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Found 13 with Last Name = 'deinum' and Initial = 'j'
TargetCoagulation factor XI(Homo sapiens (Human))
Griffith University

Curated by ChEMBL
LigandPNGBDBM50271071((2,4-Dibromo-3-{[(4-carbamimidamidobutyl)carbamoyl...)
Affinity DataIC50:  1.30E+3nMAssay Description:Inhibition of factor 11a (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlasminogen activator inhibitor 1(Homo sapiens (Human))
Griffith University

Curated by ChEMBL
LigandPNGBDBM50241599(CHEMBL453012 | sideroxylonal A)
Affinity DataIC50:  3.30E+3nMAssay Description:Inhibition of human PAI1 using tissue type plasminogen activator substrate by plasmon resonanceMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlasminogen activator inhibitor 1(Homo sapiens (Human))
Griffith University

Curated by ChEMBL
LigandPNGBDBM50241601(CHEMBL453538 | sideroxylonal C)
Affinity DataIC50:  4.70E+3nMAssay Description:Inhibition of human PAI1 using tissue type plasminogen activator substrate by plasmon resonanceMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlasminogen activator inhibitor 1(Homo sapiens (Human))
Griffith University

Curated by ChEMBL
LigandPNGBDBM50241600(CHEMBL509880 | sideroxylonal B)
Affinity DataIC50:  5.30E+3nMAssay Description:Inhibition of human PAI1 using tissue type plasminogen activator substrate by plasmon resonanceMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCoagulation factor XI(Homo sapiens (Human))
Griffith University

Curated by ChEMBL
LigandPNGBDBM50271072(2-(2-Amino-2-oxoethyl)-3,5-dibromo-4-hydroxyphenyl...)
Affinity DataIC50:  2.70E+4nMAssay Description:Inhibition of factor 11a (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-secretase 1(Homo sapiens (Human))
Astrazeneca R&D

Curated by ChEMBL
LigandPNGBDBM50226438((S)-5-((S)-1-carboxy-2-phenylethylamino)-4-((S)-2-...)
Affinity DataIC50:  3.00E+4nMAssay Description:Inhibition of BACE1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-secretase 1(Homo sapiens (Human))
Astrazeneca R&D

Curated by ChEMBL
LigandPNGBDBM16047((4S)-4-[(2S)-2-[(2R,4S,5S)-5-[(2S)-2-[(2S)-2-[(4S)...)
Affinity DataIC50:  3.00E+4nMAssay Description:Inhibition of BACE1More data for this Ligand-Target Pair
TargetPlasminogen activator inhibitor 1(Homo sapiens (Human))
Griffith University

Curated by ChEMBL
LigandPNGBDBM50241606(CHEMBL454049 | euglobal IA2)
Affinity DataIC50:  1.38E+5nMAssay Description:Inhibition of human PAI1 using tissue type plasminogen activator substrate by plasmon resonanceMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlasminogen activator inhibitor 1(Homo sapiens (Human))
Griffith University

Curated by ChEMBL
LigandPNGBDBM50241608(CHEMBL509920 | robustadial A)
Affinity DataIC50:  1.52E+5nMAssay Description:Inhibition of human PAI1 using tissue type plasminogen activator substrate by plasmon resonanceMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlasminogen activator inhibitor 1(Homo sapiens (Human))
Griffith University

Curated by ChEMBL
LigandPNGBDBM50241607(CHEMBL454050 | euglobal IIc)
Affinity DataIC50:  7.00E+5nMAssay Description:Inhibition of human PAI1 using tissue type plasminogen activator substrate by plasmon resonanceMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-secretase 1(Homo sapiens (Human))
Astrazeneca R&D

Curated by ChEMBL
LigandPNGBDBM50226439(2-amino-6-propylpyrimidin-4(3H)-one | CHEMBL235825)
Affinity DataKd:  4.45E+6nMAssay Description:Binding affinity to BACE1 expressed in HEK293 cells by Biocore ISAMore data for this Ligand-Target Pair
TargetEndothiapepsin(Cryphonectria parasitica)
Astrazeneca R&D

Curated by ChEMBL
LigandPNGBDBM50226437(2-AMINO-6-(2-PHENYLETHYL)PYRIMIDIN-4(3H)-ONE | 2-a...)
Affinity DataKd:  2.20E+5nMAssay Description:Binding affinity to endothiapepsin by Biocore ISAMore data for this Ligand-Target Pair
TargetBeta-secretase 1(Homo sapiens (Human))
Astrazeneca R&D

Curated by ChEMBL
LigandPNGBDBM50226437(2-AMINO-6-(2-PHENYLETHYL)PYRIMIDIN-4(3H)-ONE | 2-a...)
Affinity DataKd:  6.60E+5nMAssay Description:Binding affinity to BACE1 expressed in HEK293 cells by Biocore ISAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed