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Found 35 with Last Name = 'deias' and Initial = 'r'
TargetCarnitine O-palmitoyltransferase 1, liver isoform(Rattus norvegicus)
Sigma Tau Pharmaceutical Industries

Curated by ChEMBL
LigandPNGBDBM50122836(CHEMBL102993 | [3-Carboxy-2-(3-tetradecyl-ureido)-...)
Affinity DataKi:  360nMAssay Description:Inhibition of rat liver carnitine palmitoyltransferase IMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarnitine O-palmitoyltransferase 1, liver isoform(Rattus norvegicus)
Sigma Tau Pharmaceutical Industries

Curated by ChEMBL
LigandPNGBDBM50101604(CHEMBL309568 | [3-Carboxy-2-(dodecane-1-sulfonylam...)
Affinity DataIC50:  700nMAssay Description:Inhibition of [14C]-palmitoyl-CoA and carnitine binding to carnitine palmitoyltransferase I from rat liver mitochondriaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarnitine O-palmitoyltransferase 1, liver isoform(Rattus norvegicus)
Sigma Tau Pharmaceutical Industries

Curated by ChEMBL
LigandPNGBDBM50101591(CHEMBL308869 | R-[3-Carboxy-2-(undecane-1-sulfamoy...)
Affinity DataIC50:  800nMAssay Description:Inhibition of [14C]-palmitoyl-CoA and carnitine binding to carnitine palmitoyltransferase I from rat liver mitochondriaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarnitine O-palmitoyltransferase 1, liver isoform(Rattus norvegicus)
Sigma Tau Pharmaceutical Industries

Curated by ChEMBL
LigandPNGBDBM50122839(CHEMBL106227 | [3-Carboxy-2-(3-tetradecyl-ureido)-...)
Affinity DataIC50:  1.10E+3nMAssay Description:Inhibition of [14C]-palmitoyl-CoA and carnitine binding to carnitine palmitoyltransferase I from rat liver mitochondriaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarnitine O-palmitoyltransferase 1, liver isoform(Rattus norvegicus)
Sigma Tau Pharmaceutical Industries

Curated by ChEMBL
LigandPNGBDBM50122834(CHEMBL105314 | [3-Carboxy-2-(3-dodecyl-ureido)-pro...)
Affinity DataIC50:  1.80E+3nMAssay Description:Inhibition of [14C]-palmitoyl-CoA and carnitine binding to carnitine palmitoyltransferase I from rat liver mitochondriaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarnitine O-palmitoyltransferase 1, liver isoform(Rattus norvegicus)
Sigma Tau Pharmaceutical Industries

Curated by ChEMBL
LigandPNGBDBM50122828(CHEMBL106274 | [3-Carboxy-2-(3-undecyl-ureido)-pro...)
Affinity DataIC50:  3.20E+3nMAssay Description:Inhibition of [14C]-palmitoyl-CoA and carnitine binding to carnitine palmitoyltransferase I from rat liver mitochondriaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarnitine O-palmitoyltransferase 1, muscle isoform(Rattus norvegicus)
Sigma Tau Pharmaceutical Industries

Curated by ChEMBL
LigandPNGBDBM50101604(CHEMBL309568 | [3-Carboxy-2-(dodecane-1-sulfonylam...)
Affinity DataIC50:  3.40E+3nMAssay Description:In vitro inhibition of [14C]-palmitoyl-CoA and carnitine binding to carnitine palmitoyltransferase I of rat heart mitochondriaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarnitine O-palmitoyltransferase 1, muscle isoform(Rattus norvegicus)
Sigma Tau Pharmaceutical Industries

Curated by ChEMBL
LigandPNGBDBM50101591(CHEMBL308869 | R-[3-Carboxy-2-(undecane-1-sulfamoy...)
Affinity DataIC50:  5.80E+3nMAssay Description:In vitro inhibition of [14C]-palmitoyl-CoA and carnitine binding to carnitine palmitoyltransferase I of rat heart mitochondriaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarnitine O-palmitoyltransferase 1, liver isoform(Rattus norvegicus)
Sigma Tau Pharmaceutical Industries

Curated by ChEMBL
LigandPNGBDBM50101600(CHEMBL305897 | [3-Carboxy-2-(undecane-1-sulfamoyla...)
Affinity DataIC50:  6.00E+3nMAssay Description:Inhibition of [14C]-palmitoyl-CoA and carnitine binding to carnitine palmitoyltransferase I from rat liver mitochondriaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarnitine O-palmitoyltransferase 1, liver isoform(Rattus norvegicus)
Sigma Tau Pharmaceutical Industries

Curated by ChEMBL
LigandPNGBDBM50101598(CHEMBL307495 | [3-Carboxy-2-(dodecane-1-sulfonylam...)
Affinity DataIC50:  6.00E+3nMAssay Description:Inhibition of [14C]-palmitoyl-CoA and carnitine binding to carnitine palmitoyltransferase I from rat liver mitochondriaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarnitine O-palmitoyltransferase 1, liver isoform(Rattus norvegicus)
Sigma Tau Pharmaceutical Industries

Curated by ChEMBL
LigandPNGBDBM50122833((3-Carboxy-2-octyloxycarbonylamino-propyl)-trimeth...)
Affinity DataIC50:  9.50E+3nMAssay Description:Inhibition of [14C]-palmitoyl-CoA and carnitine binding to carnitine palmitoyltransferase I from rat liver mitochondriaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarnitine O-palmitoyltransferase 1, muscle isoform(Rattus norvegicus)
Sigma Tau Pharmaceutical Industries

Curated by ChEMBL
LigandPNGBDBM50101600(CHEMBL305897 | [3-Carboxy-2-(undecane-1-sulfamoyla...)
Affinity DataIC50: >1.00E+4nMAssay Description:In vitro inhibition of [14C]-palmitoyl-CoA and carnitine binding to carnitine palmitoyltransferase I of rat heart mitochondriaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarnitine O-palmitoyltransferase 1, muscle isoform(Rattus norvegicus)
Sigma Tau Pharmaceutical Industries

Curated by ChEMBL
LigandPNGBDBM50101598(CHEMBL307495 | [3-Carboxy-2-(dodecane-1-sulfonylam...)
Affinity DataIC50: >1.00E+4nMAssay Description:In vitro inhibition of [14C]-palmitoyl-CoA and carnitine binding to carnitine palmitoyltransferase I of rat heart mitochondriaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarnitine O-palmitoyltransferase 1, liver isoform(Rattus norvegicus)
Sigma Tau Pharmaceutical Industries

Curated by ChEMBL
LigandPNGBDBM50122827(CHEMBL105330 | [3-Carboxy-2-(3-nonyl-ureido)-propy...)
Affinity DataIC50:  3.13E+4nMAssay Description:Inhibition of [14C]-palmitoyl-CoA and carnitine binding to carnitine palmitoyltransferase I from rat liver mitochondriaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarnitine O-palmitoyltransferase 1, muscle isoform(Rattus norvegicus)
Sigma Tau Pharmaceutical Industries

Curated by ChEMBL
LigandPNGBDBM50122839(CHEMBL106227 | [3-Carboxy-2-(3-tetradecyl-ureido)-...)
Affinity DataIC50:  4.34E+4nMAssay Description:In vitro inhibition of [14C]-palmitoyl-CoA and carnitine binding to carnitine palmitoyltransferase I of rat heart mitochondriaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarnitine O-palmitoyltransferase 1, liver isoform(Rattus norvegicus)
Sigma Tau Pharmaceutical Industries

Curated by ChEMBL
LigandPNGBDBM50122837(CHEMBL319635 | [3-Carboxy-2-(3-heptyl-ureido)-prop...)
Affinity DataIC50:  4.36E+4nMAssay Description:Inhibition of [14C]-palmitoyl-CoA and carnitine binding to carnitine palmitoyltransferase I from rat liver mitochondriaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarnitine O-palmitoyltransferase 1, muscle isoform(Rattus norvegicus)
Sigma Tau Pharmaceutical Industries

Curated by ChEMBL
LigandPNGBDBM50122827(CHEMBL105330 | [3-Carboxy-2-(3-nonyl-ureido)-propy...)
Affinity DataIC50:  4.62E+4nMAssay Description:In vitro inhibition of [14C]-palmitoyl-CoA and carnitine binding to carnitine palmitoyltransferase I of rat heart mitochondriaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarnitine O-palmitoyltransferase 1, liver isoform(Rattus norvegicus)
Sigma Tau Pharmaceutical Industries

Curated by ChEMBL
LigandPNGBDBM50122836(CHEMBL102993 | [3-Carboxy-2-(3-tetradecyl-ureido)-...)
Affinity DataIC50:  5.88E+4nMAssay Description:Inhibition of [14C]-palmitoyl-CoA and carnitine binding to carnitine palmitoyltransferase I from rat liver mitochondriaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarnitine O-palmitoyltransferase 1, muscle isoform(Rattus norvegicus)
Sigma Tau Pharmaceutical Industries

Curated by ChEMBL
LigandPNGBDBM50122833((3-Carboxy-2-octyloxycarbonylamino-propyl)-trimeth...)
Affinity DataIC50:  8.01E+4nMAssay Description:In vitro inhibition of [14C]-palmitoyl-CoA and carnitine binding to carnitine palmitoyltransferase I of rat heart mitochondriaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarnitine O-palmitoyltransferase 1, muscle isoform(Rattus norvegicus)
Sigma Tau Pharmaceutical Industries

Curated by ChEMBL
LigandPNGBDBM50122828(CHEMBL106274 | [3-Carboxy-2-(3-undecyl-ureido)-pro...)
Affinity DataIC50:  1.18E+5nMAssay Description:In vitro inhibition of [14C]-palmitoyl-CoA and carnitine binding to carnitine palmitoyltransferase I of rat heart mitochondriaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarnitine O-palmitoyltransferase 1, muscle isoform(Rattus norvegicus)
Sigma Tau Pharmaceutical Industries

Curated by ChEMBL
LigandPNGBDBM50122834(CHEMBL105314 | [3-Carboxy-2-(3-dodecyl-ureido)-pro...)
Affinity DataIC50: >1.20E+5nMAssay Description:In vitro inhibition of [14C]-palmitoyl-CoA and carnitine binding to carnitine palmitoyltransferase I of rat heart mitochondriaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarnitine O-palmitoyltransferase 1, muscle isoform(Rattus norvegicus)
Sigma Tau Pharmaceutical Industries

Curated by ChEMBL
LigandPNGBDBM50122836(CHEMBL102993 | [3-Carboxy-2-(3-tetradecyl-ureido)-...)
Affinity DataIC50:  1.67E+5nMAssay Description:In vitro inhibition of [14C]-palmitoyl-CoA and carnitine binding to carnitine palmitoyltransferase I of rat heart mitochondriaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarnitine O-palmitoyltransferase 1, muscle isoform(Rattus norvegicus)
Sigma Tau Pharmaceutical Industries

Curated by ChEMBL
LigandPNGBDBM50122829((3-Carboxy-2-octyloxycarbonylamino-propyl)-trimeth...)
Affinity DataIC50: >3.00E+5nMAssay Description:In vitro inhibition of [14C]-palmitoyl-CoA and carnitine binding to carnitine palmitoyltransferase I of rat heart mitochondriaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarnitine O-palmitoyltransferase 1, liver isoform(Rattus norvegicus)
Sigma Tau Pharmaceutical Industries

Curated by ChEMBL
LigandPNGBDBM50122829((3-Carboxy-2-octyloxycarbonylamino-propyl)-trimeth...)
Affinity DataIC50: >3.00E+5nMAssay Description:Inhibition of [14C]-palmitoyl-CoA and carnitine binding to carnitine palmitoyltransferase I from rat liver mitochondriaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarnitine O-palmitoyltransferase 1, liver isoform(Rattus norvegicus)
Sigma Tau Pharmaceutical Industries

Curated by ChEMBL
LigandPNGBDBM50122835(CHEMBL105727 | [3-Carboxy-2-(3-nonyl-ureido)-propy...)
Affinity DataIC50: >3.00E+5nMAssay Description:Inhibition of [14C]-palmitoyl-CoA and carnitine binding to carnitine palmitoyltransferase I from rat liver mitochondriaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarnitine O-palmitoyltransferase 1, muscle isoform(Rattus norvegicus)
Sigma Tau Pharmaceutical Industries

