4R transfected in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanocortin receptor 4(Homo sapiens (Human))
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50186119((R)-N-((R)-3-(4-chlorophenyl)-1-(4-(1-cycloheptyl-...)
Affinity DataKi:  13nMAssay Description:Inhibition of [125]I-NDP-alpha-MSH binding to human MC4R transfected in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanocortin receptor 4(Homo sapiens (Human))
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50186133(3,4-Dihydro-1H-isoquinoline-2-carboxylic acid ((R)...)
Affinity DataKi:  14nMAssay Description:Inhibition of [125]I-NDP-alpha-MSH binding to human MC4R transfected in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanocortin receptor 4(Homo sapiens (Human))
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50174056(CHEMBL381015 | Diethyl-[(S)-2-(2-fluoro-phenyl)-2-...)
Affinity DataKi:  14nMAssay Description:Inhibition of [125I]-NDP MSH binding to human Melanocortin 4 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanocortin receptor 4(Homo sapiens (Human))
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50139027((R)-1,2,3,4-Tetrahydro-isoquinoline-3-carboxylic a...)
Affinity DataKi:  14nMAssay Description:Inhibition of [125I]-NDP MSH binding to human Melanocortin 4 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanocortin receptor 4(Homo sapiens (Human))
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50186132(CHEMBL378411 | N-((R)-3-(4-chlorophenyl)-1-(4-(1-c...)
Affinity DataKi:  18nMAssay Description:Inhibition of [125]I-NDP-alpha-MSH binding to human MC4R transfected in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanocortin receptor 4(Homo sapiens (Human))
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50186126(CHEMBL379051 | N-((R)-3-(4-chlorophenyl)-1-(4-(2,6...)
Affinity DataKi:  18nMAssay Description:Inhibition of [125]I-NDP-alpha-MSH binding to human MC4R transfected in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanocortin receptor 4(Homo sapiens (Human))
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50186132(CHEMBL378411 | N-((R)-3-(4-chlorophenyl)-1-(4-(1-c...)
Affinity DataKi:  18nMAssay Description:Inhibition of [125]I-NDP-alpha-MSH binding to human MC4R transfected in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanocortin receptor 4(Homo sapiens (Human))
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50174055(CHEMBL198379 | Diethyl-[2-(2-fluoro-phenyl)-2-(4-m...)
Affinity DataKi:  20nMAssay Description:Inhibition of [125I]-NDP MSH binding to human Melanocortin 4 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanocortin receptor 4(Homo sapiens (Human))
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50177561((R)-N-((R)-3-(4-chlorophenyl)-1-(4-(2-(diethylamin...)
Affinity DataKi:  20nMAssay Description:Inhibition of [125]I-NDP-alpha-MSH binding to human MC4R transfected in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanocortin receptor 4(Homo sapiens (Human))
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50186134(CHEMBL209559 | N-((R)-3-(4-chlorophenyl)-1-(4-(1-c...)
Affinity DataKi:  26nMAssay Description:Inhibition of [125]I-NDP-alpha-MSH binding to human MC4R transfected in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanocortin receptor 4(Homo sapiens (Human))
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50186130(CHEMBL211078 | N-((R)-3-(4-chlorophenyl)-1-(4-(dic...)
Affinity DataKi:  35nMAssay Description:Inhibition of [125]I-NDP-alpha-MSH binding to human MC4R transfected in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanocortin receptor 4(Homo sapiens (Human))
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50174062(CHEMBL371896 | Diethyl-[2-(4-methyl-piperazin-1-yl...)
Affinity DataKi:  40nMAssay Description:Inhibition of [125I]-NDP MSH binding to human Melanocortin 4 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanocortin receptor 4(Homo sapiens (Human))
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50174050(CHEMBL365184 | Diethyl-[2-(4-methyl-piperazin-1-yl...)
Affinity DataKi:  40nMAssay Description:Inhibition of [125I]-NDP MSH binding to human Melanocortin 4 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanocortin receptor 4(Homo sapiens (Human))
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50174045(CHEMBL373042 | Diethyl-[(R)-2-(4-methyl-piperazin-...)
Affinity DataKi:  50nMAssay Description:Inhibition of [125I]-NDP MSH binding to human Melanocortin 4 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanocortin receptor 4(Homo sapiens (Human))
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50186118(CHEMBL209325 | N-((R)-3-(4-chlorophenyl)-1-(4-(1-c...)
Affinity DataKi:  54nMAssay Description:Inhibition of [125]I-NDP-alpha-MSH binding to human MC4R transfected in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanocortin receptor 4(Homo sapiens (Human))
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50174060(CHEMBL198320 | [2-(2-Chloro-phenyl)-2-(4-methyl-pi...)
Affinity DataKi:  70nMAssay Description:Inhibition of [125I]-NDP MSH binding to human Melanocortin 4 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanocortin receptor 4(Homo sapiens (Human))
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50174053(CHEMBL198378 | Diethyl-[2-(4-methyl-piperazin-1-yl...)
Affinity DataKi:  70nMAssay Description:Inhibition of [125I]-NDP MSH binding to human Melanocortin 4 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanocortin receptor 4(Homo sapiens (Human))
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50186136((R)-N-((R)-3-(4-chlorophenyl)-1-(4-(1-((diethylami...)
