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Found 192 with Last Name = 'dodo' and Initial = 'k'
TargetAndrogen receptor(Homo sapiens (Human))
The University Of Tokyo

Curated by ChEMBL
LigandPNGBDBM50253371(CHEMBL522172 | N4-Isobutyl-6-(2-naphthalen-1-yl-et...)
Affinity DataKi:  1.50E+3nMAssay Description:Inhibition of ARMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEstrogen receptor(Homo sapiens (Human))
The University Of Tokyo

Curated by ChEMBL
LigandPNGBDBM50313149(6-(2-benzylpyridin-4-yl)-3-hydroxy-5-isobutyl-1-(n...)
Affinity DataKi:  4.20E+3nMAssay Description:Inhibition of ERMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEstrogen receptor(Homo sapiens (Human))
The University Of Tokyo

Curated by ChEMBL
LigandPNGBDBM50313148(CHEMBL1087884 | N2,N4,6-triisobutylpyrimidine-2,4-...)
Affinity DataKi:  2.90E+4nMAssay Description:Inhibition of ERMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVitamin D3 receptor(Homo sapiens (Human))
The University Of Tokyo

Curated by ChEMBL
LigandPNGBDBM50313152((3R,5S)-5-((R)-2-((1R,3aS,7aR,E)-4-((Z)-2-((3S,5R)...)
Affinity DataIC50:  220nMAssay Description:Antagonist activity at human recombinant VDR LBD expressed in HEK293 cells assessed as inhibition of 3 nM 1,25-(OH)2D3-induced transcriptional activa...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetM-phase inducer phosphatase 1(Homo sapiens (Human))
The University Of Tokyo

Curated by ChEMBL
LigandPNGBDBM50147586((S)-4-{2-[(3R,7S)-1-((2R,3R)-1,5-Dimethyl-hexyl)-4...)
Affinity DataIC50:  440nMAssay Description:Concentration required to inhibit human Cell division cycle 25A activityMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetM-phase inducer phosphatase 1(Homo sapiens (Human))
The University Of Tokyo

Curated by ChEMBL
LigandPNGBDBM50147585((R)-4-{2-[(3R,7R)-1-((2R,3R)-1,5-Dimethyl-hexyl)-4...)
Affinity DataIC50:  480nMAssay Description:Concentration required to inhibit human Cell division cycle 25A activityMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetM-phase inducer phosphatase 1(Homo sapiens (Human))
The University Of Tokyo

Curated by ChEMBL
LigandPNGBDBM50147582(4-{(R)-2-[(3aR,4S)-1-((1R,2R)-1,5-Dimethyl-hexyl)-...)
Affinity DataIC50:  860nMAssay Description:Concentration required to inhibit human Cell division cycle 25A activityMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetM-phase inducer phosphatase 1(Homo sapiens (Human))
The University Of Tokyo

Curated by ChEMBL
LigandPNGBDBM50147583((S)-4-Methylene-3-{2-[(R)-7a-(R)-methyl-1-((R)-5-m...)
Affinity DataIC50:  890nMAssay Description:Concentration required to inhibit human Cell division cycle 25A activity; Value ranges from 0.44 uM to 0.89 uMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetM-phase inducer phosphatase 1(Homo sapiens (Human))
The University Of Tokyo

Curated by ChEMBL
LigandPNGBDBM50147587((S)-4-{2-[(3R,7R)-1-((2R,3R)-1,5-Dimethyl-hexyl)-4...)
Affinity DataIC50:  890nMAssay Description:Concentration required to inhibit human Cell division cycle 25A activityMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetM-phase inducer phosphatase 2(Homo sapiens (Human))
The University Of Tokyo

Curated by ChEMBL
LigandPNGBDBM50147585((R)-4-{2-[(3R,7R)-1-((2R,3R)-1,5-Dimethyl-hexyl)-4...)
Affinity DataIC50:  1.44E+3nMAssay Description:Concentration required to inhibit human Cell division cycle 25B activityMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetM-phase inducer phosphatase 2(Homo sapiens (Human))
The University Of Tokyo

Curated by ChEMBL
LigandPNGBDBM50147587((S)-4-{2-[(3R,7R)-1-((2R,3R)-1,5-Dimethyl-hexyl)-4...)
Affinity DataIC50:  1.62E+3nMAssay Description:Concentration required to inhibit human Cell division cycle 25B activityMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetM-phase inducer phosphatase 2(Homo sapiens (Human))
The University Of Tokyo

Curated by ChEMBL
LigandPNGBDBM50147582(4-{(R)-2-[(3aR,4S)-1-((1R,2R)-1,5-Dimethyl-hexyl)-...)
Affinity DataIC50:  1.88E+3nMAssay Description:Concentration required to inhibit human Cell division cycle 25B activityMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetM-phase inducer phosphatase 2(Homo sapiens (Human))
The University Of Tokyo

Curated by ChEMBL
LigandPNGBDBM50147586((S)-4-{2-[(3R,7S)-1-((2R,3R)-1,5-Dimethyl-hexyl)-4...)
Affinity DataIC50:  1.90E+3nMAssay Description:Concentration required to inhibit human Cell division cycle 25B activityMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOxysterols receptor LXR-alpha(Homo sapiens (Human))
University of Tokyo

LigandPNGBDBM23843(5,16,25-trimethoxy-14-oxapentacyclo[20.2.2.2^{10,1...)
Affinity DataIC50:  2.00E+3nMT: 2°CAssay Description:Human embryonic kidney (HEK) 293 cells were cultured in D-MEM medium. Transfections were performed by the calcium phosphate coprecipitation method. T...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOxysterols receptor LXR-alpha(Homo sapiens (Human))
University of Tokyo

LigandPNGBDBM23844(16,25-dimethoxy-14-oxapentacyclo[20.2.2.2^{10,13}....)
Affinity DataIC50:  2.20E+3nMT: 2°CAssay Description:Human embryonic kidney (HEK) 293 cells were cultured in D-MEM medium. Transfections were performed by the calcium phosphate coprecipitation method. T...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone-lysine N-methyltransferase EHMT2(Homo sapiens (Human))
Riken Advanced Science Institute

Curated by ChEMBL
LigandPNGBDBM50315537(CHEMBL1089316 | chaetocin)
Affinity DataIC50:  2.40E+3nMAssay Description:Inhibition of protein lysine methyltransferase G9a (unknown origin) by ELISA assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOxysterols receptor LXR-alpha(Homo sapiens (Human))
University of Tokyo

LigandPNGBDBM23848(25-methoxy-14-oxapentacyclo[20.2.2.2^{10,13}.1^{15...)
Affinity DataIC50:  2.50E+3nMAssay Description:Human embryonic kidney (HEK) 293 cells were cultured in D-MEM medium. Transfections were performed by the calcium phosphate coprecipitation method. T...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOxysterols receptor LXR-alpha(Homo sapiens (Human))
University of Tokyo

LigandPNGBDBM23842(2-[2,6-bis(propan-2-yl)phenyl]-3-sulfanylidene-2,3...)
Affinity DataIC50:  3.10E+3nMT: 2°CAssay Description:Human embryonic kidney (HEK) 293 cells were cultured in D-MEM medium. Transfections were performed by the calcium phosphate coprecipitation method. T...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOxysterols receptor LXR-alpha(Homo sapiens (Human))
University of Tokyo

LigandPNGBDBM23853(14-oxapentacyclo[20.2.2.2^{10,13}.1^{15,19}.0^{2,7...)
Affinity DataIC50:  3.20E+3nMAssay Description:Human embryonic kidney (HEK) 293 cells were cultured in D-MEM medium. Transfections were performed by the calcium phosphate coprecipitation method. T...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone-lysine N-methyltransferase EHMT2(Homo sapiens (Human))
Riken Advanced Science Institute

Curated by ChEMBL
LigandPNGBDBM50425308(CHEMBL2311579)
Affinity DataIC50:  3.30E+3nMAssay Description:Inhibition of protein lysine methyltransferase G9a (unknown origin) by modified ELISA assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVitamin D3 receptor(Homo sapiens (Human))
The University Of Tokyo

