Affinity DataIC50: 220nMAssay Description:Antagonist activity at human recombinant VDR LBD expressed in HEK293 cells assessed as inhibition of 3 nM 1,25-(OH)2D3-induced transcriptional activa...More data for this Ligand-Target Pair
Affinity DataIC50: 440nMAssay Description:Concentration required to inhibit human Cell division cycle 25A activityMore data for this Ligand-Target Pair
Affinity DataIC50: 480nMAssay Description:Concentration required to inhibit human Cell division cycle 25A activityMore data for this Ligand-Target Pair
Affinity DataIC50: 860nMAssay Description:Concentration required to inhibit human Cell division cycle 25A activityMore data for this Ligand-Target Pair
Affinity DataIC50: 890nMAssay Description:Concentration required to inhibit human Cell division cycle 25A activity; Value ranges from 0.44 uM to 0.89 uMMore data for this Ligand-Target Pair
Affinity DataIC50: 890nMAssay Description:Concentration required to inhibit human Cell division cycle 25A activityMore data for this Ligand-Target Pair
Affinity DataIC50: 1.44E+3nMAssay Description:Concentration required to inhibit human Cell division cycle 25B activityMore data for this Ligand-Target Pair
Affinity DataIC50: 1.62E+3nMAssay Description:Concentration required to inhibit human Cell division cycle 25B activityMore data for this Ligand-Target Pair
Affinity DataIC50: 1.88E+3nMAssay Description:Concentration required to inhibit human Cell division cycle 25B activityMore data for this Ligand-Target Pair
Affinity DataIC50: 1.90E+3nMAssay Description:Concentration required to inhibit human Cell division cycle 25B activityMore data for this Ligand-Target Pair
Affinity DataIC50: 2.00E+3nMT: 2°CAssay Description:Human embryonic kidney (HEK) 293 cells were cultured in D-MEM medium. Transfections were performed by the calcium phosphate coprecipitation method. T...More data for this Ligand-Target Pair
Affinity DataIC50: 2.20E+3nMT: 2°CAssay Description:Human embryonic kidney (HEK) 293 cells were cultured in D-MEM medium. Transfections were performed by the calcium phosphate coprecipitation method. T...More data for this Ligand-Target Pair
TargetHistone-lysine N-methyltransferase EHMT2(Homo sapiens (Human))
Riken Advanced Science Institute
Curated by ChEMBL
Riken Advanced Science Institute
Curated by ChEMBL
Affinity DataIC50: 2.40E+3nMAssay Description:Inhibition of protein lysine methyltransferase G9a (unknown origin) by ELISA assayMore data for this Ligand-Target Pair
Affinity DataIC50: 2.50E+3nMAssay Description:Human embryonic kidney (HEK) 293 cells were cultured in D-MEM medium. Transfections were performed by the calcium phosphate coprecipitation method. T...More data for this Ligand-Target Pair
Affinity DataIC50: 3.10E+3nMT: 2°CAssay Description:Human embryonic kidney (HEK) 293 cells were cultured in D-MEM medium. Transfections were performed by the calcium phosphate coprecipitation method. T...More data for this Ligand-Target Pair
Affinity DataIC50: 3.20E+3nMAssay Description:Human embryonic kidney (HEK) 293 cells were cultured in D-MEM medium. Transfections were performed by the calcium phosphate coprecipitation method. T...More data for this Ligand-Target Pair
TargetHistone-lysine N-methyltransferase EHMT2(Homo sapiens (Human))
Riken Advanced Science Institute
Curated by ChEMBL
Riken Advanced Science Institute
Curated by ChEMBL
Affinity DataIC50: 3.30E+3nMAssay Description:Inhibition of protein lysine methyltransferase G9a (unknown origin) by modified ELISA assayMore data for this Ligand-Target Pair