Affinity DataKi:  70nMAssay Description:Inhibition of [125]I-NDP-alpha-MSH binding to human MC4R transfected in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanocortin receptor 4(Homo sapiens (Human))
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50174065(CHEMBL448473 | Diethyl-[2-(4-methyl-piperazin-1-yl...)
Affinity DataKi:  90nMAssay Description:Inhibition of [125I]-NDP MSH binding to human Melanocortin 4 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanocortin receptor 4(Homo sapiens (Human))
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50174061(CHEMBL197288 | [2-(2,4-Difluoro-phenyl)-2-(4-methy...)
Affinity DataKi:  100nMAssay Description:Inhibition of [125I]-NDP MSH binding to human Melanocortin 4 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanocortin receptor 4(Homo sapiens (Human))
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50174048(CHEMBL197820 | N-Ethyl-N-[2-(2-fluoro-phenyl)-2-(4...)
Affinity DataKi:  106nMAssay Description:Inhibition of [125I]-NDP MSH binding to human Melanocortin 4 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanocortin receptor 4(Homo sapiens (Human))
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50174057(CHEMBL194464 | Diethyl-[2-(4-methyl-piperazin-1-yl...)
Affinity DataKi:  110nMAssay Description:Inhibition of [125I]-NDP MSH binding to human Melanocortin 4 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanocortin receptor 4(Homo sapiens (Human))
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50174054(CHEMBL199192 | Diethyl-[(R)-2-(2-fluoro-phenyl)-2-...)
Affinity DataKi:  111nMAssay Description:Inhibition of [125I]-NDP MSH binding to human Melanocortin 4 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanocortin receptor 4(Homo sapiens (Human))
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50174051(CHEMBL198319 | N,N-Diethyl-2-(2-fluoro-phenyl)-2-(...)
Affinity DataKi:  125nMAssay Description:Inhibition of [125I]-NDP MSH binding to human Melanocortin 4 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanocortin receptor 4(Homo sapiens (Human))
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50174047(CHEMBL195998 | Diethyl-[2-(4-methyl-piperazin-1-yl...)
Affinity DataKi:  130nMAssay Description:Inhibition of [125I]-NDP MSH binding to human Melanocortin 4 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanocortin receptor 4(Homo sapiens (Human))
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50186129(2-{4-[(R)-3-(4-chloro-phenyl)-2-(2-2,3-dihydro-1H-...)
Affinity DataKi:  148nMAssay Description:Inhibition of [125]I-NDP-alpha-MSH binding to human MC4R transfected in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanocortin receptor 4(Homo sapiens (Human))
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50174052(CHEMBL199071 | [2-(2,6-Difluoro-phenyl)-2-(4-methy...)
Affinity DataKi:  150nMAssay Description:Inhibition of [125I]-NDP MSH binding to human Melanocortin 4 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanocortin receptor 4(Homo sapiens (Human))
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50174059(CHEMBL194761 | Diethyl-[2-(4-methyl-piperazin-1-yl...)
Affinity DataKi:  150nMAssay Description:Inhibition of [125I]-NDP MSH binding to human Melanocortin 4 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanocortin receptor 4(Homo sapiens (Human))
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50174068(CHEMBL198607 | N-Ethyl-N-[2-(2-fluoro-phenyl)-2-(4...)
Affinity DataKi:  157nMAssay Description:Inhibition of [125I]-NDP MSH binding to human Melanocortin 4 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanocortin receptor 4(Homo sapiens (Human))
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50174043(CHEMBL371105 | Diethyl-[2-(2-methoxy-phenyl)-2-(4-...)
Affinity DataKi:  190nMAssay Description:Inhibition of [125I]-NDP MSH binding to human Melanocortin 4 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanocortin receptor 4(Homo sapiens (Human))
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50174046(CHEMBL197859 | Diethyl-[(S)-2-(4-methyl-piperazin-...)
Affinity DataKi:  190nMAssay Description:Inhibition of [125I]-NDP MSH binding to human Melanocortin 4 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanocortin receptor 4(Homo sapiens (Human))
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50174049(CHEMBL199003 | Diethyl-[2-(4-methyl-piperazin-1-yl...)
Affinity DataKi:  200nMAssay Description:Inhibition of [125I]-NDP MSH binding to human Melanocortin 4 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanocortin receptor 4(Homo sapiens (Human))
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50174058(CHEMBL198606 | Ethyl-[2-(2-fluoro-phenyl)-2-(4-met...)
Affinity DataKi:  261nMAssay Description:Inhibition of [125I]-NDP MSH binding to human Melanocortin 4 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanocortin receptor 4(Homo sapiens (Human))
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50186123(CHEMBL378568 | N-((R)-3-(4-chlorophenyl)-1-(4-(1,3...)
Affinity DataKi:  326nMAssay Description:Inhibition of [125]I-NDP-alpha-MSH binding to human MC4R transfected in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanocortin receptor 4(Homo sapiens (Human))
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50174063(CHEMBL198665 | N-[2-(2-Fluoro-phenyl)-2-(4-methyl-...)
Affinity DataKi:  467nMAssay Description:Inhibition of [125I]-NDP MSH binding to human Melanocortin 4 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanocortin receptor 4(Homo sapiens (Human))
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50174067(CHEMBL198544 | N-[2-(2-Fluoro-phenyl)-2-(4-methyl-...)
Affinity DataKi:  472nMAssay Description:Inhibition of [125I]-NDP MSH binding to human Melanocortin 4 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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