Compile Data Set for Download or QSAR
maximum 50k data
Found 37 with Last Name = 'dinda' and Initial = 'b'
TargetD(3) dopamine receptor(Rattus norvegicus (Rat))TBA
LigandPNGBDBM50610253(CHEMBL5283620)
Affinity DataKi:  1.30nMAssay Description:Displacement of [3H]-spiroperidol from rat D3 receptor expressed in HEK293 cells assessed as inhibition constant by Cheng-Prusoff equation analysisMore data for this Ligand-Target Pair
Ligand Info
In DepthDetails PubMed
TargetD(3) dopamine receptor(Rattus norvegicus (Rat))TBA
LigandPNGBDBM50610247(CHEMBL5276671)
Affinity DataKi:  1.80nMAssay Description:Displacement of [3H]-spiroperidol from rat D3 receptor expressed in HEK293 cells assessed as inhibition constant by Cheng-Prusoff equation analysisMore data for this Ligand-Target Pair
Ligand Info
In DepthDetails PubMed
TargetD(2) dopamine receptor(Rattus norvegicus (rat))TBA
LigandPNGBDBM50610247(CHEMBL5276671)
Affinity DataKi:  2nMAssay Description:Displacement of [3H]-spiroperidol from rat D2L receptor expressed in HEK293 cells assessed as inhibition constant by Cheng-Prusoff equation analysisMore data for this Ligand-Target Pair
Ligand Info
In DepthDetails PubMed
TargetD(3) dopamine receptor(Rattus norvegicus (Rat))TBA
LigandPNGBDBM50115277((2R,3R)-6-Dipropylamino-5,6,7,8-tetrahydro-naphtha...)
Affinity DataKi:  2.10nMAssay Description:Displacement of [3H]-spiroperidol from rat D3 receptor expressed in HEK293 cells assessed as inhibition constant by Cheng-Prusoff equation analysisMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetD(3) dopamine receptor(Rattus norvegicus (Rat))TBA
LigandPNGBDBM50610250(CHEMBL5267221)
Affinity DataKi:  2.20nMAssay Description:Displacement of [3H]-spiroperidol from rat D3 receptor expressed in HEK293 cells assessed as inhibition constant by Cheng-Prusoff equation analysisMore data for this Ligand-Target Pair
Ligand Info
In DepthDetails PubMed
TargetD(3) dopamine receptor(Rattus norvegicus (Rat))TBA
LigandPNGBDBM50610248(CHEMBL5274131)
Affinity DataKi:  3.60nMAssay Description:Displacement of [3H]-spiroperidol from rat D3 receptor expressed in HEK293 cells assessed as inhibition constant by Cheng-Prusoff equation analysisMore data for this Ligand-Target Pair
Ligand Info
In DepthDetails PubMed
TargetD(2) dopamine receptor(Rattus norvegicus (rat))TBA
LigandPNGBDBM50610249(CHEMBL5282690)
Affinity DataKi:  3.90nMAssay Description:Displacement of [3H]-spiroperidol from rat D2L receptor expressed in HEK293 cells assessed as inhibition constant by Cheng-Prusoff equation analysisMore data for this Ligand-Target Pair
Ligand Info
In DepthDetails PubMed
TargetD(3) dopamine receptor(Rattus norvegicus (Rat))TBA
LigandPNGBDBM50610249(CHEMBL5282690)
Affinity DataKi:  3.90nMAssay Description:Displacement of [3H]-spiroperidol from rat D3 receptor expressed in HEK293 cells assessed as inhibition constant by Cheng-Prusoff equation analysisMore data for this Ligand-Target Pair
Ligand Info
In DepthDetails PubMed
TargetD(2) dopamine receptor(Rattus norvegicus (rat))TBA
LigandPNGBDBM50610250(CHEMBL5267221)
Affinity DataKi:  4.90nMAssay Description:Displacement of [3H]-spiroperidol from rat D2L receptor expressed in HEK293 cells assessed as inhibition constant by Cheng-Prusoff equation analysisMore data for this Ligand-Target Pair
Ligand Info
In DepthDetails PubMed
TargetD(3) dopamine receptor(Rattus norvegicus (Rat))TBA