Curated by ChEMBL
LigandPNGBDBM50122837(CHEMBL319635 | [3-Carboxy-2-(3-heptyl-ureido)-prop...)
Affinity DataIC50: >3.00E+5nMAssay Description:In vitro inhibition of [14C]-palmitoyl-CoA and carnitine binding to carnitine palmitoyltransferase I of rat heart mitochondriaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarnitine O-palmitoyltransferase 1, muscle isoform(Rattus norvegicus)
Sigma Tau Pharmaceutical Industries

Curated by ChEMBL
LigandPNGBDBM50122835(CHEMBL105727 | [3-Carboxy-2-(3-nonyl-ureido)-propy...)
Affinity DataIC50: >3.00E+5nMAssay Description:In vitro inhibition of [14C]-palmitoyl-CoA and carnitine binding to carnitine palmitoyltransferase I of rat heart mitochondriaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUracil nucleotide/cysteinyl leukotriene receptor(Homo sapiens (Human))
Tampere University

Curated by ChEMBL
LigandPNGBDBM50580105(CHEMBL5086989)
Affinity DataEC50:  2.63E+4nMAssay Description:Agonist activity at human GPR17 in human SNB-19 cells assessed as decrease in calcium ion levels incubated for 2 hrs by Calcium Fura 2 Dynamic assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetUracil nucleotide/cysteinyl leukotriene receptor(Homo sapiens (Human))
Tampere University

Curated by ChEMBL
LigandPNGBDBM50580104(CHEMBL5083629)
Affinity DataEC50:  4.19E+4nMAssay Description:Agonist activity at human GPR17 in human LN-229 cells assessed as decrease in calcium ion levels incubated for 2 hrs by Calcium Fura 2 Dynamic assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetUracil nucleotide/cysteinyl leukotriene receptor(Homo sapiens (Human))
Tampere University

Curated by ChEMBL
LigandPNGBDBM50580105(CHEMBL5086989)
Affinity DataEC50:  2.69E+4nMAssay Description:Agonist activity at human GPR17 in human LN-229 cells assessed as decrease in calcium ion levels incubated for 2 hrs by Calcium Fura 2 Dynamic assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetUracil nucleotide/cysteinyl leukotriene receptor(Homo sapiens (Human))
Tampere University

Curated by ChEMBL
LigandPNGBDBM50580105(CHEMBL5086989)
Affinity DataEC50:  1.77E+4nMAssay Description:Inverse agonist at human GPR17 in human SNB-19 cells assessed as intracellular cAMP levels incubated for 2 hrs by cAMP Glo Dynamic assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetUracil nucleotide/cysteinyl leukotriene receptor(Homo sapiens (Human))
Tampere University

Curated by ChEMBL
LigandPNGBDBM50580105(CHEMBL5086989)
Affinity DataEC50:  1.66E+4nMAssay Description:Inverse agonist at human GPR17 in human LN-229 cells assessed as intracellular cAMP levels incubated for 2 hrs by cAMP Glo Dynamic assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetUracil nucleotide/cysteinyl leukotriene receptor(Homo sapiens (Human))
Tampere University

Curated by ChEMBL
LigandPNGBDBM50580104(CHEMBL5083629)
Affinity DataEC50:  1.92E+4nMAssay Description:Agonist activity at human GPR17 in human SNB-19 cells assessed as decrease in intracellular cAMP levels incubated for 2 hrs by cAMP Glo Dynamic assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetUracil nucleotide/cysteinyl leukotriene receptor(Homo sapiens (Human))
Tampere University

Curated by ChEMBL
LigandPNGBDBM50580104(CHEMBL5083629)
Affinity DataEC50:  7.67E+3nMAssay Description:Agonist activity at human GPR17 in human SNB-19 cells assessed as decrease in calcium ion levels incubated for 2 hrs by Calcium Fura 2 Dynamic assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetUracil nucleotide/cysteinyl leukotriene receptor(Homo sapiens (Human))
Tampere University

Curated by ChEMBL
LigandPNGBDBM50580104(CHEMBL5083629)
Affinity DataEC50:  5.97E+4nMAssay Description:Agonist activity at human GPR17 in human LN-229 cells assessed as decrease in intracellular cAMP levels incubated for 2 hrs by cAMP Glo Dynamic assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed