Affinity DataKi: 0.0230nMAssay Description:Inhibition of specific binding of [3H]-BK (1 nM) to rat Bradykinin receptor B2 by 50% in NG108-15 cell membranesMore data for this Ligand-Target Pair
Affinity DataKi: 0.310nMAssay Description:Inhibition of specific binding of [3H]-BK (1 nM) to rat Bradykinin receptor B2 by 50% in NG108-15 cell membranesMore data for this Ligand-Target Pair
Affinity DataKi: 0.5nMAssay Description:Inhibition of specific binding of [3H]-BK (1 nM) to rat Bradykinin receptor B2 by 50% in NG108-15 cell membranesMore data for this Ligand-Target Pair
Affinity DataKi: 0.5nMAssay Description:Inhibition of binding of [3H]-BK to rat bradykinin B2 receptor expressed in NG108-15 neuroblastoma-glioma hybrid cell membranesMore data for this Ligand-Target Pair
Affinity DataKi: 0.600nMAssay Description:Inhibition of binding of [3H]-BK to rat bradykinin B2 receptor expressed in NG108-15 neuroblastoma-glioma hybrid cell membranesMore data for this Ligand-Target Pair
Affinity DataKi: 0.600nMAssay Description:Inhibition of specific binding of [3H]-BK (1 nM) to rat Bradykinin receptor B2 by 50% in NG108-15 cell membranesMore data for this Ligand-Target Pair
TargetB2 bradykinin receptor(Homo sapiens (Human))
Novartis Institute For Medical Sciences
Curated by ChEMBL
Novartis Institute For Medical Sciences
Curated by ChEMBL
Affinity DataKi: 0.790nMAssay Description:Displacement of [3H]BK (1 nM) from human Bradykinin receptor B2 expressed in Cos-7 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 1nMAssay Description:Binding affinity for Bradykinin receptor B1 expressed in HEK293 cellsMore data for this Ligand-Target Pair
TargetB2 bradykinin receptor(Homo sapiens (Human))
Novartis Institute For Medical Sciences
Curated by ChEMBL
Novartis Institute For Medical Sciences
Curated by ChEMBL
Affinity DataKi: 1.47nMAssay Description:Displacement of [3H]BK (1 nM) from human Bradykinin receptor B2 expressed in Cos-7 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 1.80nMAssay Description:Inhibition of binding of [3H]-BK to rat bradykinin B2 receptor expressed in NG108-15 neuroblastoma-glioma hybrid cell membranesMore data for this Ligand-Target Pair
TargetB2 bradykinin receptor(Homo sapiens (Human))
Novartis Institute For Medical Sciences
Curated by ChEMBL
Novartis Institute For Medical Sciences
Curated by ChEMBL
Affinity DataKi: 2.79nMAssay Description:Displacement of [3H]BK (1 nM) from human Bradykinin receptor B2 expressed in Cos-7 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 4nMAssay Description:Inhibition of binding of [3H]-BK to rat bradykinin B2 receptor expressed in NG108-15 neuroblastoma-glioma hybrid cell membranesMore data for this Ligand-Target Pair
TargetB2 bradykinin receptor(Homo sapiens (Human))
Novartis Institute For Medical Sciences
Curated by ChEMBL
Novartis Institute For Medical Sciences
Curated by ChEMBL
Affinity DataKi: 4.67nMAssay Description:Displacement of [3H]BK (1 nM) from human Bradykinin receptor B2 expressed in Cos-7 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 5.46nMAssay Description:Inhibition of specific binding of [3H]-BK (1 nM) to rat Bradykinin receptor B2 by 50% in NG108-15 cell membranesMore data for this Ligand-Target Pair
Affinity DataKi: 7.30nMAssay Description:Inhibition of specific binding of [3H]-BK (1 nM) to rat Bradykinin receptor B2 by 50% in NG108-15 cell membranesMore data for this Ligand-Target Pair
Affinity DataKi: 10nMAssay Description:Binding affinity for Bradykinin receptor B1 expressed in HEK293 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 10nMAssay Description:Binding affinity for Bradykinin receptor B1 expressed in HEK293 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 10nMAssay Description:Binding affinity for Bradykinin receptor B1 expressed in HEK293 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 10nMAssay Description:Binding affinity for Bradykinin receptor B1 expressed in HEK293 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 10.7nMAssay Description:Inhibition of specific binding of [3H]-BK (1 nM) to rat Bradykinin receptor B2 by 50% in NG108-15 cell membranesMore data for this Ligand-Target Pair
Affinity DataKi: 14.5nMAssay Description:Inhibition of specific binding of [3H]-BK (1 nM) to rat Bradykinin receptor B2 by 50% in NG108-15 cell membranesMore data for this Ligand-Target Pair
TargetB2 bradykinin receptor(Homo sapiens (Human))
Novartis Institute For Medical Sciences
Curated by ChEMBL
Novartis Institute For Medical Sciences
Curated by ChEMBL
Affinity DataKi: 34.1nMAssay Description:Displacement of [3H]BK (1 nM) from human Bradykinin receptor B2 expressed in Cos-7 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 38nMAssay Description:Inhibition of binding of [3H]-BK to rat bradykinin B2 receptor expressed in NG108-15 neuroblastoma-glioma hybrid cell membranesMore data for this Ligand-Target Pair
Affinity DataKi: 64.5nMAssay Description:Inhibition of specific binding of [3H]-BK (1 nM) to rat Bradykinin receptor B2 by 50% in NG108-15 cell membranesMore data for this Ligand-Target Pair
TargetB2 bradykinin receptor(Homo sapiens (Human))
Novartis Institute For Medical Sciences
Curated by ChEMBL
Novartis Institute For Medical Sciences
Curated by ChEMBL
Affinity DataKi: 95nMAssay Description:Displacement of [3H]BK (1 nM) from human Bradykinin receptor B2 expressed in Cos-7 cellsMore data for this Ligand-Target Pair
TargetB2 bradykinin receptor(Homo sapiens (Human))
Novartis Institute For Medical Sciences
Curated by ChEMBL
Novartis Institute For Medical Sciences
Curated by ChEMBL
Affinity DataKi: 119nMAssay Description:Displacement of [3H]BK (1 nM) from human Bradykinin receptor B2 expressed in Cos-7 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 130nMAssay Description:Binding affinity for Bradykinin receptor B1 expressed in HEK293 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 140nMAssay Description:Binding affinity for Bradykinin receptor B1 expressed in HEK293 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 148nMAssay Description:Inhibition of binding of [3H]-BK to rat bradykinin B2 receptor expressed in NG108-15 neuroblastoma-glioma hybrid cell membranesMore data for this Ligand-Target Pair
Affinity DataKi: 176nMAssay Description:Inhibition of specific binding of [3H]-BK (1 nM) to rat Bradykinin receptor B2 by 50% in NG108-15 cell membranesMore data for this Ligand-Target Pair
Affinity DataKi: 230nMAssay Description:Binding affinity for Bradykinin receptor B1 expressed in HEK293 cellsMore data for this Ligand-Target Pair
TargetB2 bradykinin receptor(Homo sapiens (Human))
Novartis Institute For Medical Sciences
Curated by ChEMBL
Novartis Institute For Medical Sciences
Curated by ChEMBL
Affinity DataKi: 237nMAssay Description:Displacement of [3H]BK (1 nM) from human Bradykinin receptor B2 expressed in Cos-7 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 250nMAssay Description:Binding affinity for Bradykinin receptor B1 expressed in HEK293 cellsMore data for this Ligand-Target Pair
TargetB2 bradykinin receptor(Homo sapiens (Human))
Novartis Institute For Medical Sciences
Curated by ChEMBL
Novartis Institute For Medical Sciences
Curated by ChEMBL
Affinity DataKi: 253nMAssay Description:Displacement of [3H]BK (1 nM) from human Bradykinin receptor B2 expressed in Cos-7 cellsMore data for this Ligand-Target Pair
TargetB2 bradykinin receptor(Homo sapiens (Human))
Novartis Institute For Medical Sciences
Curated by ChEMBL
Novartis Institute For Medical Sciences
Curated by ChEMBL
Affinity DataKi: 299nMAssay Description:Displacement of [3H]BK (1 nM) from human Bradykinin receptor B2 expressed in Cos-7 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 310nMAssay Description:Inhibition of binding of [3H]-BK to rat bradykinin B2 receptor expressed in NG108-15 neuroblastoma-glioma hybrid cell membranesMore data for this Ligand-Target Pair