Affinity DataIC50: 3.30E+3nMAssay Description:Antagonist activity at human recombinant VDR LBD expressed in HEK293 cells assessed as inhibition of 300 nM 1,25-(OH)2D3-induced transcriptional acti...More data for this Ligand-Target Pair
Affinity DataIC50: 3.60E+3nMT: 2°CAssay Description:Human embryonic kidney (HEK) 293 cells were cultured in D-MEM medium. Transfections were performed by the calcium phosphate coprecipitation method. T...More data for this Ligand-Target Pair
Affinity DataIC50: 4.40E+3nMAssay Description:Human embryonic kidney (HEK) 293 cells were cultured in D-MEM medium. Transfections were performed by the calcium phosphate coprecipitation method. T...More data for this Ligand-Target Pair
Affinity DataIC50: 4.80E+3nMpH: 7.0 T: 2°CAssay Description:The alpha-glucosidase inhibitory activity of test compounds was determined in a 96-well plate format. The reaction mixture containing enzyme and chro...More data for this Ligand-Target Pair
Affinity DataIC50: 4.90E+3nMpH: 7.0 T: 2°CAssay Description:The alpha-glucosidase inhibitory activity of test compounds was determined in a 96-well plate format. The reaction mixture containing enzyme and chro...More data for this Ligand-Target Pair
Affinity DataIC50: 4.90E+3nMT: 2°CAssay Description:Human embryonic kidney (HEK) 293 cells were cultured in D-MEM medium. Transfections were performed by the calcium phosphate coprecipitation method. T...More data for this Ligand-Target Pair
Affinity DataIC50: 5.10E+3nMpH: 7.0 T: 2°CAssay Description:The alpha-glucosidase inhibitory activity of test compounds was determined in a 96-well plate format. The reaction mixture containing enzyme and chro...More data for this Ligand-Target Pair
TargetHistone-lysine N-methyltransferase EHMT2(Homo sapiens (Human))
Riken Advanced Science Institute
Curated by ChEMBL
Riken Advanced Science Institute
Curated by ChEMBL
Affinity DataIC50: 5.20E+3nMAssay Description:Inhibition of protein lysine methyltransferase G9a (unknown origin) by modified ELISA assayMore data for this Ligand-Target Pair
TargetHistone-lysine N-methyltransferase EHMT2(Homo sapiens (Human))
Riken Advanced Science Institute
Curated by ChEMBL
Riken Advanced Science Institute
Curated by ChEMBL
Affinity DataIC50: 5.30E+3nMAssay Description:Inhibition of protein lysine methyltransferase G9a (unknown origin) by modified ELISA assayMore data for this Ligand-Target Pair
Affinity DataIC50: 5.50E+3nMAssay Description:Concentration required to inhibit human Cell division cycle 25A activityMore data for this Ligand-Target Pair
Affinity DataIC50: 5.70E+3nMAssay Description:Human embryonic kidney (HEK) 293 cells were cultured in D-MEM medium. Transfections were performed by the calcium phosphate coprecipitation method. T...More data for this Ligand-Target Pair
TargetHistone-lysine N-methyltransferase EHMT2(Homo sapiens (Human))
Riken Advanced Science Institute
Curated by ChEMBL
Riken Advanced Science Institute
Curated by ChEMBL
Affinity DataIC50: 6.40E+3nMAssay Description:Inhibition of protein lysine methyltransferase G9a (unknown origin) by modified ELISA assayMore data for this Ligand-Target Pair
Affinity DataIC50: 6.60E+3nMAssay Description:Human embryonic kidney (HEK) 293 cells were cultured in D-MEM medium. Transfections were performed by the calcium phosphate coprecipitation method. T...More data for this Ligand-Target Pair
Affinity DataIC50: 6.60E+3nMAssay Description:Human embryonic kidney (HEK) 293 cells were cultured in D-MEM medium. Transfections were performed by the calcium phosphate coprecipitation method. T...More data for this Ligand-Target Pair
Affinity DataIC50: 7.10E+3nMAssay Description:Human embryonic kidney (HEK) 293 cells were cultured in D-MEM medium. Transfections were performed by the calcium phosphate coprecipitation method. T...More data for this Ligand-Target Pair
