Affinity DataKi: 0.320nMAssay Description:Displacement of [125I]-BH-JMV-179 from wild type human CCK1 receptor expressed in COS7 cells after 60 mins by gamma countingMore data for this Ligand-Target Pair
Affinity DataKi: 2.30nMAssay Description:Displacement of [125I]BH-(Thr,-Nle)-CCK-9 from human CCK1 receptor expressed in COS-7 cells after 60 mins by gamma countingMore data for this Ligand-Target Pair
Affinity DataKi: 3.90nMAssay Description:Displacement of [125I]BH-(Thr,-Nle)-CCK-9 from human CCK1 receptor expressed in COS-7 cells after 60 mins by gamma countingMore data for this Ligand-Target Pair
Affinity DataKi: 5.80nMAssay Description:Displacement of [3H]-SR-27897 from wild type human CCK1 receptor expressed in COS7 cells after 60 mins by gamma countingMore data for this Ligand-Target Pair
Affinity DataKi: 10.4nMAssay Description:Displacement of [125I]BH-(Thr,-Nle)-CCK-9 from human CCK1 receptor expressed in COS-7 cells after 60 mins by gamma countingMore data for this Ligand-Target Pair
Affinity DataKi: 59.8nMAssay Description:Displacement of [125I]BH-(Thr,-Nle)-CCK-9 from human CCK1 receptor expressed in COS-7 cells after 60 mins by gamma countingMore data for this Ligand-Target Pair
TargetGastrin/cholecystokinin type B receptor(Homo sapiens (Human))
University Of Trieste
Curated by ChEMBL
University Of Trieste
Curated by ChEMBL
Affinity DataKi: 169nMAssay Description:Displacement of [125I]BH-(Thr,-Nle)-CCK-9 from human CCK2 receptor expressed in COS-7 cells after 60 mins by gamma countingMore data for this Ligand-Target Pair
Affinity DataKi: 973nMAssay Description:Displacement of [125I]BH-(Thr,-Nle)-CCK-9 from human CCK1 receptor expressed in COS-7 cells after 60 mins by gamma countingMore data for this Ligand-Target Pair
TargetGastrin/cholecystokinin type B receptor(Homo sapiens (Human))
University Of Trieste
Curated by ChEMBL
University Of Trieste
Curated by ChEMBL
Affinity DataKi: 1.00E+3nMAssay Description:Displacement of [125I]BH-(Thr,-Nle)-CCK-9 from human CCK2 receptor expressed in COS-7 cells after 60 mins by gamma countingMore data for this Ligand-Target Pair
TargetGastrin/cholecystokinin type B receptor(Homo sapiens (Human))
University Of Trieste
Curated by ChEMBL
University Of Trieste
Curated by ChEMBL
Affinity DataKi: 1.00E+3nMAssay Description:Displacement of [125I]BH-(Thr,-Nle)-CCK-9 from human CCK2 receptor expressed in COS-7 cells after 60 mins by gamma countingMore data for this Ligand-Target Pair
TargetGastrin/cholecystokinin type B receptor(Homo sapiens (Human))
University Of Trieste
Curated by ChEMBL
University Of Trieste
Curated by ChEMBL
Affinity DataKi: 1.53E+4nMAssay Description:Displacement of [125I]BH-(Thr,-Nle)-CCK-9 from human CCK2 receptor expressed in COS-7 cells after 60 mins by gamma countingMore data for this Ligand-Target Pair
TargetGastrin/cholecystokinin type B receptor(Homo sapiens (Human))
University Of Trieste
Curated by ChEMBL
University Of Trieste
Curated by ChEMBL
Affinity DataKi: 2.20E+4nMAssay Description:Displacement of [125I]BH-(Thr,-Nle)-CCK-9 from human CCK2 receptor expressed in COS-7 cells after 60 mins by gamma countingMore data for this Ligand-Target Pair
Affinity DataIC50: 0.0900nMAssay Description:Inhibition of 71 pM [125I]BH-(Thr,Nle)CCK-9 binding to rat cholecystokinin 1 receptorMore data for this Ligand-Target Pair
