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Found 127 with Last Name = 'de souza' and Initial = 'eb'
TargetCorticotropin-releasing factor receptor 1(Homo sapiens (Human))
Neurocrine Biosciences

Curated by ChEMBL
LigandPNGBDBM50054245(5-Chloro-N-cyclopropylmethyl-2-methyl-N-propyl-N''...)
Affinity DataKi:  1.70nMAssay Description:Inhibition of [125I]-CRF binding to human Corticotropin releasing factor receptor 1 tested at 6-12 dosesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCorticotropin-releasing factor receptor 1(Homo sapiens (Human))
Neurocrine Biosciences

Curated by ChEMBL
LigandPNGBDBM50074349((2-Bromo-4-isopropyl-phenyl)-ethyl-[4-(1-ethyl-pro...)
Affinity DataKi:  2nMAssay Description:Binding affinity for human recombinant corticotropin releasing factor receptor 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCorticotropin-releasing factor receptor 1(Homo sapiens (Human))
Neurocrine Biosciences

Curated by ChEMBL
LigandPNGBDBM50054252(5-Bromo-N-cyclopropylmethyl-2-methyl-N-propyl-N'-(...)
Affinity DataKi:  2nMAssay Description:Inhibition of [125I]-CRF binding to human Corticotropin releasing factor receptor 1 tested at 6-12 dosesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCorticotropin-releasing factor receptor 1(Homo sapiens (Human))
Neurocrine Biosciences

Curated by ChEMBL
LigandPNGBDBM50054250(CHEMBL306482 | N-Cyclopropylmethyl-2,5-dimethyl-N-...)
Affinity DataKi:  2.30nMAssay Description:Inhibition of [125I]-CRF binding to human Corticotropin releasing factor receptor 1 tested at 6-12 dosesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCorticotropin-releasing factor receptor 1(Homo sapiens (Human))
Neurocrine Biosciences

Curated by ChEMBL
LigandPNGBDBM50054248(2,5-Dimethyl-N,N-dipropyl-N'-(2,4,6-trichloro-phen...)
Affinity DataKi:  2.5nMAssay Description:Inhibition of [125I]-CRF binding to human Corticotropin releasing factor receptor 1 tested at 6-12 dosesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCorticotropin-releasing factor receptor 1(Homo sapiens (Human))
Neurocrine Biosciences

Curated by ChEMBL
LigandPNGBDBM50074354(CHEMBL168131 | N,N-Diallyl-N'-(2-bromo-4-dimethyla...)
Affinity DataKi:  3nMAssay Description:Binding affinity for human recombinant corticotropin releasing factor receptor 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCorticotropin-releasing factor receptor 1(Homo sapiens (Human))
Neurocrine Biosciences

Curated by ChEMBL
LigandPNGBDBM50054253(CHEMBL77716 | N-Cyclopropylmethyl-5-ethyl-2-methyl...)
Affinity DataKi:  3.80nMAssay Description:Inhibition of [125I]-CRF binding to human Corticotropin releasing factor receptor 1 tested at 6-12 dosesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCorticotropin-releasing factor receptor 1(Homo sapiens (Human))
Neurocrine Biosciences

Curated by ChEMBL
LigandPNGBDBM50074404(CHEMBL168844 | N-(2-Bromo-4-isopropyl-phenyl)-N-et...)
Affinity DataKi:  4nMAssay Description:Binding affinity for human recombinant corticotropin releasing factor receptor 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCorticotropin-releasing factor receptor 1(Homo sapiens (Human))
Neurocrine Biosciences

Curated by ChEMBL
LigandPNGBDBM50074332(CHEMBL167463 | N,N-Diallyl-N'-(2-bromo-4-trifluoro...)
Affinity DataKi:  4nMAssay Description:Binding affinity for human recombinant corticotropin releasing factor receptor 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCorticotropin-releasing factor receptor 1(Homo sapiens (Human))
Neurocrine Biosciences