Affinity DataKi: 540nMAssay Description:Inhibition of binding of [3H]-BK to rat bradykinin B2 receptor expressed in NG108-15 neuroblastoma-glioma hybrid cell membranesMore data for this Ligand-Target Pair
TargetB2 bradykinin receptor(Homo sapiens (Human))
Novartis Institute For Medical Sciences
Curated by ChEMBL
Novartis Institute For Medical Sciences
Curated by ChEMBL
Affinity DataKi: 645nMAssay Description:Displacement of [3H]BK (1 nM) from human Bradykinin receptor B2 expressed in Cos-7 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 654nMAssay Description:Inhibition of specific binding of [3H]-BK (1 nM) to rat Bradykinin receptor B2 by 50% in NG108-15 cell membranesMore data for this Ligand-Target Pair
TargetB2 bradykinin receptor(Homo sapiens (Human))
Novartis Institute For Medical Sciences
Curated by ChEMBL
Novartis Institute For Medical Sciences
Curated by ChEMBL
Affinity DataKi: 772nMAssay Description:Displacement of [3H]BK (1 nM) from human Bradykinin receptor B2 expressed in Cos-7 cellsMore data for this Ligand-Target Pair
Affinity DataKi: >1.00E+3nMAssay Description:Binding affinity for Bradykinin receptor B1 expressed in HEK293 cellsMore data for this Ligand-Target Pair
TargetB2 bradykinin receptor(Homo sapiens (Human))
Novartis Institute For Medical Sciences
Curated by ChEMBL
Novartis Institute For Medical Sciences
Curated by ChEMBL
Affinity DataKi: 1.40E+3nMAssay Description:Binding affinity for Bradykinin receptor B2 expressed in COS7 cellsMore data for this Ligand-Target Pair
TargetB2 bradykinin receptor(Homo sapiens (Human))
Novartis Institute For Medical Sciences
Curated by ChEMBL
Novartis Institute For Medical Sciences
Curated by ChEMBL
Affinity DataKi: 1.43E+3nMAssay Description:Displacement of [3H]BK (1 nM) from human Bradykinin receptor B2 expressed in Cos-7 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 1.60E+3nMAssay Description:Inhibition of binding of [3H]-BK to rat bradykinin B2 receptor expressed in NG108-15 neuroblastoma-glioma hybrid cell membranesMore data for this Ligand-Target Pair
TargetAdenosine receptor A1(Homo sapiens (Human))
Novartis Institutes Of Biomedical Research
Curated by ChEMBL
Novartis Institutes Of Biomedical Research
Curated by ChEMBL
Affinity DataKi: 2.30E+3nMAssay Description:Inhibition of adenosine A1 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 3.00E+3nMAssay Description:Binding affinity for Bradykinin receptor B1 expressed in HEK293 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 7.10E+3nMAssay Description:Inhibition of binding of [3H]-BK to rat bradykinin B2 receptor expressed in NG108-15 neuroblastoma-glioma hybrid cell membranesMore data for this Ligand-Target Pair
TargetB2 bradykinin receptor(Homo sapiens (Human))
Novartis Institute For Medical Sciences
Curated by ChEMBL
Novartis Institute For Medical Sciences
Curated by ChEMBL
Affinity DataKi: 8.90E+3nMAssay Description:Binding affinity towards human bradykinin B2 receptor (membranes from Cos-7 cells expressing human B2 receptor) using [3H]-BK as radioligandMore data for this Ligand-Target Pair
TargetB2 bradykinin receptor(Homo sapiens (Human))
Novartis Institute For Medical Sciences
Curated by ChEMBL
Novartis Institute For Medical Sciences
Curated by ChEMBL
Affinity DataKi: 9.20E+3nMAssay Description:Binding affinity towards human bradykinin B2 receptor (membranes from Cos-7 cells expressing human B2 receptor) using [3H]-BK as radioligandMore data for this Ligand-Target Pair
TargetB2 bradykinin receptor(Homo sapiens (Human))
Novartis Institute For Medical Sciences
Curated by ChEMBL
Novartis Institute For Medical Sciences
Curated by ChEMBL
Affinity DataKi: 1.19E+4nMAssay Description:Binding affinity towards human bradykinin B2 receptor (membranes from Cos-7 cells expressing human B2 receptor) using [3H]-BK as radioligandMore data for this Ligand-Target Pair