Affinity DataIC50: 0.0900nMAssay Description:Inhibition of 71 pM [125I]BH-(Thr,Nle)CCK-9 binding to rat cholecystokinin 1 receptorMore data for this Ligand-Target Pair
Affinity DataIC50: 0.590nMAssay Description:Inhibition of 71 pM [125I]BH-(Thr,Nle)CCK-9 binding to rat cholecystokinin 1 receptorMore data for this Ligand-Target Pair
Affinity DataIC50: 0.590nMAssay Description:Inhibition of 71 pM [125I]BH-(Thr,Nle)CCK-9 binding to rat cholecystokinin 1 receptorMore data for this Ligand-Target Pair
Affinity DataIC50: 1.59nMAssay Description:Inhibition of 71 pM [125I]BH-(Thr,Nle)CCK-9 binding to rat cholecystokinin 1 receptorMore data for this Ligand-Target Pair
Affinity DataIC50: 2.10nMAssay Description:Inhibition of CCK binding to Cos-7 cells expressing human cholecystokinin 1 receptorMore data for this Ligand-Target Pair
Affinity DataIC50: 3.60nMAssay Description:Inhibition of CCK-Induced inositol phosphate in Cos-7 cells expressing mutant CCK1R (S348A)More data for this Ligand-Target Pair
Affinity DataIC50: 3.80nMAssay Description:Inhibition of CCK binding to Cos-7 cells expressing human cholecystokinin 1 receptorMore data for this Ligand-Target Pair
Affinity DataIC50: 5.20nMAssay Description:Inhibition of CCK-Induced inositol phosphate in Cos-7 cells expressing mutant CCK1R (M195L)More data for this Ligand-Target Pair
Affinity DataIC50: 5.20nMAssay Description:Inhibition of CCK binding to Cos-7 cells expressing human cholecystokinin 1 receptorMore data for this Ligand-Target Pair
Affinity DataIC50: 5.70nMAssay Description:Inhibition of CCK-Induced inositol phosphate in Cos-7 cells expressing mutant CCK1R (S348A)More data for this Ligand-Target Pair
Affinity DataIC50: 5.80nMAssay Description:Inhibition of CCK-Induced inositol phosphate in Cos-7 cells expressing mutant CCK1R (M195L)More data for this Ligand-Target Pair
Affinity DataIC50: 7.30nMAssay Description:Inhibition of CCK-Induced inositol phosphate production in Cos-7 cells expressing human CCK1RMore data for this Ligand-Target Pair
Affinity DataIC50: 7.90nMAssay Description:Inhibition of CCK-Induced inositol phosphate in Cos-7 cells expressing mutant CCK1R (S342A)More data for this Ligand-Target Pair
Affinity DataIC50: 8.80nMAssay Description:Inhibition of CCK-Induced inositol phosphate production in Cos-7 cells expressing human CCK1RMore data for this Ligand-Target Pair
Affinity DataIC50: 8.90nMAssay Description:Inhibition of CCK-Induced inositol phosphate in Cos-7 cells expressing mutant CCK1R (R197M)More data for this Ligand-Target Pair
Affinity DataIC50: 9.30nMAssay Description:Inhibition of CCK-induced inositol phosphate in Cos-7 cells expressing mutant CCK1R (I329A)More data for this Ligand-Target Pair
Affinity DataIC50: 9.5nMAssay Description:Displacement of [125I]-BH-CCK8 from CCK1 receptor in Sprague-Dawley rat pancreatic acini after 120 hrs by gamma-countingMore data for this Ligand-Target Pair
Affinity DataIC50: 11.8nMAssay Description:Inhibition of CCK-Induced inositol phosphate in Cos-7 cells expressing mutant CCK1R (R197M)More data for this Ligand-Target Pair
Affinity DataIC50: 15.7nMAssay Description:Displacement of [125I]-BH-CCK8 from CCK1 receptor in Sprague-Dawley rat pancreatic acini after 120 hrs by gamma-countingMore data for this Ligand-Target Pair
