Affinity DataIC50: 800nMAssay Description:Inhibition of EG5 (unknown origin)More data for this Ligand-Target Pair
TargetDNA topoisomerase 2-alpha(Homo sapiens (Human))
Dr. Babasaheb Ambedkar Marathwada University
Curated by ChEMBL
Dr. Babasaheb Ambedkar Marathwada University
Curated by ChEMBL
Affinity DataIC50: 990nMAssay Description:Inhibition of human topoisomerase-2 alpha in human A498 cells assessed as decrease in relaxation of supercoiled DNA at 10 uMMore data for this Ligand-Target Pair
TargetDNA topoisomerase 2-alpha(Homo sapiens (Human))
Dr. Babasaheb Ambedkar Marathwada University
Curated by ChEMBL
Dr. Babasaheb Ambedkar Marathwada University
Curated by ChEMBL
Affinity DataIC50: 1.03E+4nMAssay Description:Inhibition of human topoisomerase-2 alpha in human A498 cells assessed as decrease in relaxation of supercoiled DNA at 10 uMMore data for this Ligand-Target Pair
TargetDNA topoisomerase 2-alpha(Homo sapiens (Human))
Dr. Babasaheb Ambedkar Marathwada University
Curated by ChEMBL
Dr. Babasaheb Ambedkar Marathwada University
Curated by ChEMBL
Affinity DataIC50: 1.24E+4nMAssay Description:Inhibition of human topoisomerase-2 alpha in human A498 cells assessed as decrease in relaxation of supercoiled DNA at 10 uMMore data for this Ligand-Target Pair
TargetDNA topoisomerase 2-alpha(Homo sapiens (Human))
Dr. Babasaheb Ambedkar Marathwada University
Curated by ChEMBL
Dr. Babasaheb Ambedkar Marathwada University
Curated by ChEMBL
Affinity DataIC50: 1.67E+4nMAssay Description:Inhibition of human topoisomerase-2 alpha in human A498 cells assessed as decrease in relaxation of supercoiled DNA at 10 uMMore data for this Ligand-Target Pair
TargetDNA topoisomerase 2-alpha(Homo sapiens (Human))
Dr. Babasaheb Ambedkar Marathwada University
Curated by ChEMBL
Dr. Babasaheb Ambedkar Marathwada University
Curated by ChEMBL
Affinity DataIC50: 1.71E+4nMAssay Description:Inhibition of human topoisomerase-2 alpha in human A498 cells assessed as decrease in relaxation of supercoiled DNA at 10 uMMore data for this Ligand-Target Pair
TargetDNA topoisomerase 2-alpha(Homo sapiens (Human))
Dr. Babasaheb Ambedkar Marathwada University
Curated by ChEMBL
Dr. Babasaheb Ambedkar Marathwada University
Curated by ChEMBL
Affinity DataIC50: 2.64E+4nMAssay Description:Inhibition of human topoisomerase-2 alpha in human A498 cells assessed as decrease in relaxation of supercoiled DNA at 10 uMMore data for this Ligand-Target Pair
TargetDNA topoisomerase 2-alpha(Homo sapiens (Human))
Dr. Babasaheb Ambedkar Marathwada University
Curated by ChEMBL
Dr. Babasaheb Ambedkar Marathwada University
Curated by ChEMBL
Affinity DataIC50: 3.99E+4nMAssay Description:Inhibition of human topoisomerase-2 alpha in human A498 cells assessed as decrease in relaxation of supercoiled DNA at 10 uMMore data for this Ligand-Target Pair
TargetDNA topoisomerase 2-alpha(Homo sapiens (Human))
Dr. Babasaheb Ambedkar Marathwada University
Curated by ChEMBL
Dr. Babasaheb Ambedkar Marathwada University
Curated by ChEMBL
Affinity DataIC50: 4.84E+4nMAssay Description:Inhibition of human topoisomerase-2 alpha in human A498 cells assessed as decrease in relaxation of supercoiled DNA at 10 uMMore data for this Ligand-Target Pair