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Found 59 with Last Name = 'de ryck' and Initial = 'm'
TargetCannabinoid receptor 1(Homo sapiens (Human))
Ucb Pharma

Curated by ChEMBL
LigandPNGBDBM50234380(CHEMBL245876 | quinolin-8-yl 4-methyl-3-(piperidin...)
Affinity DataIC50:  0.790nMAssay Description:Binding affinity to human recombinant CB1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Ucb Pharma

Curated by ChEMBL
LigandPNGBDBM50423205(CHEMBL245878)
Affinity DataIC50:  1.30nMAssay Description:Binding affinity to human recombinant CB1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Ucb Pharma

Curated by ChEMBL
LigandPNGBDBM50072775(2-((1R,2R,5R)-5-hydroxy-2-(3-hydroxypropyl)cyclohe...)
Affinity DataIC50:  2.5nMAssay Description:Binding affinity to human recombinant CB1 receptorMore data for this Ligand-Target Pair
TargetCannabinoid receptor 1(Homo sapiens (Human))
Ucb Pharma

Curated by ChEMBL
LigandPNGBDBM50423209(CHEMBL247331)
Affinity DataIC50:  16nMAssay Description:Binding affinity to human recombinant CB1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Ucb Pharma

Curated by ChEMBL
LigandPNGBDBM50423204(CHEMBL246922)
Affinity DataIC50:  32nMAssay Description:Binding affinity to human recombinant CB1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAurora kinase B(Homo sapiens (Human))
University Of Dundee

Curated by ChEMBL
LigandPNGBDBM50463653(CHEMBL4241707)
Affinity DataIC50:  40nMAssay Description:Inhibition of aurora B (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Ucb Pharma

Curated by ChEMBL
LigandPNGBDBM50423207(CHEMBL393018)
Affinity DataIC50:  40nMAssay Description:Binding affinity to human recombinant CB1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Ucb Pharma

Curated by ChEMBL
LigandPNGBDBM50423202(CHEMBL393224)
Affinity DataIC50:  50nMAssay Description:Binding affinity to human recombinant CB1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Ucb Pharma

Curated by ChEMBL
LigandPNGBDBM50463653(CHEMBL4241707)
Affinity DataIC50:  63nMAssay Description:Inhibition of CB1 (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Ucb Pharma

Curated by ChEMBL
LigandPNGBDBM21281((11R)-2-methyl-11-(morpholin-4-ylmethyl)-3-(naphth...)
Affinity DataIC50:  63nMAssay Description:Binding affinity to human recombinant CB1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase 15(Homo sapiens (Human))
University Of Dundee

Curated by ChEMBL
LigandPNGBDBM50548060(CHEMBL4762609)
Affinity DataIC50:  110nMAssay Description:Inhibition of human ERK8 (2 to 544 residues) incubated for 5 mins in presence of [gamma33P]ATP by scintillation counting analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCyclin-dependent kinase 2(Homo sapiens (Human))
University Of Dundee

Curated by ChEMBL
LigandPNGBDBM50384600(CHEMBL2036792 | US9744172, Compound UNC00000563A)
Affinity DataIC50:  114nMAssay Description:Inhibition of CDK2 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Ucb Pharma

Curated by ChEMBL
LigandPNGBDBM50423216(CHEMBL247332)
Affinity DataIC50:  158nMAssay Description:Binding affinity to human recombinant CB1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCyclin-dependent kinase 4(Homo sapiens (Human))
University Of Dundee

Curated by ChEMBL
LigandPNGBDBM50384600(CHEMBL2036792 | US9744172, Compound UNC00000563A)
Affinity DataIC50:  199nMAssay Description:Inhibition of CDK4 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Ucb Pharma

Curated by ChEMBL
LigandPNGBDBM50423208(CHEMBL246302)
Affinity DataIC50:  200nMAssay Description:Binding affinity to human recombinant CB1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Ucb Pharma

Curated by ChEMBL
LigandPNGBDBM50423214(CHEMBL427873)
Affinity DataIC50:  398nMAssay Description:Binding affinity to human recombinant CB1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase 11(Homo sapiens (Human))
University Of Dundee

Curated by ChEMBL
LigandPNGBDBM50548060(CHEMBL4762609)
Affinity DataIC50:  550nMAssay Description:Inhibition of human p38beta MAPK (1 to 364 residues) incubated for 5 mins in presence of [gamma33P]ATP by scintillation counting analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Ucb Pharma

Curated by ChEMBL
LigandPNGBDBM50423213(CHEMBL248344)
Affinity DataIC50:  1.26E+3nMAssay Description:Binding affinity to human recombinant CB1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Ucb Pharma

Curated by ChEMBL
LigandPNGBDBM50423217(CHEMBL246923)
Affinity DataIC50:  1.26E+3nMAssay Description:Binding affinity to human recombinant CB1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Ucb Pharma

Curated by ChEMBL
LigandPNGBDBM50423203(CHEMBL246095)
Affinity DataIC50:  1.59E+3nMAssay Description:Binding affinity to human recombinant CB1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Ucb Pharma

Curated by ChEMBL
LigandPNGBDBM50423201(CHEMBL246303)
Affinity DataIC50:  1.59E+3nMAssay Description:Binding affinity to human recombinant CB1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Ucb Pharma

Curated by ChEMBL
LigandPNGBDBM50423206(CHEMBL395672)
Affinity DataIC50:  2.00E+3nMAssay Description:Binding affinity to human recombinant CB1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Ucb Pharma

Curated by ChEMBL
LigandPNGBDBM70185(4-methyl-N-(5-methyl-2-pyridinyl)-3-(1-piperidinyl...)
Affinity DataIC50:  3.16E+3nMAssay Description:Binding affinity to human recombinant CB1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Ucb Pharma

Curated by ChEMBL
LigandPNGBDBM50234402(4-methyl-N-phenyl-3-(piperidin-1-ylsulfonyl)benzam...)
Affinity DataIC50:  3.16E+3nMAssay Description:Binding affinity to human recombinant CB1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Ucb Pharma

Curated by ChEMBL
LigandPNGBDBM50423200(CHEMBL246713)
Affinity DataIC50:  3.16E+3nMAssay Description:Binding affinity to human recombinant CB1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Ucb Pharma

Curated by ChEMBL
LigandPNGBDBM50423211(CHEMBL245891)
Affinity DataIC50:  3.98E+3nMAssay Description:Binding affinity to human recombinant CB1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] A(Homo sapiens (Human))
University Of Dundee

Curated by ChEMBL
LigandPNGBDBM50542902(CHEMBL4645906)
Affinity DataIC50:  3.98E+3nMAssay Description:Inhibition of MAOA (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
University Of Dundee

Curated by ChEMBL
LigandPNGBDBM50463653(CHEMBL4241707)
Affinity DataIC50:  3.98E+3nMAssay Description:Inhibition of human ERGMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
University Of Dundee

Curated by ChEMBL
LigandPNGBDBM50613723(CHEMBL5268330)
Affinity DataIC50:  5.00E+3nMAssay Description:Inhibition of hERG potassium channel by Q-patch clamp assayMore data for this Ligand-Target Pair
Ligand Info
In DepthDetails PubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
University Of Dundee

Curated by ChEMBL
LigandPNGBDBM50463654(CHEMBL4241692)
Affinity DataIC50:  5.01E+3nMAssay Description:Inhibition of human ERGMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Ucb Pharma

Curated by ChEMBL
LigandPNGBDBM50423215(CHEMBL246093)
Affinity DataIC50:  5.01E+3nMAssay Description:Binding affinity to human recombinant CB1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
University Of Dundee

Curated by ChEMBL
LigandPNGBDBM50613719(CHEMBL5281165)
Affinity DataIC50:  6.00E+3nMAssay Description:Inhibition of hERG potassium channel by Q-patch clamp assayMore data for this Ligand-Target Pair
Ligand Info
In DepthDetails PubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Ucb Pharma

Curated by ChEMBL
LigandPNGBDBM50423212(CHEMBL248345)
Affinity DataIC50:  6.31E+3nMAssay Description:Binding affinity to human recombinant CB1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCytochrome P450 3A4(Homo sapiens (Human))
University Of Dundee

Curated by ChEMBL
LigandPNGBDBM50517286(CHEMBL4516798)
Affinity DataIC50:  6.31E+3nMAssay Description:Inhibition of CYP3A4 in human liver microsomes using midazolam as substrate preincubated for 20 mins followed by substrate addition and measured afte...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
University Of Dundee

Curated by ChEMBL
LigandPNGBDBM50613721(CHEMBL5275547)
Affinity DataIC50:  7.00E+3nMAssay Description:Inhibition of hERG potassium channel by Q-patch clamp assayMore data for this Ligand-Target Pair
Ligand Info
In DepthDetails PubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Ucb Pharma

Curated by ChEMBL
LigandPNGBDBM50423210(CHEMBL248140)
Affinity DataIC50:  7.94E+3nMAssay Description:Binding affinity to human recombinant CB1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSterol 14-alpha demethylase(Trypanosoma cruzi)
University Of Dundee

Curated by ChEMBL
LigandPNGBDBM50463655(CHEMBL546608 | TCMDC-124726)
Affinity DataIC50: <1.00E+4nMAssay Description:Inhibition of Trypanosoma cruzi CYP51More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCytochrome P450 2D6(Homo sapiens (Human))TBA
LigandPNGBDBM50613725(CHEMBL5268278)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of CYP2D6 (unknown origin)More data for this Ligand-Target Pair
Ligand Info
In DepthDetails PubMed
TargetCytochrome P450 2C9(Homo sapiens (Human))TBA
LigandPNGBDBM50613725(CHEMBL5268278)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of CYP2C9 (unknown origin)More data for this Ligand-Target Pair
Ligand Info
In DepthDetails PubMed
TargetCytochrome P450 2C19(Homo sapiens (Human))TBA
LigandPNGBDBM50613725(CHEMBL5268278)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of CYP2C19 (unknown origin)More data for this Ligand-Target Pair
Ligand Info
In DepthDetails PubMed
TargetCytochrome P450 1A2(Homo sapiens (Human))TBA
LigandPNGBDBM50613725(CHEMBL5268278)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of CYP1A2 (unknown origin)More data for this Ligand-Target Pair
Ligand Info
In DepthDetails PubMed
TargetCytochrome P450 3A4(Homo sapiens (Human))
University Of Dundee

Curated by ChEMBL
LigandPNGBDBM50613725(CHEMBL5268278)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of CYP3A4 (unknown origin)More data for this Ligand-Target Pair
Ligand Info
In DepthDetails PubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
University Of Dundee

Curated by ChEMBL
LigandPNGBDBM50517286(CHEMBL4516798)
Affinity DataIC50:  1.75E+4nMAssay Description:Inhibition of human ERG by patch clamp assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
University Of Dundee

Curated by ChEMBL
LigandPNGBDBM50613720(CHEMBL5283073)
Affinity DataIC50:  1.80E+4nMAssay Description:Inhibition of hERG potassium channel by Q-patch clamp assayMore data for this Ligand-Target Pair
Ligand Info
In DepthDetails PubMed
TargetCyclin-dependent kinase 4(Homo sapiens (Human))
University Of Dundee

Curated by ChEMBL
LigandPNGBDBM50517285(CHEMBL4572962)
Affinity DataIC50: >2.00E+4nMAssay Description:Inhibition of human CDK4 by kinobeads-based assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
University Of Dundee

Curated by ChEMBL
LigandPNGBDBM50613716(CHEMBL5283476)
Affinity DataIC50:  2.30E+4nMAssay Description:Inhibition of hERG potassium channel by Q-patch clamp assayMore data for this Ligand-Target Pair
Ligand Info
In DepthDetails PubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
University Of Dundee

Curated by ChEMBL
LigandPNGBDBM50613725(CHEMBL5268278)
Affinity DataIC50:  2.40E+4nMAssay Description:Inhibition of hERG potassium channel by Q-patch clamp assayMore data for this Ligand-Target Pair
Ligand Info
In DepthDetails PubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
University Of Dundee

Curated by ChEMBL
LigandPNGBDBM50613718(CHEMBL5286709)
Affinity DataIC50: >3.00E+4nMAssay Description:Inhibition of hERG potassium channel by Q-patch clamp assayMore data for this Ligand-Target Pair
Ligand Info
In DepthDetails PubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
University Of Dundee

Curated by ChEMBL
LigandPNGBDBM50613726(CHEMBL5272922)
Affinity DataIC50: >3.00E+4nMAssay Description:Inhibition of hERG potassium channel by Q-patch clamp assayMore data for this Ligand-Target Pair
Ligand Info
In DepthDetails PubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
University Of Dundee

Curated by ChEMBL
LigandPNGBDBM50517285(CHEMBL4572962)
Affinity DataIC50: >3.00E+4nMAssay Description:Inhibition of human ERG by patch clamp assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
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