Affinity DataIC50: 23nMAssay Description:Inhibition of CCK-Induced inositol phosphate in Cos-7 cells expressing mutant CCK1R (R197M)More data for this Ligand-Target Pair
Affinity DataIC50: 23.3nMAssay Description:Inhibition of CCK-induced inositol phosphate in Cos-7 cells expressing mutant CCK1R (F107A)More data for this Ligand-Target Pair
Affinity DataIC50: 24.9nMAssay Description:Inhibition of CCK-Induced inositol phosphate in Cos-7 cells expressing mutant CCK1R (T117A)More data for this Ligand-Target Pair
Affinity DataIC50: 26.8nMAssay Description:Inhibition of CCK-induced inositol phosphate in Cos-7 cells expressing mutant CCK1R (F107A)More data for this Ligand-Target Pair
Affinity DataIC50: 27.5nMAssay Description:Inhibition of CCK-Induced inositol phosphate in Cos-7 cells expressing mutant CCK1R (S342A)More data for this Ligand-Target Pair
Affinity DataIC50: 28.4nMAssay Description:Inhibition of CCK-Induced inositol phosphate in Cos-7 cells expressing mutant CCK1R (T117A)More data for this Ligand-Target Pair
Affinity DataIC50: 31.5nMAssay Description:Inhibition of CCK-induced inositol phosphate in Cos-7 cells expressing mutant CCK1R (F107A)More data for this Ligand-Target Pair
Affinity DataIC50: 33.2nMAssay Description:Inhibition of CCK-Induced inositol phosphate in Cos-7 cells expressing mutant CCK1R (S342A)More data for this Ligand-Target Pair
Affinity DataIC50: 35.2nMAssay Description:Inhibition of CCK-Induced inositol phosphate production in Cos-7 cells expressing human CCK1RMore data for this Ligand-Target Pair
Affinity DataIC50: 35.2nMAssay Description:Inhibition of CCK-Induced inositol phosphate in Cos-7 cells expressing mutant CCK1R (M195L)More data for this Ligand-Target Pair
Affinity DataIC50: 36.6nMAssay Description:Inhibition of CCK-Induced inositol phosphate in Cos-7 cells expressing mutant CCK1R (S348A)More data for this Ligand-Target Pair
Affinity DataIC50: 71.6nMAssay Description:Inhibition of CCK-Induced inositol phosphate in Cos-7 cells expressing mutant CCK1R (T117A)More data for this Ligand-Target Pair
Affinity DataIC50: 107nMAssay Description:Displacement of [125I]-BH-CCK8 from CCK1 receptor in Sprague-Dawley rat pancreatic acini after 120 hrs by gamma-countingMore data for this Ligand-Target Pair
Affinity DataIC50: 129nMAssay Description:Inhibition of CCK-induced inositol phosphate in Cos-7 cells expressing mutant CCK1R (I329A)More data for this Ligand-Target Pair
Affinity DataIC50: 183nMAssay Description:Inhibition of CCK-Induced inositol phosphate in Cos-7 cells expressing mutant CCK1R (I329F)More data for this Ligand-Target Pair
Affinity DataIC50: 197nMAssay Description:Displacement of [125I]-BH-CCK8 from CCK1 receptor in Sprague-Dawley rat pancreatic acini after 120 hrs by gamma-countingMore data for this Ligand-Target Pair
Affinity DataIC50: 227nMAssay Description:Inhibition of CCK-Induced inositol phosphate in Cos-7 cells expressing mutant CCK1R (I352A)More data for this Ligand-Target Pair
Affinity DataIC50: 313nMAssay Description:Displacement of [125I]-BH-CCK8 from CCK1 receptor in Sprague-Dawley rat pancreatic acini after 120 hrs by gamma-countingMore data for this Ligand-Target Pair