Curated by ChEMBL
LigandPNGBDBM50074391(CHEMBL424555 | N,N-Diallyl-N'-(2-bromo-4-isopropyl...)
Affinity DataKi:  4nMAssay Description:Binding affinity for human recombinant corticotropin releasing factor receptor 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCorticotropin-releasing factor receptor 1(Homo sapiens (Human))
Neurocrine Biosciences

Curated by ChEMBL
LigandPNGBDBM50074338(2-Bromo-N*1*-(4,6-dimethyl-pyrimidin-2-yl)-N*1*-et...)
Affinity DataKi:  5nMAssay Description:Binding affinity for human recombinant corticotropin releasing factor receptor 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCorticotropin-releasing factor receptor 1(Homo sapiens (Human))
Neurocrine Biosciences

Curated by ChEMBL
LigandPNGBDBM50074375(CHEMBL354395 | N,N-Bis-cyclopropylmethyl-N'-(4-dim...)
Affinity DataKi:  5nMAssay Description:Binding affinity for human recombinant corticotropin releasing factor receptor 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCorticotropin-releasing factor receptor 1(Homo sapiens (Human))
Neurocrine Biosciences

Curated by ChEMBL
LigandPNGBDBM50074336(1-{3-Bromo-4-[(4-diethylamino-6-methyl-pyrimidin-2...)
Affinity DataKi:  5nMAssay Description:Binding affinity for human recombinant corticotropin releasing factor receptor 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCorticotropin-releasing factor receptor 1(Homo sapiens (Human))
Neurocrine Biosciences

Curated by ChEMBL
LigandPNGBDBM50074384(CHEMBL167428 | N-Cyclopropylmethyl-N'-(4-dimethyla...)
Affinity DataKi:  5nMAssay Description:Binding affinity for human recombinant corticotropin releasing factor receptor 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCorticotropin-releasing factor receptor 1(Homo sapiens (Human))
Neurocrine Biosciences

Curated by ChEMBL
LigandPNGBDBM50074330(3-({4-[(4-Dimethylamino-2-trifluoromethyl-phenyl)-...)
Affinity DataKi:  5nMAssay Description:Binding affinity for human recombinant corticotropin releasing factor receptor 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCorticotropin-releasing factor receptor 1(Homo sapiens (Human))
Neurocrine Biosciences

Curated by ChEMBL
LigandPNGBDBM50074333(CHEMBL353877 | N*2*-(2-Bromo-4-isopropyl-phenyl)-N...)
Affinity DataKi:  5nMAssay Description:Binding affinity for human recombinant corticotropin releasing factor receptor 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCorticotropin-releasing factor receptor 1(Homo sapiens (Human))
Neurocrine Biosciences

Curated by ChEMBL
LigandPNGBDBM50074401(CHEMBL166345 | N-Allyl-N'-(2-bromo-4-isopropyl-phe...)
Affinity DataKi:  5nMAssay Description:Binding affinity for human recombinant corticotropin releasing factor receptor 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCorticotropin-releasing factor receptor 1(Homo sapiens (Human))
Neurocrine Biosciences

Curated by ChEMBL
LigandPNGBDBM50074399(CHEMBL354367 | N-(2-Bromo-4-trifluoromethoxy-pheny...)
Affinity DataKi:  5nMAssay Description:Binding affinity for human recombinant corticotropin releasing factor receptor 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCorticotropin-releasing factor receptor 1(Homo sapiens (Human))
Neurocrine Biosciences

Curated by ChEMBL
LigandPNGBDBM50074397(CHEMBL166388 | N-(2-Bromo-4-isopropyl-phenyl)-N'-b...)
Affinity DataKi:  5nMAssay Description:Binding affinity for human recombinant corticotropin releasing factor receptor 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCorticotropin-releasing factor receptor 1(Homo sapiens (Human))
Neurocrine Biosciences

