TargetCarnitine O-palmitoyltransferase 1, liver isoform(Rattus norvegicus)
Sigma Tau Pharmaceutical Industries
Curated by ChEMBL
Sigma Tau Pharmaceutical Industries
Curated by ChEMBL
Affinity DataKi: 360nMAssay Description:Inhibition of rat liver carnitine palmitoyltransferase IMore data for this Ligand-Target Pair
TargetCarnitine O-palmitoyltransferase 1, liver isoform(Rattus norvegicus)
Sigma Tau Pharmaceutical Industries
Curated by ChEMBL
Sigma Tau Pharmaceutical Industries
Curated by ChEMBL
Affinity DataIC50: 700nMAssay Description:Inhibition of [14C]-palmitoyl-CoA and carnitine binding to carnitine palmitoyltransferase I from rat liver mitochondriaMore data for this Ligand-Target Pair
TargetCarnitine O-palmitoyltransferase 1, liver isoform(Rattus norvegicus)
Sigma Tau Pharmaceutical Industries
Curated by ChEMBL
Sigma Tau Pharmaceutical Industries
Curated by ChEMBL
Affinity DataIC50: 800nMAssay Description:Inhibition of [14C]-palmitoyl-CoA and carnitine binding to carnitine palmitoyltransferase I from rat liver mitochondriaMore data for this Ligand-Target Pair
TargetCarnitine O-palmitoyltransferase 1, liver isoform(Rattus norvegicus)
Sigma Tau Pharmaceutical Industries
Curated by ChEMBL
Sigma Tau Pharmaceutical Industries
Curated by ChEMBL
Affinity DataIC50: 1.10E+3nMAssay Description:Inhibition of [14C]-palmitoyl-CoA and carnitine binding to carnitine palmitoyltransferase I from rat liver mitochondriaMore data for this Ligand-Target Pair
TargetCarnitine O-palmitoyltransferase 1, liver isoform(Rattus norvegicus)
Sigma Tau Pharmaceutical Industries
Curated by ChEMBL
Sigma Tau Pharmaceutical Industries
Curated by ChEMBL
Affinity DataIC50: 1.80E+3nMAssay Description:Inhibition of [14C]-palmitoyl-CoA and carnitine binding to carnitine palmitoyltransferase I from rat liver mitochondriaMore data for this Ligand-Target Pair
TargetCarnitine O-palmitoyltransferase 1, liver isoform(Rattus norvegicus)
Sigma Tau Pharmaceutical Industries
Curated by ChEMBL
Sigma Tau Pharmaceutical Industries
Curated by ChEMBL
Affinity DataIC50: 3.20E+3nMAssay Description:Inhibition of [14C]-palmitoyl-CoA and carnitine binding to carnitine palmitoyltransferase I from rat liver mitochondriaMore data for this Ligand-Target Pair
TargetCarnitine O-palmitoyltransferase 1, muscle isoform(Rattus norvegicus)
Sigma Tau Pharmaceutical Industries
Curated by ChEMBL
Sigma Tau Pharmaceutical Industries
Curated by ChEMBL
Affinity DataIC50: 3.40E+3nMAssay Description:In vitro inhibition of [14C]-palmitoyl-CoA and carnitine binding to carnitine palmitoyltransferase I of rat heart mitochondriaMore data for this Ligand-Target Pair
TargetCarnitine O-palmitoyltransferase 1, muscle isoform(Rattus norvegicus)
Sigma Tau Pharmaceutical Industries
Curated by ChEMBL
Sigma Tau Pharmaceutical Industries
Curated by ChEMBL
Affinity DataIC50: 5.80E+3nMAssay Description:In vitro inhibition of [14C]-palmitoyl-CoA and carnitine binding to carnitine palmitoyltransferase I of rat heart mitochondriaMore data for this Ligand-Target Pair
TargetCarnitine O-palmitoyltransferase 1, liver isoform(Rattus norvegicus)
Sigma Tau Pharmaceutical Industries
Curated by ChEMBL
Sigma Tau Pharmaceutical Industries
Curated by ChEMBL
Affinity DataIC50: 6.00E+3nMAssay Description:Inhibition of [14C]-palmitoyl-CoA and carnitine binding to carnitine palmitoyltransferase I from rat liver mitochondriaMore data for this Ligand-Target Pair
TargetCarnitine O-palmitoyltransferase 1, liver isoform(Rattus norvegicus)
Sigma Tau Pharmaceutical Industries
Curated by ChEMBL
Sigma Tau Pharmaceutical Industries
Curated by ChEMBL
Affinity DataIC50: 6.00E+3nMAssay Description:Inhibition of [14C]-palmitoyl-CoA and carnitine binding to carnitine palmitoyltransferase I from rat liver mitochondriaMore data for this Ligand-Target Pair
TargetCarnitine O-palmitoyltransferase 1, liver isoform(Rattus norvegicus)
Sigma Tau Pharmaceutical Industries
Curated by ChEMBL
Sigma Tau Pharmaceutical Industries
Curated by ChEMBL
Affinity DataIC50: 9.50E+3nMAssay Description:Inhibition of [14C]-palmitoyl-CoA and carnitine binding to carnitine palmitoyltransferase I from rat liver mitochondriaMore data for this Ligand-Target Pair
TargetCarnitine O-palmitoyltransferase 1, muscle isoform(Rattus norvegicus)
Sigma Tau Pharmaceutical Industries
Curated by ChEMBL
Sigma Tau Pharmaceutical Industries
Curated by ChEMBL
Affinity DataIC50: >1.00E+4nMAssay Description:In vitro inhibition of [14C]-palmitoyl-CoA and carnitine binding to carnitine palmitoyltransferase I of rat heart mitochondriaMore data for this Ligand-Target Pair
TargetCarnitine O-palmitoyltransferase 1, muscle isoform(Rattus norvegicus)
Sigma Tau Pharmaceutical Industries
Curated by ChEMBL
Sigma Tau Pharmaceutical Industries
Curated by ChEMBL
Affinity DataIC50: >1.00E+4nMAssay Description:In vitro inhibition of [14C]-palmitoyl-CoA and carnitine binding to carnitine palmitoyltransferase I of rat heart mitochondriaMore data for this Ligand-Target Pair
TargetCarnitine O-palmitoyltransferase 1, liver isoform(Rattus norvegicus)
Sigma Tau Pharmaceutical Industries
Curated by ChEMBL
Sigma Tau Pharmaceutical Industries
Curated by ChEMBL
Affinity DataIC50: 3.13E+4nMAssay Description:Inhibition of [14C]-palmitoyl-CoA and carnitine binding to carnitine palmitoyltransferase I from rat liver mitochondriaMore data for this Ligand-Target Pair
TargetCarnitine O-palmitoyltransferase 1, muscle isoform(Rattus norvegicus)
Sigma Tau Pharmaceutical Industries
Curated by ChEMBL
Sigma Tau Pharmaceutical Industries
Curated by ChEMBL
Affinity DataIC50: 4.34E+4nMAssay Description:In vitro inhibition of [14C]-palmitoyl-CoA and carnitine binding to carnitine palmitoyltransferase I of rat heart mitochondriaMore data for this Ligand-Target Pair
TargetCarnitine O-palmitoyltransferase 1, liver isoform(Rattus norvegicus)
Sigma Tau Pharmaceutical Industries
Curated by ChEMBL
Sigma Tau Pharmaceutical Industries
Curated by ChEMBL
Affinity DataIC50: 4.36E+4nMAssay Description:Inhibition of [14C]-palmitoyl-CoA and carnitine binding to carnitine palmitoyltransferase I from rat liver mitochondriaMore data for this Ligand-Target Pair
TargetCarnitine O-palmitoyltransferase 1, muscle isoform(Rattus norvegicus)
Sigma Tau Pharmaceutical Industries
Curated by ChEMBL
Sigma Tau Pharmaceutical Industries
Curated by ChEMBL
Affinity DataIC50: 4.62E+4nMAssay Description:In vitro inhibition of [14C]-palmitoyl-CoA and carnitine binding to carnitine palmitoyltransferase I of rat heart mitochondriaMore data for this Ligand-Target Pair
TargetCarnitine O-palmitoyltransferase 1, liver isoform(Rattus norvegicus)
Sigma Tau Pharmaceutical Industries
Curated by ChEMBL
Sigma Tau Pharmaceutical Industries
Curated by ChEMBL
Affinity DataIC50: 5.88E+4nMAssay Description:Inhibition of [14C]-palmitoyl-CoA and carnitine binding to carnitine palmitoyltransferase I from rat liver mitochondriaMore data for this Ligand-Target Pair
TargetCarnitine O-palmitoyltransferase 1, muscle isoform(Rattus norvegicus)
Sigma Tau Pharmaceutical Industries
Curated by ChEMBL
Sigma Tau Pharmaceutical Industries
Curated by ChEMBL
Affinity DataIC50: 8.01E+4nMAssay Description:In vitro inhibition of [14C]-palmitoyl-CoA and carnitine binding to carnitine palmitoyltransferase I of rat heart mitochondriaMore data for this Ligand-Target Pair
TargetCarnitine O-palmitoyltransferase 1, muscle isoform(Rattus norvegicus)
Sigma Tau Pharmaceutical Industries
Curated by ChEMBL
Sigma Tau Pharmaceutical Industries
Curated by ChEMBL
Affinity DataIC50: 1.18E+5nMAssay Description:In vitro inhibition of [14C]-palmitoyl-CoA and carnitine binding to carnitine palmitoyltransferase I of rat heart mitochondriaMore data for this Ligand-Target Pair
TargetCarnitine O-palmitoyltransferase 1, muscle isoform(Rattus norvegicus)
Sigma Tau Pharmaceutical Industries
Curated by ChEMBL
Sigma Tau Pharmaceutical Industries
Curated by ChEMBL
Affinity DataIC50: >1.20E+5nMAssay Description:In vitro inhibition of [14C]-palmitoyl-CoA and carnitine binding to carnitine palmitoyltransferase I of rat heart mitochondriaMore data for this Ligand-Target Pair
TargetCarnitine O-palmitoyltransferase 1, muscle isoform(Rattus norvegicus)
Sigma Tau Pharmaceutical Industries
Curated by ChEMBL
Sigma Tau Pharmaceutical Industries
Curated by ChEMBL
Affinity DataIC50: 1.67E+5nMAssay Description:In vitro inhibition of [14C]-palmitoyl-CoA and carnitine binding to carnitine palmitoyltransferase I of rat heart mitochondriaMore data for this Ligand-Target Pair
TargetCarnitine O-palmitoyltransferase 1, muscle isoform(Rattus norvegicus)
Sigma Tau Pharmaceutical Industries
Curated by ChEMBL
Sigma Tau Pharmaceutical Industries
Curated by ChEMBL
Affinity DataIC50: >3.00E+5nMAssay Description:In vitro inhibition of [14C]-palmitoyl-CoA and carnitine binding to carnitine palmitoyltransferase I of rat heart mitochondriaMore data for this Ligand-Target Pair
TargetCarnitine O-palmitoyltransferase 1, liver isoform(Rattus norvegicus)
Sigma Tau Pharmaceutical Industries
Curated by ChEMBL
Sigma Tau Pharmaceutical Industries
Curated by ChEMBL
Affinity DataIC50: >3.00E+5nMAssay Description:Inhibition of [14C]-palmitoyl-CoA and carnitine binding to carnitine palmitoyltransferase I from rat liver mitochondriaMore data for this Ligand-Target Pair
TargetCarnitine O-palmitoyltransferase 1, liver isoform(Rattus norvegicus)
Sigma Tau Pharmaceutical Industries
Curated by ChEMBL
Sigma Tau Pharmaceutical Industries
Curated by ChEMBL
Affinity DataIC50: >3.00E+5nMAssay Description:Inhibition of [14C]-palmitoyl-CoA and carnitine binding to carnitine palmitoyltransferase I from rat liver mitochondriaMore data for this Ligand-Target Pair
TargetCarnitine O-palmitoyltransferase 1, muscle isoform(Rattus norvegicus)
Sigma Tau Pharmaceutical Industries
Curated by ChEMBL
Sigma Tau Pharmaceutical Industries
Curated by ChEMBL
Affinity DataIC50: >3.00E+5nMAssay Description:In vitro inhibition of [14C]-palmitoyl-CoA and carnitine binding to carnitine palmitoyltransferase I of rat heart mitochondriaMore data for this Ligand-Target Pair
TargetCarnitine O-palmitoyltransferase 1, muscle isoform(Rattus norvegicus)
Sigma Tau Pharmaceutical Industries
Curated by ChEMBL
Sigma Tau Pharmaceutical Industries
Curated by ChEMBL
Affinity DataIC50: >3.00E+5nMAssay Description:In vitro inhibition of [14C]-palmitoyl-CoA and carnitine binding to carnitine palmitoyltransferase I of rat heart mitochondriaMore data for this Ligand-Target Pair
TargetUracil nucleotide/cysteinyl leukotriene receptor(Homo sapiens (Human))
Tampere University
Curated by ChEMBL
Tampere University
Curated by ChEMBL
Affinity DataEC50: 2.63E+4nMAssay Description:Agonist activity at human GPR17 in human SNB-19 cells assessed as decrease in calcium ion levels incubated for 2 hrs by Calcium Fura 2 Dynamic assayMore data for this Ligand-Target Pair
TargetUracil nucleotide/cysteinyl leukotriene receptor(Homo sapiens (Human))
Tampere University
Curated by ChEMBL
Tampere University
Curated by ChEMBL
Affinity DataEC50: 4.19E+4nMAssay Description:Agonist activity at human GPR17 in human LN-229 cells assessed as decrease in calcium ion levels incubated for 2 hrs by Calcium Fura 2 Dynamic assayMore data for this Ligand-Target Pair
TargetUracil nucleotide/cysteinyl leukotriene receptor(Homo sapiens (Human))
Tampere University
Curated by ChEMBL
Tampere University
Curated by ChEMBL
Affinity DataEC50: 2.69E+4nMAssay Description:Agonist activity at human GPR17 in human LN-229 cells assessed as decrease in calcium ion levels incubated for 2 hrs by Calcium Fura 2 Dynamic assayMore data for this Ligand-Target Pair
TargetUracil nucleotide/cysteinyl leukotriene receptor(Homo sapiens (Human))
Tampere University
Curated by ChEMBL
Tampere University
Curated by ChEMBL
Affinity DataEC50: 1.77E+4nMAssay Description:Inverse agonist at human GPR17 in human SNB-19 cells assessed as intracellular cAMP levels incubated for 2 hrs by cAMP Glo Dynamic assayMore data for this Ligand-Target Pair
TargetUracil nucleotide/cysteinyl leukotriene receptor(Homo sapiens (Human))
Tampere University
Curated by ChEMBL
Tampere University
Curated by ChEMBL
Affinity DataEC50: 1.66E+4nMAssay Description:Inverse agonist at human GPR17 in human LN-229 cells assessed as intracellular cAMP levels incubated for 2 hrs by cAMP Glo Dynamic assayMore data for this Ligand-Target Pair
TargetUracil nucleotide/cysteinyl leukotriene receptor(Homo sapiens (Human))
Tampere University
Curated by ChEMBL
Tampere University
Curated by ChEMBL
Affinity DataEC50: 1.92E+4nMAssay Description:Agonist activity at human GPR17 in human SNB-19 cells assessed as decrease in intracellular cAMP levels incubated for 2 hrs by cAMP Glo Dynamic assayMore data for this Ligand-Target Pair
TargetUracil nucleotide/cysteinyl leukotriene receptor(Homo sapiens (Human))
Tampere University
Curated by ChEMBL
Tampere University
Curated by ChEMBL
Affinity DataEC50: 7.67E+3nMAssay Description:Agonist activity at human GPR17 in human SNB-19 cells assessed as decrease in calcium ion levels incubated for 2 hrs by Calcium Fura 2 Dynamic assayMore data for this Ligand-Target Pair
TargetUracil nucleotide/cysteinyl leukotriene receptor(Homo sapiens (Human))
Tampere University
Curated by ChEMBL
Tampere University
Curated by ChEMBL
Affinity DataEC50: 5.97E+4nMAssay Description:Agonist activity at human GPR17 in human LN-229 cells assessed as decrease in intracellular cAMP levels incubated for 2 hrs by cAMP Glo Dynamic assayMore data for this Ligand-Target Pair