TargetHistone-lysine N-methyltransferase EHMT2(Homo sapiens (Human))
Riken Advanced Science Institute
Curated by ChEMBL
Riken Advanced Science Institute
Curated by ChEMBL
Affinity DataIC50: 7.20E+3nMAssay Description:Inhibition of protein lysine methyltransferase G9a (unknown origin) by modified ELISA assayMore data for this Ligand-Target Pair
TargetHistone-lysine N-methyltransferase EHMT2(Homo sapiens (Human))
Riken Advanced Science Institute
Curated by ChEMBL
Riken Advanced Science Institute
Curated by ChEMBL
Affinity DataIC50: 7.20E+3nMAssay Description:Inhibition of protein lysine methyltransferase G9a (unknown origin) by modified ELISA assayMore data for this Ligand-Target Pair
Affinity DataIC50: 7.30E+3nMAssay Description:Human embryonic kidney (HEK) 293 cells were cultured in D-MEM medium. Transfections were performed by the calcium phosphate coprecipitation method. T...More data for this Ligand-Target Pair
Affinity DataIC50: 7.60E+3nMAssay Description:Human embryonic kidney (HEK) 293 cells were cultured in D-MEM medium. Transfections were performed by the calcium phosphate coprecipitation method. T...More data for this Ligand-Target Pair
Affinity DataIC50: 7.60E+3nMAssay Description:Human embryonic kidney (HEK) 293 cells were cultured in D-MEM medium. Transfections were performed by the calcium phosphate coprecipitation method. T...More data for this Ligand-Target Pair
Affinity DataIC50: 7.70E+3nMAssay Description:Concentration required for the inhibitory activity against human Cell division cycle 25AMore data for this Ligand-Target Pair
Affinity DataIC50: 8.00E+3nMAssay Description:Concentration required to inhibit human Cell division cycle 25B activityMore data for this Ligand-Target Pair
Affinity DataIC50: 8.00E+3nMpH: 7.0 T: 2°CAssay Description:The alpha-glucosidase inhibitory activity of test compounds was determined in a 96-well plate format. The reaction mixture containing enzyme and chro...More data for this Ligand-Target Pair
Affinity DataIC50: 8.40E+3nMAssay Description:Human embryonic kidney (HEK) 293 cells were cultured in D-MEM medium. Transfections were performed by the calcium phosphate coprecipitation method. T...More data for this Ligand-Target Pair
Affinity DataIC50: 8.60E+3nMpH: 7.0 T: 2°CAssay Description:The alpha-glucosidase inhibitory activity of test compounds was determined in a 96-well plate format. The reaction mixture containing enzyme and chro...More data for this Ligand-Target Pair
Affinity DataIC50: 9.00E+3nMAssay Description:Concentration required for the inhibitory activity against human Cell division cycle 25AMore data for this Ligand-Target Pair
Affinity DataIC50: 9.40E+3nMAssay Description:Concentration required to inhibit human Cell division cycle 25A activityMore data for this Ligand-Target Pair
Affinity DataIC50: 9.80E+3nMT: 2°CAssay Description:Human embryonic kidney (HEK) 293 cells were cultured in D-MEM medium. Transfections were performed by the calcium phosphate coprecipitation method. T...More data for this Ligand-Target Pair
Affinity DataIC50: 9.90E+3nMpH: 7.0 T: 2°CAssay Description:The alpha-glucosidase inhibitory activity of test compounds was determined in a 96-well plate format. The reaction mixture containing enzyme and chro...More data for this Ligand-Target Pair
Affinity DataIC50: 1.00E+4nMAssay Description:Human embryonic kidney (HEK) 293 cells were cultured in D-MEM medium. Transfections were performed by the calcium phosphate coprecipitation method. T...More data for this Ligand-Target Pair