Curated by ChEMBL
LigandPNGBDBM50074347((Butyl-{4-[(4-dimethylamino-2-trifluoromethyl-phen...)
Affinity DataKi:  6nMAssay Description:Binding affinity for human recombinant corticotropin releasing factor receptor 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCorticotropin-releasing factor receptor 1(Homo sapiens (Human))
Neurocrine Biosciences

Curated by ChEMBL
LigandPNGBDBM50074388(CHEMBL168497 | N-(4-Dimethylamino-2-trifluoromethy...)
Affinity DataKi:  6nMAssay Description:Binding affinity for human recombinant corticotropin releasing factor receptor 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCorticotropin-releasing factor receptor 1(Homo sapiens (Human))
Neurocrine Biosciences

Curated by ChEMBL
LigandPNGBDBM50074339(CHEMBL424538 | N-(2-Bromo-4-dimethylamino-phenyl)-...)
Affinity DataKi:  6nMAssay Description:Binding affinity for human recombinant corticotropin releasing factor receptor 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCorticotropin-releasing factor receptor 1(Homo sapiens (Human))
Neurocrine Biosciences

Curated by ChEMBL
LigandPNGBDBM50074335(3-({4-[(4-Dimethylamino-2-methyl-phenyl)-ethyl-ami...)
Affinity DataKi:  7nMAssay Description:Binding affinity for human recombinant corticotropin releasing factor receptor 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCorticotropin-releasing factor receptor 1(Homo sapiens (Human))
Neurocrine Biosciences

Curated by ChEMBL
LigandPNGBDBM50074381(CHEMBL168169 | N-(4-Dimethylamino-2-methyl-phenyl)...)
Affinity DataKi:  7nMAssay Description:Binding affinity for human recombinant corticotropin releasing factor receptor 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCorticotropin-releasing factor receptor 1(Homo sapiens (Human))
Neurocrine Biosciences

Curated by ChEMBL
LigandPNGBDBM50074394(3-(Butyl-{4-[(4-dimethylamino-2-methyl-phenyl)-eth...)
Affinity DataKi:  8nMAssay Description:Binding affinity for human recombinant corticotropin releasing factor receptor 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCorticotropin-releasing factor receptor 1(Homo sapiens (Human))
Neurocrine Biosciences

Curated by ChEMBL
LigandPNGBDBM50074368(1-(3-Bromo-4-{[4-(butyl-ethyl-amino)-6-methyl-pyri...)
Affinity DataKi:  8nMAssay Description:Binding affinity for human recombinant corticotropin releasing factor receptor 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCorticotropin-releasing factor receptor 1(Homo sapiens (Human))
Neurocrine Biosciences

Curated by ChEMBL
LigandPNGBDBM50074407((Butyl-{4-[(4-dimethylamino-2-methyl-phenyl)-ethyl...)
Affinity DataKi:  8nMAssay Description:Binding affinity for human recombinant corticotropin releasing factor receptor 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCorticotropin-releasing factor receptor 1(Homo sapiens (Human))
Neurocrine Biosciences

Curated by ChEMBL
LigandPNGBDBM50074366(CHEMBL10203 | N*2*-(2-Bromo-4-isopropyl-phenyl)-N*...)
Affinity DataKi:  9nMAssay Description:Binding affinity for human recombinant corticotropin releasing factor receptor 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCorticotropin-releasing factor receptor 1(Homo sapiens (Human))
Neurocrine Biosciences

Curated by ChEMBL
LigandPNGBDBM50074383(CHEMBL268993 | N*2*-(2-Bromo-4-isopropyl-phenyl)-N...)
Affinity DataKi:  9nMAssay Description:Binding affinity for human recombinant corticotropin releasing factor receptor 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCorticotropin-releasing factor receptor 1(Homo sapiens (Human))
Neurocrine Biosciences

Curated by ChEMBL
LigandPNGBDBM50074393(CHEMBL353973 | N*2*-(2-Bromo-4-iodo-phenyl)-N*2*,N...)
Affinity DataKi:  9nMAssay Description:Binding affinity for human recombinant corticotropin releasing factor receptor 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCorticotropin-releasing factor receptor 1(Homo sapiens (Human))
Neurocrine Biosciences

Curated by ChEMBL
LigandPNGBDBM50074360(CHEMBL352378 | N*2*-(2-Chloro-4,6-dimethoxy-phenyl...)
Affinity DataKi:  10nMAssay Description:Binding affinity for human recombinant corticotropin releasing factor receptor 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCorticotropin-releasing factor receptor 1(Homo sapiens (Human))
Neurocrine Biosciences

Curated by ChEMBL
LigandPNGBDBM50074400(CHEMBL167122 | N-(2-Bromo-4,6-dimethoxy-phenyl)-N,...)
Affinity DataKi:  10nMAssay Description:Binding affinity for human recombinant corticotropin releasing factor receptor 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCorticotropin-releasing factor receptor 1(Homo sapiens (Human))
Neurocrine Biosciences

Curated by ChEMBL
LigandPNGBDBM50074413(CHEMBL169094 | N*2*-(4-Dimethylamino-2-trifluorome...)
Affinity DataKi:  11nMAssay Description:Binding affinity for human recombinant corticotropin releasing factor receptor 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCorticotropin-releasing factor receptor 1(Homo sapiens (Human))
Neurocrine Biosciences

Curated by ChEMBL
LigandPNGBDBM50074331(CHEMBL167444 | N*2*-(2-Bromo-4-isopropyl-phenyl)-N...)
Affinity DataKi:  11nMAssay Description:Binding affinity for human recombinant corticotropin releasing factor receptor 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCorticotropin-releasing factor receptor 1(Homo sapiens (Human))
Neurocrine Biosciences

Curated by ChEMBL
LigandPNGBDBM50074411((2-Bromo-4,6-dimethoxy-phenyl)-(4,6-dimethyl-pyrim...)
Affinity DataKi:  12nMAssay Description:Binding affinity for human recombinant corticotropin releasing factor receptor 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCorticotropin-releasing factor receptor 1(Homo sapiens (Human))
Neurocrine Biosciences

Curated by ChEMBL
LigandPNGBDBM50074403(CHEMBL166835 | N-Butyl-N'-ethyl-N-(2-methoxy-ethyl...)
Affinity DataKi:  13nMAssay Description:Binding affinity for human recombinant corticotropin releasing factor receptor 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCorticotropin-releasing factor receptor 1(Homo sapiens (Human))
Neurocrine Biosciences

Curated by ChEMBL
LigandPNGBDBM50074379(CHEMBL165531 | N*2*-(2-Bromo-4-iodo-phenyl)-N*4*-b...)
Affinity DataKi:  14nMAssay Description:Binding affinity for human recombinant corticotropin releasing factor receptor 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCorticotropin-releasing factor receptor 1(Homo sapiens (Human))
Neurocrine Biosciences

Curated by ChEMBL
LigandPNGBDBM50074363(CHEMBL166235 | N*4*-Benzyl-N*2*-(2-bromo-4-isoprop...)
Affinity DataKi:  14nMAssay Description:Binding affinity for human recombinant corticotropin releasing factor receptor 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCorticotropin-releasing factor receptor 1(Homo sapiens (Human))
Neurocrine Biosciences

Curated by ChEMBL
LigandPNGBDBM50074342(CHEMBL354584 | N*2*-(2,6-Dichloro-4-methoxy-phenyl...)
Affinity DataKi:  15nMAssay Description:Binding affinity for human recombinant corticotropin releasing factor receptor 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCorticotropin-releasing factor receptor 1(Homo sapiens (Human))
Neurocrine Biosciences

Curated by ChEMBL
LigandPNGBDBM50074344(1-{3-Bromo-4-[(4-diethylamino-6-methyl-[1,3,5]tria...)
Affinity DataKi:  17nMAssay Description:Binding affinity for human recombinant corticotropin releasing factor receptor 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCorticotropin-releasing factor receptor 1(Homo sapiens (Human))
Neurocrine Biosciences