Curated by ChEMBL
LigandPNGBDBM50313152((3R,5S)-5-((R)-2-((1R,3aS,7aR,E)-4-((Z)-2-((3S,5R)...)
Affinity DataIC50:  3.30E+3nMAssay Description:Antagonist activity at human recombinant VDR LBD expressed in HEK293 cells assessed as inhibition of 300 nM 1,25-(OH)2D3-induced transcriptional acti...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOxysterols receptor LXR-alpha(Homo sapiens (Human))
University of Tokyo

LigandPNGBDBM23845(5,16-dimethoxy-14-oxapentacyclo[20.2.2.2^{10,13}.1...)
Affinity DataIC50:  3.60E+3nMT: 2°CAssay Description:Human embryonic kidney (HEK) 293 cells were cultured in D-MEM medium. Transfections were performed by the calcium phosphate coprecipitation method. T...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOxysterols receptor LXR-alpha(Homo sapiens (Human))
University of Tokyo

LigandPNGBDBM23850(14-oxapentacyclo[20.2.2.2^{10,13}.1^{15,19}.0^{2,7...)
Affinity DataIC50:  4.40E+3nMAssay Description:Human embryonic kidney (HEK) 293 cells were cultured in D-MEM medium. Transfections were performed by the calcium phosphate coprecipitation method. T...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-glucosidase MAL32(Saccharomyces cerevisiae)
University of Tokyo

LigandPNGBDBM19992(2-[3-[3-[[2-chloro-3-(trifluoromethyl)phenyl]methy...)
Affinity DataIC50:  4.80E+3nMpH: 7.0 T: 2°CAssay Description:The alpha-glucosidase inhibitory activity of test compounds was determined in a 96-well plate format. The reaction mixture containing enzyme and chro...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-glucosidase MAL32(Saccharomyces cerevisiae)
University of Tokyo

LigandPNGBDBM23850(14-oxapentacyclo[20.2.2.2^{10,13}.1^{15,19}.0^{2,7...)
Affinity DataIC50:  4.90E+3nMpH: 7.0 T: 2°CAssay Description:The alpha-glucosidase inhibitory activity of test compounds was determined in a 96-well plate format. The reaction mixture containing enzyme and chro...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOxysterols receptor LXR-alpha(Homo sapiens (Human))
University of Tokyo

LigandPNGBDBM23839(14-oxapentacyclo[20.2.2.2^{10,13}.1^{15,19}.0^{2,7...)
Affinity DataIC50:  4.90E+3nMT: 2°CAssay Description:Human embryonic kidney (HEK) 293 cells were cultured in D-MEM medium. Transfections were performed by the calcium phosphate coprecipitation method. T...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-glucosidase MAL32(Saccharomyces cerevisiae)
University of Tokyo

LigandPNGBDBM23851(14-oxapentacyclo[20.2.2.2^{10,13}.1^{15,19}.0^{2,7...)
Affinity DataIC50:  5.10E+3nMpH: 7.0 T: 2°CAssay Description:The alpha-glucosidase inhibitory activity of test compounds was determined in a 96-well plate format. The reaction mixture containing enzyme and chro...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone-lysine N-methyltransferase EHMT2(Homo sapiens (Human))
Riken Advanced Science Institute

Curated by ChEMBL
LigandPNGBDBM50425305(CHEMBL2315521)
Affinity DataIC50:  5.20E+3nMAssay Description:Inhibition of protein lysine methyltransferase G9a (unknown origin) by modified ELISA assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone-lysine N-methyltransferase EHMT2(Homo sapiens (Human))
Riken Advanced Science Institute

Curated by ChEMBL
LigandPNGBDBM50425304(CHEMBL2315522)
Affinity DataIC50:  5.30E+3nMAssay Description:Inhibition of protein lysine methyltransferase G9a (unknown origin) by modified ELISA assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetM-phase inducer phosphatase 1(Homo sapiens (Human))
The University Of Tokyo

Curated by ChEMBL
LigandPNGBDBM50087141((E)-2-((1R,7aR)-7a-methyl-1-((R)-6-methylheptan-2-...)
Affinity DataIC50:  5.50E+3nMAssay Description:Concentration required to inhibit human Cell division cycle 25A activityMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOxysterols receptor LXR-alpha(Homo sapiens (Human))
University of Tokyo

