TargetSerine/threonine-protein kinase PLK1(Homo sapiens (Human))
University Of Massachusetts-Boston
Curated by ChEMBL
University Of Massachusetts-Boston
Curated by ChEMBL
Affinity DataIC50: 1.10nMAssay Description:Inhibition of human recombinant PLK1 by Z-Lyte assayMore data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase PLK1(Homo sapiens (Human))
University Of Massachusetts-Boston
Curated by ChEMBL
University Of Massachusetts-Boston
Curated by ChEMBL
Affinity DataIC50: 4nMAssay Description:Inhibition of human recombinant PLK1 by Z-Lyte assayMore data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase PLK1(Homo sapiens (Human))
University Of Massachusetts-Boston
Curated by ChEMBL
University Of Massachusetts-Boston
Curated by ChEMBL
Affinity DataIC50: 4nMAssay Description:Inhibition of human recombinant PLK1 by Z-Lyte assayMore data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase PLK1(Homo sapiens (Human))
University Of Massachusetts-Boston
Curated by ChEMBL
University Of Massachusetts-Boston
Curated by ChEMBL
Affinity DataIC50: 4nMAssay Description:Inhibition of human recombinant PLK1 by Z-Lyte assayMore data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase PLK1(Homo sapiens (Human))
University Of Massachusetts-Boston
Curated by ChEMBL
University Of Massachusetts-Boston
Curated by ChEMBL
Affinity DataIC50: 8.40nMAssay Description:Inhibition of human recombinant PLK1 by Z-Lyte assayMore data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase PLK1(Homo sapiens (Human))
University Of Massachusetts-Boston
Curated by ChEMBL
University Of Massachusetts-Boston
Curated by ChEMBL
Affinity DataIC50: 8.60nMAssay Description:Inhibition of human recombinant PLK1 by Z-Lyte assayMore data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase PLK1(Homo sapiens (Human))
University Of Massachusetts-Boston
Curated by ChEMBL
University Of Massachusetts-Boston
Curated by ChEMBL
Affinity DataIC50: 8.70nMAssay Description:Inhibition of human recombinant PLK1 by Z-Lyte assayMore data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase PLK1(Homo sapiens (Human))
University Of Massachusetts-Boston
Curated by ChEMBL
University Of Massachusetts-Boston
Curated by ChEMBL
Affinity DataIC50: 9nMAssay Description:Inhibition of human recombinant PLK1 by Z-Lyte assayMore data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase PLK1(Homo sapiens (Human))
University Of Massachusetts-Boston
Curated by ChEMBL
University Of Massachusetts-Boston
Curated by ChEMBL
Affinity DataIC50: 9.90nMAssay Description:Inhibition of human recombinant PLK1 by Z-Lyte assayMore data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase PLK1(Homo sapiens (Human))
University Of Massachusetts-Boston
Curated by ChEMBL
University Of Massachusetts-Boston
Curated by ChEMBL
Affinity DataIC50: 21nMAssay Description:Inhibition of human recombinant PLK1 by Z-Lyte assayMore data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase PLK1(Homo sapiens (Human))
University Of Massachusetts-Boston
Curated by ChEMBL
University Of Massachusetts-Boston
Curated by ChEMBL
Affinity DataIC50: 25nMAssay Description:Inhibition of human recombinant PLK1 by Z-Lyte assayMore data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase PLK1(Homo sapiens (Human))
University Of Massachusetts-Boston
Curated by ChEMBL
University Of Massachusetts-Boston
Curated by ChEMBL
Affinity DataIC50: 27nMAssay Description:Inhibition of human recombinant PLK1 by Z-Lyte assayMore data for this Ligand-Target Pair
Affinity DataIC50: 28nMAssay Description:Inhibition of His-tagged CBP (unknown origin) using biotinylated-H3K56ac peptide as substrate incubated for 1 hr by AlphaScreen assayMore data for this Ligand-Target Pair
TargetBromodomain-containing protein 4(Homo sapiens (Human))
University Of Massachusetts-Boston
Curated by ChEMBL
University Of Massachusetts-Boston
Curated by ChEMBL
Affinity DataIC50: 28nMAssay Description:Inhibition of BRD4-BD1 (unknown origin) incubated for 1 hr by AlphaScreen biotin-JQ1 competition assayMore data for this Ligand-Target Pair
TargetBromodomain-containing protein 4(Homo sapiens (Human))
University Of Massachusetts-Boston
Curated by ChEMBL
University Of Massachusetts-Boston
Curated by ChEMBL
Affinity DataIC50: 32nMAssay Description:Inhibition of BRD4-BD1 (unknown origin) incubated for 1 hr by AlphaScreen biotin-JQ1 competition assayMore data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase PLK1(Homo sapiens (Human))
University Of Massachusetts-Boston
Curated by ChEMBL
University Of Massachusetts-Boston
Curated by ChEMBL
Affinity DataIC50: 33nMAssay Description:Inhibition of human recombinant PLK1 by Z-Lyte assayMore data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase PLK1(Homo sapiens (Human))
University Of Massachusetts-Boston
Curated by ChEMBL
University Of Massachusetts-Boston
Curated by ChEMBL
Affinity DataIC50: 37nMAssay Description:Inhibition of human recombinant PLK1 by Z-Lyte assayMore data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase PLK1(Homo sapiens (Human))
University Of Massachusetts-Boston
Curated by ChEMBL
University Of Massachusetts-Boston
Curated by ChEMBL
Affinity DataIC50: 40nMAssay Description:Inhibition of human recombinant PLK1 by Z-Lyte assayMore data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase PLK1(Homo sapiens (Human))
University Of Massachusetts-Boston
Curated by ChEMBL
University Of Massachusetts-Boston
Curated by ChEMBL
Affinity DataIC50: 47nMAssay Description:Inhibition of human recombinant PLK1 by Z-Lyte assayMore data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase PLK1(Homo sapiens (Human))
University Of Massachusetts-Boston
Curated by ChEMBL
University Of Massachusetts-Boston
Curated by ChEMBL
Affinity DataIC50: 54nMAssay Description:Inhibition of human recombinant PLK1 by Z-Lyte assayMore data for this Ligand-Target Pair
TargetBromodomain-containing protein 4(Homo sapiens (Human))
University Of Massachusetts-Boston
Curated by ChEMBL
University Of Massachusetts-Boston
Curated by ChEMBL
Affinity DataIC50: 59nMAssay Description:Inhibition of BRD4-BD1 (unknown origin) incubated for 1 hr by AlphaScreen biotin-JQ1 competition assayMore data for this Ligand-Target Pair
Affinity DataIC50: 64nMAssay Description:Inhibition of human CBP by FRET assayMore data for this Ligand-Target Pair
Affinity DataIC50: 72nMAssay Description:Inhibition of His-tagged CBP (unknown origin) using biotinylated-H3K56ac peptide as substrate incubated for 1 hr by AlphaScreen assayMore data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase PLK1(Homo sapiens (Human))
University Of Massachusetts-Boston
Curated by ChEMBL
University Of Massachusetts-Boston
Curated by ChEMBL
Affinity DataIC50: 78nMAssay Description:Inhibition of human recombinant PLK1 by Z-Lyte assayMore data for this Ligand-Target Pair
TargetBromodomain-containing protein 4(Homo sapiens (Human))
University Of Massachusetts-Boston
Curated by ChEMBL
University Of Massachusetts-Boston
Curated by ChEMBL
Affinity DataIC50: 84nMAssay Description:Inhibition of BRD4-BD1 (unknown origin) incubated for 1 hr by AlphaScreen biotin-JQ1 competition assayMore data for this Ligand-Target Pair
TargetBromodomain-containing protein 4(Homo sapiens (Human))
University Of Massachusetts-Boston
Curated by ChEMBL
University Of Massachusetts-Boston
Curated by ChEMBL
Affinity DataIC50: 94nMAssay Description:Inhibition of BRD4-BD1 (unknown origin) incubated for 1 hr by AlphaScreen biotin-JQ1 competition assayMore data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase PLK1(Homo sapiens (Human))
University Of Massachusetts-Boston
Curated by ChEMBL
University Of Massachusetts-Boston
Curated by ChEMBL
Affinity DataIC50: 95nMAssay Description:Inhibition of human recombinant PLK1 by Z-Lyte assayMore data for this Ligand-Target Pair
TargetBromodomain-containing protein 4(Homo sapiens (Human))
University Of Massachusetts-Boston
Curated by ChEMBL
University Of Massachusetts-Boston
Curated by ChEMBL
Affinity DataIC50: 95nMAssay Description:Inhibition of BRD4-BD1 (unknown origin) incubated for 1 hr by AlphaScreen biotin-JQ1 competition assayMore data for this Ligand-Target Pair
TargetBromodomain testis-specific protein(Homo sapiens (Human))
University Of Massachusetts-Boston
Curated by ChEMBL
University Of Massachusetts-Boston
Curated by ChEMBL
Affinity DataIC50: 102nMAssay Description:Inhibition of BRDT-BD1 (unknown origin) incubated for 1 hr by AlphaScreen biotin-JQ1 competition assayMore data for this Ligand-Target Pair
TargetBromodomain testis-specific protein(Homo sapiens (Human))
University Of Massachusetts-Boston
Curated by ChEMBL
University Of Massachusetts-Boston
Curated by ChEMBL
Affinity DataIC50: 103nMAssay Description:Inhibition of BRDT-BD1 (unknown origin) incubated for 1 hr by AlphaScreen biotin-JQ1 competition assayMore data for this Ligand-Target Pair
TargetBromodomain-containing protein 4(Homo sapiens (Human))
University Of Massachusetts-Boston
Curated by ChEMBL
University Of Massachusetts-Boston
Curated by ChEMBL
Affinity DataIC50: 104nMAssay Description:Inhibition of BRD4-BD1 (unknown origin) incubated for 1 hr by AlphaScreen biotin-JQ1 competition assayMore data for this Ligand-Target Pair
TargetBromodomain-containing protein 4(Homo sapiens (Human))
University Of Massachusetts-Boston
Curated by ChEMBL
University Of Massachusetts-Boston
Curated by ChEMBL
Affinity DataIC50: 107nMAssay Description:Inhibition of BRD4-BD1 (unknown origin) incubated for 1 hr by AlphaScreen biotin-JQ1 competition assayMore data for this Ligand-Target Pair
TargetBromodomain-containing protein 4(Homo sapiens (Human))
University Of Massachusetts-Boston
Curated by ChEMBL
University Of Massachusetts-Boston
Curated by ChEMBL
Affinity DataIC50: 107nMAssay Description:Inhibition of BRD4-BD1 (unknown origin) incubated for 1 hr by AlphaScreen biotin-JQ1 competition assayMore data for this Ligand-Target Pair
TargetBromodomain-containing protein 4(Homo sapiens (Human))
University Of Massachusetts-Boston
Curated by ChEMBL
University Of Massachusetts-Boston
Curated by ChEMBL
Affinity DataIC50: 109nMAssay Description:Inhibition of BRD4-BD1 (unknown origin) incubated for 1 hr by AlphaScreen biotin-JQ1 competition assayMore data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase PLK1(Homo sapiens (Human))
University Of Massachusetts-Boston
Curated by ChEMBL
University Of Massachusetts-Boston
Curated by ChEMBL
Affinity DataIC50: 127nMAssay Description:Inhibition of human recombinant PLK1 by Z-Lyte assayMore data for this Ligand-Target Pair
Affinity DataIC50: 130nMAssay Description:Inhibition of CBP (unknown origin) by FRET assayMore data for this Ligand-Target Pair
Affinity DataIC50: 159nMAssay Description:Inhibition of His-tagged CBP (unknown origin) using biotinylated-H3K56ac peptide as substrate incubated for 1 hr by AlphaScreen assayMore data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase PLK1(Homo sapiens (Human))
University Of Massachusetts-Boston
Curated by ChEMBL
University Of Massachusetts-Boston
Curated by ChEMBL
Affinity DataIC50: 160nMAssay Description:Inhibition of human recombinant PLK1 by Z-Lyte assayMore data for this Ligand-Target Pair
TargetBromodomain-containing protein 4(Homo sapiens (Human))
University Of Massachusetts-Boston
Curated by ChEMBL
University Of Massachusetts-Boston
Curated by ChEMBL
Affinity DataIC50: 183nMAssay Description:Inhibition of BRD4-BD1 (unknown origin) incubated for 1 hr by AlphaScreen biotin-JQ1 competition assayMore data for this Ligand-Target Pair
TargetBromodomain-containing protein 4(Homo sapiens (Human))
University Of Massachusetts-Boston
Curated by ChEMBL
University Of Massachusetts-Boston
Curated by ChEMBL
Affinity DataIC50: 186nMAssay Description:Inhibition of BRD4-BD1 (unknown origin) incubated for 1 hr by AlphaScreen biotin-JQ1 competition assayMore data for this Ligand-Target Pair
TargetBromodomain-containing protein 4(Homo sapiens (Human))
University Of Massachusetts-Boston
Curated by ChEMBL
University Of Massachusetts-Boston
Curated by ChEMBL
Affinity DataIC50: 205nMAssay Description:Inhibition of BRD4-BD1 (unknown origin) incubated for 1 hr by AlphaScreen biotin-JQ1 competition assayMore data for this Ligand-Target Pair
Affinity DataIC50: 214nMAssay Description:Inhibition of His-tagged CBP (unknown origin) using biotinylated-H3K56ac peptide as substrate incubated for 1 hr by AlphaScreen assayMore data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase PLK1(Homo sapiens (Human))
University Of Massachusetts-Boston
Curated by ChEMBL
University Of Massachusetts-Boston
Curated by ChEMBL
Affinity DataIC50: 218nMAssay Description:Inhibition of human recombinant PLK1 by Z-Lyte assayMore data for this Ligand-Target Pair
TargetBromodomain testis-specific protein(Homo sapiens (Human))
University Of Massachusetts-Boston
Curated by ChEMBL
University Of Massachusetts-Boston
Curated by ChEMBL
Affinity DataIC50: 229nMAssay Description:Inhibition of BRDT-BD1 (unknown origin) incubated for 1 hr by AlphaScreen biotin-JQ1 competition assayMore data for this Ligand-Target Pair
TargetBromodomain testis-specific protein(Homo sapiens (Human))
University Of Massachusetts-Boston
Curated by ChEMBL
University Of Massachusetts-Boston
Curated by ChEMBL
Affinity DataIC50: 245nMAssay Description:Inhibition of BRDT-BD1 (unknown origin) incubated for 1 hr by AlphaScreen biotin-JQ1 competition assayMore data for this Ligand-Target Pair
TargetBromodomain-containing protein 4(Homo sapiens (Human))
University Of Massachusetts-Boston
Curated by ChEMBL
University Of Massachusetts-Boston
Curated by ChEMBL
Affinity DataIC50: 253nMAssay Description:Inhibition of BRD4-BD1 (unknown origin) incubated for 1 hr by AlphaScreen biotin-JQ1 competition assayMore data for this Ligand-Target Pair
TargetBromodomain testis-specific protein(Homo sapiens (Human))
University Of Massachusetts-Boston
Curated by ChEMBL
University Of Massachusetts-Boston
Curated by ChEMBL
Affinity DataIC50: 289nMAssay Description:Inhibition of BRDT-BD1 (unknown origin) incubated for 1 hr by AlphaScreen biotin-JQ1 competition assayMore data for this Ligand-Target Pair
Affinity DataIC50: 290nMAssay Description:Inhibition of His-tagged CBP (unknown origin) using biotinylated-H3K56ac peptide as substrate incubated for 1 hr by AlphaScreen assayMore data for this Ligand-Target Pair
TargetBromodomain-containing protein 4(Homo sapiens (Human))
University Of Massachusetts-Boston
Curated by ChEMBL
University Of Massachusetts-Boston
Curated by ChEMBL
Affinity DataIC50: 310nMAssay Description:Inhibition of BRD4-BD1 (unknown origin) incubated for 1 hr by AlphaScreen biotin-JQ1 competition assayMore data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase PLK1(Homo sapiens (Human))
University Of Massachusetts-Boston
Curated by ChEMBL
University Of Massachusetts-Boston
Curated by ChEMBL
Affinity DataIC50: 322nMAssay Description:Inhibition of human recombinant PLK1 by Z-Lyte assayMore data for this Ligand-Target Pair