Compile Data Set for Download or QSAR
maximum 50k data
Found 32 with Last Name = 'dimilo' and Initial = 'e'
TargetAlpha-1A adrenergic receptor(Homo sapiens (Human))
Marquette University

Curated by ChEMBL
LigandPNGBDBM50529214(CHEMBL343822)
Affinity DataKi:  1.10E+3nMAssay Description:Inhibition of alpha1A adrenergic receptor (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1A/Alpha-1B/Alpha-1D adrenergic receptor(Homo sapiens (Human))
Marquette University

Curated by ChEMBL
LigandPNGBDBM50529212(CHEMBL4471453)
Affinity DataKi:  1.80E+3nMAssay Description:Inhibition of alpha1 adrenergic receptor (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProtein polybromo-1(Homo sapiens (Human))
Marquette University

Curated by ChEMBL
LigandPNGBDBM50529212(CHEMBL4471453)
Affinity DataKi:  2.50E+3nMAssay Description:Inhibition of PBR receptor (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAlpha-1A/Alpha-1B/Alpha-1D adrenergic receptor(Homo sapiens (Human))
Marquette University

Curated by ChEMBL
LigandPNGBDBM50529214(CHEMBL343822)
Affinity DataKi:  3.90E+3nMAssay Description:Inhibition of alpha1 adrenergic receptor (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1A/Alpha-1B/Alpha-1D adrenergic receptor(Homo sapiens (Human))
Marquette University

Curated by ChEMBL
LigandPNGBDBM50529213(CHEMBL4465132)
Affinity DataKi: >1.00E+4nMAssay Description:Inhibition of alpha1 adrenergic receptor (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetD(3) dopamine receptor(Homo sapiens (Human))
Marquette University

Curated by ChEMBL
LigandPNGBDBM50529213(CHEMBL4465132)
Affinity DataKi: >1.00E+4nMAssay Description:Inhibition of D3 receptor (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily KQT member 2(Homo sapiens (Human))
Marquette University

Curated by ChEMBL
LigandPNGBDBM50529214(CHEMBL343822)
Affinity DataIC50:  48nMAssay Description:Inhibition of Kv7.2 in human HEK293 cells incubated for 1 hr by thallium flux assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily KQT member 2(Homo sapiens (Human))
Marquette University

Curated by ChEMBL
LigandPNGBDBM50529215(CHEBI:35046 | CHEMBL342375)
Affinity DataIC50:  55nMAssay Description:Inhibition of Kv7.2 in human HEK293 cells incubated for 1 hr by thallium flux assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily KQT member 2(Homo sapiens (Human))
Marquette University

Curated by ChEMBL
LigandPNGBDBM50529213(CHEMBL4465132)
Affinity DataIC50:  160nMAssay Description:Inhibition of Kv7.2 in human HEK293 cells incubated for 1 hr by thallium flux assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProteinase-activated receptor 1(Homo sapiens (Human))
Marquette University

Curated by ChEMBL
LigandPNGBDBM50512562(CHEMBL4438936)
Affinity DataIC50:  200nMAssay Description:Negative allosteric modulation of PAR1 in human EAhy926 cells assessed as reduction in TFLLRN-NH2-induced intracellular calcium mobilization incubate...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily KQT member 2(Homo sapiens (Human))
Marquette University

Curated by ChEMBL
LigandPNGBDBM50529212(CHEMBL4471453)
Affinity DataIC50:  200nMAssay Description:Inhibition of Kv7.2 in human HEK293 cells incubated for 1 hr by thallium flux assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProteinase-activated receptor 1(Homo sapiens (Human))
Marquette University

Curated by ChEMBL
LigandPNGBDBM50512562(CHEMBL4438936)
Affinity DataIC50:  220nMAssay Description:Negative allosteric modulation of PAR1 in human EAhy926 cells assessed as reduction in TFLLRN-NH2-induced intracellular calcium mobilization incubate...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProteinase-activated receptor 1(Homo sapiens (Human))
Marquette University

Curated by ChEMBL
LigandPNGBDBM50512565(CHEMBL4451525)
Affinity DataIC50:  316nMAssay Description:Negative allosteric modulation of PAR1 in human EAhy926 cells assessed as reduction in TFLLRN-NH2-induced intracellular calcium mobilization incubate...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProteinase-activated receptor 1(Homo sapiens (Human))
Marquette University

Curated by ChEMBL
LigandPNGBDBM50512565(CHEMBL4451525)
Affinity DataIC50:  320nMAssay Description:Negative allosteric modulation of PAR1 in human EAhy926 cells assessed as reduction in TFLLRN-NH2-induced intracellular calcium mobilization incubate...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProteinase-activated receptor 1(Homo sapiens (Human))
Marquette University

Curated by ChEMBL
LigandPNGBDBM50512563(CHEMBL4514779)
Affinity DataIC50:  370nMAssay Description:Negative allosteric modulation of PAR1 in human EAhy926 cells assessed as reduction in TFLLRN-NH2-induced intracellular calcium mobilization incubate...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProteinase-activated receptor 1(Homo sapiens (Human))
Marquette University

Curated by ChEMBL
LigandPNGBDBM50512563(CHEMBL4514779)
Affinity DataIC50:  370nMAssay Description:Negative allosteric modulation of PAR1 in human EAhy926 cells assessed as reduction in TFLLRN-NH2-induced intracellular calcium mobilization incubate...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProteinase-activated receptor 1(Homo sapiens (Human))
Marquette University

