Affinity DataIC50: 260nMAssay Description:HIV integrase inhibitory potency of the compound was evaluated as IC50 on 3' processing of target DNA.More data for this Ligand-Target Pair
Affinity DataIC50: 300nMAssay Description:HIV integrase inhibitory potency of the compound was evaluated as IC50 on 3' processing of target DNA.More data for this Ligand-Target Pair
Affinity DataIC50: 300nMAssay Description:Inhibitory activity against Integrase in 3'-end- processingMore data for this Ligand-Target Pair
Affinity DataIC50: 300nMAssay Description:Inhibition of human immunodeficiency virus-1 (HIV-1) integrase.Checked by AuthorMore data for this Ligand-Target Pair
Affinity DataIC50: 400nMAssay Description:In vitro anti-HIV integrase activity of the compound was tested against integration(strand transfer) of target plasmid.More data for this Ligand-Target Pair
Affinity DataIC50: 400nMAssay Description:Inhibitory activity against Integrase in strand transfer(integration)More data for this Ligand-Target Pair
Affinity DataIC50: 600nMAssay Description:In vitro anti-HIV integrase activity of the compound was tested against integration(strand transfer) of target plasmid.More data for this Ligand-Target Pair
Affinity DataIC50: 700nMAssay Description:In vitro inhibition of recombinant integrase activity in a standard 3'-processing assay.More data for this Ligand-Target Pair
Affinity DataIC50: 700nMAssay Description:Inhibitory activity against Integrase in 3'-end- processingMore data for this Ligand-Target Pair
Affinity DataIC50: 800nMAssay Description:HIV integrase inhibitory potency of the compound was evaluated as IC50 on 3' processing of target DNA.More data for this Ligand-Target Pair
Affinity DataIC50: 900nMAssay Description:In vitro inhibition of recombinant integrase activity in a standard 3'-processing assay.More data for this Ligand-Target Pair
Affinity DataIC50: 900nMAssay Description:Inhibitory activity against HIV-1 Integrase in 3'-end- processingMore data for this Ligand-Target Pair
Affinity DataIC50: 1.00E+3nMAssay Description:In vitro anti-HIV integrase activity of the compound was tested against integration(strand transfer) of target plasmid.More data for this Ligand-Target Pair
Affinity DataIC50: 1.00E+3nMAssay Description:Inhibitory activity against Integrase in strand transfer(integration)More data for this Ligand-Target Pair
Affinity DataIC50: 1.00E+3nMAssay Description:In vitro inhibitory concentration against HIV-1 recombinant integrase activity in strand transfer assayMore data for this Ligand-Target Pair
Affinity DataIC50: 1.00E+3nMAssay Description:Inhibition of PIM1More data for this Ligand-Target Pair
Affinity DataIC50: 1.00E+3nMAssay Description:Inhibition of PIM1More data for this Ligand-Target Pair
TargetDual specificity tyrosine-phosphorylation-regulated kinase 2(Homo sapiens (Human))
Universit£
Curated by ChEMBL
Universit£
Curated by ChEMBL
Affinity DataIC50: 1.10E+3nMAssay Description:Inhibition of DYRK2More data for this Ligand-Target Pair
Affinity DataIC50: 1.20E+3nMAssay Description:Inhibitory activity against HIV-1 Integrase in strand transfer(integration)More data for this Ligand-Target Pair
Affinity DataIC50: 1.20E+3nMAssay Description:Inhibitory activity against HIV-1 Integrase in 3'-end- processingMore data for this Ligand-Target Pair
Affinity DataIC50: 1.20E+3nMAssay Description:Inhibitory activity against HIV-1 Integrase in strand transfer(integration)More data for this Ligand-Target Pair
Affinity DataIC50: 1.30E+3nMAssay Description:Inhibitory activity against HIV-1 Integrase in 3'-end- processingMore data for this Ligand-Target Pair
TargetDual specificity tyrosine-phosphorylation-regulated kinase 1A(Mus musculus)
Universit£
Curated by ChEMBL
Universit£
Curated by ChEMBL
Affinity DataIC50: 1.30E+3nMAssay Description:Inhibition of mouse DYRK1A expressed in Escherichia coli after 20 minsMore data for this Ligand-Target Pair
Affinity DataIC50: 1.40E+3nMAssay Description:Inhibitory activity against HIV-1 Integrase in 3'-end- processingMore data for this Ligand-Target Pair
Affinity DataIC50: 1.50E+3nMAssay Description:In vitro inhibition of recombinant integrase activity in a standard 3'-processing assay.More data for this Ligand-Target Pair
Affinity DataIC50: 1.50E+3nMAssay Description:Inhibitory activity against Integrase in strand transfer(integration)More data for this Ligand-Target Pair
Affinity DataIC50: 1.60E+3nMAssay Description:Inhibitory activity against HIV-1 Integrase in 3'-end- processingMore data for this Ligand-Target Pair
Affinity DataIC50: 1.60E+3nMAssay Description:Inhibitory activity against HIV-1 Integrase in strand transfer(integration)More data for this Ligand-Target Pair
Affinity DataIC50: 1.70E+3nMAssay Description:Inhibitory activity against Integrase in strand transfer(integration)More data for this Ligand-Target Pair
Affinity DataIC50: 1.70E+3nMAssay Description:Inhibitory activity against HIV-1 Integrase in strand transfer(integration)More data for this Ligand-Target Pair
Affinity DataIC50: 1.70E+3nMAssay Description:Inhibition of PIM1More data for this Ligand-Target Pair
Affinity DataIC50: 1.90E+3nMAssay Description:Inhibitory activity against HIV-1 Integrase in 3'-end- processing was tested in CEM cellsMore data for this Ligand-Target Pair
Affinity DataIC50: 2.00E+3nMAssay Description:In vitro inhibitory concentration against HIV-1 recombinant integrase activity in standard 3'-processing assayMore data for this Ligand-Target Pair
Affinity DataIC50: 2.00E+3nMAssay Description:Inhibition of PIM1More data for this Ligand-Target Pair
Affinity DataIC50: 2.00E+3nMAssay Description:Inhibition of PIM1More data for this Ligand-Target Pair
Affinity DataIC50: 2.10E+3nMAssay Description:Inhibitory activity against HIV-1 Integrase in strand transfer(integration)More data for this Ligand-Target Pair
Affinity DataIC50: 2.10E+3nMAssay Description:Inhibition of PIM1More data for this Ligand-Target Pair
Affinity DataIC50: 2.10E+3nMAssay Description:Inhibition of PIM1More data for this Ligand-Target Pair
TargetGag-Pol polyprotein(Rous sarcoma virus (strain Prague C) (RSV-PrC))
Cnrs Umr 8532
Curated by ChEMBL
Cnrs Umr 8532
Curated by ChEMBL
Affinity DataIC50: 2.10E+3nMAssay Description:Inhibition of rous sarcoma virus (RSV) Integrase.Checked by AuthorMore data for this Ligand-Target Pair
Affinity DataIC50: 2.20E+3nMAssay Description:HIV integrase inhibitory potency of the compound was evaluated as IC50 on 3' processing of target DNA.More data for this Ligand-Target Pair
Affinity DataIC50: 2.20E+3nMAssay Description:Inhibitory activity against HIV-1 Integrase in strand transfer(integration)More data for this Ligand-Target Pair
Affinity DataIC50: 2.30E+3nMAssay Description:In vitro inhibition of recombinant integrase activity in a standard 3'-processing assay.More data for this Ligand-Target Pair
Affinity DataIC50: 2.30E+3nMAssay Description:Inhibitory activity against Integrase in 3'-end- processingMore data for this Ligand-Target Pair