LigandPNGBDBM50610251(CHEMBL5272529)
Affinity DataKi:  5.20nMAssay Description:Displacement of [3H]-spiroperidol from rat D3 receptor expressed in HEK293 cells assessed as inhibition constant by Cheng-Prusoff equation analysisMore data for this Ligand-Target Pair
Ligand Info
In DepthDetails PubMed
TargetD(3) dopamine receptor(Rattus norvegicus (Rat))TBA
LigandPNGBDBM50610252(CHEMBL5266134)
Affinity DataKi:  6.90nMAssay Description:Displacement of [3H]-spiroperidol from rat D3 receptor expressed in HEK293 cells assessed as inhibition constant by Cheng-Prusoff equation analysisMore data for this Ligand-Target Pair
Ligand Info
In DepthDetails PubMed
TargetD(2) dopamine receptor(Rattus norvegicus (rat))TBA
LigandPNGBDBM50610251(CHEMBL5272529)
Affinity DataKi:  7.60nMAssay Description:Displacement of [3H]-spiroperidol from rat D2L receptor expressed in HEK293 cells assessed as inhibition constant by Cheng-Prusoff equation analysisMore data for this Ligand-Target Pair
Ligand Info
In DepthDetails PubMed
TargetD(2) dopamine receptor(Rattus norvegicus (rat))TBA
LigandPNGBDBM50610253(CHEMBL5283620)
Affinity DataKi:  8.30nMAssay Description:Displacement of [3H]-spiroperidol from rat D2L receptor expressed in HEK293 cells assessed as inhibition constant by Cheng-Prusoff equation analysisMore data for this Ligand-Target Pair
Ligand Info
In DepthDetails PubMed
TargetD(2) dopamine receptor(Rattus norvegicus (rat))TBA
LigandPNGBDBM50610248(CHEMBL5274131)
Affinity DataKi:  12nMAssay Description:Displacement of [3H]-spiroperidol from rat D2L receptor expressed in HEK293 cells assessed as inhibition constant by Cheng-Prusoff equation analysisMore data for this Ligand-Target Pair
Ligand Info
In DepthDetails PubMed
TargetD(2) dopamine receptor(Rattus norvegicus (rat))TBA
LigandPNGBDBM50610252(CHEMBL5266134)
Affinity DataKi:  55nMAssay Description:Displacement of [3H]-spiroperidol from rat D2L receptor expressed in HEK293 cells assessed as inhibition constant by Cheng-Prusoff equation analysisMore data for this Ligand-Target Pair
Ligand Info
In DepthDetails PubMed
TargetD(3) dopamine receptor(Rattus norvegicus (Rat))TBA
LigandPNGBDBM50610254(CHEMBL5265882)
Affinity DataKi:  115nMAssay Description:Displacement of [3H]-spiroperidol from rat D3 receptor expressed in HEK293 cells assessed as inhibition constant by Cheng-Prusoff equation analysisMore data for this Ligand-Target Pair
Ligand Info
In DepthDetails PubMed
TargetD(2) dopamine receptor(Rattus norvegicus (rat))TBA
LigandPNGBDBM50115277((2R,3R)-6-Dipropylamino-5,6,7,8-tetrahydro-naphtha...)
Affinity DataKi:  153nMAssay Description:Displacement of [3H]-spiroperidol from rat D2L receptor expressed in HEK293 cells assessed as inhibition constant by Cheng-Prusoff equation analysisMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetCytochrome P450 1A2(Homo sapiens (Human))
Tripura University

Curated by ChEMBL
LigandPNGBDBM50242173((2S,3S,4S,5R,6S)-6-(5,6-dihydroxy-4-oxo-2-phenyl-4...)
Affinity DataKi:  2.54E+4nMAssay Description:Mixed-type inhibition of CYP1A2 in pooled human liver microsomes using varying levels of phenacetin as substrate pretreated for 5 mins followed by su...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCytochrome P450 3A4(Homo sapiens (Human))
Tripura University

Curated by ChEMBL
LigandPNGBDBM50009001(5,6,7-Trihydroxyflavone | 5,6,7-trihydroxy-2-pheny...)
Affinity DataIC50:  9.20E+3nMAssay Description:Inhibition of human CYP3A4 expressed in baculovirus infected insect cells using 7-benzyloxy-4-trifluoromethylcoumarin as substrate measured after 45 ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Homo sapiens (Human))TBA
LigandPNGBDBM50610255(CHEMBL5275212)
Affinity DataEC50:  1.70nMAssay Description:Agonist activity at human D2 receptor expressed in CHO cells assessed as stimulation of [35S]GTPgammaS binding by Perkin elmer analysisMore data for this Ligand-Target Pair
Ligand Info
In DepthDetails PubMed
TargetD(2) dopamine receptor(Homo sapiens (Human))TBA
LigandPNGBDBM50610247(CHEMBL5276671)
Affinity DataEC50:  0.440nMAssay Description:Agonist activity at human D2 receptor expressed in CHO cells assessed as stimulation of [35S]GTPgammaS binding by Perkin elmer analysisMore data for this Ligand-Target Pair
Ligand Info
In DepthDetails PubMed
TargetD(2) dopamine receptor(Homo sapiens (Human))TBA
LigandPNGBDBM50610250(CHEMBL5267221)
Affinity DataEC50:  13nMAssay Description:Agonist activity at human D2 receptor expressed in CHO cells assessed as stimulation of [35S]GTPgammaS binding by Perkin elmer analysisMore data for this Ligand-Target Pair
Ligand Info
In DepthDetails PubMed
TargetD(2) dopamine receptor(Homo sapiens (Human))TBA
LigandPNGBDBM50610251(CHEMBL5272529)
Affinity DataEC50:  7.70nMAssay Description:Agonist activity at human D2 receptor expressed in CHO cells assessed as stimulation of [35S]GTPgammaS binding by Perkin elmer analysisMore data for this Ligand-Target Pair
Ligand Info
In DepthDetails PubMed
TargetD(2) dopamine receptor(Homo sapiens (Human))TBA
LigandPNGBDBM50610252(CHEMBL5266134)
Affinity DataEC50:  34nMAssay Description:Agonist activity at human D2 receptor expressed in CHO cells assessed as stimulation of [35S]GTPgammaS binding by Perkin elmer analysisMore data for this Ligand-Target Pair
Ligand Info
In DepthDetails PubMed
TargetD(2) dopamine receptor(Homo sapiens (Human))TBA
LigandPNGBDBM50610253(CHEMBL5283620)
Affinity DataEC50:  5.30nMAssay Description:Agonist activity at human D2 receptor expressed in CHO cells assessed as stimulation of [35S]GTPgammaS binding by Perkin elmer analysisMore data for this Ligand-Target Pair
Ligand Info
In DepthDetails PubMed
TargetD(2) dopamine receptor(Homo sapiens (Human))TBA
LigandPNGBDBM55121(3-HYDROXYTYRAMINE HYDROCHLORIDE | 4-(2-aminoethyl)...)
Affinity DataEC50:  200nMAssay Description:Agonist activity at human D2 receptor expressed in CHO cells assessed as stimulation of [35S]GTPgammaS binding by Perkin elmer analysisMore data for this Ligand-Target Pair
In DepthDetails PubMedDrugBank

TargetD(2) dopamine receptor(Homo sapiens (Human))TBA
LigandPNGBDBM50116766((-)-Pramipexole | (6S)-N(6)-propyl-4,5,6,7-tetrahy...)
Affinity DataEC50:  251nMAssay Description:Agonist activity at human D2 receptor expressed in CHO cells assessed as stimulation of [35S]GTPgammaS binding by Perkin elmer analysisMore data for this Ligand-Target Pair
In DepthDetails PubMedDrugBank

TargetD(3) dopamine receptor(Homo sapiens)TBA
LigandPNGBDBM50115277((2R,3R)-6-Dipropylamino-5,6,7,8-tetrahydro-naphtha...)
Affinity DataEC50:  0.630nMAssay Description:Agonist activity at human D3 receptor expressed in CHO cells assessed as stimulation of [35S]GTPgammaS binding by Perkin elmer analysisMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetD(3) dopamine receptor(Homo sapiens)TBA
LigandPNGBDBM50610255(CHEMBL5275212)
Affinity DataEC50:  0.530nMAssay Description:Agonist activity at human D3 receptor expressed in CHO cells assessed as stimulation of [35S]GTPgammaS binding by Perkin elmer analysisMore data for this Ligand-Target Pair
Ligand Info
In DepthDetails PubMed
TargetD(3) dopamine receptor(Homo sapiens)TBA
LigandPNGBDBM50610247(CHEMBL5276671)
Affinity DataEC50:  0.940nMAssay Description:Agonist activity at human D3 receptor expressed in CHO cells assessed as stimulation of [35S]GTPgammaS binding by Perkin elmer analysisMore data for this Ligand-Target Pair
Ligand Info
In DepthDetails PubMed
TargetD(3) dopamine receptor(Homo sapiens)TBA
LigandPNGBDBM50610250(CHEMBL5267221)
Affinity DataEC50:  13nMAssay Description:Agonist activity at human D3 receptor expressed in CHO cells assessed as stimulation of [35S]GTPgammaS binding by Perkin elmer analysisMore data for this Ligand-Target Pair
Ligand Info
In DepthDetails PubMed
TargetD(3) dopamine receptor(Homo sapiens)TBA
LigandPNGBDBM50610251(CHEMBL5272529)
Affinity DataEC50:  1.5nMAssay Description:Agonist activity at human D3 receptor expressed in CHO cells assessed as stimulation of [35S]GTPgammaS binding by Perkin elmer analysisMore data for this Ligand-Target Pair
Ligand Info
In DepthDetails PubMed
TargetD(3) dopamine receptor(Homo sapiens)TBA
LigandPNGBDBM50610252(CHEMBL5266134)
Affinity DataEC50:  5.40nMAssay Description:Agonist activity at human D3 receptor expressed in CHO cells assessed as stimulation of [35S]GTPgammaS binding by Perkin elmer analysisMore data for this Ligand-Target Pair
Ligand Info
In DepthDetails PubMed
TargetD(3) dopamine receptor(Homo sapiens)TBA
LigandPNGBDBM50610253(CHEMBL5283620)
Affinity DataEC50:  0.860nMAssay Description:Agonist activity at human D3 receptor expressed in CHO cells assessed as stimulation of [35S]GTPgammaS binding by Perkin elmer analysisMore data for this Ligand-Target Pair
Ligand Info
In DepthDetails PubMed
TargetD(3) dopamine receptor(Homo sapiens)TBA
LigandPNGBDBM55121(3-HYDROXYTYRAMINE HYDROCHLORIDE | 4-(2-aminoethyl)...)
Affinity DataEC50:  6.10nMAssay Description:Agonist activity at human D3 receptor expressed in CHO cells assessed as stimulation of [35S]GTPgammaS binding by Perkin elmer analysisMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetD(3) dopamine receptor(Homo sapiens)TBA
LigandPNGBDBM50116766((-)-Pramipexole | (6S)-N(6)-propyl-4,5,6,7-tetrahy...)
Affinity DataEC50:  4.10nMAssay Description:Agonist activity at human D3 receptor expressed in CHO cells assessed as stimulation of [35S]GTPgammaS binding by Perkin elmer analysisMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetD(2) dopamine receptor(Homo sapiens (Human))TBA
LigandPNGBDBM50115277((2R,3R)-6-Dipropylamino-5,6,7,8-tetrahydro-naphtha...)
Affinity DataEC50:  41nMAssay Description:Agonist activity at human D2 receptor expressed in CHO cells assessed as stimulation of [35S]GTPgammaS binding by Perkin elmer analysisMore data for this Ligand-Target Pair
In DepthDetails PubMed