Curated by ChEMBL
LigandPNGBDBM50512561(CHEMBL4448258)
Affinity DataIC50:  380nMAssay Description:Negative allosteric modulation of PAR1 in human EAhy926 cells assessed as reduction in TFLLRN-NH2-induced intracellular calcium mobilization incubate...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProteinase-activated receptor 1(Homo sapiens (Human))
Marquette University

Curated by ChEMBL
LigandPNGBDBM50512564(CHEMBL4594058)
Affinity DataIC50:  398nMAssay Description:Negative allosteric modulation of PAR1 in human EAhy926 cells assessed as reduction in TFLLRN-NH2-induced intracellular calcium mobilization incubate...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProteinase-activated receptor 1(Homo sapiens (Human))
Marquette University

Curated by ChEMBL
LigandPNGBDBM50512561(CHEMBL4448258)
Affinity DataIC50:  398nMAssay Description:Negative allosteric modulation of PAR1 in human EAhy926 cells assessed as reduction in TFLLRN-NH2-induced intracellular calcium mobilization incubate...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProteinase-activated receptor 1(Homo sapiens (Human))
Marquette University

Curated by ChEMBL
LigandPNGBDBM50512564(CHEMBL4594058)
Affinity DataIC50:  420nMAssay Description:Negative allosteric modulation of PAR1 in human EAhy926 cells assessed as reduction in TFLLRN-NH2-induced intracellular calcium mobilization incubate...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily KQT member 2(Homo sapiens (Human))
Marquette University

Curated by ChEMBL
LigandPNGBDBM50529217(CHEMBL4447214)
Affinity DataIC50:  540nMAssay Description:Inhibition of Kv7.2 in human HEK293 cells incubated for 1 hr by thallium flux assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProteinase-activated receptor 1(Homo sapiens (Human))
Marquette University

Curated by ChEMBL
LigandPNGBDBM50386391(CHEMBL1411333)
Affinity DataIC50:  794nMAssay Description:Negative allosteric modulation of PAR1 in human EAhy926 cells assessed as reduction in TFLLRN-NH2-induced intracellular calcium mobilization incubate...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProteinase-activated receptor 1(Homo sapiens (Human))
Marquette University

Curated by ChEMBL
LigandPNGBDBM50386391(CHEMBL1411333)
Affinity DataIC50:  794nMAssay Description:Negative allosteric modulation of PAR1 in human EAhy926 cells assessed as reduction in TFLLRN-NH2-induced intracellular calcium mobilization incubate...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProteinase-activated receptor 1(Homo sapiens (Human))
Marquette University

Curated by ChEMBL
LigandPNGBDBM50386408(CHEMBL2047297)
Affinity DataIC50:  1.00E+3nMAssay Description:Negative allosteric modulation of PAR1 in human EAhy926 cells assessed as reduction in TFLLRN-NH2-induced intracellular calcium mobilization incubate...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProteinase-activated receptor 1(Homo sapiens (Human))
Marquette University

Curated by ChEMBL
LigandPNGBDBM50386404(CHEMBL1332325)
Affinity DataIC50:  3.16E+3nMAssay Description:Negative allosteric modulation of PAR1 in human EAhy926 cells assessed as reduction in TFLLRN-NH2-induced intracellular calcium mobilization incubate...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily KQT member 2(Homo sapiens (Human))
Marquette University

Curated by ChEMBL
LigandPNGBDBM50529216(CHEMBL4444584)
Affinity DataIC50:  5.60E+3nMAssay Description:Inhibition of Kv7.2 in human HEK293 cells incubated for 1 hr by thallium flux assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily KQT member 2(Homo sapiens (Human))
Marquette University

Curated by ChEMBL
LigandPNGBDBM50529218(CHEMBL4473641)
Affinity DataIC50:  1.00E+4nMAssay Description:Inhibition of Kv7.2 in human HEK293 cells incubated for 1 hr by thallium flux assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProteinase-activated receptor 1(Homo sapiens (Human))
Marquette University

Curated by ChEMBL
LigandPNGBDBM50461683(CHEMBL4227184)
Affinity DataIC50: <1.00E+4nMAssay Description:Negative allosteric modulation of PAR1 in human EAhy926 cells assessed as reduction in TFLLRN-NH2-induced intracellular calcium mobilization incubate...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
Target1,3-beta-glucan synthase component GSC2(Saccharomyces cerevisiae)
Marquette University

Curated by ChEMBL
LigandPNGBDBM50529212(CHEMBL4471453)
Affinity DataIC50:  1.20E+4nMAssay Description:Inhibition of ERG in human HEK293 cells incubated for 1 hr by thallium flux assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
Target1,3-beta-glucan synthase component GSC2(Saccharomyces cerevisiae)
Marquette University

Curated by ChEMBL
LigandPNGBDBM50529213(CHEMBL4465132)
Affinity DataIC50: >3.20E+4nMAssay Description:Inhibition of ERG in human HEK293 cells incubated for 1 hr by thallium flux assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
Target1,3-beta-glucan synthase component GSC2(Saccharomyces cerevisiae)
Marquette University

Curated by ChEMBL
LigandPNGBDBM50529214(CHEMBL343822)
Affinity DataIC50:  3.20E+4nMAssay Description:Inhibition of ERG in human HEK293 cells incubated for 1 hr by thallium flux assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target1,3-beta-glucan synthase component GSC2(Saccharomyces cerevisiae)
Marquette University

Curated by ChEMBL
LigandPNGBDBM50529215(CHEBI:35046 | CHEMBL342375)
Affinity DataIC50: >3.20E+4nMAssay Description:Inhibition of ERG in human HEK293 cells incubated for 1 hr by thallium flux assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed