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Found 1446 with Last Name = 'deodhar' and Initial = 'm'
TargetAmine oxidase [flavin-containing] B(Homo sapiens (Human))
Pharmaxis

Curated by ChEMBL
LigandPNGBDBM50589703(CHEMBL5196906)
Affinity DataKi:  8nMAssay Description:Time dependent inhibition of human recombinant MAO-B assessed as inhibition constantMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetLysyl oxidase homolog 2(Homo sapiens (Human))
Pharmaxis

Curated by ChEMBL
LigandPNGBDBM50505638(CHEMBL4457578)
Affinity DataKi:  83nMAssay Description:Time-dependent inhibition of recombinant human C-terminal His-tagged LOLX2 (1-774 residues) expressed in mouse myeloma cells assessed as apparent inh...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetRetina-specific copper amine oxidase(Homo sapiens (Human))
Pharmaxis

Curated by ChEMBL
LigandPNGBDBM50589703(CHEMBL5196906)
Affinity DataKi:  710nMAssay Description:Time dependent inhibition of human recombinant SSAO assessed as inhibition constantMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetMembrane primary amine oxidase(Homo sapiens (Human))
Pharmaxis

Curated by ChEMBL
LigandPNGBDBM50246766(CHEMBL489079 | Mofegiline | US9302986, Mofegiline)
Affinity DataKi:  1.61E+3nMAssay Description:Inhibition of human SSAO/VAP1 measuring H2O2 production by Kitz and Wilson plot analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMembrane primary amine oxidase(Homo sapiens (Human))
Pharmaxis

Curated by ChEMBL
LigandPNGBDBM50384084(CHEMBL2029546)
Affinity DataKi:  1.64E+3nMAssay Description:Inhibition of human SSAO/VAP1 measuring H2O2 production by Kitz and Wilson plot analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] B(Mus musculus)
Pharmaxis

Curated by ChEMBL
LigandPNGBDBM50589703(CHEMBL5196906)
Affinity DataIC50:  0.400nMAssay Description:Inhibition of mouse muscle MAO-BMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetAmine oxidase [flavin-containing] B(Homo sapiens (Human))
Pharmaxis

Curated by ChEMBL
LigandPNGBDBM50246766(CHEMBL489079 | Mofegiline | US9302986, Mofegiline)
Affinity DataIC50:  2nMAssay Description:Inhibition of human recombinant MAO-BMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetAmine oxidase [flavin-containing] B(Homo sapiens (Human))
Pharmaxis

Curated by ChEMBL
LigandPNGBDBM50589702(CHEMBL5186190)
Affinity DataIC50:  2nMAssay Description:Inhibition of human recombinant MAO-BMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetAmine oxidase [flavin-containing] B(Homo sapiens (Human))
Pharmaxis

Curated by ChEMBL
LigandPNGBDBM50589700(CHEMBL5204901)
Affinity DataIC50:  2nMAssay Description:Inhibition of human recombinant MAO-BMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetAmine oxidase [flavin-containing] B(Homo sapiens (Human))
Pharmaxis

Curated by ChEMBL
LigandPNGBDBM50589699(CHEMBL5197971)
Affinity DataIC50:  3nMAssay Description:Inhibition of human recombinant MAO-BMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetAmine oxidase [flavin-containing] B(Homo sapiens (Human))
Pharmaxis

Curated by ChEMBL
LigandPNGBDBM50589698(CHEMBL5199917)
Affinity DataIC50:  3nMAssay Description:Inhibition of human recombinant MAO-BMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetRetina-specific copper amine oxidase(Homo sapiens (Human))
Pharmaxis

Curated by ChEMBL
LigandPNGBDBM50589695(CHEMBL5198317)
Affinity DataIC50:  4nMAssay Description:Inhibition of recombinant human SSAOMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetAmine oxidase [flavin-containing] B(Homo sapiens (Human))
Pharmaxis

Curated by ChEMBL
LigandPNGBDBM50589695(CHEMBL5198317)
Affinity DataIC50:  4nMAssay Description:Inhibition of human recombinant MAO-BMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetRetina-specific copper amine oxidase(Homo sapiens (Human))
Pharmaxis

Curated by ChEMBL
LigandPNGBDBM50589700(CHEMBL5204901)
Affinity DataIC50:  5nMAssay Description:Inhibition of recombinant human SSAOMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetAmine oxidase [flavin-containing] B(Homo sapiens (Human))
Pharmaxis

Curated by ChEMBL
LigandPNGBDBM50246766(CHEMBL489079 | Mofegiline | US9302986, Mofegiline)
Affinity DataIC50:  5nMpH: 7.4 T: 2°CAssay Description:Recombinant human MAO-B (0.06 mg/mL; Sigma Aldrich) was used as source of MAO-B enzyme activities. The assay was performed in a similar way as for hu...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetMembrane primary amine oxidase(Rattus norvegicus (Rat))
Pharmaxis

Curated by ChEMBL
LigandPNGBDBM50589703(CHEMBL5196906)
Affinity DataIC50:  5nMAssay Description:Inhibition of rat SSAOMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetLysyl oxidase homolog 2(Homo sapiens (Human))
Pharmaxis

Curated by ChEMBL
LigandPNGBDBM50505638(CHEMBL4457578)
Affinity DataIC50:  5nMAssay Description:Inhibition of recombinant human C-terminal His-tagged LOLX2 (1-774 residues) expressed in mouse myeloma cells using putrescine as substrate preincuba...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetLysyl oxidase homolog 2(Homo sapiens (Human))
Pharmaxis

Curated by ChEMBL
LigandPNGBDBM50505638(CHEMBL4457578)
Affinity DataIC50:  5nMAssay Description:Inhibition of recombinant human C-terminal His-tagged LOLX2 (1-774 residues) expressed in mouse myeloma cells using putrescine as substrate preincuba...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetLysyl oxidase homolog 2(Homo sapiens (Human))
Pharmaxis

Curated by ChEMBL
LigandPNGBDBM50505633(CHEMBL4448713)
Affinity DataIC50:  5nMAssay Description:Inhibition of recombinant human C-terminal His-tagged LOLX2 (1-774 residues) expressed in mouse myeloma cells using putrescine as substrate preincuba...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] B(Homo sapiens (Human))
Pharmaxis

Curated by ChEMBL
LigandPNGBDBM50589703(CHEMBL5196906)
Affinity DataIC50:  5nMAssay Description:Inhibition of human recombinant MAO-BMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetRetina-specific copper amine oxidase(Homo sapiens (Human))
Pharmaxis

Curated by ChEMBL
LigandPNGBDBM50589696(CHEMBL5201033)
Affinity DataIC50:  6nMAssay Description:Inhibition of recombinant human SSAOMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetLysyl oxidase homolog 2(Rattus norvegicus)
Pharmaxis

Curated by ChEMBL
LigandPNGBDBM50505638(CHEMBL4457578)
Affinity DataIC50:  6nMAssay Description:Inhibition of recombinant rat LOLX2 using putrescine as substrate preincubated with enzyme for 30 mins followed by substrate addition and measured ev...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetLysyl oxidase homolog 2(Mus musculus)
Pharmaxis

Curated by ChEMBL
LigandPNGBDBM50505638(CHEMBL4457578)
Affinity DataIC50:  6nMAssay Description:Inhibition of recombinant mouse C-terminal His-tagged LOLX2 (26-776 residues) expressed in mouse myeloma cells using putrescine as substrate preincub...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] B(Homo sapiens (Human))
Pharmaxis

Curated by ChEMBL
LigandPNGBDBM50589696(CHEMBL5201033)
Affinity DataIC50:  9nMAssay Description:Inhibition of human recombinant MAO-BMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetLysyl oxidase homolog 2(Homo sapiens (Human))
Pharmaxis

Curated by ChEMBL
LigandPNGBDBM50505638(CHEMBL4457578)
Affinity DataIC50:  9nMAssay Description:Inhibition of LOXL2 in human IMR90 cells using putrescine as substrate preincubated with enzyme for 30 mins followed by substrate addition and measur...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetRetina-specific copper amine oxidase(Homo sapiens (Human))
Pharmaxis

Curated by ChEMBL
LigandPNGBDBM50246766(CHEMBL489079 | Mofegiline | US9302986, Mofegiline)
Affinity DataIC50:  10nMAssay Description:Inhibition of recombinant human SSAOMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetMembrane primary amine oxidase(Mus musculus)
Pharmaxis

Curated by ChEMBL
LigandPNGBDBM50246766(CHEMBL489079 | Mofegiline | US9302986, Mofegiline)
Affinity DataIC50:  10nMAssay Description:Inhibition of SSAO/VAP1 in mouse adipocytes measuring H2O2 production by Resorufin/Amplex Red assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] B(Homo sapiens (Human))
Pharmaxis

Curated by ChEMBL
LigandPNGBDBM50384098(CHEMBL2029537)
Affinity DataIC50:  10nMAssay Description:Inhibition of human recombinant MAO-B assessed as H2O2 production by Resorufin/Amplex Red assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] B(Homo sapiens (Human))
Pharmaxis

Curated by ChEMBL
LigandPNGBDBM50246766(CHEMBL489079 | Mofegiline | US9302986, Mofegiline)
Affinity DataIC50:  10nMAssay Description:Inhibition of human recombinant MAO-B assessed as H2O2 production by Resorufin/Amplex Red assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMembrane primary amine oxidase(Homo sapiens (Human))
Pharmaxis

Curated by ChEMBL
LigandPNGBDBM50384084(CHEMBL2029546)
Affinity DataIC50:  10nMAssay Description:Inhibition of human recombinant SSAO/VAP1 assessed as H2O2 production by Resorufin/Amplex Red assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRetina-specific copper amine oxidase(Homo sapiens (Human))
Pharmaxis

Curated by ChEMBL
LigandPNGBDBM50589702(CHEMBL5186190)
Affinity DataIC50:  11nMAssay Description:Inhibition of recombinant human SSAOMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetRetina-specific copper amine oxidase(Homo sapiens (Human))
Pharmaxis

Curated by ChEMBL
LigandPNGBDBM50589699(CHEMBL5197971)
Affinity DataIC50:  12nMAssay Description:Inhibition of recombinant human SSAOMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetLysyl oxidase homolog 2(Homo sapiens (Human))
Pharmaxis

Curated by ChEMBL
LigandPNGBDBM50505638(CHEMBL4457578)
Affinity DataIC50:  13nMAssay Description:Inhibition of recombinant human LOXL2 assessed as inhibition of collagen cross linking compound replenishment for 5 days and measured on day 7 by UPL...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] B(Homo sapiens (Human))
Pharmaxis

Curated by ChEMBL
LigandPNGBDBM50589697(CHEMBL5194056)
Affinity DataIC50:  13nMAssay Description:Inhibition of human recombinant MAO-BMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetLysyl oxidase homolog 2(Homo sapiens (Human))
Pharmaxis

Curated by ChEMBL
LigandPNGBDBM50505640(CHEMBL4556859)
Affinity DataIC50:  13nMAssay Description:Inhibition of recombinant human C-terminal His-tagged LOLX2 (1-774 residues) expressed in mouse myeloma cells using putrescine as substrate preincuba...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetLysyl oxidase homolog 2(Homo sapiens (Human))
Pharmaxis

Curated by ChEMBL
LigandPNGBDBM50505638(CHEMBL4457578)
Affinity DataIC50:  13nMAssay Description:Inhibition of recombinant human C-terminal His-tagged LOLX2 (1-774 residues) expressed in mouse myeloma cells assessed as inhibition of collagen oxid...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetLysyl oxidase homolog 3(Homo sapiens (Human))
Pharmaxis

Curated by ChEMBL
LigandPNGBDBM50505638(CHEMBL4457578)
Affinity DataIC50:  16nMAssay Description:Inhibition of recombinant C-terminal His-tagged human LOXL3 (1 to 753 residues) expressed in CHO cells using putrescine as substrate preincubated wit...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetRetina-specific copper amine oxidase(Homo sapiens (Human))
Pharmaxis

Curated by ChEMBL
LigandPNGBDBM50589697(CHEMBL5194056)
Affinity DataIC50:  19nMAssay Description:Inhibition of recombinant human SSAOMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetRetina-specific copper amine oxidase(Homo sapiens (Human))
Pharmaxis

Curated by ChEMBL
LigandPNGBDBM50589703(CHEMBL5196906)
Affinity DataIC50:  19nMAssay Description:Inhibition of recombinant human SSAOMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetLysyl oxidase homolog 2(Homo sapiens (Human))
Pharmaxis

Curated by ChEMBL
LigandPNGBDBM50505653(CHEMBL4458907)
Affinity DataIC50:  20nMAssay Description:Inhibition of recombinant human C-terminal His-tagged LOLX2 (1-774 residues) expressed in mouse myeloma cells using putrescine as substrate preincuba...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetLysyl oxidase homolog 2(Homo sapiens (Human))
Pharmaxis

Curated by ChEMBL
LigandPNGBDBM50505658(CHEMBL4581458)
Affinity DataIC50:  20nMAssay Description:Inhibition of recombinant human C-terminal His-tagged LOLX2 (1-774 residues) expressed in mouse myeloma cells using putrescine as substrate preincuba...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLysyl oxidase homolog 2(Homo sapiens (Human))
Pharmaxis

Curated by ChEMBL
LigandPNGBDBM50505647(CHEMBL4531065)
Affinity DataIC50:  20nMAssay Description:Inhibition of recombinant human C-terminal His-tagged LOLX2 (1-774 residues) expressed in mouse myeloma cells using putrescine as substrate preincuba...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetMembrane primary amine oxidase(Homo sapiens (Human))
Pharmaxis

Curated by ChEMBL
LigandPNGBDBM50246766(CHEMBL489079 | Mofegiline | US9302986, Mofegiline)
Affinity DataIC50:  20nMAssay Description:Inhibition of human recombinant SSAO/VAP1 assessed as H2O2 production by Resorufin/Amplex Red assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLysyl oxidase homolog 2(Homo sapiens (Human))
Pharmaxis

Curated by ChEMBL
LigandPNGBDBM50505657(CHEMBL4467234)
Affinity DataIC50:  20nMAssay Description:Inhibition of recombinant human C-terminal His-tagged LOLX2 (1-774 residues) expressed in mouse myeloma cells using putrescine as substrate preincuba...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetMembrane primary amine oxidase(Homo sapiens (Human))
Pharmaxis

Curated by ChEMBL
LigandPNGBDBM50384083(CHEMBL2029545)
Affinity DataIC50:  20nMAssay Description:Inhibition of human recombinant SSAO/VAP1 assessed as H2O2 production by Resorufin/Amplex Red assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMembrane primary amine oxidase(Homo sapiens (Human))
Pharmaxis

Curated by ChEMBL
LigandPNGBDBM50384095(CHEMBL2029534)
Affinity DataIC50:  20nMAssay Description:Inhibition of human recombinant SSAO/VAP1 assessed as H2O2 production by Resorufin/Amplex Red assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLysyl oxidase homolog 2(Homo sapiens (Human))
Pharmaxis

Curated by ChEMBL
LigandPNGBDBM50505643(CHEMBL4582216)
Affinity DataIC50:  25nMAssay Description:Inhibition of recombinant human C-terminal His-tagged LOLX2 (1-774 residues) expressed in mouse myeloma cells using putrescine as substrate preincuba...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] B(Homo sapiens (Human))
Pharmaxis

Curated by ChEMBL
LigandPNGBDBM50589701(CHEMBL5186898)
Affinity DataIC50:  26nMAssay Description:Inhibition of human recombinant MAO-BMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetRetina-specific copper amine oxidase(Homo sapiens (Human))
Pharmaxis

Curated by ChEMBL
LigandPNGBDBM50589703(CHEMBL5196906)
Affinity DataIC50:  29nMAssay Description:Inhibition of SSAO in HMEC cellsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetMembrane primary amine oxidase(Homo sapiens (Human))
Pharmaxis

Curated by ChEMBL
LigandPNGBDBM50384087(CHEMBL2029549)
Affinity DataIC50:  30nMAssay Description:Inhibition of human recombinant SSAO/VAP1 assessed as H2O2 production by Resorufin/Amplex Red assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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