LigandPNGBDBM23852(14-oxapentacyclo[20.2.2.2^{10,13}.1^{15,19}.0^{2,7...)
Affinity DataIC50:  5.70E+3nMAssay Description:Human embryonic kidney (HEK) 293 cells were cultured in D-MEM medium. Transfections were performed by the calcium phosphate coprecipitation method. T...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone-lysine N-methyltransferase EHMT2(Homo sapiens (Human))
Riken Advanced Science Institute

Curated by ChEMBL
LigandPNGBDBM50396029(CHEMBL1222849)
Affinity DataIC50:  6.40E+3nMAssay Description:Inhibition of protein lysine methyltransferase G9a (unknown origin) by modified ELISA assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOxysterols receptor LXR-beta(Homo sapiens (Human))
University of Tokyo

LigandPNGBDBM23839(14-oxapentacyclo[20.2.2.2^{10,13}.1^{15,19}.0^{2,7...)
Affinity DataIC50:  6.60E+3nMAssay Description:Human embryonic kidney (HEK) 293 cells were cultured in D-MEM medium. Transfections were performed by the calcium phosphate coprecipitation method. T...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOxysterols receptor LXR-alpha(Homo sapiens (Human))
University of Tokyo

LigandPNGBDBM23849(14-oxapentacyclo[20.2.2.2^{10,13}.1^{15,19}.0^{2,7...)
Affinity DataIC50:  6.60E+3nMAssay Description:Human embryonic kidney (HEK) 293 cells were cultured in D-MEM medium. Transfections were performed by the calcium phosphate coprecipitation method. T...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOxysterols receptor LXR-alpha(Homo sapiens (Human))
University of Tokyo

LigandPNGBDBM23854(14-oxapentacyclo[20.2.2.2^{10,13}.1^{15,19}.0^{2,7...)
Affinity DataIC50:  7.10E+3nMAssay Description:Human embryonic kidney (HEK) 293 cells were cultured in D-MEM medium. Transfections were performed by the calcium phosphate coprecipitation method. T...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone-lysine N-methyltransferase EHMT2(Homo sapiens (Human))
Riken Advanced Science Institute

Curated by ChEMBL
LigandPNGBDBM50315537(CHEMBL1089316 | chaetocin)
Affinity DataIC50:  7.20E+3nMAssay Description:Inhibition of protein lysine methyltransferase G9a (unknown origin) by modified ELISA assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone-lysine N-methyltransferase EHMT2(Homo sapiens (Human))
Riken Advanced Science Institute

Curated by ChEMBL
LigandPNGBDBM50425311(CHEMBL2315526)
Affinity DataIC50:  7.20E+3nMAssay Description:Inhibition of protein lysine methyltransferase G9a (unknown origin) by modified ELISA assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOxysterols receptor LXR-beta(Homo sapiens (Human))
University of Tokyo

LigandPNGBDBM23853(14-oxapentacyclo[20.2.2.2^{10,13}.1^{15,19}.0^{2,7...)
Affinity DataIC50:  7.30E+3nMAssay Description:Human embryonic kidney (HEK) 293 cells were cultured in D-MEM medium. Transfections were performed by the calcium phosphate coprecipitation method. T...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOxysterols receptor LXR-alpha(Homo sapiens (Human))
University of Tokyo

LigandPNGBDBM23847(16-methoxy-14-oxapentacyclo[20.2.2.2^{10,13}.1^{15...)
Affinity DataIC50:  7.60E+3nMAssay Description:Human embryonic kidney (HEK) 293 cells were cultured in D-MEM medium. Transfections were performed by the calcium phosphate coprecipitation method. T...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOxysterols receptor LXR-beta(Homo sapiens (Human))
University of Tokyo

LigandPNGBDBM23850(14-oxapentacyclo[20.2.2.2^{10,13}.1^{15,19}.0^{2,7...)
Affinity DataIC50:  7.60E+3nMAssay Description:Human embryonic kidney (HEK) 293 cells were cultured in D-MEM medium. Transfections were performed by the calcium phosphate coprecipitation method. T...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetM-phase inducer phosphatase 1(Homo sapiens (Human))
The University Of Tokyo

Curated by ChEMBL
LigandPNGBDBM50087141((E)-2-((1R,7aR)-7a-methyl-1-((R)-6-methylheptan-2-...)
Affinity DataIC50:  7.70E+3nMAssay Description:Concentration required for the inhibitory activity against human Cell division cycle 25AMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetM-phase inducer phosphatase 2(Homo sapiens (Human))
The University Of Tokyo

Curated by ChEMBL
LigandPNGBDBM50087141((E)-2-((1R,7aR)-7a-methyl-1-((R)-6-methylheptan-2-...)
Affinity DataIC50:  8.00E+3nMAssay Description:Concentration required to inhibit human Cell division cycle 25B activityMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-glucosidase MAL32(Saccharomyces cerevisiae)
University of Tokyo

LigandPNGBDBM23842(2-[2,6-bis(propan-2-yl)phenyl]-3-sulfanylidene-2,3...)
Affinity DataIC50:  8.00E+3nMpH: 7.0 T: 2°CAssay Description:The alpha-glucosidase inhibitory activity of test compounds was determined in a 96-well plate format. The reaction mixture containing enzyme and chro...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOxysterols receptor LXR-alpha(Homo sapiens (Human))
University of Tokyo

LigandPNGBDBM23851(14-oxapentacyclo[20.2.2.2^{10,13}.1^{15,19}.0^{2,7...)
Affinity DataIC50:  8.40E+3nMAssay Description:Human embryonic kidney (HEK) 293 cells were cultured in D-MEM medium. Transfections were performed by the calcium phosphate coprecipitation method. T...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-glucosidase MAL32(Saccharomyces cerevisiae)
University of Tokyo

LigandPNGBDBM23849(14-oxapentacyclo[20.2.2.2^{10,13}.1^{15,19}.0^{2,7...)
Affinity DataIC50:  8.60E+3nMpH: 7.0 T: 2°CAssay Description:The alpha-glucosidase inhibitory activity of test compounds was determined in a 96-well plate format. The reaction mixture containing enzyme and chro...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetM-phase inducer phosphatase 1(Homo sapiens (Human))
The University Of Tokyo

Curated by ChEMBL
LigandPNGBDBM50087143(4-[(1R,7aR)-1-((R)-1,5-Dimethyl-hexyl)-7a-methyl-o...)
Affinity DataIC50:  9.00E+3nMAssay Description:Concentration required for the inhibitory activity against human Cell division cycle 25AMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetM-phase inducer phosphatase 1(Homo sapiens (Human))
The University Of Tokyo

Curated by ChEMBL
LigandPNGBDBM50341997(CHEMBL1765353 | Dysidiolide)
Affinity DataIC50:  9.40E+3nMAssay Description:Concentration required to inhibit human Cell division cycle 25A activityMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOxysterols receptor LXR-alpha(Homo sapiens (Human))
University of Tokyo

LigandPNGBDBM23840(2-[2-(2-phenylethyl)phenyl]-2,3-dihydro-1H-isoindo...)
Affinity DataIC50:  9.80E+3nMT: 2°CAssay Description:Human embryonic kidney (HEK) 293 cells were cultured in D-MEM medium. Transfections were performed by the calcium phosphate coprecipitation method. T...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-glucosidase MAL32(Saccharomyces cerevisiae)
University of Tokyo

LigandPNGBDBM23839(14-oxapentacyclo[20.2.2.2^{10,13}.1^{15,19}.0^{2,7...)
Affinity DataIC50:  9.90E+3nMpH: 7.0 T: 2°CAssay Description:The alpha-glucosidase inhibitory activity of test compounds was determined in a 96-well plate format. The reaction mixture containing enzyme and chro...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOxysterols receptor LXR-beta(Homo sapiens (Human))
University of Tokyo

LigandPNGBDBM23851(14-oxapentacyclo[20.2.2.2^{10,13}.1^{15,19}.0^{2,7...)
Affinity DataIC50:  1.00E+4nMAssay Description:Human embryonic kidney (HEK) 293 cells were cultured in D-MEM medium. Transfections were performed by the calcium phosphate coprecipitation method. T...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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