Curated by ChEMBL
LigandPNGBDBM50074359(CHEMBL354791 | N*4*-Benzyl-N*2*-(2-bromo-4-isoprop...)
Affinity DataKi:  17nMAssay Description:Binding affinity for human recombinant corticotropin releasing factor receptor 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCorticotropin-releasing factor receptor 1(Homo sapiens (Human))
Neurocrine Biosciences

Curated by ChEMBL
LigandPNGBDBM50074374(CHEMBL355055 | N-(2-Bromo-4-isopropyl-phenyl)-N-et...)
Affinity DataKi:  18nMAssay Description:Binding affinity for human recombinant corticotropin releasing factor receptor 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCorticotropin-releasing factor receptor 1(Homo sapiens (Human))
Neurocrine Biosciences

Curated by ChEMBL
LigandPNGBDBM50074364(CHEMBL350356 | N*2*-(2-Bromo-4-isopropyl-phenyl)-N...)
Affinity DataKi:  19nMAssay Description:Binding affinity for human recombinant corticotropin releasing factor receptor 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCorticotropin-releasing factor receptor 1(Homo sapiens (Human))
Neurocrine Biosciences

Curated by ChEMBL
LigandPNGBDBM50074378(CHEMBL165991 | N-(4-Dimethylamino-2-trifluoromethy...)
Affinity DataKi:  20nMAssay Description:Binding affinity for human recombinant corticotropin releasing factor receptor 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCorticotropin-releasing factor receptor 1(Homo sapiens (Human))
Neurocrine Biosciences

Curated by ChEMBL
LigandPNGBDBM50074356(CHEMBL168360 | N*1*-(4,6-Dimethyl-pyrimidin-2-yl)-...)
Affinity DataKi:  20nMAssay Description:Binding affinity for human recombinant corticotropin releasing factor receptor 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCorticotropin-releasing factor receptor 1(Homo sapiens (Human))
Neurocrine Biosciences

Curated by ChEMBL
LigandPNGBDBM50074414(CHEMBL167737 | N*2*-(2-Bromo-4-isopropyl-phenyl)-N...)
Affinity DataKi:  22nMAssay Description:Binding affinity for human recombinant corticotropin releasing factor receptor 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCorticotropin-releasing factor receptor 1(Homo sapiens (Human))
Neurocrine Biosciences

Curated by ChEMBL
LigandPNGBDBM50074372((2-Bromo-4-isopropyl-phenyl)-ethyl-(4-methyl-6-mor...)
Affinity DataKi:  22nMAssay Description:Binding affinity for human recombinant corticotropin releasing factor receptor 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCorticotropin-releasing factor receptor 1(Homo sapiens (Human))
Neurocrine Biosciences

Curated by ChEMBL
LigandPNGBDBM50074387(CHEMBL166890 | N*2*-(2-Bromo-4-isopropyl-phenyl)-N...)
Affinity DataKi:  22nMAssay Description:Binding affinity for human recombinant corticotropin releasing factor receptor 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCorticotropin-releasing factor receptor 1(Homo sapiens (Human))
Neurocrine Biosciences

Curated by ChEMBL
LigandPNGBDBM50074387(CHEMBL166890 | N*2*-(2-Bromo-4-isopropyl-phenyl)-N...)
Affinity DataKi:  22nMAssay Description:Binding affinity for human recombinant corticotropin releasing factor receptor 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCorticotropin-releasing factor receptor 1(Homo sapiens (Human))
Neurocrine Biosciences

Curated by ChEMBL
LigandPNGBDBM50074367(CHEMBL165473 | N-Butyl-N,N'-diethyl-6-methyl-N'-(2...)
Affinity DataKi:  23nMAssay Description:Binding affinity for human recombinant corticotropin releasing factor receptor 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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