Affinity DataIC50: 0.200nMAssay Description:In vitro kinase enzyme assay using Jak3, Jak2, Jak1, and Tyk2.More data for this Ligand-Target Pair
Affinity DataIC50: 0.300nMAssay Description:In vitro kinase enzyme assay using Jak3, Jak2, Jak1, and Tyk2.More data for this Ligand-Target Pair
Affinity DataIC50: 0.600nMAssay Description:In vitro kinase enzyme assay using Jak3, Jak2, Jak1, and Tyk2.More data for this Ligand-Target Pair
Affinity DataIC50: 5.30nMAssay Description:Compound was evaluated in vitro for beta-adrenergic activity against beta-1 adrenergic receptor by the inhibition of insulin stimulated [14C]- glucos...More data for this Ligand-Target Pair
Affinity DataIC50: 30nMAssay Description:Compound was evaluated for its binding affinity towards Beta-2 adrenergic receptor in rat soleus membrane by displacing (-)-isoproterenol (50 microM)More data for this Ligand-Target Pair
Affinity DataIC50: 45nMAssay Description:In vitro kinase enzyme assay using Jak3, Jak2, Jak1, and Tyk2.More data for this Ligand-Target Pair
Affinity DataIC50: 59nMAssay Description:Compound was evaluated for its binding affinity towards Beta-1 adrenergic receptor in rat heart membrane by displacing [125I]- iodocyanopindololMore data for this Ligand-Target Pair
Affinity DataIC50: 136nMAssay Description:In vitro kinase enzyme assay using Jak3, Jak2, Jak1, and Tyk2.More data for this Ligand-Target Pair
Affinity DataIC50: 175nMAssay Description:In vitro kinase enzyme assay using Jak3, Jak2, Jak1, and Tyk2.More data for this Ligand-Target Pair
Affinity DataIC50: 190nMAssay Description:Compound was evaluated in vitro for beta-adrenergic activity against beta-1 adrenergic receptor by the inhibition of insulin stimulated [14C]- glucos...More data for this Ligand-Target Pair
Affinity DataIC50: 270nMAssay Description:In vitro kinase enzyme assay using Jak3, Jak2, Jak1, and Tyk2.More data for this Ligand-Target Pair
Affinity DataIC50: 330nMAssay Description:In vitro kinase enzyme assay using Jak3, Jak2, Jak1, and Tyk2.More data for this Ligand-Target Pair
Affinity DataIC50: 500nMAssay Description:Compound was evaluated in vitro for beta-adrenergic activity against beta-1 adrenergic receptor by the inhibition of insulin stimulated [14C]- glucos...More data for this Ligand-Target Pair
Affinity DataIC50: 500nMAssay Description:In vitro kinase enzyme assay using Jak3, Jak2, Jak1, and Tyk2.More data for this Ligand-Target Pair
Affinity DataIC50: 600nMAssay Description:Compound was evaluated for its binding affinity towards beta-1 adrenergic receptor in rat heart membrane by displacing [125I]- iodocyanopindololMore data for this Ligand-Target Pair
Affinity DataIC50: 1.00E+3nMAssay Description:Compound was evaluated for its binding affinity towards beta-2 adrenergic receptor in rat soleus membrane by displacing(-)-isoproterenol (50 microM)More data for this Ligand-Target Pair
Affinity DataIC50: 1.30E+3nMAssay Description:Compound was evaluated for its binding affinity towards Beta-2 adrenergic receptor in rat soleus membrane by displacing (-)-isoproterenol (50 microM)More data for this Ligand-Target Pair
Affinity DataIC50: 2.70E+3nMAssay Description:In vitro kinase enzyme assay using Jak3, Jak2, Jak1, and Tyk2.More data for this Ligand-Target Pair
Affinity DataIC50: 3.30E+3nMAssay Description:Compound was evaluated for its binding affinity towards Beta-1 adrenergic receptor in rat heart membrane by displacing [125I]- iodocyanopindololMore data for this Ligand-Target Pair
Affinity DataIC50: >1.00E+4nMAssay Description:In vitro kinase enzyme assay using Jak3, Jak2, Jak1, and Tyk2.More data for this Ligand-Target Pair
Affinity DataIC50: >1.00E+4nMAssay Description:In vitro kinase enzyme assay using Jak3, Jak2, Jak1, and Tyk2.More data for this Ligand-Target Pair
Affinity DataIC50: >1.00E+4nMAssay Description:In vitro kinase enzyme assay using Jak3, Jak2, Jak1, and Tyk2.More data for this Ligand-Target Pair
Affinity DataIC50: >1.00E+4nMAssay Description:In vitro kinase enzyme assay using Jak3, Jak2, Jak1, and Tyk2.More data for this Ligand-Target Pair
Affinity DataIC50: >1.00E+4nMAssay Description:In vitro kinase enzyme assay using Jak3, Jak2, Jak1, and Tyk2.More data for this Ligand-Target Pair
Affinity DataIC50: >1.00E+4nMAssay Description:In vitro kinase enzyme assay using Jak3, Jak2, Jak1, and Tyk2.More data for this Ligand-Target Pair
Affinity DataIC50: >1.00E+4nMAssay Description:In vitro kinase enzyme assay using Jak3, Jak2, Jak1, and Tyk2.More data for this Ligand-Target Pair
Affinity DataIC50: >1.00E+4nMAssay Description:In vitro kinase enzyme assay using Jak3, Jak2, Jak1, and Tyk2.More data for this Ligand-Target Pair
Affinity DataIC50: >1.00E+4nMAssay Description:In vitro kinase enzyme assay using Jak3, Jak2, Jak1, and Tyk2.More data for this Ligand-Target Pair
Affinity DataIC50: >1.00E+4nMAssay Description:In vitro kinase enzyme assay using Jak3, Jak2, Jak1, and Tyk2.More data for this Ligand-Target Pair
Affinity DataIC50: >1.00E+4nMAssay Description:In vitro kinase enzyme assay using Jak3, Jak2, Jak1, and Tyk2.More data for this Ligand-Target Pair
Affinity DataIC50: >1.00E+4nMAssay Description:In vitro kinase enzyme assay using Jak3, Jak2, Jak1, and Tyk2.More data for this Ligand-Target Pair
Affinity DataIC50: >1.00E+4nMAssay Description:In vitro kinase enzyme assay using Jak3, Jak2, Jak1, and Tyk2.More data for this Ligand-Target Pair
Affinity DataIC50: >1.00E+4nMAssay Description:In vitro kinase enzyme assay using Jak3, Jak2, Jak1, and Tyk2.More data for this Ligand-Target Pair
Affinity DataIC50: >1.00E+4nMAssay Description:In vitro kinase enzyme assay using Jak3, Jak2, Jak1, and Tyk2.More data for this Ligand-Target Pair
Affinity DataIC50: >1.00E+4nMAssay Description:In vitro kinase enzyme assay using Jak3, Jak2, Jak1, and Tyk2.More data for this Ligand-Target Pair
Affinity DataIC50: >1.00E+4nMAssay Description:In vitro kinase enzyme assay using Jak3, Jak2, Jak1, and Tyk2.More data for this Ligand-Target Pair
Affinity DataIC50: >1.00E+4nMAssay Description:In vitro kinase enzyme assay using Jak3, Jak2, Jak1, and Tyk2.More data for this Ligand-Target Pair
Affinity DataIC50: >1.00E+4nMAssay Description:In vitro kinase enzyme assay using Jak3, Jak2, Jak1, and Tyk2.More data for this Ligand-Target Pair
Affinity DataIC50: >1.00E+4nMAssay Description:In vitro kinase enzyme assay using Jak3, Jak2, Jak1, and Tyk2.More data for this Ligand-Target Pair
Affinity DataIC50: >1.00E+4nMAssay Description:In vitro kinase enzyme assay using Jak3, Jak2, Jak1, and Tyk2.More data for this Ligand-Target Pair
Affinity DataIC50: >1.00E+4nMAssay Description:In vitro kinase enzyme assay using Jak3, Jak2, Jak1, and Tyk2.More data for this Ligand-Target Pair
Affinity DataIC50: >1.00E+4nMAssay Description:In vitro kinase enzyme assay using Jak3, Jak2, Jak1, and Tyk2.More data for this Ligand-Target Pair
Affinity DataIC50: >1.00E+4nMAssay Description:In vitro kinase enzyme assay using Jak3, Jak2, Jak1, and Tyk2.More data for this Ligand-Target Pair
Affinity DataIC50: >1.00E+4nMAssay Description:In vitro kinase enzyme assay using Jak3, Jak2, Jak1, and Tyk2.More data for this Ligand-Target Pair
Affinity DataIC50: >1.00E+4nMAssay Description:In vitro kinase enzyme assay using Jak3, Jak2, Jak1, and Tyk2.More data for this Ligand-Target Pair
Affinity DataIC50: >1.00E+4nMAssay Description:In vitro kinase enzyme assay using Jak3, Jak2, Jak1, and Tyk2.More data for this Ligand-Target Pair
Affinity DataIC50: >1.00E+4nMAssay Description:In vitro kinase enzyme assay using Jak3, Jak2, Jak1, and Tyk2.More data for this Ligand-Target Pair
Affinity DataIC50: >1.00E+4nMAssay Description:In vitro kinase enzyme assay using Jak3, Jak2, Jak1, and Tyk2.More data for this Ligand-Target Pair
Affinity DataIC50: >1.00E+4nMAssay Description:In vitro kinase enzyme assay using Jak3, Jak2, Jak1, and Tyk2.More data for this Ligand-Target Pair
Affinity DataIC50: >1.00E+4nMAssay Description:In vitro kinase enzyme assay using Jak3, Jak2, Jak1, and Tyk2.More data for this Ligand-Target Pair